Method of preserving organic materials from fungal attack and a
composition for use in such a method
    1.
    发明授权
    Method of preserving organic materials from fungal attack and a composition for use in such a method 失效
    从真菌侵袭中保存有机材料的方法和用于这种方法的组合物

    公开(公告)号:US4421766A

    公开(公告)日:1983-12-20

    申请号:US338141

    申请日:1982-01-08

    摘要: A variety of organic materials susceptible to fungal attack (especially wood and wood-based materials) can be protected from such attack and fungi growing on such materials can be eradicated by treating them, e.g. by applying to the surfaces or impregnating, with one or more compounds of formula (I): ##STR1## (wherein X represents a halogen atom and R represents a hydroxy group, an alkoxy gorup, a substituted or unsubstituted phenoxy group, an amino group, a mono- or di- alkylamino group, a phenylamino or benzylamino group which is unsubstituted or has one or two substituents on the benzene ring of the phenyl or benzyl moiety, or a 3-halo-2,3-diiodoallyloxy group). An anti-fungal composition contains one or more of these compounds in admixture with a carrier or adjuvant.

    摘要翻译: 可以保护易受真菌侵袭的各种有机材料(特别是木材和木质材料),免受这种攻击,并且可以通过对这些材料进行处理来消除在这些材料上生长的真菌。 (I)(其中X表示卤素原子,R表示羟基,烷氧基羰基,取代或未取代的苯氧基,烷氧基羰基,取代或未取代的苯氧基, 氨基,单或二烷基氨基,苯基氨基或苄基氨基,或苯基或苄基部分的苯环上未取代或具有一个或两个取代基,或3-卤代-2,3-二碘代乙酰氧基 )。 抗真菌组合物含有一种或多种这些化合物与载体或佐剂的混合物。

    Pyridine sulfonamides and their use as anticoccidial agents
    6.
    发明授权
    Pyridine sulfonamides and their use as anticoccidial agents 失效
    吡啶磺酰亚胺及其作为抗焦虑剂

    公开(公告)号:US4094982A

    公开(公告)日:1978-06-13

    申请号:US681154

    申请日:1976-04-28

    CPC分类号: C07D213/70

    摘要: Pyridine derivatives having the formula ##STR1## wherein R.sub.1 represents hydrogen atom, amino group or a group ##STR2## in which R.sub.5 and R.sub.6 may be the same or different and each represents an alkyl group of 1 to 4 carbon atoms or R.sub.5 is hydrogen atom and R.sub.6 represents an alkyl group of 1 to 4 carbon atoms, an alkenyl group of 3 or 4 carbon atoms or a benzyl group optionally substituted with halogen, cyano, alkyl of 1 to 4 carbon atoms or alkoxy of 1 to 4 carbon atoms;R.sub.2 represents nitro group, amino group or an alkylamino group of 1 to 3 carbon atoms;R.sub.3 and R.sub.4 individually represent hydrogen atom, an alkyl group of 1 to 4 carbon atoms, an alkoxyalkyl group which has 1 to 4 carbon atoms in the alkoxy moiety and 2 to 4 carbon atoms in the alkyl moiety, an alkenyl group of 3 or 4 carbon atoms, an alkanoyl group of 1 to 18 carbon atoms or a benzyl group optionally substituted with halogen, cyano, alkyl of 1 to 4 carbon atoms or alkoxy of 1 to 4 carbon atoms; provided that when R.sub.1 is hydrogen atom and R.sub.2 is nitro group, R.sub.3 and R.sub.4 may be the same or different and each represents said alkyl group or said alkoxyalkyl group or R.sub.3 is hydrogen atom and R.sub.4 is hydrogen atom, said alkyl group, said alkoxyalkyl group, said alkenyl group, said alkanoyl group or said benzyl group, when R.sub.1 is hydrogen atom and R.sub.2 is amino group or said alkylamino group, R.sub.3 and R.sub.4 individually is hydrogen atom or they may be the same or different and each represents said alkyl group, when R.sub.1 is amino group and R.sub.2 is nitro group, R.sub.3 and R.sub.4 may be the same or different and each represents said alkyl group or R.sub. 3 is hydrogen atom and R.sub.4 is said alkyl group or said alkenyl group, and when R.sub.1 is said group ##STR3## and R.sub.2 is nitro group, R.sub.3 and R.sub.4 are the same as defined above with respect to the R.sub.5 and R.sub.6.They are highly effective in the treatment of coccidiosis, especially that caused by the protozoa belonging to the species Eimeria tenella or E. necatrix.

    Pyridine derivatives and their use as anticoccidial agents
    7.
    发明授权
    Pyridine derivatives and their use as anticoccidial agents 失效
    吡啶衍生物及其作为抗球虫药的用途

    公开(公告)号:US4054663A

    公开(公告)日:1977-10-18

    申请号:US639697

    申请日:1975-12-11

    摘要: Pyridine derivatives having the formula ##STR1## wherein R.sub.1 is an alkyl group having 1 to 3 carbon atoms; R.sub.2 is hydrogen atom or an alkyl group having 1 to 3 carbon atoms; R.sub.3 is hydrogen atom, an alkyl group having 1 to 4 carbon atoms, an alkenyl group having 3 or 4 carbon atoms, an alkyl group having 1 or 2 carbon atoms and hydroxy as a substituent, an alkanoyl group having 1 to 18 carbon atoms, an alkenoyl group having 3 to 11 carbon atoms, an aromatic acyl group having 6 or 10 carbon atoms in the aromatic ring and optionally alkyl, alkoxy, acetylamino, cyano or halogen as a substituent, a heterocyclic acyl group, an alkylcarbamoyl group having 1 to 4 carbon atoms in the alkyl moiety, an allylcarbamoyl group or hydroxy group; n is an integer of 0 to 2 inclusive; and, when n is 2, R.sub.1 's may be the same or different; provided that when R.sub.2 is said alkyl group having 1 to 3 carbon atoms, R.sub.3 is said alkyl group having 1 to 4 carbon atoms.They are highly effective in the treatment of coccidiosis.

    摘要翻译: 具有式“IMAGE”的吡啶衍生物,其中R 1是具有1至3个碳原子的烷基; R2是氢原子或碳原子数1〜3的烷基; R3是氢原子,碳原子数1〜4的烷基,碳原子数3〜4的烯基,碳原子数1〜2的烷基,羟基作为取代基,碳原子数1〜18的烷酰基, 具有3至11个碳原子的烯酰基,芳环中具有6或10个碳原子的芳族酰基和任选的烷基,烷氧基,乙酰氨基,氰基或卤素作为取代基,杂环酰基,烷基氨基甲酰基具有1至 烷基部分中的4个碳原子,烯丙基氨基甲酰基或羟基; n为0〜2的整数, 并且当n为2时,R 1可以相同或不同; 条件是当R 2为所述具有1至3个碳原子的烷基时,R 3为所述具有1至4个碳原子的烷基。

    1,2,4-triazinone derivatives, their preparation and use
    9.
    发明授权
    1,2,4-triazinone derivatives, their preparation and use 失效
    1,2,4-三嗪酮衍生物,其制备和用途

    公开(公告)号:US4898862A

    公开(公告)日:1990-02-06

    申请号:US26290

    申请日:1987-03-16

    摘要: Compounds of formula (I): ##STR1## (in which: R.sup.1 is hydrogen or alkl; R.sup.2 is a variety of groups or atoms; R.sup.3 is optionally substituted hydroxy or --(NH).sub.n --NR.sup.5 R.sup.6, wherein R.sup.5 and R.sup.6 are a variety of groups or atoms, preferably alkyl substituted by heterocyclic, and n is 0 or 1; Q is oxygen or sulfur; and A is a C.sub.1 -C.sub.6 alkylene group) have valuable cardiotionic activity and may be used for the treatment of cardiac disorders. They may be prepared from corresponding compounds containing a benzene ring with a group --QH at the 1-position and a group --CO--CHR.sup.1 --NH--COOR.sup.7 at the 4-position by ring closure and introduction of the group of formula --A--CO--R.sup.3 in any order.

    摘要翻译: 式(I)化合物:其中:R 1是氢或烷基; R 2是各种基团或基团; R 3是任选取代的羟基或 - (NH)n -NR 5 R 6,其中R 5和R 6 是各种基团或原子,优选被杂环取代的烷基,n为0或1; Q为氧或硫; A为C1-C6亚烷基)具有有价值的心血管活性,可用于治疗心脏 疾病 它们可以由相应的化合物制备,所述化合物含有1-环基团-QH的苯环和通过闭环在4-位上的-CO-CHR1-NH-COOR7基团,并引入式-A- CO-R3以任何顺序。

    Pyridine derivatives and their use as anticoccidial agents
    10.
    发明授权
    Pyridine derivatives and their use as anticoccidial agents 失效
    吡啶衍生物及其用作抗焦虑剂

    公开(公告)号:US4098893A

    公开(公告)日:1978-07-04

    申请号:US816215

    申请日:1977-07-15

    摘要: Pyridine derivatives having the formula ##STR1## wherein R.sub.1 is an alkyl group having 1 to 3 carbon atoms; R.sub.2 is hydrogen atom or an alkyl group having 1 to 3 carbon atoms; R.sub.3 is hydrogen atom, an alkyl group having 1 to 4 carbon atoms, an alkenyl group having 3 or 4 carbon atoms, an alkyl group having 1 or 2 carbon atoms and hydroxy as a substituent, an alkanoyl group having 1 to 18 carbon atoms, an alkenoyl group having 3 to 11 carbon atoms, an aromatic acyl group having 6 or 10 carbon atoms in the aromatic ring and optionally alkyl, alkoxy, acetylamino, cyano or halogen as a substituent, a heterocyclic acyl group, an alkylcarbamoyl group having 1 to 4 carbon atoms in the alkyl moiety, an allylcarbamoyl group or hydroxy group; n is an integer of 0 to 2 inclusive; and, when n is 2, R.sub.1 's may be the same or different; provided that when R.sub.2 is said alkyl group having 1 to 3 carbon atoms, R.sub.3 is said alkyl group having 1 to 4 carbon atoms.They are highly effective in the treatment of coccidiosis.