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1.发明公开NEUE 2-ARYL-THIAZOL-4-CARBONSÄUREAMID-DERIVATE, DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL 有权NEW 2-芳基噻唑-4-羧酸酰胺衍生物，生产和使用AS DRUGS
公开(公告)号：EP2240457A1
公开(公告)日：2010-10-20
申请号：EP08877913.7
申请日：2008-12-02
发明人： BOTHE, Ulrich , VON BONIN, Arne , NGUYEN, Duy , BÖMER, Ulf , GUENTHER, Judith
IPC分类号： C07D277/32
CPC分类号： C07D277/56 , C07D417/04 , C07D417/12 , C07D417/14 , C07D495/04
摘要： The invention relates to 2-aryl thiazole-4-carboxamide derivatives of formula (I), the use thereof as a medicament for treating various diseases, and methods for the production thereof.
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2.发明公开CYANOQUINOLINE DERIVATIVES, THEIR PREPARATION, THEIR USE, AND MEDICAMENTS COMPRISING THEM 审中-公开CYANOCHINOLINDERIVATE，生产，使用和药物它们含有
公开(公告)号：EP2035433A1
公开(公告)日：2009-03-18
申请号：EP07764743.6
申请日：2007-06-15
发明人： PRIEN, Olaf , EIS, Knut , SCHWEDE, Wolfgang , GUENTHER, Judith , ZOPF, Dieter
IPC分类号： C07D495/04 , A61P35/00 , A61K31/435
CPC分类号： C07D495/04
摘要： The present invention relates to a quinoline derivative having the general formula (A) : in which R1, R2, X, Y and Z are indicated in the description and the claims, the use of the compounds of the general formula (A) for the treatment of various disorders, and the preparation of compounds of the general formula (A).
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3.发明授权NEUE 2-ARYL-THIAZOL-4-CARBONSÄUREAMID-DERIVATE, DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL 有权NEW 2-芳基噻唑-4-羧酸酰胺衍生物，生产和使用AS DRUGS
公开(公告)号：EP2240457B1
公开(公告)日：2011-05-11
申请号：EP08877913.7
申请日：2008-12-02
发明人： BOTHE, Ulrich , VON BONIN, Arne , NGUYEN, Duy , BÖMER, Ulf , GUENTHER, Judith
IPC分类号： C07D277/32
CPC分类号： C07D277/56 , C07D417/04 , C07D417/12 , C07D417/14 , C07D495/04
摘要： The invention relates to 2-aryl thiazole-4-carboxamide derivatives of formula (I), the use thereof as a medicament for treating various diseases, and methods for the production thereof.
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4.发明公开QUINAZOLINE DERIVATIVES, THEIR PREPARATION, THEIR USE AS TYROSINE KINASE INHIBITORS AND MEDICAMENTS COMPRISING THEM 审中-公开喹唑啉衍生物，生产，它们的使用药物和酪氨酸激酶抑制剂，含
公开(公告)号：EP2041143A1
公开(公告)日：2009-04-01
申请号：EP07764744.4
申请日：2007-06-15
发明人： PRIEN, Olaf , EIS, Knut , SCHWEDE, Wolfgang , GUENTHER, Judith , ZOPF, Dieter , BRITTAIN, Dominic, E., A.
IPC分类号： C07D495/04 , A61K31/517 , A61P25/00 , A61P25/16 , A61P25/28 , A61P29/00
CPC分类号： C07D513/04 , C07D239/70 , C07D487/04 , C07D491/04 , C07D495/04
摘要： The present invention relates to a quinazoline derivative having the general formula (A): in which R1, R2, X, Y and Z are indicated in the description and the claims, the use of the compounds of the general formula (A) for the treatment of various disorders, and the preparation of compounds of the general formula (A).
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5.发明公开
公开(公告)号：EP2035434A1
公开(公告)日：2009-03-18
申请号：EP07764746.9
申请日：2007-06-15
发明人： PRIEN, Olaf , EIS, Knut , NGUYEN, Duy , HUWE, Christoph , SCHWEDE, Wolfgang , GUENTHER, Judith , ZOPF, Dieter
IPC分类号： C07D495/04 , A61P35/00 , A61K31/435
CPC分类号： C07D513/04 , C07D495/04
摘要： The present invention relates to a quinoline derivative having the general formula (A) : in which R1, R2, W, X, Y and Z are indicated in the description and the claims, the use of the compounds of the general formula (A) for the treatment of various disorders, and the preparation of compounds of the general formula (A).
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6.发明公开NEUE 2-SUBSTITUIERTE TIAZOL-4-CARBONSÄUREAMID-DERIVATE, DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL 有权NEW 2-取代Tiazole -4-羧酸酰胺衍生物，生产和使用AS DRUGS
公开(公告)号：EP2231654A1
公开(公告)日：2010-09-29
申请号：EP08859757.0
申请日：2008-11-28
发明人： BOTHE, Ulrich , VON BONIN, Arne , NGUYEN, Duy , BÖMER, Ulf , GUENTHER, Judith
IPC分类号： C07D417/14 , C07D417/04 , A61K31/427 , A61P35/00 , A61P37/08
CPC分类号： C07D417/14 , C07D417/04
摘要： The invention relates to 2-substituted thiazole-4-carboxamide derivatives of formula (I), the use thereof as a medicament for treating various diseases, and methods for the production thereof.
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7.发明公开NEUE 2-HETARYLTHIAZOL-4-CARBONSÄUREAMID-DERIVATE, DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL 有权新的2 HETARYLTHIAZOL -4-羧酸酰胺衍生物，生产和使用AS DRUGS
公开(公告)号：EP2231652A1
公开(公告)日：2010-09-29
申请号：EP08859392.6
申请日：2008-12-02
发明人： BOTHE, Ulrich , VON BONIN, Arne , NGUYEN, Duy , BÖMER, Ulf , GUENTHER, Judith
IPC分类号： C07D417/04 , C07D417/14 , C07D495/02 , A61K31/427 , A61P1/16 , A61P35/00 , A61P11/00 , A61P17/00 , A61P19/02 , A61P27/02 , A61P37/00
CPC分类号： C07D417/04 , C07D417/14 , C07D495/02
摘要： The invention relates to 2-hetaryl thiazole-4-carboxamide derivatives of formula (I), the use thereof as a medicament for treating various diseases, and methods for the production thereof.
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8.发明公开SUBSTITUTED PHENYLAMINO-BENZENE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH MITOGEN EXTRACELLULAR KINASE ACTIVITY 审中-公开取代PHENYLAMINBENZEN衍生物用于治疗和过度增生细胞外MITROGENKINASE活动诱发的疾病
公开(公告)号：EP2155659A1
公开(公告)日：2010-02-24
申请号：EP08749469.6
申请日：2008-05-09
发明人： RUDOLPH, Joachim , DUMAS, Jaques , LI, Yingfu , AUCLAIR, Daniel , LOBELL, Mario , HITCHCOCK, Marion , HARTUNG, Ingo , KOPPITZ, Marcus , BRITTAIN, Dominic , PUEHLER, Florian , PETERSEN, Kirstin , GUENTHER, Judith , BADER, Benjamin
IPC分类号： C07C217/92 , C07C233/65 , C07C255/59 , C07C271/16 , C07C307/10 , C07D211/22 , C07D317/22 , C07D497/04 , C07D295/088 , A61K31/136 , A61K31/4465 , A61K31/277 , A61K31/167 , A61K31/357 , A61K31/495
CPC分类号： C07D233/60 , C07C217/92 , C07C237/30 , C07C237/44 , C07C243/38 , C07C255/58 , C07C255/59 , C07C271/16 , C07C271/28 , C07C271/44 , C07C275/28 , C07C275/36 , C07C307/02 , C07C307/10 , C07C309/66 , C07C311/08 , C07C311/09 , C07C311/17 , C07C311/48 , C07C2601/08 , C07C2601/10 , C07D205/04 , C07D207/08 , C07D207/27 , C07D207/48 , C07D209/08 , C07D211/22 , C07D211/46 , C07D211/96 , C07D213/30 , C07D213/34 , C07D213/68 , C07D231/18 , C07D233/84 , C07D265/30 , C07D277/22 , C07D295/088 , C07D295/185 , C07D295/26 , C07D317/22 , C07D317/64 , C07D327/04 , C07D403/12
摘要： This invention relates to novel substituted phenylamino-benzene compounds, pharmaceutical compositions containing such compounds and the use of those compounds or compositions for treating hyper- proliferative and/or angiogenesis disorders, as a sole agent or in combination with other active ingredients.
摘要翻译： 本发明涉及新的substituiertem苯氨基苯化合物，药物组合物含有受试化合物和用于治疗过度增殖和/或血管生成病症，作为唯一的药物或与其它活性成分组合使用这些化合物或组合物。
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9.发明公开NOVEL SULPHOXIMINE-SUBSTITUTED QUINAZOLINE AND QUINAZOLINE DERIVATIVES AS KINASE INHIBITORS 审中-公开新SULPHOXIMIN - 取代喹唑啉和喹唑啉衍生物作为激酶抑制剂
公开(公告)号：EP2152672A1
公开(公告)日：2010-02-17
申请号：EP08749502.4
申请日：2008-05-23
发明人： EIS, Knut , PRIEN, Olaf , LUECKING, Ulrich , GUENTHER, Judith , ZOPF, Dieter , BROHM, Dirk , VÖHRINGER, Verena , WOLTERING, Elisabeth , BECK, Hartmut , LOBELL, Mario , LI, Volkhart, Min-Jian , GRESCHAT, Susanne
IPC分类号： C07D215/233 , C07D215/42 , C07D215/44 , C07D239/94 , C07D401/12 , A61K31/4706 , A61K31/4709 , A61K31/47 , A61P35/00 , A61P25/28
CPC分类号： C07D239/86 , C07D215/44 , C07D409/04
摘要： The present invention relates to a quinoline or quinazoline derivative having the general formula (A): in which R3, R4, W, Y and Q are indicated in the description and the claims, the use of the compounds of the general formula (A) for the treatment of various disorders, and the preparation of compounds of the general formula (A).
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10.发明公开OXO-SUBSTITUIERTE IMIDAZO[1,2b]PYRIDAZINE, DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL 审中-公开OXO-SUBSTITUIERTE IMIDAZO [1,2b]吡咯烷酮，DEREN HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL
公开(公告)号：EP2044071A1
公开(公告)日：2009-04-08
申请号：EP07726169.1
申请日：2007-06-20
发明人： PRIEN, Olaf , EIS, Knut , BADER, Benjamin , GUENTHER, Judith , BONIN VON, Arne
IPC分类号： C07D487/04 , A61K31/5025 , A61P11/00 , A61P17/00 , A61P35/00 , A61P37/00
CPC分类号： C07D487/04
摘要： The invention relates to novel kinase inhibitors of general formula (I), wherein Q and R1 are defined as in the claims. The invention also relates to methods for producing said inhibitors, to intermediates for producing the same and to uses thereof.
摘要翻译： 本发明涉及通式（I）的新型激酶抑制剂：其中Q和R 1在权利要求书中定义，制备这种抑制剂的方法，制备这种抑制剂的中间体和这种抑制剂的用途。
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