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    Pesticidal compounds
    3.
    发明授权
    Pesticidal compounds 失效
    杀虫化合物

    公开(公告)号：US6043286A

    公开(公告)日：2000-03-28

    申请号：US891079

    申请日：1997-07-10

    申请人： Bhupinder Pall Singh Khambay ,  Duncan Batty

    发明人： Bhupinder Pall Singh Khambay ,  Duncan Batty

    IPC分类号： A01N35/06 ,  A01N35/10 ,  A01N37/02 ,  A01N37/10 ,  C07C46/00 ,  C07C50/32 ,  C07C69/013 ,  C07C251/46 ,  A01N33/02 ,  C07C50/00 ,  C07C50/12

    CPC分类号： C07C251/46 ,  A01N35/06 ,  A01N35/10 ,  A01N37/02 ,  A01N37/10 ,  C07C46/00 ,  C07C50/32 ,  C07C69/013 ,  C07C2101/14 ,  C07C2101/18

    摘要： Pesticidal as a pesticide against whitefly, Lepidoptera and certain fungi is provided of compound of general formula (I) ##STR1## or a salt thereof is provided, in which n represents an integer from 0 to 4; m represents an integer 0 or 1;each R independently represents a halogen atom or a nitro, cyano, hydroxyl, alkyl, alkenyl, haloalkyl, haloalkenyl, alkoxy, haloalkoxy, haloalkenoxy, amino, alkylamino, dialkylamino, alkoxycarbonyl, carboxyl, alkanoyl, alkylthio, alkylsulphinyl, alkylsulphonyl, carbamoyl, alkylamido, cycloalkyl, aryl or aralkyl group;R.sup.1 and R.sup.2 each independently represent an optionally substituted alkoxy group or together represent a group .dbd.O, .dbd.S or .dbd.N--OR.sup.9, where R.sup.9 represents a hydrogen atom or an optionally substituted alkyl group;R.sup.3 represents a hydroxyl group, or a group --OL where L is a leaving group, or a group which in vivo is transformed into a group --OL.sup.1 where L.sup.1 is a leaving group;R.sup.7 and R.sup.8 independently represent an optionally substituted alkoxy group or together represent a group .dbd.O, .dbd.S or .dbd.N--OR.sup.9, where R.sup.9 is as previously defined;wherein R.sub.4 and R.sub.5 independently represent a halogen atom or an optionally substituted alkyl or alkenyl group, or together with the interjacent carbon atom represent an optionally substituted cycloalkyl or cycloalkenyl ring; andA represents a straight or branched chain alkyl or alkenyl group, which may be optionally substituted, an acyclic carbon chain of which links the 3 position of the naphthalene ring shown and the moiety --CHR.sup.4 R.sup.5 and wherein A does not include a quaternary carbon atom in that chain; andwherein the total number of carbon atoms in the longest carbon chain running from the 3-position of the naphthalene ring shown is no more than 8.

    摘要翻译： 提供了杀虫剂作为粉虱，鳞翅目和某些真菌的杀虫剂，提供通式（I）的化合物或其盐，其中n表示0至4的整数; m表示整数0或1; 每个R独立地表示卤素原子或硝基，氰基，羟基，烷基，烯基，卤代烷基，卤代烯基，烷氧基，卤代烷氧基，卤代烯氧基，氨基，烷基氨基，二烷基氨基，烷氧基羰基，羧基，烷酰基，烷硫基，烷基亚磺酰基，烷基磺酰基，氨基甲酰基， ，环烷基，芳基或芳烷基; R 1和R 2各自独立地表示任选取代的烷氧基或一起表示基团= O，= S或= N-OR 9，其中R 9表示氢原子或任选取代的烷基; R3表示羟基或其中L为离去基团的基团-OL，或将体内转化为基团-OL1的基团，其中L1为离去基团; R 7和R 8独立地表示任选取代的烷氧基或一起表示基团= O，= S或= N-OR 9，其中R 9如前所定义; 其中R 4和R 5独立地表示卤原子或任选取代的烷基或烯基，或与中间碳原子一起表示任选取代的环烷基或环烯基环; 并且A表示直链或支链烷基或烯基，其可以是任选取代的，其连接所示萘环的3位和部分-CHR 4 R 5的无环碳链，其中A不包括季碳原子 那条链 并且其中从所示的萘环的3位运行的最长碳链中的碳原子总数不大于8。

    SHIKONIN, ALKANNIN; AND RACEMIC PARENT NUCLEUS CABONYL OXIME DERIVATIVES AND APPLICATIONS THEREOF
    7.
    发明申请
    SHIKONIN, ALKANNIN; AND RACEMIC PARENT NUCLEUS CABONYL OXIME DERIVATIVES AND APPLICATIONS THEREOF 审中-公开
    SHIKONIN，阿尔坎宁 和种族主义核仁CABONYL OXIME衍生物及其应用

    公开(公告)号：US20150344415A1

    公开(公告)日：2015-12-03

    申请号：US14759024

    申请日：2013-06-25

    申请人： SHANGHAI JIAO TONG UNIVERSITY

    发明人： Shaoshun Li ,  Rubing Wang ,  Xiaogang Zheng ,  Xu Zhang

    IPC分类号： C07C251/34 ,  C07D333/40 ,  C07C249/08 ,  C07D213/79

    CPC分类号： C07C251/34 ,  A61K31/15 ,  A61K31/222 ,  C07C249/08 ,  C07C251/46 ,  C07D213/79 ,  C07D333/40

    摘要： A structural formula of a shikonin naphthazarin parent nucleus hydroxyl methylation carbonyl oxime derivative is shown in Formula (I) or (II); a structural formula of an alkannin naphthazarin parent nucleus hydroxyl methylation carbonyl oxime derivative is shown in Formula (III) or (IV); and a structural formula of a racemic shikonin naphthazarin parent nucleus hydroxyl methylation carbonyl oxime derivative is shown in Formula (V) or (VI), wherein R1 is alkane, olefin, arene, or substituting arene comprising 1 to 6 carbon atoms; and R2 is alkane, olefin, arene, or substituting arene comprising 1 to 6 carbon atoms or is H. The shikonin, alkannin, and racemic oxime derivatives of the present invention have novel structures, and in-vitro experiments show that the present invention has good growth inhibitory activity against tumor cells and can be used in tumor treatment.

    摘要翻译： 紫草素萘甲酰胺母核羟基甲基化羰基肟衍生物的结构式如式（I）或（II）所示; 式（III）或（IV）中示出了链烷烃萘氮杂环母体核羟基甲基化羰基肟衍生物的结构式。 （V）或（VI）所示，其中R 1为烷烃，烯烃，芳烃，或以1-6个碳原子取代的芳烃;式（Ⅴ）或（Ⅵ）表示外消旋的紫草素萘甲脒母核羟基甲基化羰基肟衍生物的结构式。 R2是烷烃，烯烃，芳烃或代替含有1至6个碳原子的芳烃或为H。本发明的紫草素，链烷酸和外消旋肟衍生物具有新颖的结构，体外实验表明本发明具有 对肿瘤细胞有良好的生长抑制活性，可用于肿瘤治疗。