公开(公告)号：US4551531A

公开(公告)日：1985-11-05

申请号：US641140

申请日：1984-07-26

申请人： Willy Meyer ,  Karl Gass ,  Werner Topfl ,  Rolf Schurter ,  Georg Pissiotas

发明人： Willy Meyer ,  Karl Gass ,  Werner Topfl ,  Rolf Schurter ,  Georg Pissiotas

IPC分类号： C07D239/47 ,  A01N47/36 ,  A01P13/00 ,  C07D239/42 ,  C07D239/46 ,  C07D239/48 ,  C07D239/52 ,  C07D239/54 ,  C07D239/545 ,  C07D239/56 ,  C07D251/46 ,  C07D521/00

CPC分类号： C07D239/47 ,  A01N47/36 ,  C07D239/48 ,  C07D239/52 ,  C07D239/545 ,  C07D239/56 ,  C07D251/46 ,  C07D521/00

摘要： The invention relates to N-arylsulfonyl-N'-pyrimidinyl ureas of the general formula ##STR1## and to the salts thereof with amines, alkali metal hydroxides or alkaline earth metal hydroxides or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.In the formula, R.sub.18 is hydrogen, alkyl or alkoxy, X is an unsubstituted or substituted phenyl radical or an unsubstituted or substituted naphthyl radical, Y is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, C.sub.1 -C.sub.3 alkylthio, C.sub.2 -C.sub.3 alkoxyalkyl, halogen or an unsubstituted amino group and Z is oxygen or sulfur.

摘要翻译： 本发明涉及通式为（I）的N-芳基磺酰基-N'-嘧啶基脲，以及其与胺，碱金属氢氧化物或碱土金属氢氧化物或季铵碱的盐。 这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。 式中，R 18为氢，烷基或烷氧基，X为未取代或取代的苯基或未取代或取代的萘基，Y为C1-C3烷基，C1-C3卤代烷基，C1-C3烷氧基，C1-C3卤代烷氧基，C1-C3烷硫基， C 2 -C 3烷氧基烷基，卤素或未取代的氨基，Z是氧或硫。

公开(公告)号：US4478635A

公开(公告)日：1984-10-23

申请号：US455175

申请日：1983-01-03

申请人： Willy Meyer ,  Karl Gass ,  Werner Topfl ,  Rolf Schurter ,  Georg Pissiotas

发明人： Willy Meyer ,  Karl Gass ,  Werner Topfl ,  Rolf Schurter ,  Georg Pissiotas

IPC分类号： A01N47/36 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D239/56 ,  C07D251/46 ,  C07D239/69 ,  A01N43/54

CPC分类号： C07D239/47 ,  A01N47/36 ,  C07D239/48 ,  C07D239/52 ,  C07D239/56 ,  C07D251/46

摘要： The invention relates to N-arylsulfonyl-N'-pyrimidinyl ureas of the general formula ##STR1## and to the salts thereof with amines, alkali metal hydroxides or alkaline earth metal hydroxides or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.In the formula, R.sub.18 is hydrogen, alkyl or alkoxy, X is an unsubstituted or substituted phenyl radical or an unsubstituted or substituted naphthyl radical, Y is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, C.sub.1 -C.sub.3 alkylthio, C.sub.2 -C.sub.3 alkoxyalkyl, halogen or an unsubstituted amino group and Z is oxygen or sulfur.

摘要翻译： 本发明涉及通式为（I）的N-芳基磺酰基-N'-嘧啶基脲，以及其与胺，碱金属氢氧化物或碱土金属氢氧化物或季铵碱的盐。 这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。 式中，R 18为氢，烷基或烷氧基，X为未取代或取代的苯基或未取代或取代的萘基，Y为C1-C3烷基，C1-C3卤代烷基，C1-C3烷氧基，C1-C3卤代烷氧基，C1-C3烷硫基， C 2 -C 3烷氧基烷基，卤素或未取代的氨基，Z是氧或硫。

公开(公告)号：US4664695A

公开(公告)日：1987-05-12

申请号：US717637

申请日：1985-03-29

申请人： Rolf Schurter ,  Rudolph C. Thummel ,  Werner Topfl ,  Willy Meyer ,  Dieter Durr

发明人： Rolf Schurter ,  Rudolph C. Thummel ,  Werner Topfl ,  Willy Meyer ,  Dieter Durr

IPC分类号： C07D249/16 ,  A01N47/36 ,  C07C67/00 ,  C07C301/00 ,  C07C311/39 ,  C07D207/38 ,  C07D207/40 ,  C07D207/404 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D251/16 ,  C07D251/18 ,  C07D251/22 ,  C07D251/46 ,  C07D251/52 ,  C07D275/02 ,  C07D521/00 ,  C07D239/69 ,  A01N43/54 ,  C07D401/12 ,  C07D417/12

CPC分类号： C07D207/404 ,  A01N47/36 ,  C07D207/38 ,  C07D239/42 ,  C07D239/47 ,  C07D251/16 ,  C07D275/02 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinylureas of the general formula I ##STR1## and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and growth regulating properties when applied pre- and postemergence.The symbols in formula I have the following meanings:R.sub.1 is hydrogen, halogen, nitro, cyano, or an alkyl, alkoxy, alkylthio, alkylsulfonyl, alkylcarbonyl, alkylcarbamoyl or alkoxycarbonyl group, each unsubstituted or substituted by halogen or alkoxy,R.sub.2 is hydrogen, halogen, alkyl, or an alkyl, alkoxy or alkylthio group, each unsubstituted or substituted by halogen or alkoxy,R.sub.3 is alkyl, haloalkyl, alkoxy or haloalkoxy,R.sub.4 is hydrogen, halogen, R.sub.3, alkylamino or dialkylamino,R.sub.5 is hydrogen, alkyl or alkoxy, andX is an alkenylamino, cycloalkylamino or cycloalkenylamino group which may be further substituted, or is a carbamoylamido or sulfonylamino group as defined in the description, or is a 5- or 6-membered saturated heterocyclic ring system which is bonded through the nitrogen atom and which may contain a further oxygen, sulfur or nitrogen atom in the ring and must contain at least one oxo group.

摘要翻译： 具有通式I（I）的N-苯基磺酰基-N'-嘧啶基和这些化合物与胺，碱金属碱或碱土金属碱或季铵碱的盐具有良好的选择性除草和生长调节性质 应用于芽前和芽后。 式I中的符号具有以下含义：R 1是氢，卤素，硝基，氰基或烷基，烷氧基，烷硫基，烷基磺酰基，烷基羰基，烷基氨基甲酰基或烷氧基羰基，各自未被取代或被卤素或烷氧基取代， 卤素，烷基或烷基，烷氧基或烷硫基，各自未被取代或被卤素或烷氧基取代，R3是烷基，卤代烷基，烷氧基或卤代烷氧基，R4是氢，卤素，R3，烷基氨基或二烷基氨基，R5是氢，烷基或 烷氧基，X是可以被进一步取代的链烯基氨基，环烷基氨基或环烯基氨基，或者是说明书中定义的氨基甲酰氨基或磺酰氨基，或是通过氮键合的5或6元饱和杂环体系 原子，并且其可以在环中含有另外的氧，硫或氮原子，并且必须含有至少一个氧代基团。

公开(公告)号：US4632695A

公开(公告)日：1986-12-30

申请号：US806168

申请日：1985-12-06

申请人： Rolf Schurter ,  Rudolph C. Thummel ,  Werner Topfl ,  Willy Meyer ,  Dieter Durr

发明人： Rolf Schurter ,  Rudolph C. Thummel ,  Werner Topfl ,  Willy Meyer ,  Dieter Durr

IPC分类号： C07D249/16 ,  A01N47/36 ,  C07C67/00 ,  C07C301/00 ,  C07C311/39 ,  C07D207/38 ,  C07D207/40 ,  C07D207/404 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D251/16 ,  C07D251/18 ,  C07D251/22 ,  C07D251/46 ,  C07D251/52 ,  C07D275/02 ,  C07D521/00 ,  A01N43/66 ,  A01N43/70

CPC分类号： C07D207/404 ,  A01N47/36 ,  C07D207/38 ,  C07D239/42 ,  C07D239/47 ,  C07D251/16 ,  C07D275/02 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-triazinylureas of the general formula I ##STR1## and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and growth regulating properties when applied pre- and postemergence. The symbols in formula I have the following meanings:R.sub.1 is hydrogen, halogen, nitro, cyano, or an alkyl, alkoxy, alkylthio, alkylsulfonyl, alkylcarbonyl, alkylcarbamoyl or alkoxycarbonyl group, each unsubstituted or substituted by halogen or alkoxy,R.sub.2 is hydrogen, halogen, alkyl, or an alkyl, alkoxy or alkylthio group, each unsubstituted or substituted by halogen or alkoxy,R.sub.3 is alkyl, haloalkyl, alkoxy or haloalkoxy,R.sub.4 is hydrogen, halogen, R.sub.3, alkylamino or dialkylamino,R.sub.5 is hydrogen, alkyl or alkoxy, andX is an alkenylamino, cycloalkylamino or cycloalkenylamino group which may be further substituted, or is a carbamoylamido or sulfonylamino group as defined in the description, or is a 5- or 6-membered saturated heterocyclic ring system which is bonded through the nitrogen atom and which may contain a further oxygen, sulfur or nitrogen atom in the ring and must contain at least one oxo group.

摘要翻译： 具有通式I（I）的N-苯基磺酰基-N'-三嗪基和这些化合物与胺，碱金属碱或碱土金属碱或季铵碱的盐具有良好的选择性除草和生长调节性质 应用于芽前和芽后。 式I中的符号具有以下含义：R 1是氢，卤素，硝基，氰基或烷基，烷氧基，烷硫基，烷基磺酰基，烷基羰基，烷基氨基甲酰基或烷氧基羰基，各自未被取代或被卤素或烷氧基取代， 卤素，烷基或烷基，烷氧基或烷硫基，各自未被取代或被卤素或烷氧基取代，R3是烷基，卤代烷基，烷氧基或卤代烷氧基，R4是氢，卤素，R3，烷基氨基或二烷基氨基，R5是氢，烷基或 烷氧基，X是可以被进一步取代的链烯基氨基，环烷基氨基或环烯基氨基，或者是说明书中定义的氨基甲酰氨基或磺酰氨基，或是通过氮键合的5或6元饱和杂环体系 原子，并且其可以在环中含有另外的氧，硫或氮原子，并且必须含有至少一个氧代基团。

公开(公告)号：US4487951A

公开(公告)日：1984-12-11

申请号：US571976

申请日：1984-01-19

申请人： Werner F/o/ ry ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

发明人： Werner F/o/ ry ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

IPC分类号： A01N47/24 ,  A01N47/08 ,  A01N47/22 ,  A01N47/36 ,  C07C303/36 ,  C07C311/16 ,  C07C311/53 ,  C07C323/67 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D239/56 ,  C07D251/16 ,  C07D251/22 ,  C07D251/40 ,  C07D251/46 ,  C07D251/52 ,  C07D521/00 ,  C07C143/83

CPC分类号： C07C311/65 ,  A01N47/36 ,  C07D239/47 ,  C07D239/48 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, with alkali or alkaline-earth metal bases or with quaternary ammonium bases, have good pre- and post-emergence selective, herbicidal and growth-regulating properties.The symbols in this formula are as follows:A is a C.sub.3 -C.sub.6 -alkynyl group,E is the methine group or nitrogen,X is oxygen, sulfur or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is the number one or two,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl or C.sub.2 -C.sub.5 -alkenyl or a group --Y--R.sub.5,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.1 -C.sub.4 -haloalkyl, or a group --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, halogen or alkoxyalkyl having at most 4 carbon atoms,R.sub.5 and R.sub.6 are each C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl,R.sub.7 and R.sub.8 independently of one another are each hydrogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, andY is oxygen, sulfur or a sulfinyl or sulfonyl bridge.

摘要翻译： 具有通式（I）的N-苯基磺酰基-N'-嘧啶基 - 和 - 三嗪基脲和这些化合物与胺与碱金属或碱土金属碱或季铵碱的盐具有良好的前和后 芽后选择性，除草和生长调节性质。 该式中的符号如下：A是C 3 -C 6炔基，E是次甲基或氮，X是氧，硫或亚磺酰基或磺酰基桥，Z是氧或硫，m是第一个 或两个，R 1是氢，卤素，C 1 -C 5 - 烷基或C 2 -C 5 - 烯基或基团-Y-R 5，R 2是氢，卤素，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 1 -C 4 - 卤代烷基或基团-Y-R 5，-COOR 6，-NO 2或-CO-NR 7 -R 8，R 3和R 4彼此独立地为氢，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，卤素或至多4个碳原子的烷氧基烷基，R 5和R 6各自为C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6炔基，R 7和R 8独立地为 各自为氢，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6 - 炔基，Y为氧，硫或亚磺酰基或磺酰基桥。

公开(公告)号：US4443243A

公开(公告)日：1984-04-17

申请号：US396959

申请日：1982-07-09

申请人： Werner Fory ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

发明人： Werner Fory ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

IPC分类号： A01N47/24 ,  A01N47/08 ,  A01N47/22 ,  A01N47/36 ,  C07C303/36 ,  C07C311/16 ,  C07C311/53 ,  C07C323/67 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D239/56 ,  C07D251/16 ,  C07D251/22 ,  C07D251/40 ,  C07D251/46 ,  C07D251/52 ,  C07D521/00 ,  C07D251/44 ,  A01N43/66 ,  C07D251/42

CPC分类号： C07C311/65 ,  A01N47/36 ,  C07D239/47 ,  C07D239/48 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, with alkali or alkaline-earth metal bases or with quaternary ammonium bases, have good pre- and post-emergence selective, herbicidal and growth-regulating properties.The symbols in this formula are as follows:A is a C.sub.3 -C.sub.6 -alkynyl group,E is the methine group or nitrogen,X is oxygen, sulfur or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is the number one or two,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl or C.sub.2 -C.sub.5 -alkenyl or a group --Y--R.sub.5,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.1 -C.sub.4 -haloalkyl, or a group --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, halogen or alkoxyalkyl having at most 4 carbon atoms,R.sub.5 and R.sub.6 are each C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl,R.sub.7 and R.sub.8 independently of one another are each hydrogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, andY is oxygen, sulfur or a sulfinyl or sulfonyl bridge.

摘要翻译： 具有通式（I）的N-苯基磺酰基-N'-嘧啶基 - 和 - 三嗪基脲和这些化合物与胺与碱金属或碱土金属碱或季铵碱的盐具有良好的前和后 芽后选择性，除草和生长调节性质。 该式中的符号如下：A是C 3 -C 6炔基，E是次甲基或氮，X是氧，硫或亚磺酰基或磺酰基桥，Z是氧或硫，m是第一个 或两个，R 1是氢，卤素，C 1 -C 5 - 烷基或C 2 -C 5 - 烯基或基团-Y-R 5，R 2是氢，卤素，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 1 -C 4 - 卤代烷基或基团-Y-R 5，-COOR 6，-NO 2或-CO-NR 7 -R 8，R 3和R 4彼此独立地为氢，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，卤素或至多4个碳原子的烷氧基烷基，R 5和R 6各自为C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6炔基，R 7和R 8 各自独立地为氢，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6 - 炔基，Y为氧，硫或亚磺酰基或磺酰基桥。

公开(公告)号：US4523944A

公开(公告)日：1985-06-18

申请号：US571985

申请日：1984-01-19

申请人： Werner Fory ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

发明人： Werner Fory ,  Karl Gass ,  Willy Meyer ,  Rolf Schurter

IPC分类号： A01N43/54 ,  A01N47/36 ,  C07D239/42 ,  C07D239/48 ,  C07D251/22 ,  C07D521/00

CPC分类号： C07D239/48 ,  A01N47/36 ,  C07C317/00 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, with alkali or alkaline-earth metal bases or with quaternary ammonium bases, have good pre- and post-emergence selective, herbicidal and growth-regulating properties.The symbols in this formula are as follows:A is a C.sub.3 -C.sub.6 -alkynyl group,E is the methine group or nitrogen,X is oxygen, sulfur or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is the number one or two,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl or C.sub.2 -C.sub.5 -alkenyl or a group --Y--R.sub.5,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.1 -C.sub.4 -haloalkyl, or a group --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, halogen or alkoxyalkyl having at most 4 carbon atoms,R.sub.5 and R.sub.6 are each C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl,R.sub.7 and R.sub.8 independently of one another are each hydrogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, andY is oxygen, sulfur or a sulfinyl or sulfonyl bridge.

摘要翻译： 具有通式（I）的N-苯基磺酰基-N'-嘧啶基 - 和 - 三嗪基脲和这些化合物与胺与碱金属或碱土金属碱或季铵碱的盐具有良好的前和后 芽后选择性，除草和生长调节性质。 该式中的符号如下：A是C 3 -C 6炔基，E是次甲基或氮，X是氧，硫或亚磺酰基或磺酰基桥，Z是氧或硫，m是第一个 或两个，R 1是氢，卤素，C 1 -C 5 - 烷基或C 2 -C 5 - 烯基或基团-Y-R 5，R 2是氢，卤素，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 1 -C 4 - 卤代烷基或基团-Y-R 5，-COOR 6，-NO 2或-CO-NR 7 -R 8，R 3和R 4彼此独立地为氢，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，卤素或至多4个碳原子的烷氧基烷基，R 5和R 6各自为C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6炔基，R 7和R 8 各自独立地为氢，C 1 -C 5 - 烷基，C 2 -C 5 - 烯基或C 2 -C 6 - 炔基，Y为氧，硫或亚磺酰基或磺酰基桥。

公开(公告)号：US4835311A

公开(公告)日：1989-05-30

申请号：US141820

申请日：1988-01-11

申请人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

发明人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

IPC分类号： C07D251/16 ,  A01N47/36 ,  C07D211/22 ,  C07D213/30 ,  C07D213/64 ,  C07D213/643 ,  C07D239/42 ,  C07D251/46 ,  C07D251/52 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D521/00

CPC分类号： C07D213/30 ,  C07D213/643 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinylureas and -N'-triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, alkali metal bases and alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and plant growth regulating properties when applied pre- and postemergence.In the formulaR.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.5 alkenyl or C.sub.1 -C.sub.4 alkoxycarbonyl,R.sub.2 is C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms,R.sub.3 is halogen, hydrogen, --NR.sub.4 R.sub.5, C.sub.1 -C.sub.3 alkyl, unsubstituted or substituted by 1 to 3 halogen atoms of C.sub.1 -C.sub.4 alkoxy, or is C.sub.1 -C.sub.3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms,R.sub.4 is hydrogen or methyl,R.sub.5 is hydrogen, C.sub.1 -C.sub.2 alkyl or methoxy,A is C.sub.1 -C.sub.4 alkylene or C.sub.2 -C.sub.4 alkenylene, each unsubstituted or substituted by C.sub.1 -C.sub.4 alkyl,m is 0 or 1,E is nitrogen or the methine group,X is oxygen, sulfur, --SO-- or --SO.sub.2 --, andQ is hydroxyl, cyano or radicals selected from the group consisting of 5- or 6-membered heterocyclic rings and fused homologues, amines, acetals, esters, ketones, phenyls, sulfonic acid and carboxylic acids, which radicals may be further substituted and have functional structures.

摘要翻译： 具有通式“IMAGE”的N-苯基磺酰基-N'-嘧啶基脲和-N'-三嗪基脲以及这些化合物与胺，碱金属碱和碱土金属碱或季铵碱的盐具有良好的选择性除草和植物 应用芽前和芽后的生长调节性质。 式中R 1为氢，卤素，硝基，C 1 -C 4卤代烷基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 2 -C 5烯基或C 1 -C 4烷氧基羰基，R 2为C 1 -C 3烷基或C 1 -C 3烷氧基，各自未被取代或被1至3个卤素 原子，R3是卤素，氢，-NR4R5，C1-C3烷基，未取代或被C1-C4烷氧基的1至3个卤素原子取代，或是未被取代或被甲氧基，乙氧基或1至3个卤素原子取代的C1-C3烷氧基， R4是氢或甲基，R5是氢，C1-C2烷基或甲氧基，A是C1-C4亚烷基或C2-C4亚烯基，各自未被取代或被C1-C4烷基取代，m是0或1，E是氮或次甲基，X 是氧，硫，-SO-或-SO 2 - ，Q是羟基，氰基或选自5-或6-元杂环和稠合同系物，胺，缩醛，酯，酮，苯基，磺酸的基团 酸和羧酸，该基团可以进一步被取代并具有官能结构。

公开(公告)号：US4648899A

公开(公告)日：1987-03-10

申请号：US855060

申请日：1986-04-23

申请人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

发明人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

IPC分类号： C07D251/16 ,  A01N47/36 ,  C07D211/22 ,  C07D213/30 ,  C07D213/64 ,  C07D213/643 ,  C07D239/42 ,  C07D251/46 ,  C07D251/52 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D521/00 ,  A01N43/70 ,  C07D251/42

CPC分类号： C07D213/30 ,  C07D213/643 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinylureas and -N'-triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, alkali metal bases and alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and plant growth regulating properties when applied pre- and postemergence.In the formulaR.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.5 alkenyl or C.sub.1 -C.sub.4 alkoxycarbonyl,R.sub.2 is C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms,R.sub.3 is halogen, hydrogen, --NR.sub.4 R.sub.5, C.sub.1 -C.sub.3 alkyl, unsubstituted or substituted by 1 to 3 halogen atoms or C.sub.1 -C.sub.4 alkoxy, or is C.sub.1 -C.sub.3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms,R.sub.4 is hydrogen or methyl,R.sub.5 is hydrogen, C.sub.1 -C.sub.2 alkyl or methoxy,A is C.sub.1 -C.sub.4 alkylene or C.sub.2 -C.sub.4 alkenylene, each unsubstituted or substituted by C.sub.1 -C.sub.4 alkyl,m is 0 or 1,E is nitrogen or the methine group,X is oxygen, sulfur, --SO--, or --SO.sub.2 --, andQ is hydroxyl, cyano or radicals selected from the group consisting of 5- or 6-membered heterocyclic rings and fused homologues, amines, acetals, esters, ketones, phenyls, sulfonic acid and carboxylic acids, which radicals may be further substituted and have functional structures.

摘要翻译： 具有通式“IMAGE”的N-苯基磺酰基-N'-嘧啶基脲和-N'-三嗪基脲和这些化合物与胺，碱金属碱和碱土金属碱或季铵碱的盐具有良好的选择性除草和植物 应用芽前和芽后的生长调节性质。 式中R 1为氢，卤素，硝基，C 1 -C 4卤代烷基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 2 -C 5烯基或C 1 -C 4烷氧基羰基，R 2为C 1 -C 3烷基或C 1 -C 3烷氧基，各自未被取代或被1至3个卤素 原子，R 3是卤素，氢，-NR 4 R 5，未被取代或被1至3个卤素原子或C 1 -C 4烷氧基取代的C 1 -C 3烷基，或是未被取代或被甲氧基，乙氧基或1至3个卤素原子取代的C 1 -C 3烷氧基， R4是氢或甲基，R5是氢，C1-C2烷基或甲氧基，A是C1-C4亚烷基或C2-C4亚烯基，各自未被取代或被C1-C4烷基取代，m是0或1，E是氮或次甲基，X 是氧，硫，-SO-或-SO 2 - ，Q是羟基，氰基或选自5-或6-元杂环和稠合同系物，胺，缩醛，酯，酮，苯基， 磺酸和羧酸，该基团可进一步被取代并具有官能结构。

公开(公告)号：US4618363A

公开(公告)日：1986-10-21

申请号：US458799

申请日：1983-01-18

申请人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

发明人： Karl Gass ,  Werner Fory ,  Willy Meyer ,  Werner Topfl

IPC分类号： C07D251/16 ,  A01N47/36 ,  C07D211/22 ,  C07D213/30 ,  C07D213/64 ,  C07D213/643 ,  C07D239/42 ,  C07D251/46 ,  C07D251/52 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D521/00 ,  A01N43/66 ,  A01N43/70

CPC分类号： C07D213/30 ,  C07D213/643 ,  C07D301/14 ,  C07D303/22 ,  C07D307/12 ,  C07D309/06 ,  C07D317/22 ,  C07D333/16 ,  C07D521/00

摘要： N-Phenylsulfonyl-N'-pyrimidinylureas and -N'-triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, alkali metal bases and alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and plant growth regulating properties when applied pre- and postemergence.In the formulaR.sub.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.5 alkenyl or C.sub.1 -C.sub.4 alkoxycarbonyl,R.sub.2 is C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms,R.sub.3 is halogen, hydrogen, --NR.sub.4 R.sub.5, C.sub.1 -C.sub.3 alkyl, unsubstituted or substituted by 1 to 3 halogen atoms or C.sub.1 -C.sub.4 alkoxy, or is C.sub.1 -C.sub.3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms,R.sub.4 is hydrogen or methyl,R.sub.5 is hydrogen, C.sub.1 -C.sub.2 alkyl or methoxy,A is C.sub.1 -C.sub.4 alkylene or C.sub.2 -C.sub.4 alkenylene, each unsubstituted or substituted by C.sub.1 -C.sub.4 alkyl,m is 0 or 1,E is nitrogen or the methine group,X is oxygen, sulfur, --SO-- or --SO.sub.2 --, andQ is hydroxyl, cyano or radicals selected from the group consisting of 5- or 6-membered heterocyclic rings and fused homologues, amines, acetals, esters, ketones, phenyls, sulfonic acid and carboxylic acids, which radicals may be further substituted and have functional structures.

摘要翻译： 具有通式“IMAGE”的N-苯基磺酰基-N'-嘧啶基脲和-N'-三嗪基脲和这些化合物与胺，碱金属碱和碱土金属碱或季铵碱的盐具有良好的选择性除草和植物 应用芽前和芽后的生长调节性质。 式中R 1为氢，卤素，硝基，C 1 -C 4卤代烷基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 2 -C 5烯基或C 1 -C 4烷氧基羰基，R 2为C 1 -C 3烷基或C 1 -C 3烷氧基，各自未被取代或被1至3个卤素 原子，R 3是卤素，氢，-NR 4 R 5，未被取代或被1至3个卤素原子或C 1 -C 4烷氧基取代的C 1 -C 3烷基，或是未被取代或被甲氧基，乙氧基或1至3个卤素原子取代的C 1 -C 3烷氧基， R4是氢或甲基，R5是氢，C1-C2烷基或甲氧基，A是C1-C4亚烷基或C2-C4亚烯基，各自未被取代或被C1-C4烷基取代，m是0或1，E是氮或次甲基，X 是氧，硫，-SO-或-SO 2 - ，Q是羟基，氰基或选自5-或6-元杂环和稠合同系物，胺，缩醛，酯，酮，苯基，磺酸的基团 酸和羧酸，该基团可以进一步被取代并具有官能结构。