Fungicidal 1,4-disubstituted 1-azolyl-3,3-dimethylbutane derivatives
    1.
    发明授权
    Fungicidal 1,4-disubstituted 1-azolyl-3,3-dimethylbutane derivatives 失效
    杀真菌剂1,4-二取代的1-噻唑基-3,3-二甲基丁烷衍生物

    公开(公告)号:US4968712A

    公开(公告)日:1990-11-06

    申请号:US225971

    申请日:1988-07-29

    摘要: Fungicidal 1,4-disubstituted 1-azolyl-3,3-dimethylbutane derivatives of the formula ##STR1## in which R.sup.1 represents hydrogen or halogen,R.sup.2 represents hydrogen or halogen,R.sup.3 represents hydrogen, halogen or trifluoromethoxy,R.sup.4 represents halogen, trifluoromethoxy, trifluoromethylthio, trifluoromethylsulphinyl, trifluoromethylsulphonyl, difluoromethoxy, difluorochloromethoxy, trifluorochloroethoxy, tetrafluoroethoxy, trifluoroethoxy, difluoromethylthio, trifluorochloroethylthio, tetrafuoroethylthio, difluoromethylsulphinyl, difluorochloromethylsulphinyl, trifluorochloroethylsulphinyl, tetrafluoroethylsulphinyl, difluoromethylsulphonyl, difluorochloromethylsulphonyl, trifluorochloroethylsulphonyl, tetrafluoroethylsulphonyl, difluorobromomethylthio, difluorobromomethylsulphinyl, difluorobromomethylsulphonyl or difluorochloromethylthio orR.sup.3 and R.sup.4 together represent alkylenedioxy substituted by halogen,R.sup.5 represents hydrogen or halogen,A represents a keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group andR.sup.6 and R.sup.7 identical or different and independently of one another represent hydrogen, alkyl, alkenyl, alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl or optionally substituted phenylalkyl, whereR.sup.3 represents trifluoromethoxy whenR.sup.4 represents halogen,and addition products thereof with acids and metal salts.

    摘要翻译: 式(I)的杀真菌的1,4-二取代的1-吡唑基-3,3-二甲基丁烷衍生物,其中R 1表示氢或卤素,R 2表示氢或卤素,R 3表示氢,卤素或三氟甲氧基,R 4表示卤素 三氟甲氧基,三氟甲硫基,三氟甲磺酰基,三氟甲磺酰基,二氟甲氧基,二氟氯甲氧基,三氟氯乙氧基,四氟乙氧基,三氟乙氧基,二氟甲硫基,三氟氯乙硫基,四氟乙基硫代, 和R4一起代表被卤素取代的亚烷基二氧基,R 5代表氢或卤素,A代表酮基或CH(OH) Z表示氮原子或CH基团,R 6和R 7相同或不同且彼此独立地表示氢,烷基,烯基,炔基,任选取代的环烷基,任选取代的环烷基烷基或任选取代的苯基烷基,其中当R 4表示卤素时,R 3表示三氟甲氧基 ,及其与酸和金属盐的加成产物。

    Novel substituted azolylvinyl ketones and carbinols as fungicides and
plant growth regulators
    3.
    发明授权
    Novel substituted azolylvinyl ketones and carbinols as fungicides and plant growth regulators 失效
    新型取代的唑基乙烯基酮和甲醇作为杀真菌剂和植物生长调节剂

    公开(公告)号:US4728356A

    公开(公告)日:1988-03-01

    申请号:US754788

    申请日:1985-07-12

    摘要: A substituted azolylvinyl ketone or carbinol of the formula ##STR1## in which R.sup.1 represents optionally substituted cycloalkyl with 3 to 5 carbon atoms, substituted cyclohexyl or the grouping ##STR2## wherein R.sup.3 represents optionally substituted phenyl, alkenyl, alkinyl, cyano or the grouping --Z--R.sup.4,whereinR.sup.4 represents alkyl, halogenoalkyl, optionally substituted phenyl or optionally substituted phenylalkyl andZ represents O, S, SO or SO.sub.2,n represents a number from 0 to 2,R.sup.2 represents alkyl, alkenyl, alkinyl, in each case optionally substituted phenyl or phenylalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkenyl, cycloalkenylalkyl, bicycloalkyl or bicycloalkenyl, but R.sup.2 does not represent optionally substituted phenyl at the same time as R.sup.1 represents optionally substituted cycloalkyl with 3 to 5 carbon atoms or substituted cyclohexyl or R.sup.3 represents optionally substituted phenyl,X represents the CO or CH(OH) group andY represents a nitrogen atom or the CH group,or an addition product thereof with an acid or metal salt.The products are active in combating fungi and in regulating the growth of plants.

    摘要翻译: 其中R 1表示任选取代的具有3至5个碳原子的环烷基,取代的环己基或基团,其中R 3表示任选取代的苯基,烯基,炔基,氰基或基团 - Z-R4,其中R4代表烷基,卤代烷基,任选取代的苯基或任选取代的苯基烷基,Z代表O,S,SO或SO 2,n代表0至2的数,R 2代表烷基,烯基,炔基, 取代的苯基或苯基烷基,或者在每种情况下都是任选取代的环烷基,环烷基烷基,环烯基,环烯基烷基,双环烷基或双环烯基,但R 2不同时代表任选取代的苯基,其中R 1表示任选取代的具有3至5个碳原子的环烷基或取代的环己基 或R 3表示任选取代的苯基,X表示CO或CH(OH)基团,Y表示氮气 m或CH基团,或其与酸或金属盐的加成产物。 该产品在防治真菌和调节植物生长方面发挥积极作用。