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1.INHIBITION OF P38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS 审中-公开
标题翻译: 使用对称和非对称二苯醚类尿素抑制P38激酶公开(公告)号:US20120270878A1
公开(公告)日:2012-10-25
申请号:US13539914
申请日:2012-07-02
申请人: Scott MILLER , Martin OSTERHOUT , Jacques DUMAS , Uday KHIRE , Timothy B. LOWINGER , William J. SCOTT , Roger A. SMITH , Jill E. WOOD , David E. GUNN , Holia HATOUM-MOKDAD , Marell RODRIGUEZ , Robert SIBLEY , Ming WANG , Tiffany TURNER , Catherine BRENNAN
发明人: Scott MILLER , Martin OSTERHOUT , Jacques DUMAS , Uday KHIRE , Timothy B. LOWINGER , William J. SCOTT , Roger A. SMITH , Jill E. WOOD , David E. GUNN , Holia HATOUM-MOKDAD , Marell RODRIGUEZ , Robert SIBLEY , Ming WANG , Tiffany TURNER , Catherine BRENNAN
IPC分类号: A61K31/17 , A61K31/4436 , A61K31/4409 , A61K31/428 , A61P41/00 , A61P29/00 , A61P19/02 , A61P19/10 , A61P11/00 , A61P1/00 , A61K31/5375 , A61K31/403
CPC分类号: A61K31/17 , A61K31/341 , A61K31/381 , A61K31/4035 , A61K31/44 , A61K31/5375 , Y02A50/411
摘要: This invention relates to the use of a group of aryl ureas in treating cytokine mediated diseases and proteolytic enzyme mediated diseases, and pharmaceutical compositions for use in such therapy.
摘要翻译: 本发明涉及一组芳基脲在治疗细胞因子介导的疾病和蛋白水解酶介导的疾病中的用途,以及用于这种治疗的药物组合物。
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2.INHIBITION OF P38 KINASE ACTIVITY USING SUBSTITUTED HETEROCYCLIC UREAS 审中-公开
标题翻译: 使用取代的杂环类抗生素抑制P38激酶活性公开(公告)号:US20120149706A1
公开(公告)日:2012-06-14
申请号:US13401272
申请日:2012-02-21
申请人: Jacques DUMAS , Uday KHIRE , Timothy B. Lowinger , Holger PAULSEN , Bernd RIEDL , Willian J. SCOTT , Roger A. SMITH , Jill WOOD , Holia HATOUM-MOKDAD , Wendy LEE , Aniko REDMAN , Jeffrey JOHNSON , Robert SIBLEY
发明人: Jacques DUMAS , Uday KHIRE , Timothy B. Lowinger , Holger PAULSEN , Bernd RIEDL , Willian J. SCOTT , Roger A. SMITH , Jill WOOD , Holia HATOUM-MOKDAD , Wendy LEE , Aniko REDMAN , Jeffrey JOHNSON , Robert SIBLEY
IPC分类号: A61K31/42 , C07D413/12 , A61K31/4439 , A61K31/497 , A61K31/506 , A61P37/06 , A61P29/00 , A61P37/02 , A61P19/10 , A61P19/02 , A61P11/06 , A61P1/00 , C07D261/14 , A61K31/5377
CPC分类号: C07D231/40 , A61K31/381 , A61K31/415 , A61K31/4155 , A61K31/416 , A61K31/42 , A61K31/421 , A61K31/422 , A61K31/426 , A61K31/428 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4709 , A61K31/506 , C07D261/14 , Y02A50/411
摘要: This invention relates to the use of a group of aryl ureas in treating cytokine mediated diseases, other than cancer and proteolytic enzyme mediated diseases, other than cancer, and pharmaceutical compositions for use in such therapy.
摘要翻译: 本发明涉及一组芳基脲处理细胞因子介导的疾病,除了癌症以外的癌症和蛋白水解酶介导的疾病,以及用于这种治疗的药物组合物。
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3.BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES USEFUL IN THE TREATMENT OF HYPER-PROLIFERATIVE DISORDERS 失效
标题翻译: 用于治疗高血压疾病的苯并呋喃和苯并噻吩衍生物公开(公告)号:US20090054514A1
公开(公告)日:2009-02-26
申请号:US12059984
申请日:2008-03-31
申请人: Chengzhi ZHANG , Michael BURKE , Zhi CHEN , Jacques DUMAS , Dongping FAN , Jianmei FAN , Holia HATOUM-MOKDAD , Benjamin JONES , Gaetan LADOUCEUR , Wendy LEE , Barton PHILLIPS
发明人: Chengzhi ZHANG , Michael BURKE , Zhi CHEN , Jacques DUMAS , Dongping FAN , Jianmei FAN , Holia HATOUM-MOKDAD , Benjamin JONES , Gaetan LADOUCEUR , Wendy LEE , Barton PHILLIPS
IPC分类号: A61K31/381 , C07D307/82 , A61K31/343 , A61P35/00 , C07D333/66
CPC分类号: C07D307/82 , C07D307/92 , C07D307/93 , C07D333/66 , C07D333/74 , C07D333/78 , C07D405/04 , C07D405/06 , C07D405/10 , C07D405/14 , C07D407/06 , C07D409/04 , C07D409/14 , C07D413/04 , C07D413/06 , C07D417/04 , C07D417/06 , C07D493/04
摘要: This invention relates to novel benzofuran and benzothiophene derivatives of the general formula and their use for the treatment of hyper-proliferative disorders.
摘要翻译: 本发明涉及通式的新型苯并呋喃和苯并噻吩衍生物及其用于治疗高增殖性疾病的用途。
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