摘要:
The present invention provides a compound represented by Formula: wherein ring A and ring B may be same or different and each is an optionally substituted homocyclic or heterocyclic ring and the like, each R1 may be same or different and is a hydrogen atom, an optionally substituted hydrocarbon group, an acyl group, an optionally substituted heterocyclic group or SR2, etc., X1 is a bond, an optionally substituted divalent C1-3 aliphatic hydrocarbon group or —NR3—, etc, X2 is a bond, an optionally substituted divalent C1-3 aliphatic hydrocarbon group, —NR4—, —O— or —S(O)p— (wherein p is 0, 1 or 2), each Y may be same or different and is a hydrogen atom, an optionally substituted hydrocarbon group, a halogen atom, a carboxyl group, an acyl group, an optionally substituted hydroxy group, an optionally substituted amino group, SR5, an oxo group, a thioxo group, an optionally substituted imino group, a nitro group, a cyano group, etc., each m may be same or different and is 0 or 1, n is an integer of 1 to 3, q1 is an integer of 1 to 2n+4, q2 is an integer of 0 to 2n+3, and the sum of q1 and q2 is 2n+4 or a salt thereof.
摘要:
The present invention provides a compound represented by Formula: wherein ring A and ring B may be same or different and each is an optionally substituted homocyclic or heterocyclic ring and the like, each R1 may be same or different and is a hydrogen atom, an optionally substituted hydrocarbon group, an acyl group, an optionally substituted heterocyclic group or SR2, etc., X1 is a bond, an optionally substituted divalent C1-3 aliphatic hydrocarbon group or —NR3—, etc, X2 is a bond, an optionally substituted divalent C1-3 aliphatic hydrocarbon group, —NR4—, —O— or —S(O)p— (wherein p is 0, 1 or 2), each Y may be same or different and is a hydrogen atom, an optionally substituted hydrocarbon group, a halogen atom, a carboxyl group, an acyl group, an optionally substituted hydroxy group, an optionally substituted amino group, SR5, an oxo group, a thioxo group, an optionally substituted imino group, a nitro group, a cyano group, etc., each m may be same or different and is 0 or 1, n is an integer of 1 to 3, q1 is an integer of 1 to 2n+4, q2 is an integer of 0 to 2n+3, and the sum of q1 and q2 is 2n+4 or a salt thereof.
摘要:
Compounds represented by general formula (1) or salts thereof which have a matrix metalloprotease inhibitory activity and are useful as drugs, wherein the rings A and B represent each an optionally substituted homocycle or heterocycle, etc.; R1s are the same or different and each represents hydrogen, optionally substituted hydrocarbyl, acyl, etc.; X1 represents a bond, optionally substituted divalent aliphatic hydrocarbyl, etc.; X2 represents a bond, optionally substituted divalent aliphatic hydrocarbyl, —O—, etc.; Ys are the same or different represents hydrogen, optionally substituted hydrocarbyl, oxo, etc.; m is 0 or 1; n is an integer of 1 to 3; q1 is an integer of 1 to 2n+4; and q2 is an integer of 0 to 2n+3, provided that q1+q2 is 2n+4.
摘要翻译:由通式(1)表示的化合物或其盐具有基质金属蛋白酶抑制活性,可用作药物,其中环A和B各自表示任选取代的杂环或杂环等; R 1相同或不同,各自表示氢,任选取代的烃基,酰基等; X1表示键,任选取代的二价脂族烃基等; X 2表示键,任选取代的二价脂族烃基,-O-等; Y相同或不同,表示氢,任选取代的烃基,氧代等; m为0或1; n为1〜3的整数。 q1为1〜2n + 4的整数, 并且q2为0〜2n + 3的整数,条件是q1 + q2为2n + 4。
摘要:
A digital information reproducing apparatus in accordance with a prior art that uses a semiconductor memory to realize a memory means cannot reproduce digital data which has been encoded according to a compression coding form different from the one adopted by an incorporated decoding circuit. According to the present invention, a decoding program stored in a second semiconductor memory is selected according to a compression coding form adopted for digital data stored in a first semiconductor memory. The selected decoding program is used to decode the digital data by means of an arithmetic circuit. Thus, digital information can be reproduced irrespective of a compression coding form adopted for provided digital information.
摘要:
The object of the present invention is to provide soluble β-amyloid precursor protein secretory stimulators, which are effective in treating neurodegenerative diseases as well as cerebrovascular disorder-induced neuronopathy. More specifically, the present invention provides a novel compound of the following Formula (I) or a salt or prodrug thereof: [wherein R1 and R2 each represent a hydrogen atom or a lower alkyl group, etc., Ar1 and the ring B each represent an optionally substituted aromatic group, the ring A represents an optionally substituted benzene ring, the ring C represents an optionally substituted 4- to 8-membered ring which may further be condensed with an optionally substituted ring, X represents CH or N, and Y represents CH or N].
摘要:
A multiple-processor system uses transfer blocks each having a size equal to or less than the capacity of a shared memory when transferring data from a master system to a slave system via the shared memory. Each transfer block includes a data to be transferred from the master system or a plurality of divisional data obtained by dividing the data to be transferred; information representing a writing-start address at which the data to be transferred or the plurality of divisional data starts to be written in storage for the slave system; and information representing the length of the data or the plurality of divisional data.
摘要:
A digital information reproduction apparatus for compressing frames of data so as to intermittently reproduce the data in fast-forward speed. A data re-write device retrieves a reproduction-target frame for the fast-forward reproduction and a parameter-calculation-target frame exclusively for calculation of the frame data parameters. The frames then are transferred to a RAM. A decoder determines the frame data in the RAM, calculates the parameter-calculation frame data, and decodes the reproduction frame data by use of the parameter obtained as above. The described operation prevents expending the reproduction frame data with an incorrect parameter so as to normally fast-forward reproduce the compressed data. Furthermore, the present can select a frame used in the fast forward reproduction according to a feature index so that a section subjected to the fast-forward reproduction can be easily grasped by the user.
摘要:
The present invention relates to a 11β-hydroxysteroid dehydrogenase 1 inhibitor comprising a compound represented by the formula (1): wherein each symbol is as defined in the description, or a salt thereof, or a prodrug thereof. The 11β-hydroxysteroid dehydrogenase 1 inhibitor of the present invention has a superior activity, and is useful as a pharmaceutical agent such as agents for the prophylaxis or treatment of diabetes, insulin resistance, obesity, abnormal lipid metabolism, hypertension and the like, and the like.
摘要:
There are provided with a novel N-substituted-3-halopropiolamide compound, a method of producing the compound, and a composition for controlling noxious organisms containing the compound. The present compound exhibits superior antimicrobial and antifungal effects. Pest control agents containing the compound can advantageously be used for wide applications.
摘要:
A compound having a partial structure represented by the formula (A) (wherein ring Xa represents a nitrogen-containing ring and R represents optionally substituted amino) or a salt thereof. The compound or salt is highly effective in regulating neuromedin U receptors and is useful as a preventive/therapeutic agent for hypertension, etc.