公开(公告)号：US06458748B1

公开(公告)日：2002-10-01

申请号：US09744209

申请日：2001-01-22

申请人： Takumi Yoshimura ,  Masao Nakatani ,  Masatoshi Tamaru ,  Takeshi Danjo ,  Yukimasa Ono ,  Katsutada Yanagisawa

发明人： Takumi Yoshimura ,  Masao Nakatani ,  Masatoshi Tamaru ,  Takeshi Danjo ,  Yukimasa Ono ,  Katsutada Yanagisawa

IPC分类号： C07D23952

CPC分类号： A01N43/54 ,  A01N47/02 ,  C07D239/52

摘要： The present invention provides a novel compound which is effective for the removal of a wide variety of weeds including difficult-to-control weeds emerging in paddy field and which is safe to mammals; a process for production thereof; a herbicide containing the compound as an active ingredient; and novel raw material compounds used in said process. The present invention relates to a di- or trifluoromethanesulfonyl anilide derivative represented by the following general formula: (wherein R1 is a hydrogen atom, an alkyl group or an alkoxyalkyl group; and R2 is a hydrogen atom when R1 is a hydrogen atom or an alkyl group, and is a hydrogen atom or a fluorine atom when R1 is an alkoxyalkyl group), or a salt thereof, both of said derivative and said salt having a herbicidal activity.

摘要翻译： 本发明提供了一种新颖的化合物，其有效去除各种杂草，包括难以控制的稻田中出现的杂草，对哺乳动物是安全的; 其生产方法; 含有该化合物作为活性成分的除草剂; 和所述方法中使用的新型原料化合物。本发明涉及由以下通式表示的二 - 或三氟甲磺酰苯胺衍生物：其中R1是氢原子，烷基或烷氧基烷基; R2是氢 当R 1为氢原子或烷基时为原子，当R 1为烷氧基烷基时为氢原子或氟原子）或其盐，所述衍生物和所述盐都具有除草活性。

公开(公告)号：US06841519B1

公开(公告)日：2005-01-11

申请号：US10049039

申请日：2000-08-09

申请人： Masao Nakatani ,  Kouichirou Kaku ,  Takumi Yoshimura ,  Masatoshi Tamaru ,  Hiroshi Kawasaki ,  Kazunori Kobayashi ,  Takeshige Miyazawa

发明人： Masao Nakatani ,  Kouichirou Kaku ,  Takumi Yoshimura ,  Masatoshi Tamaru ,  Hiroshi Kawasaki ,  Kazunori Kobayashi ,  Takeshige Miyazawa

IPC分类号： A01N43/80 ,  A01P13/00 ,  C07D261/04 ,  C07D261/20

CPC分类号： A01N43/80 ,  C07D261/04 ,  C07D261/20

摘要： The isoxazoline derivative of the present invention is represented by the following general formula [I]: [wherein Q is a group represented by —S(O)n—(CR5R6)m- (wherein n is an integer of 0 to 2, m is an integer of 1 to 3, and R5 and R6 are a hydrogen atom, a cyano group, an alkoxycarbonyl group, if an alkyl group or the like); R1 and R2 are a hydrogen atom, all optionally substituted alkyl group, an alkoxycarbonyl group, an optionally substituted phenyl group or the like; R3 and R4 are a hydrogen atom, an optionally substituted alkyl group, a cycloalkyl group or the like; Y is a hydrogen atom, an alkoxycarbonyl group, a carboxyl group, an alkenyl group, an optionally substituted alkyl group or an optionally substituted phenyl group]. The herbicide of the present invention contains the above isoxazoline derivative as the active ingredient.

摘要翻译： 本发明的异恶唑啉衍生物由以下通式[I]表示：[其中Q为-S（O）n - （CR 5 R 6）m - （其中n为0〜2的整数，m 为1〜3的整数，R5，R6为氢原子，氰基，烷氧基羰基，烷基等）。 R1和R2是氢原子，全部任选取代的烷基，烷氧基羰基，任意取代的苯基等; R3和R4是氢原子，任选取代的烷基，环烷基等; Y是氢原子，烷氧基羰基，羧基，烯基，任意取代的烷基或任意取代的苯基]。 本发明的除草剂含有上述异恶唑啉衍生物作为有效成分。

公开(公告)号：US20120131718A1

公开(公告)日：2012-05-31

申请号：US13148449

申请日：2010-02-08

申请人： Mitsuya Uchida ,  Osamu Tanaka ,  Kiyoshi Fukaya ,  Takumi Yoshimura ,  Toshiyo Tamura ,  Yukitoshi Takahashi

发明人： Mitsuya Uchida ,  Osamu Tanaka ,  Kiyoshi Fukaya ,  Takumi Yoshimura ,  Toshiyo Tamura ,  Yukitoshi Takahashi

IPC分类号： A41D1/00 ,  A41F19/00

CPC分类号： A62B99/00 ,  A41D13/018

摘要： An airbag device for the body instantaneously activates an airbag without malfunctions.When an absolute value of an angular velocity detected by an angular velocity sensor exceeds a predetermined angular velocity value, angular velocity values are integrated from a most recent detected value to an oldest value within a predetermined time period, and if an absolute value of a resultant value of integral exceeds a predetermined value and an acceleration detected by an acceleration sensor is smaller than a predetermined acceleration, the airbag is inflated. Based on the value of the integral of the angular velocities, a case in which an angular velocity gradually increases is distinguished from a case in which an angular velocity momentarily increases, so the airbag device effectively prevents malfunctions caused by an action other than falling over. Additionally, because it is unnecessary to intentionally delay determination to prevent malfunctions, the airbag can instantaneously be inflated.

摘要翻译： 用于身体的安全气囊装置瞬间激活安全气囊而不发生故障。 当由角速度传感器检测到的角速度的绝对值超过预定的角速度值时，角速度值在预定时间段内从最近的检测值积分到最老的值，并且如果得到的绝对值 积分值超过预定值，并且由加速度传感器检测到的加速度小于预定加速度时，气囊膨胀。 基于角速度的积分值，角速度逐渐增加的情况与角速度瞬时增加的情况不同，因此安全气囊装置有效地防止除掉落以外的动作引起的故障。 此外，由于不必有意地延迟确定以防止故障，所以气囊可以瞬间膨胀。

公开(公告)号：US5527763A

公开(公告)日：1996-06-18

申请号：US107716

申请日：1993-12-08

申请人： Masahiro Miyazaki ,  Masafumi Matsuzawa ,  Takumi Yoshimura ,  Kuniaki Shimizu ,  Shigehiko Tachikawa

发明人： Masahiro Miyazaki ,  Masafumi Matsuzawa ,  Takumi Yoshimura ,  Kuniaki Shimizu ,  Shigehiko Tachikawa

IPC分类号： A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/647 ,  A01N43/66 ,  A01N43/707 ,  A01N43/74 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D239/54 ,  C07D239/545 ,  C07D239/553 ,  C07D239/60 ,  C07D401/12 ,  C07D403/12 ,  C07D403/14 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00 ,  C07F7/10 ,  C07D239/32

CPC分类号： C07D239/54 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/66 ,  A01N43/707 ,  A01N43/74 ,  A01N43/80 ,  C07D231/12 ,  C07D233/56 ,  C07D239/545 ,  C07D239/553 ,  C07D239/60 ,  C07D249/08 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/12

摘要： A herbicide containing a pyrimidine or triazine derivative of the formula (I): ##STR1## [wherein A is a furan ring, a pyrimidine ring, a 1,2,4-triazine ring or the like which may suitably be substituted, R is a hydroxyl group or a lower alkoxy group, each of R.sup.1 and R.sup.2 which may be the same or different, is a halogen atom, a lower alkyl group or a lower alkoxy group, W is an oxygen atom or a sulfur atom, and Z is nitrogen or a methine group] and its salt, as an active ingredient, is presented. The pyrimidine or triazine derivative of the present invention has excellent herbicidal effects against noxious weeds in paddy fields, upland fields and non-agricultural fields.

摘要翻译： PCT No.PCT / JP92 / 01690 Sec。 371日期1993年12月8日第 102（e）日期1993年12月8日PCT提交1992年12月24日PCT公布。 公开号WO93 / 13078 日本时间：1993年7月8日。含有式（I）的嘧啶或三嗪衍生物的除草剂：其中A是呋喃环，嘧啶环，1,2,4-三嗪环或 R可以相同或不同，R为羟基或低级烷氧基的卤素原子，低级烷基或低级烷氧基，W为 氧原子或硫原子，Z为氮或次甲基]，其盐作为活性成分。 本发明的嘧啶或三嗪衍生物对稻田，旱田和非农田中的有害杂草具有优异的除草效果。

公开(公告)号：US5536837A

公开(公告)日：1996-07-16

申请号：US443766

申请日：1995-05-18

申请人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihisa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

发明人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihisa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

IPC分类号： A01N43/54 ,  A01N43/66 ,  A01P3/00 ,  A01P13/00 ,  C07D239/28 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  C07D239/52 ,  C07D251/20 ,  C07D239/26 ,  C07D403/12

CPC分类号： C07D239/28 ,  A01N43/54 ,  A01N43/66 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/47 ,  C07D239/52 ,  C07D251/20

摘要： The present invention provides an N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring represented by formula [I]: ##STR1## wherein R.sup.1 represents an alkyl group, an alkenyl group, or the like, R.sup.2 represents a hydrogen atom, an alkyl group, or the like, R.sup.3 and R.sup.4 represent independently an alkyl group, alkoxy group, or the like, and X and Y represent independently a methyne group or a nitrogen atom; or the salt of the same, a method for producing the same, and a biocide containing the same as an active ingredient. The N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring according to the present invention exhibits superior effects against blight caused by plant pathogenic fungi belonging to Oomycetes such as downy mildew, late blight, or the like in a low concentration as well as controls weeds occurring in paddy fields and plowed fields.

摘要翻译： 本发明提供了包括由式[I]表示的含N 6芳香环的N-磺酰基羧酰胺衍生物：其中R 1表示烷基，烯基等，R 2 代表氢原子，烷基等，R3和R4独立地表示烷基，烷氧基等，X和Y独立地表示甲炔基或氮原子; 或其盐，其制备方法，以及含有活性成分的杀生物剂。 包含根据本发明的含有N元素的6元芳环的N-磺酰基羧酰胺衍生物对低浓度的属于卵菌属的霉菌属如霜霉病，晚疫病等的植物致病真菌具有优异的抗枯萎作用 以及控制稻田和耕地中发生的杂草。

公开(公告)号：US5444060A

公开(公告)日：1995-08-22

申请号：US137190

申请日：1993-11-02

申请人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihasa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

发明人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihasa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

IPC分类号： A01N43/54 ,  A01N43/66 ,  A01P3/00 ,  A01P13/00 ,  C07D239/28 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  C07D239/52 ,  C07D251/20 ,  C07D239/26 ,  C07D401/12

CPC分类号： C07D239/28 ,  A01N43/54 ,  A01N43/66 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/47 ,  C07D239/52 ,  C07D251/20

摘要： The present invention provides an N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring represented by formula [I]: ##STR1## wherein R.sup.1 represents an alkyl group, an alkenyl group, or the like, R.sup.2 represents a hydrogen atom, an alkyl group, or the like, R.sup.3 and R.sup.4 represent independently an alkyl group, alkoxy group, or the like, and X and Y represent independently a methyne group or a nitrogen atom; or the salt of the same, a method for producing the same, and a biocide containing the same as an active ingredient. The N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring according to the present invention exhibits superior effects against blight caused by plant pathogenic fungi belonging to Oomycetes such as downy mildew, late blight, or the like in a low concentration as well as controls weeds occurring in paddy fields and plowed fields.

摘要翻译： PCT No.PCT / JP93 / 00273 Sec。 371日期：1993年11月2日 102（e）1993年11月2日PCT PCT 1993年3月3日PCT公布。 公开号WO93 / 1801200 日本1993年9月16日。本发明提供了包含式[I]表示的含N 6芳香环的N-磺酰基羧酰胺衍生物：其中R 1表示烷基， 基团等，R 2表示氢原子，烷基等，R 3和R 4分别独立地表示烷基，烷氧基等，X和Y分别独立地表示甲炔基或氮原子; 或其盐，其制备方法，以及含有活性成分的杀生物剂。 包含根据本发明的含有N元素的6元芳环的N-磺酰基羧酰胺衍生物对低浓度的属于卵菌属的霉菌属如霜霉病，晚疫病等的植物致病真菌具有优异的抗枯萎作用 以及控制稻田和耕地中发生的杂草。

公开(公告)号：US5411934A

公开(公告)日：1995-05-02

申请号：US916127

申请日：1992-07-30

申请人： Takumi Yoshimura ,  Keiji Toriyabe ,  Katsumi Masuda ,  Ryo Hanai

发明人： Takumi Yoshimura ,  Keiji Toriyabe ,  Katsumi Masuda ,  Ryo Hanai

IPC分类号： C07D239/46 ,  A01N43/54 ,  A01N43/66 ,  A01P13/00 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/52 ,  C07D239/54 ,  C07D405/12 ,  C07D409/12 ,  C07F7/08 ,  C07D239/42

CPC分类号： C07D239/26 ,  A01N43/54 ,  A01N43/66 ,  C07D239/34 ,  C07D239/47 ,  C07D239/52 ,  C07D405/12 ,  C07D409/12 ,  C07F7/0812

摘要： The present invention provides a novel alkanoic acid amide derivative of the formula, ##STR1## (wherein R.sup.1 is a hydrogen atom, an alkyl group or an alkoxyalkoxy group, R.sup.2 is a group of -SO.sub.2 R or a hydroxyl group, R.sup.5 is an alkyl group, R.sup.3 is an alkyl group, a cycloalkyl group, a cycloalkenyl group or a phenyl group, R.sup.4 is a hydrogen atom or an alkyl group, X and Y may be the same or different and are an alkoxy group, an alkylamino group or a dialkylamino group, and Z is a methine group or a nitrogen atom) and its salt, a process for preparing the same and a herbicidal composition containing the same as an effective ingredient.This compound kills annual and perennial weeds grown in paddy fields and upland fields at a small dose, and is safe to a useful crop plant.

摘要翻译： PCT No.PCT / JP91 / 01649 Sec。 371日期：1992年7月30日 102（e）日期1992年7月30日PCT 1991年11月29日PCT PCT。 第WO92 / 09584号公报 日本1992年6月19日。本发明提供了下式的新型链烷酰胺衍生物，其中R1是氢原子，烷基或烷氧基烷氧基，R2是-SO2R基团 或羟基，R5是烷基，R3是烷基，环烷基，环烯基或苯基，R4是氢原子或烷基，X和Y可以相同或不同，并且是 烷氧基，烷基氨基或二烷基氨基，Z为次甲基或氮原子）及其盐，其制备方法和含有该有机组合物的除草组合物。 这种化合物以小剂量杀死在稻田和高地田间种植的一年生和多年生杂草，对于有用的作物植物是安全的。

公开(公告)号：US09126065B2

公开(公告)日：2015-09-08

申请号：US13148449

申请日：2010-02-08

申请人： Mitsuya Uchida ,  Osamu Tanaka ,  Kiyoshi Fukaya ,  Takumi Yoshimura ,  Toshiyo Tamura ,  Yukitoshi Takahashi

发明人： Mitsuya Uchida ,  Osamu Tanaka ,  Kiyoshi Fukaya ,  Takumi Yoshimura ,  Toshiyo Tamura ,  Yukitoshi Takahashi

IPC分类号： A41D1/02 ,  A62B99/00 ,  A41D13/018

CPC分类号： A62B99/00 ,  A41D13/018

摘要： An airbag device for the body instantaneously activates an airbag without malfunctions.When an absolute value of an angular velocity detected by an angular velocity sensor exceeds a predetermined angular velocity value, angular velocity values are integrated from a most recent detected value to an oldest value within a predetermined time period, and if an absolute value of a resultant value of integral exceeds a predetermined value and an acceleration detected by an acceleration sensor is smaller than a predetermined acceleration, the airbag is inflated. Based on the value of the integral of the angular velocities, a case in which an angular velocity gradually increases is distinguished from a case in which an angular velocity momentarily increases, so the airbag device effectively prevents malfunctions caused by an action other than falling over. Additionally, because it is unnecessary to intentionally delay determination to prevent malfunctions, the airbag can instantaneously be inflated.

摘要翻译： 用于身体的安全气囊装置瞬间激活安全气囊而不发生故障。 当由角速度传感器检测到的角速度的绝对值超过预定的角速度值时，角速度值在预定时间段内从最近的检测值积分到最老的值，并且如果得到的绝对值 积分值超过预定值，并且由加速度传感器检测到的加速度小于预定加速度时，气囊膨胀。 基于角速度的积分值，角速度逐渐增加的情况与角速度瞬时增加的情况不同，因此气囊装置有效地防止除掉落以外的动作引起的故障。 此外，由于不必有意地延迟确定以防止故障，所以气囊可以瞬间膨胀。

公开(公告)号：US5478799A

公开(公告)日：1995-12-26

申请号：US443775

申请日：1995-05-18

申请人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihisa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

发明人： Ikumi Urushibata ,  Takumi Yoshimura ,  Takeshi Deguchi ,  Norihisa Yonekura ,  Junetsu Sakai ,  Shigeru Hayashi

IPC分类号： A01N43/54 ,  A01N43/66 ,  A01P3/00 ,  A01P13/00 ,  C07D239/28 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  C07D239/52 ,  C07D251/20

CPC分类号： C07D239/28 ,  A01N43/54 ,  A01N43/66 ,  C07D239/30 ,  C07D239/34 ,  C07D239/42 ,  C07D239/47 ,  C07D239/52 ,  C07D251/20

摘要： The present invention provides an N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring represented by formula [I]: ##STR1## wherein R.sup.1 represents an alkyl group, an alkenyl group, or the like, R.sup.2 represents a hydrogen atom, an alkyl group, or the like. R.sup.3 and R.sup.4 represent independently an alkyl group or a nitrogen atom; or the salt of the same, a method for producing the same, and a biocide containing the same as an active ingredient. The N-sulfonyl carboxylic amide derivative including an N-containing 6-membered aromatic ring according to the present invention exhibits superior effects against blight caused by plant pathogenic fungi belonging to Oomycetes such as downy mildew, late blight, or the like in a low concentration as well as controls weeds occurring in paddy fields and plowed fields.

摘要翻译： 本发明提供了包括由式[I]表示的含N 6芳香环的N-磺酰基羧酰胺衍生物：其中R 1表示烷基，烯基等，R 2 表示氢原子，烷基等。 R3和R4独立地表示烷基或氮原子; 或其盐，其制备方法，以及含有活性成分的杀生物剂。 包含根据本发明的含N的6元芳香环的N-磺酰基羧酰胺衍生物，对低浓度的属于软菌属如霜霉病，晚疫病等的植物致病真菌具有优异的抗枯萎作用 以及控制稻田和耕地中发生的杂草。

公开(公告)号：US5418212A

公开(公告)日：1995-05-23

申请号：US53008

申请日：1993-04-27

申请人： Takumi Yoshimura ,  Keiji Toriyabe ,  Katsumi Masuda ,  Ryo Hanai

发明人： Takumi Yoshimura ,  Keiji Toriyabe ,  Katsumi Masuda ,  Ryo Hanai

IPC分类号： A01N43/54 ,  A01N43/66 ,  C07D239/26 ,  C07D239/34 ,  C07D239/46 ,  C07D239/52 ,  C07D405/12 ,  C07D409/12 ,  C07F7/08 ,  C07D251/18 ,  C07D251/22 ,  C07D251/24

CPC分类号： C07D239/26 ,  A01N43/54 ,  A01N43/66 ,  C07D239/34 ,  C07D239/47 ,  C07D239/52 ,  C07D405/12 ,  C07D409/12 ,  C07F7/0812

摘要： The present invention provides a novel alkanoic acid amide derivative of the formula, ##STR1## (wherein R.sup.1 is a hydrogen atom, an alkyl group or an alkoxyalkoxy group, R.sup.2 is a group of --SO.sub.2 R or a hydroxyl group, R.sup.5 is an alkyl group, R.sup.3 is an alkyl group, a cycloalkyl group, a cycloalkenyl group or a phenyl group, R.sup.4 is a hydrogen atom or an alkyl group, X and Y may be the same or different and are an alkoxy group, an alkylamino group or a dialkylamino group, and Z is a methine group or a nitrogen atom) and its salt, a process for preparing the same and a herbicidal composition containing the same as an effective ingredient.This compound kills annual and perennial weeds grown in paddy fields and upland fields at a small dose, and is safe to a useful crop plant.

摘要翻译： 本发明提供下式的新型链烷酸酰胺衍生物，其中R1是氢原子，烷基或烷氧基烷氧基，R2是-SO2R基团或羟基，R5是 烷基，R3是烷基，环烷基，环烯基或苯基，R4是氢原子或烷基，X和Y可以相同或不同，是烷氧基，烷基氨基 或二烷基氨基，Z为次甲基或氮原子）及其盐，其制备方法和含有该有机组合物的除草组合物。 这种化合物以小剂量杀死在稻田和高地田间种植的一年生和多年生杂草，对于有用的作物植物是安全的。