Abstract:
Novel N-substituted amino acid derivatives of the formula: ##STR1## wherein R.sub.1 is an alkenyl group having 2 to 5 carbon atoms, a halogen-substituted alkenyl group having 2 to 5 carbon atoms or an alkynyl group having 2 to 5 carbon atoms, R.sub.2 is a methyl or ##STR2## group in which R.sub.2 ' is an alkyl group having 1 to 4 carbon atoms or a halogen-substituted alkyl group having 1 to 4 carbon atoms; and R.sub.3 is a hydrogen atom, an alkyl having 1 to 20 carbon atoms, cycloalkyl having 3 to 6 carbon atoms, benzyl, hydroxyethyl or methoxyethyl group, and inorganic or organic acid addition salts thereof, which possess useful soil fungicidal activities and can be produced by reacting a sarcosine derivative of the formula:CH.sub.3 HNCH.sub.2 COOR.sub.3 (II)wherein R.sub.3 is as defined above, with a halogen compound of the formula:R.sub.1 -- X (III)wherein R.sub.1 is as defined above and X is a halogen atom, or by reacting an N-substituted glycine derivative of the formula: ##STR3## wherein R.sub.1 and R.sub.3 are as defined above, with an acyl compound of the formula: ##STR4## wherein R.sub.2 ' is as defined above and X is a halogen atom.
Abstract:
A method of preparing N-phosphonomethylglycine comprising (a) reacting a substituted triazine with an acyl halide to form the N-carboalkoxymethyl-N-halomethyl amide of the acyl halide; reacting the said amide with a phosphite to form a phosphonate compound; and hydrolyzing said phosphonate to yield N-phosphonomethylglycine.
Abstract:
N-substituted 2-methylnaphthylamides of the general formula I ##STR1## where R is an unsubstituted or substituted furyl, isoxazolyl, oxazolyl, isothiazolyl, thiazolyl, 1,2,4-oxadiazol-3-yl, 1,2,4-thiadiazol-3-yl, 1,2,4-thiadiazol-5-yl, 1,2,5-thiadiazol-3-yl, 1,3,4-thiadiazol-2-yl or C.sub.1 -C.sub.5 -alkyl radical, or the group --CH.sub.2 --Y--R.sup.1, where Y is oxygen or sulfur and R.sup.1 is C.sub.1 -C.sub.6 -alkoxyethyl or C.sub.1 -C.sub.6 -alkoxyethoxyethyl, or R is C.sub.2 -C.sub.5 -alkenyl, C.sub.2 -C.sub.5 -alkynyl, C.sub.1 -C.sub.5 -alkoxy, C.sub.1 -C.sub.5 -alkoxycarbonyl or C.sub.3 -C.sub.7 -cycloalkyl, and fungicides containing these compounds.
Abstract:
This invention relates to 8-aza-11,12-secoprostaglandins and processes for their manufacture. These compounds have prostaglandin-like biological activity and are particularly useful as renal vasodilators.
Abstract:
A compound which is 4-(3,5-dihydroxy-3-methylpentylamide)butyric acid or its pharmaceutically acceptable salt or ester; this compound being produced by reacting a salt or an ester of gamma-aminobutyric acid with beta-hydroxy-beta-methyl-delta-valerolactone, and as required, converting the resulting compound in the form of a salt or ester to a free acid, or as required, converting the resulting compound in the form of a free acid to its pharmaceutically acceptable salt or ester; and useful as a medicament for preventing or treating an impediment in cerebral function.
Abstract:
Novel fabric softener compounds having the formula ##STR1## wherein R is hydrogen or methyl, R.sub.1 and R.sub.2 are the same or different and are selected from linear and branched chain alkyl groups having from 8 to 22 carbon atoms; R.sub.3 is selected from hydrogen, formyl, acetyl, benzoyl; R.sub.4 and R.sub.5 being the same or different and selected from lower alkyl groups having from 1 to 4 carbon atoms, -hydroxyalkyl groups having from 2 to 4 carbon atoms and R.sub.4 and R.sub.5 taken together are diethylene oxide, R.sub.6 is selected from hydrogen, lower alkyl having from 1 to 4 carbon atoms and benzyl; n is a whole number selected from 2 to 10; and A is an anion selected from methyl sulfate, ethyl sulfate, chlorides, fluorides, sulfates, acetates, bromides, iodides, benzoates and gluconates.
Abstract:
N,N-disubstituted acryl- and methacrylamides are disclosed wherein one of the amido nitrogen atom substituents is an n-propionate radical and the other of such substituents is a hydrocarbyl group. The disclosed compounds are useful as comonomers for the preparation of polyvinyl resinous systems in general.
Abstract:
1-(Bis-ethoxycarbonyl)-acetylamino-3-methyl-3-(bis-ethoxycarbonyl)-acetylaminomethyl-5-dimethyl-cyclohexane, a new blocked diisocyanate, its manufacture from isophorone diisocyanate and diethyl malonate, and its use.
Abstract:
A PROCESS FOR TRANSFORMING AN ALKYL AMINO ACID SALT OF A MINERAL ACID INTO THE CORRESPONDING N-ACYL AMINO ALKANOIC ACID COMPRISING NEUTRALIZING THE MINERAL ACID PORTION. THE AMMONIUM SALT IS SEPARATED OUT BY ADDING ALKADROXIDE, SEPARATING OUT THE THEREBY FORMED AMMONIUM SALT OF THE MINERAL ACID, AND ACYLATING THE REMAINING SOLUTION. THE AMMONIUM SALT IS SEPARATED OUT BY ADDING ALKANOC ACID TO THE NEUTRALIZED SOLUTION.