Taxane Compound Having Azetidine Ring Structure
    2.
    发明申请
    Taxane Compound Having Azetidine Ring Structure 审中-公开
    具有氮杂环丁烷环结构的紫杉烷化合物

    公开(公告)号:US20090186868A1

    公开(公告)日:2009-07-23

    申请号:US12084065

    申请日:2006-10-24

    CPC分类号: C07D493/08

    摘要: A compound represented by the general formula (1) [X1 and X2 represent hydrogen atom, a halogen atom, hydroxyl group and the like, R1 represents a phenyl group, R2 represents an alkyl group, an alkenyl group, or an alkoxy group, R3 represents hydrogen atom, a halogen atom, hydroxyl group, or an alkoxy group, R4 represents hydrogen atom, or an alkyl group, Z1 and Z2 represent hydrogen atom, a halogen atom, hydroxyl group and the like, Z3 represents cyano group, an alkyl group, an alkenyl group and the like, Z4 represents an alkyl group, an alkenyl group, an alkynyl group and the like, and represents a single bond or a double bond], which shows high antitumor effect against cancer cells including drug resistant cells.

    摘要翻译: 由通式(1)表示的化合物[X1和X2表示氢原子,卤素原子,羟基等,R1表示苯基,R2表示烷基,烯基或烷氧基,R3 表示氢原子,卤素原子,羟基或烷氧基,R4表示氢原子或烷基,Z1和Z2表示氢原子,卤素原子,羟基等,Z3表示氰基,烷基 基团,烯基等,Z4表示烷基,烯基,炔基等,并且表示单键或双键],其对包括耐药细胞在内的癌细胞显示出高抗肿瘤效果。

    Image-recording medium
    4.
    发明申请
    Image-recording medium 审中-公开
    图像记录介质

    公开(公告)号:US20050025912A1

    公开(公告)日:2005-02-03

    申请号:US10476334

    申请日:2002-05-23

    申请人: Yasuyuki Takeda

    发明人: Yasuyuki Takeda

    IPC分类号: B41M5/00 B41M5/52

    摘要: To provide an image-recording medium, which can form a high quality image thereon without yellowing (the shift of color tone) or the blotting of the ink with both the dye ink and the pigment ink. An image-recording medium having a support having breathing micropores, the surfaces and the micropores of which are made hydrophilic, and an ink-receptive layer which is provided on the surface of the support and comprises a binder and a coagulant, characterized in that the ink-receptive layer contains a cationic organic oligomer having a cationic functional group in the molecule, or a cationic polymer having a cationic functional group in the molecule as a coagulant.

    摘要翻译: 为了提供可以在其上形成高质量图像的图像记录介质,而不会变黄(色调的变化)或墨水与染料墨水和颜料墨水两者的印迹。 一种具有支持体的图像记录介质,其具有呼吸微孔,其表面和微孔被制成亲水性,以及设置在支撑体的表面上并包含粘合剂和凝结剂的油墨接收层,其特征在于, 油墨接收层含有分子中具有阳离子官能团的阳离子有机低聚物,或分子中具有阳离子官能团的阳离子聚合物作为凝结剂。

    Aminophenol derivatives
    5.
    发明授权
    Aminophenol derivatives 失效
    氨基苯酚衍生物

    公开(公告)号:US5919824A

    公开(公告)日:1999-07-06

    申请号:US894799

    申请日:1997-09-12

    摘要: Aminophenol derivatives represented by the following formula (1): ##STR1## wherein X is O or S; A is alkylene, R.sup.1 is phenyl, etc., R.sup.2 and R.sup.3 are H or alkyl; R.sup.4 is substituted carbamoylalkyl, etc.; R.sup.5 is substituted amino, etc.; their salts, and optical isomers of the derivatives and salts. Also disclosed are gastrin receptor antagonists, cholecystokinin receptor antagonists, and medicines for digestive diseases. The compounds have strong binding inhibition against gastrin receptor or CCK-A receptor and also they have higher selectivity to either group of CCK-A receptor or gastrin receptor, and therefore, the compounds are useful for preventing and treating gastrointestinal diseases including peptic ulcers as well as central nervous system diseases.

    摘要翻译: PCT No.PCT / JP96 / 00611 Sec。 371日期:1997年9月12日 102(e)1997年9月12日PCT PCT 1996年3月12日PCT公布。 公开号WO96 / 28416 日期:1996年9月19日由下式(1)表示的苯酚衍生物:其中X为O或S; A是亚烷基,R 1是苯基等,R 2和R 3是H或烷基; R4是取代的氨基甲酰基烷基等; R5是取代氨基等。 它们的盐和衍生物和盐的光学异构体。 还公开了胃泌素受体拮抗剂,胆囊收缩素受体拮抗剂和用于消化疾病的药物。 这些化合物对胃泌素受体或CCK-A受体具有强烈的结合抑制作用,并且对CCK-A受体或胃泌素受体组也具有较高的选择性,因此,该化合物也可用于预防和治疗胃肠疾病,包括消化性溃疡 作为中枢神经系统疾病。

    Printed circuit board connector
    6.
    发明授权
    Printed circuit board connector 失效
    印刷电路板连接器

    公开(公告)号:US5641291A

    公开(公告)日:1997-06-24

    申请号:US352612

    申请日:1994-12-09

    IPC分类号: H01R24/00 H01R9/22 H01R9/09

    CPC分类号: H01R12/57 Y10S439/931

    摘要: A printed circuit board connector has: an insulating housing (2); SMT type contacts (7, 11) disposed in the insulating housing and spaced apart from each other; and each contact having a lead (11) which extends to a junction surface (2a) of the housing so as to be soldered to a conductive pattern (16) formed on a printed circuit board (15). The lead (11) of each contact is a plating layer (10) formed on the junction surface (2a). The contacts (7) are pin contacts held in place by the insulating housing (2) so as to be electrically connected to the plating layer (10) formed as the leads. The contacts' leads are included in a common plane so that the reliability of electric connection and the durability of connector are improved, and the connector is rendered thinner and more compact to reduce an area required to mount it.

    摘要翻译: 印刷电路板连接器具有:绝缘壳体(2); SMT型触点(7,11)设置在绝缘壳体中并彼此间隔开; 并且每个触点具有延伸到壳体的接合表面(2a)的引线(11),以便被焊接到形成在印刷电路板(15)上的导电图案(16)。 每个触点的引线(11)是形成在接合表面(2a)上的镀层(10)。 触点(7)是通过绝缘壳体(2)保持在适当位置的销触点,以便与形成为引线的镀层(10)电连接。 接触引线被包含在共同的平面中,使得电连接的可靠性和连接器的耐久性得到改善,并且连接器变得更薄和更紧凑以减少安装所需的面积。

    Epoxy resin composition
    7.
    发明授权
    Epoxy resin composition 失效
    环氧树脂组合物

    公开(公告)号:US07727426B2

    公开(公告)日:2010-06-01

    申请号:US11991299

    申请日:2006-08-23

    IPC分类号: F21V9/00 H01L27/15 C08F20/00

    CPC分类号: C08G59/4215

    摘要: Disclosed is an epoxy resin composition which is solid at ordinary room temperature, cures with excellent light resistance and heat resistance and minimal shrinkage, and is useful for encapsulating LEDs. The epoxy resin composition is characterized by comprising as an essential component an epoxy resin having an epoxy equivalent of 300-1000 g/eq and a softening point of 65-110° C. obtained by reacting a nonaromatic polycarboxylic acid (A) having an acid value of 100-250 mgKOH/g with a nonaromatic epoxy resin (B) having an epoxy equivalent of 100-400 g/eq. The nonaromatic polycarboxylic acid (A) may be obtained by reacting 1,4-cyclohexanedimethanol, 2,2-bis(4-hydroxycyclohexyl)propane, or 3,9-bis(1,1-dimethyl-2-hydroxyethyl)-2,4,8,10-tetraoxaspiro[5,5]undecane with methylhexahydrophthalic acid or hexahydrophthalic acid.

    摘要翻译: 公开了在常温下为固体的环氧树脂组合物,具有优异的耐光性和耐热性和最小的收缩率,并且可用于封装LED。 环氧树脂组合物的特征在于,通过使具有酸的非芳香族多元羧酸(A)反应,得到环氧当量为300〜1000g / eq,软化点为65〜110℃的环氧树脂作为必要成分 与环氧当量为100-400g / eq的非芳族环氧树脂(B)的值为100-250mgKOH / g。 非芳族多元羧酸(A)可以通过使1,4-环己烷二甲醇,2,2-双(4-羟基环己基)丙烷或3,9-双(1,1-二甲基-2-羟乙基)-2, 4,8,10-四氧杂螺[5,5]十一烷与甲基六氢邻苯二甲酸或六氢邻苯二甲酸。

    Navigation system and a memory medium
    8.
    发明授权
    Navigation system and a memory medium 有权
    导航系统和存储介质

    公开(公告)号:US06807480B1

    公开(公告)日:2004-10-19

    申请号:US09632793

    申请日:2000-08-04

    IPC分类号: G01C2100

    摘要: A vicinity search using register point data in a designated area reduces search time. The vicinity search data include at least category information, names of register points and country information. The search device conducts the vicinity search by specifying any one of category information to which the register points belong, names of the register points and country information, or a combination, by option and display. The search device further uses category information with flags representing the presence and absence of the register point data, whereby the register point data are searched by referring to the flags.

    摘要翻译: 使用指定区域中的注册点数据进行的附近搜索减少搜索时间。 附近搜索数据至少包括类别信息,登记点的名称和国家信息。 搜索装置通过选项和显示来指定登记点所属类别信息,登记点名称和国家信息或组合中的任何一个进行附近搜索。 搜索装置还使用具有代表登记点数据的存在和不存在的标志的类别信息,从而通过参考标志来搜索登记点数据。

    Developer solution for positive-working resist composition
    10.
    发明授权
    Developer solution for positive-working resist composition 失效
    正性抗蚀剂组合物的显影剂溶液

    公开(公告)号:US4997748A

    公开(公告)日:1991-03-05

    申请号:US394586

    申请日:1989-08-16

    IPC分类号: G03F7/32

    CPC分类号: G03F7/322

    摘要: The developer solution of the invention is suitable for use to develop a positive-working resist composition comprising an alkali-soluble novolac resin and a naphthoquinone diazide compound and capable of giving a patterned image of the resist layer with a high contrast and increasing the effective depth of focus. The characteristic ingredient in the inventive developer solution is an alkali-soluble organic cyclic nitrogen compound such as N-hydroxyethyl piperazine, N-methyl-4-piperidone, 1,3-dimethyl-2-imidazolidinone and the like added in a specified concentration to a conventional developer solution containing tetramethyl ammonium hydroxide or choline as the water-soluble alkaline compound.

    摘要翻译: 本发明的显影剂溶液适用于开发包含碱溶性酚醛清漆树脂和萘醌二叠氮化合物的正性抗蚀剂组合物,能够以高对比度提供抗蚀剂层的图案化图像并增加有效深度 的焦点。 本发明的显影剂溶液中的特征成分是以特定浓度添加的碱溶性有机环状氮化合物,例如N-羟乙基哌嗪,N-甲基-4-哌啶酮,1,3-二甲基-2-咪唑啉酮等, 包含四甲基氢氧化铵或胆碱作为水溶性碱性化合物的常规显影剂溶液。