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    NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE
    91.
    发明申请
    NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE 审中-公开
    新型吡哩啶-4-酮和吡哩啶-4-基作为杀真菌剂

    公开(公告)号：WO9914202A3

    公开(公告)日：1999-05-14

    申请号：PCT/EP9805790

    申请日：1998-09-10

    申请人： NOVARTIS AG ,  NOVARTIS ERFIND VERWALT GMBH ,  WALTER HARALD

    发明人： WALTER HARALD

    IPC分类号： A01N43/54 ,  A01N43/90 ,  C07D239/86 ,  C07D239/90 ,  C07D239/91 ,  C07D239/92 ,  C07D471/04 ,  C07D487/04 ,  C07D495/04 ,  C07D513/04 ,  C07F7/10

    CPC分类号： C07D471/04 ,  A01N43/54 ,  A01N43/90 ,  C07D239/86 ,  C07D239/90 ,  C07D239/91 ,  C07D239/92 ,  C07D495/04 ,  C07D513/04

    摘要： Novel pyrimidin-4-one and pyrimidin-4-thione derivatives of formula (I) wherein A is phenyl, thienyl (including all 3 isomers), thiazolyl, pyridyl or pyridazinyl; X is oxygen or sulfur; R1 is hydrogen, halogen or trimethylsilyl; R2 is hydrogen, halogen or trimethylsilyl; at least one of R1 and R2 is not hydrogen; R3 is C1-C8alkyl, C1-C8alkenyl, C1-C8alkinyl which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen, C1-C6alkoxy or C1-C6haloalkoxy; O-C1-C6alkyl, O-C2-C6alkenyl, O-C2-C6alkynyl, which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen or C1-C6alkoxy; N-C1-C6alkyl; or N=CHC1-C6alkyl; R4 is C1-C8alkyl, C1-C8alkenyl, C1-C8alkinyl which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen, cyano, C1-C6alkoxy or C1-C6haloalkoxy; C1-C4alkoxy-C1-C4alkoxy; C1-C4alkoxy-C1-C4alkylthio; nitro; -CO-C1-C6alkyl; C3-C6cycloalkyl; or phenyl, which is unsubstitued or mono to tri-substituted by halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, cyano, nitro, amino, mono-C1-C6alkylamino, di-C1-C6alkylamino, C1-C6alkylthio, phenyl or phenoxy and in which the phenyl part is unsubstituted or mono to tri-substituted by halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy. The novel compounds have plant-protective properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms, in particular fungi.

    摘要翻译： 式（I）的新型嘧啶-4-酮和嘧啶-4-硫酮衍生物，其中A是苯基，噻吩基（包括所有3个异构体），噻唑基，吡啶基或哒嗪基; X是氧或硫; R1是氢，卤素或三甲基甲硅烷基; R2是氢，卤素或三甲基甲硅烷基; R1和R2中的至少一个不是氢; R3是C1-C8烷基，C1-C8链烯基，C1-C8炔基，其未被取代或被C3-C6环烷基，卤素，C1-C6烷氧基或C1-C6卤代烷氧基单取代或三取代。 O-C 1 -C 6烷基，O-C 2 -C 6烯基，O-C 2 -C 6炔基，其未被取代或被C 3 -C 6环烷基，卤素或C 1 -C 6烷氧基单取代至三取代; N-C 1 -C 6烷基; 或N = CHCl-C6烷基; R4是C1-C8烷基，C1-C8链烯基，C1-C8炔基，它们是未取代的或被C3-C6环烷基，卤素，氰基，C1-C6烷氧基或C1-C6卤代烷氧基单取代或三取代。 C1-C4烷氧基-C1-C4烷氧基; C1-C4烷氧基，C1-C4烷硫基; 硝基; -CO-C1-C6烷基; C3-C6环烷基; C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，氰基，硝基，氨基，单C 1 -C 6烷基氨基，二-C 1 -C 6烷基氨基，C 1 -C 6烷氧基 C 1-6烷硫基，苯基或苯氧基，其中苯基部分是未取代的或被卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基或C 1 -C 6卤代烷氧基单取代或三取代。 新化合物具有植物保护性质，并且适用于保护植物免受植物病原微生物特别是真菌的侵袭。

    NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE
    92.
    发明申请
    NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE 审中-公开
    嘧啶-4-酮和嘧啶-4-脯氨酸新用作杀真菌剂

    公开(公告)号：WO99014202A2

    公开(公告)日：1999-03-25

    申请号：PCT/EP1998/005790

    申请日：1998-09-10

    IPC分类号： A01N43/54 ,  A01N43/90 ,  C07D239/86 ,  C07D239/90 ,  C07D239/91 ,  C07D239/92 ,  C07D471/04 ,  C07D487/04 ,  C07D495/04 ,  C07D513/04 ,  C07D239/00

    CPC分类号： C07D471/04 ,  A01N43/54 ,  A01N43/90 ,  C07D239/86 ,  C07D239/90 ,  C07D239/91 ,  C07D239/92 ,  C07D495/04 ,  C07D513/04

    摘要： Novel pyrimidin-4-one and pyrimidin-4-thione derivatives of formula (I) wherein A is phenyl, thienyl (including all 3 isomers), thiazolyl, pyridyl or pyridazinyl; X is oxygen or sulfur; R1 is hydrogen, halogen or trimethylsilyl; R2 is hydrogen, halogen or trimethylsilyl; at least one of R1 and R2 is not hydrogen; R3 is C1-C8alkyl, C1-C8alkenyl, C1-C8alkinyl which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen, C1-C6alkoxy or C1-C6haloalkoxy; O-C1-C6alkyl, O-C2-C6alkenyl, O-C2-C6alkynyl, which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen or C1-C6alkoxy; N-C1-C6alkyl; or N=CHC1-C6alkyl; R4 is C1-C8alkyl, C1-C8alkenyl, C1-C8alkinyl which are unsubstituted or mono to tri-substituted by C3-C6cycloalkyl, halogen, cyano, C1-C6alkoxy or C1-C6haloalkoxy; C1-C4alkoxy-C1-C4alkoxy; C1-C4alkoxy-C1-C4alkylthio; nitro; -CO-C1-C6alkyl; C3-C6cycloalkyl; or phenyl, which is unsubstitued or mono to tri-substituted by halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, cyano, nitro, amino, mono-C1-C6alkylamino, di-C1-C6alkylamino, C1-C6alkylthio, phenyl or phenoxy and in which the phenyl part is unsubstituted or mono to tri-substituted by halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy. The novel compounds have plant-protective properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms, in particular fungi.

    摘要翻译： 本发明涉及新的嘧啶-4-酮和嘧啶-4-硫酮，对应于式（I）其中A是苯基，噻吩基（包括三种异构体），噻唑基，吡啶基或哒嗪基; X表示氧或硫，R 1表示氢，卤素或三甲基甲硅烷，R 2是氢，卤素或三甲基甲硅烷，R 1和R 2不表示氢的至少一种，R 3表示C1-C8链烯基，C1-C8炔基C1 C8烷基，-O-C1-C6烷基，O- C2-C6链烯基，O-（其不被C3-C6环烷基，卤素，C1-C6烷氧基或卤代烷C1-C6取代的或有一至三次） 炔基C2-C6（其不被C3-C6环烷基，卤素或C1-C6烷氧基取代的或者是一至三次），N-C1-C6烷基，或N = C1-C6烷基，R 4代表C 1烷基 C8烯基，C1-C8炔基C 1 -C 8烷氧基，C 1 -C 4（其不被C3-C6环烷基，卤素，氰基，C1-C6烷氧基或卤代烷C1-C6取代的或有一至三次） C1-C4烷氧基，C1-C4烷氧基C1-C4烷硫基，硝基，-CO-C1-C6烷基，C3-C6环烷基，或苯基（其可以不被取代或者是一至三次被卤素 ，al 凯尔C1-C6卤代烷基，C1-C6烷氧基C1-C6卤代烷氧基C1-C6烷基，氰基，硝基，氨基，单 - 烷基氨基C 1 -C 6二烷基氨基C1-C6烷硫基C1-C6烷基，苯基或苯氧基和 其中苯基部分未被取代或被卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基或C 1 -C 6卤代烷氧基取代1-3次。 这些新型化合物具有植物保护特性，并特别设计用于保护植物免受植物病原微生物（主要是真菌）侵染。

    SUBSTITUTED QUINAZOLIN(THI)ONES
    94.
    发明申请
    SUBSTITUTED QUINAZOLIN(THI)ONES 审中-公开
    取代喹唑啉（硫）

    公开(公告)号：WO1997007105A1

    公开(公告)日：1997-02-27

    申请号：PCT/EP1996003469

    申请日：1996-08-06

    申请人： BAYER AKTIENGESELLSCHAFT ,  DREWES, Mark, Wilhelm ,  ANDREE, Roland ,  DOLLINGER, Markus

    发明人： BAYER AKTIENGESELLSCHAFT

    IPC分类号： C07D239/93

    CPC分类号： C07D239/90 ,  A01N43/54 ,  C07D239/93

    摘要： The invention concerns novel substituted quinazolin(thi)ones of general formula (I) in which Q, R , R , R , R , R and R have the meanings given in the description. The invention also concerns a process for their preparation and their use as herbicides.

    摘要翻译： 本发明涉及新的取代的喹唑啉的通式（I）的（硫）这样的，其中Q，R <1>，R <2>，R <3>，R <4>，R <5>和R <6> 具有说明书中给出的含义，它们的制备方法和它们作为除草剂的用途。

    NOVEL NON-CLASSICAL FOLATE ANALOGUE INHIBITORS OF GLYCINAMIDE RIBONUCLEOTIDE FORMYLTRANSFERASE (GARFT)
    95.
    发明申请
    NOVEL NON-CLASSICAL FOLATE ANALOGUE INHIBITORS OF GLYCINAMIDE RIBONUCLEOTIDE FORMYLTRANSFERASE (GARFT) 审中-公开
    甘氨酰胺呋喃糖苷（GARFT）的新型非经典酯类化合物抑制剂

    公开(公告)号：WO1996040680A1

    公开(公告)日：1996-12-19

    申请号：PCT/US1996010449

    申请日：1996-06-07

    申请人： NAIR, Madhavan, G.

    发明人： LIU, Li

    IPC分类号： C07D401/06

    CPC分类号： C07D239/90 ,  C07D239/95

    摘要： Several new 10-formyl and 10-hydroxymethyl derivatives of 5,8,10-trideazapteroic acid are provided, as well as procedures for their preparation. These compounds were shown to be powerful inhibitors of glycinamide ribonucleotide formyltransferase (GARFT), an enzyme that mediates the de novo biosynthesis of purine nucleotides that are required for DNA synthesis and cell division. Due to their ability to interfere with nucleotide biosynthesis and to penetrate microbial cells they are anti-microbial agents and are useful for the treatment of Pneumocystis carinii infection in AIDS and other infections responding to folate based antimicrobial agents.

    摘要翻译： 提供了5,8,10-十三碳八烯酸的几种新的10-甲酰基和10-羟甲基衍生物及其制备方法。 这些化合物被证明是强大的甘氨酰胺核糖核苷酸甲酰转移酶抑制剂（GARFT），其是介导DNA合成和细胞分裂所需的嘌呤核苷酸的从头生物合成的酶。 由于它们干扰核苷酸生物合成和渗透微生物细胞的能力，它们是抗微生物剂，并且可用于治疗艾滋病卡氏肺囊虫感染和对叶酸类抗微生物剂的其它感染。

    PYRIMIDINE DERIVATIVE
    97.
    发明申请
    PYRIMIDINE DERIVATIVE 审中-公开
    吡啶衍生物

    公开(公告)号：WO1994008975A1

    公开(公告)日：1994-04-28

    申请号：PCT/JP1993001478

    申请日：1993-10-14

    申请人： NIPPON SODA CO., LTD. ,  YAMADA, Hirokazu ,  TANAKA, Katsunori ,  ADACHI, Hiroyuki ,  YAMADA, Shigeo ,  SHIMODA, Susumu ,  HASHIMOTO, Sho ,  UMEDA, Nobuhiro

    发明人： NIPPON SODA CO., LTD.

    IPC分类号： C07D239/26

    CPC分类号： C07D239/28 ,  A01N43/54 ,  A01N43/90 ,  A01N47/24 ,  A01N57/24 ,  C07D239/34 ,  C07D239/36 ,  C07D239/38 ,  C07D239/40 ,  C07D239/42 ,  C07D239/47 ,  C07D239/86 ,  C07D239/90 ,  C07D239/91 ,  C07D239/93 ,  C07D471/04 ,  C07D487/04 ,  C07D491/04 ,  C07D495/04 ,  C07F7/0812 ,  C07F9/6512 ,  C07F9/6561

    摘要： A compound represented by general formula (I) and excellent in herbicidal and agrohorticultural antibacterial activities, wherein R and R represent each hydrogen, alkyl, etc., or alternatively they may be combined together to represent oxo, thioxo, etc., or a spiro ring selected from among (a), (b), etc.; R and R represent each hydrogen, halogen, alkyl, etc., and R represents hydrogen, halogen, amino, etc., provided that R and R are different from each other when R is hydrogen and that R may be combined with R or R and the pyrimidine ring to represent a condensed ring represented by (c) or (d); R and R represent each hydrogen, halogen, alkyl, etc., provided that the case wherein both R and R represent hydrogen is excluded; R represents halogen, alkyl, etc.; and n represents 0, 1, 2 or 3; provided that when both R and R represent hydrogen, then R is combined with R or R and the pyrimidine group to represent the above condensed ring.

    摘要翻译： 由通式（I）表示的化合物，除草和农业园艺抗菌活性优异，其中R 1和R 2代表每个氢，烷基等，或者它们可以组合在一起代表氧代，硫代， 或选自（a），（b）等的螺环; R 3和R 5分别表示氢，卤素，烷基等，R 4表示氢，卤素，氨基等，条件是R 3和R 5不同于 另外当R 4为氢时，R 4可以与R 3或R 5结合，嘧啶环表示（c）或（d）所示的稠环; R 6和R 7各自代表氢，卤素，烷基等，条件是其中R 6和R 7均表示氢的情况除外; R 8表示卤素，烷基等; n表示0,1,2或3; 条件是当R 1和R 2都表示氢时，则R 4与R 3或R 5和嘧啶基团组合以代表上述稠环。

    PROPENOIC ACID DERIVATIVES USEFUL AS FUNGICIDES
    98.
    发明申请
    PROPENOIC ACID DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
    丙烯酸衍生物作为防腐剂有用

    公开(公告)号：WO1994008968A1

    公开(公告)日：1994-04-28

    申请号：PCT/GB1993001990

    申请日：1993-09-22

    申请人： ZENECA LIMITED ,  DE FRAINE, Paul, John ,  PILKINGTON, Brian, Leslie

    发明人： ZENECA LIMITED

    IPC分类号： C07D217/14

    CPC分类号： C07D239/26 ,  A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  C07C251/60 ,  C07C2601/08 ,  C07C2601/14 ,  C07D213/64 ,  C07D217/14 ,  C07D239/90 ,  C07D401/04 ,  C07D487/04 ,  C07D495/04

    摘要： A fungicidal compound having formula (I), wherein either: A is hydrogen, halogen, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, phenoxy, nitro or cyano; and one of R and R is optionally substituted isoquinoline while the other is hydrogen, C1-4 alkyl, C1-4 haloalkyl, halogen or cyano; or A is hydrogen, R is methyl and R is 4-t &cir& _e &cir& _r &cir& _t &cir& _-butylpyrid-2-yl, 4t &cir& _e &cir& _r &cir& _t &cir& _-butylpyrimidin-2-yl, 5-methyl-6-i &cir& _s &cir& _o &cir& _-propoxypyrimidin-4-yl or 4-(C1-4 chlorofluoroalkyl)pyrid-2-yl.

    摘要翻译： 具有式（I）的杀真菌化合物，其中：A是氢，卤素，羟基，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基，C 1-4卤代烷氧基，C 1-4烷基羰基，C 1-4烷氧基羰基， 苯氧基，硝基或氰基; R 1和R 2之一是任选取代的异喹啉，而另一个是氢，C 1-4烷基，C 1-4卤代烷基，卤素或氰基; 或A为氢，R 2为甲基，R 1为4-叔丁基 - 吡啶-2-基，4'，“ - ” - “和” ，5-甲基-6-氨基嘧啶-4-基或4-（C1-4氯氟代烷基）吡啶-2-基。