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公开(公告)号:US09127004B2
公开(公告)日:2015-09-08
申请号:US14298182
申请日:2014-06-06
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dhond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dhond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: C07D487/00 , A61K31/44 , C07D471/08 , A61K31/424 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , C07D519/00 , C07D498/04
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
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2.1,6-Diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US20140088068A1
公开(公告)日:2014-03-27
申请号:US14113980
申请日:2012-08-24
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: C07D471/08 , A61K31/43 , A61K31/424 , A61K31/496 , A61K31/439 , C07D519/00 , A61K31/5383 , A61K31/5377 , A61K31/4545 , A61K31/546
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
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3.1,6-diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US09006230B2
公开(公告)日:2015-04-14
申请号:US14113980
申请日:2012-08-24
申请人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
发明人: Sachin Bhagwat , Prasad Keshav Deshpande , Satish Bhawsar , Vijaykumar Jagdishwar Patil , Ravikumar Tadiparthi , Shivaji Sampatrao Pawar , Sunil Bhaginath Jadhav , Sanjay Kisan Dabhade , Vikas Vitthalrao Deshmukh , Bharat Dond , Satish Birajdar , Mohammad Usman Shaikh , Deepak Dekhane , Piyush Ambalal Patel
IPC分类号: A61K31/00 , C07D233/10 , C07D243/00 , C07D471/08 , A61K31/424 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , C07D519/00 , C07D498/04
CPC分类号: C07D471/08 , A61K31/424 , A61K31/43 , A61K31/431 , A61K31/439 , A61K31/4545 , A61K31/46 , A61K31/496 , A61K31/5377 , A61K31/5383 , A61K31/546 , A61K45/06 , C07D498/04 , C07D519/00 , A61K2300/00
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed.
摘要翻译: 公开了式(I)化合物及其制备和用于预防或治疗细菌感染的方法。
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4.1,6-diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US08822450B2
公开(公告)日:2014-09-02
申请号:US14111592
申请日:2012-08-24
申请人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawsar , Sachin Bhagwat , Mohammed Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
发明人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawsar , Sachin Bhagwat , Mohammed Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
IPC分类号: C07D471/08 , A61K31/542 , A61K31/529 , A61K31/429 , A61K45/06 , A61K31/407 , A61K31/496 , A61K31/167 , A61K31/427
CPC分类号: A61K31/5377 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/529 , A61K31/542 , A61K31/546 , A61K45/06 , C07D471/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infection is disclosed.
摘要翻译: 公开了式(I)化合物,其制备和用于预防或治疗细菌感染。
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5.1,6- Diazabicyclo [3,2,1] octan-7-one derivatives and their use in the treatment of bacterial infections 有权
标题翻译: 1,6-二氮杂双环[3,2,1]辛-7-酮衍生物及其在细菌感染治疗中的应用公开(公告)号:US20140148431A1
公开(公告)日:2014-05-29
申请号:US14111592
申请日:2012-08-24
申请人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawsar , Sachin Bhagwat , Mohammed Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
发明人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawsar , Sachin Bhagwat , Mohammed Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
IPC分类号: A61K31/542 , A61K31/529 , A61K31/429 , A61K45/06 , A61K31/407 , A61K31/496 , A61K31/167 , C07D471/08 , A61K31/427
CPC分类号: A61K31/5377 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/529 , A61K31/542 , A61K31/546 , A61K45/06 , C07D471/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infection is disclosed.
摘要翻译: 公开了式(I)化合物,其制备和用于预防或治疗细菌感染。
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公开(公告)号:US08217058B2
公开(公告)日:2012-07-10
申请号:US12225744
申请日:2007-05-08
申请人: Mahesh Vithalbhai Patel , Mahesh Phansalkar , Vijaykumar Jagdishwar Patil , Milind Dattatraya Sindkhedkar , Prasad Keshav Deshpande
发明人: Mahesh Vithalbhai Patel , Mahesh Phansalkar , Vijaykumar Jagdishwar Patil , Milind Dattatraya Sindkhedkar , Prasad Keshav Deshpande
IPC分类号: A61K31/445 , C07D413/10
CPC分类号: C07D413/10 , A23K20/137
摘要: The present invention relates to certain substituted piperidino phenyloxazolidinones. Specifically, the invention relates to geminally disubstituted piperidino phenyloxazolidinones having antimicrobial activity with improved pharmacokinetic profile. The invention also relates to processes for the preparation of compounds of the present invention, pharmaceutical compositions containing the compounds of the present invention and the methods for treating or preventing microbial infections using the compounds of the present invention.
摘要翻译: 本发明涉及某些取代的哌啶子基苯基恶唑烷酮。 具体地,本发明涉及具有改善的药代动力学特征的具有抗微生物活性的双重取代的哌啶子基苯基恶唑烷酮。 本发明还涉及制备本发明化合物的方法,含有本发明化合物的药物组合物以及使用本发明化合物治疗或预防微生物感染的方法。
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公开(公告)号:US20100056581A1
公开(公告)日:2010-03-04
申请号:US12225744
申请日:2007-05-08
申请人: Mahesh Vithalbhai Patel , Mahesh Phansalkar , Vijaykumar Jagdishwar Patil , Milind Dattatraya Sindkhedkar , Prasad Keshav Deshpande
发明人: Mahesh Vithalbhai Patel , Mahesh Phansalkar , Vijaykumar Jagdishwar Patil , Milind Dattatraya Sindkhedkar , Prasad Keshav Deshpande
IPC分类号: A61K31/437 , C07D413/10 , A61P31/00 , A61P31/04
CPC分类号: C07D413/10 , A23K20/137
摘要: The present invention relates to certain substituted piperidino phenyloxazolidinones. Specifically, the invention relates to geminally disubstituted piperidino phenyloxazolidinones having antimicrobial activity with improved pharmacokinetic profile. The invention also relates to processes for the preparation of compounds of the present invention, pharmaceutical compositions containing the compounds of the present invention and the methods for treating or preventing microbial infections using the compounds of the present invention.
摘要翻译: 本发明涉及某些取代的哌啶子基苯基恶唑烷酮。 具体地,本发明涉及具有改善的药代动力学特征的具有抗微生物活性的双重取代的哌啶子基苯基恶唑烷酮。 本发明还涉及制备本发明化合物的方法,含有本发明化合物的药物组合物以及使用本发明化合物治疗或预防微生物感染的方法。
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公开(公告)号:US08987297B2
公开(公告)日:2015-03-24
申请号:US14452652
申请日:2014-08-06
申请人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
发明人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
IPC分类号: A61K31/439 , A61K31/407 , A61K31/167 , C07D471/08 , A61K31/427 , A61K31/429 , A61K31/496 , A61K31/529 , A61K31/542 , A61K45/06
CPC分类号: A61K31/5377 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/529 , A61K31/542 , A61K31/546 , A61K45/06 , C07D471/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infection is disclosed.
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公开(公告)号:US09132133B2
公开(公告)日:2015-09-15
申请号:US14609704
申请日:2015-01-30
申请人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
发明人: Mahesh Vithalbhai Patel , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
IPC分类号: A61K31/439 , A61K31/5377 , C07D471/08 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/496 , A61K31/529 , A61K31/542 , A61K45/06 , A61K31/43 , A61K31/546
CPC分类号: A61K31/5377 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/529 , A61K31/542 , A61K31/546 , A61K45/06 , C07D471/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infection is disclosed.
摘要翻译: 公开了式(I)化合物,其制备和用于预防或治疗细菌感染。
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公开(公告)号:US20150174133A1
公开(公告)日:2015-06-25
申请号:US14609704
申请日:2015-01-30
申请人: Mahesh Vithalbhai PATEL , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
发明人: Mahesh Vithalbhai PATEL , Prasad Keshav Deshpande , Satish Bhawasar , Sachin Bhagwat , Mohammad Alam Jafri , Amit Mishra , Laxmikant Pavase , Sunil Gupta , Rajesh Kale , Sanjeev Joshi
IPC分类号: A61K31/5377 , A61K31/496 , A61K31/43 , A61K31/427 , A61K31/407 , A61K31/439 , A61K31/546
CPC分类号: A61K31/5377 , A61K31/167 , A61K31/407 , A61K31/427 , A61K31/429 , A61K31/43 , A61K31/439 , A61K31/4545 , A61K31/496 , A61K31/529 , A61K31/542 , A61K31/546 , A61K45/06 , C07D471/08
摘要: Compounds of Formula (I), their preparation and use in preventing or treating bacterial infection is disclosed.
摘要翻译: 公开了式(I)化合物,其制备和用于预防或治疗细菌感染。
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