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1.发明公开DIHYDRO-PYRROLOPYRIDIN-, DIHYDRO-PYRROLOPYRIDAZIN- UND DIHYDRO-PYRROLOPYRIMIDIN-DERIVATE UND IHRE VERWENDUNG 审中-公开二氢PYRROLOPYRIDIN-，二氢PYRROLOPYRIDAZIN-和二氢吡咯衍生物及其
公开(公告)号：EP2029589A1
公开(公告)日：2009-03-04
申请号：EP07725591.7
申请日：2007-05-25
申请人： Bayer HealthCare AG
IPC分类号： C07D471/04 , C07D487/04 , A61P7/02 , A61K31/437 , A61K31/519
CPC分类号： C07D487/04 , C07D471/04
摘要： The invention relates to novel dihydro-pyrrolopyridine-, dihydro-pyrrolopyridazine- and dihydro-pyrrolopyrimidine-derivatives, to methods for the production thereof, to the use thereof for treating and/or preventing diseases, and to the use thereof for producing medicaments for treating and/or preventing diseases, in particular thromboembolic diseases.
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2.发明授权
公开(公告)号：EP1751153B1
公开(公告)日：2008-12-03
申请号：EP05740054.1
申请日：2005-03-30
申请人： Bayer HealthCare AG
发明人： SCHIROK, Hartmut , RADTKE, Martin , MITTENDORF, Joachim , KAST, Raimund , STASCH, Johannes-Peter , GNOTH, Mark, Jean , MÜNTER, Klaus , LANG, Dieter , FIGUEROA, PEREZ, Santiago , THUTEWOHL, Michael , BENNABI, Samir , EHMKE, Heimo
IPC分类号： C07D471/04 , A61K31/437 , A61P9/00
CPC分类号： C07D471/04
摘要： The invention relates to hetaryloxy-substituted phenylamino pyrimidines, a method for the production thereof, and the use thereof for producing medicaments utilized for the treatment and/or prevention of diseases in humans and animals, particularly cardiovascular diseases.
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3.发明公开
公开(公告)号：EP1751153A1
公开(公告)日：2007-02-14
申请号：EP05740054.1
申请日：2005-03-30
申请人： Bayer HealthCare AG
发明人： SCHIROK, Hartmut , RADTKE, Martin , MITTENDORF, Joachim , KAST, Raimund , STASCH, Johannes-Peter , GNOTH, Mark, Jean , MÜNTER, Klaus , LANG, Dieter , FIGUEROA, PEREZ, Santiago , THUTEWOHL, Michael , BENNABI, Samir , EHMKE, Heimo
IPC分类号： C07D471/04 , A61K31/437 , A61P9/00
CPC分类号： C07D471/04
摘要： The invention relates to hetaryloxy-substituted phenylamino pyrimidines, a method for the production thereof, and the use thereof for producing medicaments utilized for the treatment and/or prevention of diseases in humans and animals, particularly cardiovascular diseases.
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4.发明公开PYRAZOLINE ALS PAR-1-ANTAGONISTEN ZUR BEHANDLUNG VON HERZ-KREISLAUF-ERKRANKUNGEN 审中-公开吡唑啉ALS PAR-1拮抗剂用于治疗心血管疾病的治疗
公开(公告)号：EP1648447A1
公开(公告)日：2006-04-26
申请号：EP04740582.4
申请日：2004-07-02
申请人： Bayer HealthCare AG
发明人： ALLERHEILIGEN, Swen , BROHM, Dirk , DIEDRICHS, Nicole , FRÖHLEN, Britta-Nicole , GERDES, Christoph , GNOTH, Mark, Jean , HECKROTH, Heike , HÜBSCH, Walter , PERZBORN, Elisabeth , STAHL, Elke , VÖHRINGER, Verena
IPC分类号： A61K31/4155 , A61P9/00 , C07D403/04 , C07D409/14 , C07D405/14 , C07D401/14 , C07D413/04 , C07D417/04 , C07D403/14 , C07D401/04 , C07D417/14 , C07D413/14
CPC分类号： C07D401/04 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/04 , C07D417/14
摘要： The invention relates to pyrazolines of formula (I), where E = methylene, NH, O or S and R2 = a group of formula (II), methods for the production and use thereof for the production of medicaments for the treatment and/or prophylaxis of diseases, in particular, cardiovascular diseases, such as thromboembolitic diseases.
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公开(公告)号：EP2079708A2
公开(公告)日：2009-07-22
申请号：EP07818862.0
申请日：2007-10-10
申请人： Bayer HealthCare AG
发明人： BAUSER, Marcus , BUCHMÜLLER, Anja , VON DEGENFELD, Georges , DITTRICH-WENGENROTH, Elke , GERDES, Christoph , GNOTH, Mark, Jean , GOTTSCHLING, Dirk , HEITMEIER, Stefan , HENDRIX, Martin , KÖBBERLING, Johannes , LANG, Dieter , RESTER, Ulrich , SAATMANN, Uwe , TERSTEEGEN, Adrian , BRÜNS, Astrid
IPC分类号： C07D233/88
CPC分类号： C07D233/88 , C07D277/20 , C07D401/14 , C07D403/04 , C07D405/14 , C07D417/12
摘要： The invention relates to acyl aminoimidazoles and acyl aminothiazoles, to a method for producing same and to the use thereof for producing medicaments for the treatment and/or prevention of diseases, in particular cardiovascular diseases, preferably thromboembolic diseases.
摘要翻译： 本发明涉及酰基氨基咪唑和酰基氨基噻唑，其制备方法及其用于制备用于治疗和/或预防疾病，特别是心血管疾病，优选血栓栓塞性疾病的药物。
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6.发明公开SUBSTITUIERTE (OXAZOLIDINON-5-YL-METHYL) -2-THIOPHEN-CARBOXAMIDE UND IHRE VERWENDUNG IM GEBIET DER BLUTGERINNUNG 有权SUBSTITUIERTE（恶唑烷酮-5-基 - 甲基）-2-噻吩 - 甲酰胺和IHRE VERWENDUNG IM GEBIET DER BLUTGERINNUNG
公开(公告)号：EP2173744A1
公开(公告)日：2010-04-14
申请号：EP08759099.8
申请日：2008-06-07
申请人： Bayer HealthCare AG
发明人： ALLERHEILIGEN, Swen , BAUSER, Marcus , SCHIROK, Hartmut , RESTER, Ulrich , HEITMEIER, Stefan , GERDES, Christoph , VON DEGENFELD, Georges , DITTRICH-WENGENROTH, Elke , SAATMANN, Uwe , STRASSBURGER, Julia , MÜNTER, Klaus , GNOTH, Mark, Jean , LANG, Dieter
IPC分类号： C07D413/14 , A61K31/4439 , A61P7/00
CPC分类号： C07D413/14
摘要： The invention relates to novel substituted oxazolidinones, methods for the production thereof, use thereof for treating and/or for the prophylaxis of diseases and use thereof for producing medicaments for treating and/or for the prophylaxis of diseases, in particular thromboembolic disorders.
摘要翻译： 本发明涉及新的取代的恶唑烷酮，其制备方法，其用于治疗和/或预防疾病的用途以及用于制备用于治疗和/或预防疾病，特别是血栓栓塞性疾病的药物的用途。
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7.发明公开SUBSTITUIERTE (OXAZOLIDINON-5-YL-METHYL) -2-THIOPHEN-CARBOXAMIDE UND IHRE VERWENDUNG IM GEBIET DER BLUTGERINNUNG 有权取代的（恶唑烷酮-5-基 - 甲基）-2-噻吩甲酰胺和它们在血液凝固领域
公开(公告)号：EP2170877A1
公开(公告)日：2010-04-07
申请号：EP08773372.1
申请日：2008-06-07
申请人： Bayer HealthCare AG
发明人： ALLERHEILIGEN, Swen , BAUSER, Marcus , HEIMBACH, Dirk , HEITMEIER, Stefan , GNOTH, Mark, Jean , GERDES, Christoph , VON DEGENFELD, Georges , RÖHRIG, Susanne , RESTER, Ulrich , DITTRICH-WENGENROTH, Elke , SAATMANN, Uwe , TERSTEEGEN, Adrian
IPC分类号： C07D413/14 , A61K31/4439 , A61P7/00
CPC分类号： C07D413/14
摘要： The invention relates to novel substituted oxazolidinones, methods for the production thereof, use thereof for treating and/or for the prophylaxis of diseases and use thereof for producing medicaments for treating and/or for the prophylaxis of diseases, in particular thromboembolic disorders.
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8.发明公开PHENYL SUBSTITUIERTE PIPERAZIN-DERIVATE ALS HEMMER VOM PLAMINOGEN AKTIVATOR INHIBITOR-I (PAI-I) 审中-公开苯基取代的哌嗪衍生物作为激活物抑制物纤溶酶原-I（PAI-I）抑制剂
公开(公告)号：EP1907363A1
公开(公告)日：2008-04-09
申请号：EP06762520.2
申请日：2006-07-11
申请人： Bayer HealthCare AG
发明人： WILMEN, Andreas , STRASSBURGER, Julia , GNOTH, Mark, Jean , GERDES, Christoph , FRÖHLEN, Britta-Nicole , SIEGEL, Stephan
IPC分类号： C07D213/82 , C07D213/81 , A61K31/444 , A61P7/02
CPC分类号： C07D213/81 , C07D213/82
摘要： The invention relates to substituted pyridocarboxamides, to a method for the production thereof and to the use thereof in the production of medicaments for the treatment and/or prophylaxis of illnesses in humans and animals, in particular thrombotic diseases.
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9.发明公开2- (HETEROARYL) ALKYL-INDAZOLE-6-PHENYL UND THIENYLMETHYLAMIDE ALS THROMBININHIBITOREN 审中-公开2-（异丁基）烷基 - 吲哚-6-基苯甲酰甲基硫代吗啉
公开(公告)号：EP2044031A1
公开(公告)日：2009-04-08
申请号：EP07764989.5
申请日：2007-07-02
申请人： Bayer HealthCare AG
发明人： SIEGEL, Stephan , SCHNEIDER, Dirk , BUCHMÜLLER, Anja , DITTRICH-WENGENROTH, Elke , GERDES, Christoph , GNOTH, Mark, Jean , HEITMEIER, Stefan , HENDRIX, Martin c/o Bayer Healthcare LLC , RESTER, Ulrich , SAATMANN, Uwe
IPC分类号： C07D231/52 , C07D417/06 , C07D401/06 , C07D413/06 , C07D403/06 , C07D401/14 , A61K31/416 , A61K31/421 , A61K31/427 , A61K31/4196 , A61K31/4402 , A61K31/445 , A61K31/5377
CPC分类号： C07D403/06 , C07D231/52 , C07D231/56 , C07D401/06 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/06 , C07D417/06
摘要： The invention relates to substituted indazols and methods for the production thereof, as well as to the utilization thereof in the production of drugs to treat and/or prevent illnesses, in particular illnesses of the cardiovascular system and, preferably, thrombo-embolic illnesses.
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10.发明公开SUBSTITUIERTE PYRIDOCARBOXAMIDE ALS HEMMER VOM PLASMINOGEN AKTIVATOR INHIBITOR-1 (PAI-I) 审中-公开取代PYRIDOCARBOXAMIDE纤溶酶原激活物抑制剂-1的抑制剂（PAI-I）
公开(公告)号：EP1910295A1
公开(公告)日：2008-04-16
申请号：EP06818239.3
申请日：2006-07-20
申请人： Bayer HealthCare AG
发明人： SIEGEL, Stephan , FRÖHLEN, Britta-Nicole , GERDES, Christoph , GNOTH, Mark, Jean , STRASSBURGER, Julia , WILMEN, Andreas
IPC分类号： C07D213/82 , C07D213/81 , A61K31/44 , A61P7/02
CPC分类号： C07D213/81 , C07D213/82
摘要： The invention relates to substituted pyridocarboxamides, to a process for preparing them and to their use for producing medicaments for the treatment and/or prophylaxis of diseases in humans and animals, particularly of thrombotic disorders.
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