SUBSTITUTED QUINAZOLINE DERIVATIVES
    54.
    发明授权
    SUBSTITUTED QUINAZOLINE DERIVATIVES 有权
    取代衍生物Chinazolines

    公开(公告)号:EP1100788B1

    公开(公告)日:2005-11-09

    申请号:EP99939658.3

    申请日:1999-07-28

    申请人: Wyeth

    摘要: This invention provides a process for preparing compounds of formula (1) wherein: X is phenyl optionally substituted with one or more substituents selected from the group consisting of halogen, alkyl of 1-6 carbon atoms, alkoxy of 1-6 carbon atoms, hydroxy, trifluoromethyl, cyano, nitro, carboxy, carboalkoxy of 2-7 carbon atoms, carboalkyl of 2-7 carbon atoms, amino, and alkanoylamino of 1-6 carbon atoms; R and R1 are each, independently, hydrogen, halogen, alkyl of 1-6 carbon atoms, alkoxy of 1-6 carbon atoms, hydroxy, or trifluoromethyl; R2 is hydrogen, alkyl of 1-6 carbon atoms, alkoxy of 1-6 carbon atoms, hydroxy, trifluoromethyl; Y is (2) or (3); R3 is independently hydrogen, alkyl of 1-6 carbon atoms, carboxy, carboalkoxy of 1-6 carbon atoms, phenyl, or carboalkyl of 2-7 carbon atoms; n = 2-4; or a pharmaceutically acceptable salt thereof, with the proviso that each R3 of Y may be the same or different.

    N-BIPHENYLAMIDES AND FUNGICIDAL COMPOSITIONS CONTAINING THE SAME
    57.
    发明公开
    N-BIPHENYLAMIDES AND FUNGICIDAL COMPOSITIONS CONTAINING THE SAME 审中-公开
    N-BIPHENYLAMIDE UND DIEE ENTHALTENDE FUNGIZIDE ZUSAMMENSETZUNGEN

    公开(公告)号:EP1486483A1

    公开(公告)日:2004-12-15

    申请号:EP03707030.7

    申请日:2003-02-25

    摘要: A N-biphenylamide compound of the formula (1):
    wherein R 1 , R 2 , R 3 , R 4 and R 5 independently represent a hydrogen atom, halogen atom or the like, R 6 represents C1-C6 alkyl and the like, R 7 represents a hydrogen atom or C1-C3 alkyl,
    R 8 represents a hydrogen atom or C1-C3 alkyl,
    R 9 and R 10 independently represents a halogen atom, C1-C6 alkyl, C1-C6 alkoxy or the like,
    R 11 , R 12 and R 13 independently represent a hydrogen atom, halogen atom or the like, R 14 , R 15 , R 16 and R 17 independently is a hydrogen atom, halogen atom or the like, X 1 represents an oxygen atom or sulfur atom, X 2 represents an oxygen atom or sulfur atom;
    has excellent effect aginst plant diseases.

    摘要翻译: 式(1)的N-联苯酰胺化合物:其中R 1,R 2,R 3,R 4和R 5独立地表示氢原子,卤素原子或 R 6表示C 1 -C 6烷基等,R 7表示氢原子或C 1 -C 3烷基,R 8表示氢原子或C 1 -C 3烷基,R 9和R 8, R 10独立地表示卤素原子,C 1 -C 6烷基,C 1 -C 6烷氧基等,R 11,R 12和R 13独立地表示氢原子,卤素原子等,R 14 R 15,R 16和R 17独立地为氢原子,卤素原子等,X 1表示氧原子或硫原子,X 2表示氧原子或硫原子 原子; 具有优良的植物病害效果。