Thiazolidinedione derivatives, method for preparing the derivatives and
pharmaceutical compositions containing same
    1.
    发明授权
    Thiazolidinedione derivatives, method for preparing the derivatives and pharmaceutical compositions containing same 失效
    噻唑烷二酮衍生物,制备衍生物的方法和含有它们的药物组合物

    公开(公告)号:US5811439A

    公开(公告)日:1998-09-22

    申请号:US768937

    申请日:1996-12-18

    CPC分类号: C07D417/06 C07D417/14

    摘要: A thiazolidinedione derivative represented by the following general formula (I): ##STR1## �wherein the dotted line represents a single bond or a double bond, the thiazolidinedione ring residue is linked to either of 2-, 3-, 4-, 5- and 6-positions on the indole ring and R represents a group selected from the group consisting of hydrogen atom and alkyl, alkenyl, alkynyl, phenyl, aralkyl, heterocycloalkyl, arylsulfonyl and arylaminocarbonyl groups! or a pharmaceutically acceptable salt thereof exhibits excellent effects of reducing the blood sugar level and of reducing the lipid concentration in blood and is accordingly useful as a therapeutic agent for treating diabates mellitus. These derivatives and pharmaceutically acceptable salt thereof are almost free of any side effect.

    摘要翻译: 由下列通式(I)表示的噻唑烷二酮衍生物:其中虚线代表单键或双键,噻唑烷二酮环残基与2-,3-,4- 在吲哚环上的5-和6-位,R表示选自氢原子和烷基,烯基,炔基,苯基,芳烷基,杂环烷基,芳基磺酰基和芳基氨基羰基的基团]或其药学上可接受的盐显示出优异的 降低血糖水平和降低血液中的脂质浓度的效果,因此可用作治疗二倍体的治疗剂。 这些衍生物及其药学上可接受的盐几乎没有副作用。

    Amino acid derivative having anti-CCK activity
    2.
    发明授权
    Amino acid derivative having anti-CCK activity 失效
    具有抗CCK活性的氨基酸衍生物

    公开(公告)号:US5716958A

    公开(公告)日:1998-02-10

    申请号:US513018

    申请日:1995-08-09

    摘要: A compound represented by the formula (1): ##STR1## wherein, m is an integer of 1 to 3; n is an integer 0 or 1; A represents CH or N atom, and forms together with the N atom bonded to the carbonyl group a piperidine ring or a piperazine ring; R.sub.1 independently represents a straight or branched chain alkyl group having 1 to 4 carbon atoms; a cycloalkyl group having 3 to 8 carbon atoms; a phenyl group, unsubstituted or substituted with a halogen atom or with an alkoxy group having 1 to 4 carbon atoms; or a pyridyl group; or two R.sub.1, together with the group >CH-- to which they bind, form a dibenzo cycloheptenyl group or a fluorenyl group; R.sub.2 represents a phenyl group substituted with a carboxyl or substituted carboxyl group; a pyridyl group substituted with a carboxyl or substituted carboxyl group, a pyrazyl group substituted with a carboxyl or substituted carboxyl group, an oxazolyl substituted with a carboxyl or substituted carboxyl group, a triazolyl substituted with one or two carboxyl or substituted carboxyl groups, or a phosphonopyridyl group; and R.sub.3 represents an indolyl group unsubstituted or substituted with a substituent selected from the group consisting of a halogen atom, a hydroxy group, an alkoxy group having 1 to 4 carbon atoms and methoxycarbonyl ethyl group and the pharmaceutically acceptable salts thereof.

    摘要翻译: 由式(1)表示的化合物:其中,m为1〜3的整数, n是整数0或1; A表示CH或N原子,并与与羰基键合的N原子一起形成哌啶环或哌嗪环; R1独立地表示具有1至4个碳原子的直链或支链烷基; 具有3-8个碳原子的环烷基; 未取代或被卤素原子或具有1至4个碳原子的烷氧基取代的苯基; 或吡啶基; 或两个R 1与它们所结合的基团> CH-一起形成二苯并环庚烯基或芴基; R2表示被羧基或取代羧基取代的苯基; 被羧基或取代羧基取代的吡啶基,被羧基或取代羧基取代的吡唑基,被羧基或取代羧基取代的恶唑基,被一个或两个羧基或取代羧基取代的三唑基,或 膦酰吡啶基; R3表示未取代或被选自卤素原子,羟基,具有1〜4个碳原子的烷氧基和甲氧基羰基乙基的取代基取代的吲哚基及其药学上可接受的盐。

    Contact/non-contact type hybrid IC card, communication method, program and communication system
    3.
    发明授权
    Contact/non-contact type hybrid IC card, communication method, program and communication system 有权
    接触/非接触式混合IC卡,通讯方式,程序通讯系统

    公开(公告)号:US09058553B2

    公开(公告)日:2015-06-16

    申请号:US12477632

    申请日:2009-06-03

    申请人: Tadashi Morita

    发明人: Tadashi Morita

    IPC分类号: G06K19/00 G06K19/077

    摘要: A contact/non-contact type hybrid IC card is provided which includes a non-contact interface to communicate in a non-contact manner with a non-contact type reader/writer through an antenna, a contact interface to communicate in a contact manner with a contact type reader/writer through a contact terminal, a storage unit to store personal identification information input from the contact type reader/writer through the contact interface during a contact communication mode by the contact interface, and a control unit to remove a limitation of a prescribed function in a non-contact communication mode by the non-contact interface based on the personal identification information stored in the storage unit during the contact communication mode and switch a communication mode from the contact communication mode to the non-contact communication mode with the limitation of the prescribed function being removed.

    摘要翻译: 提供一种接触/非接触式混合IC卡,其包括非接触式接口,以非接触方式通过天线与非接触式读取器/写入器进行通信,接触界面以接触方式与 通过接触终端的接触型读取器/写入器,存储单元,用于通过接触界面在接触通信模式期间通过接触接口存储从接触型读取器/写入器输入的个人识别信息;以及控制单元, 基于在接触通信模式期间存储在存储单元中的个人识别信息,通过非接触式接口在非接触通信模式中的规定功能,并且将通信模式从接触通信模式切换到非接触通信模式, 规定功能的限制被删除。

    Information processing system, information processor, information processing method, and program

    公开(公告)号:US09001048B2

    公开(公告)日:2015-04-07

    申请号:US12430601

    申请日:2009-04-27

    申请人: Tadashi Morita

    发明人: Tadashi Morita

    IPC分类号: G09G5/00 G06F3/0488

    CPC分类号: G06F3/0488

    摘要: An information processing system includes a first information processor to process data to be displayed in a first display unit and a second information processor to indicate the data displayed in the first display unit. The first information processor includes a first display control unit to control the data to be displayed; a first communication unit to receive operation information from the second information processor and transmit data information about a piece of data indicated by the second information processor; and a first detecting unit to detect a position on the first display unit indicated by the second information processor. The second information processor includes an accepting unit to accept an operation by a user; a second communication unit to transmit operation information to the first information processor and receive the data information from the first information processor; and a received data storage unit to store the data information.

    WIRELESS COMMUNICATION DEVICE
    5.
    发明申请
    WIRELESS COMMUNICATION DEVICE 有权
    无线通信设备

    公开(公告)号:US20140064264A1

    公开(公告)日:2014-03-06

    申请号:US14009743

    申请日:2013-01-23

    IPC分类号: H04W56/00

    摘要: A WiGig wireless device partially performs a masking processing on a preamble of a transmission signal frame and generates a repetition pattern of the same pulse capable of being used in a correlation detection of a sensor. That is, a repetition pattern of a Golay code is output by intermittently performing the masking processing on the Golay code sequence. The sensor performs the correlation detection using a pulse compression technology, thereby detecting the antenna radiation pattern even in an environment where a reflected wave is generated, by separating the direct wave and the reflected wave.

    摘要翻译: WiGig无线设备部分地对发送信号帧的前导码进行掩蔽处理,并且生成能够用于传感器的相关检测的相同脉冲的重复模式。 也就是说,通过对Golay码序列间歇地执行掩蔽处理来输出Golay码的重复图案。 传感器使用脉冲压缩技术执行相关检测,从而即使在产生反射波的环境中也可以通过分离直接波和反射波来检测天线辐射图。

    Delta sigma ADC
    6.
    发明授权
    Delta sigma ADC 有权
    Delta西格玛ADC

    公开(公告)号:US08466821B2

    公开(公告)日:2013-06-18

    申请号:US13256524

    申请日:2011-01-07

    申请人: Tadashi Morita

    发明人: Tadashi Morita

    IPC分类号: H03M3/00

    CPC分类号: H03M3/47

    摘要: A ΔΣADC is provided that is capable of suppressing increase of a circuit scale without losing noise shaping function even when a switching speed of a switch for performing time-division process is lower than a sampling rate of the ΔΣADC. For a code values provided by a comparator (105), the ΔΣADC (100) has a first storage section (106-1) and a second storage section (106-2) respectively for signal sequences (a first signal sequence and a second signal sequence) constituting a time-divisionally combined signal. Then, one of the two storage sections (i.e. the first storage section (106-1) and the second storage section (106-2)) that corresponds to a branch selection signal is configured to store the code value obtained from the comparator (105). On the other hand, one of the two storage sections (i.e. the first storage section (106-1) and the second storage section (106-2)) that is not the storage section corresponding to the branch selection signal is configured to hold the already stored code value.

    摘要翻译: 提供了一种DeltaSigmaADC,即使当用于执行时分处理的开关的切换速度低于DeltaSigmaADC的采样率时,也能够抑制电路规模的增加而不失去噪声整形功能。 对于由比较器(105)提供的代码值,DeltaSigmaADC(100)具有分别用于信号序列的第一存储部分(106-1)和第二存储部分(106-2)(第一信号序列和第二信号 序列)构成时分组合信号。 然后,对应于分支选择信号的两个存储部分(即,第一存储部分(106-1)和第二存储部分(106-2))之一被配置为存储从比较器(105)获得的代码值 )。 另一方面,不是与分支选择信号对应的存储部的两个存储部(即,第一存储部(106-1)和第二存储部106-2)中的一个被配置为保持 已经存储的代码值。

    WIRELESS DEVICE AND RECEIVING METHOD
    7.
    发明申请
    WIRELESS DEVICE AND RECEIVING METHOD 有权
    无线设备和接收方法

    公开(公告)号:US20130142294A1

    公开(公告)日:2013-06-06

    申请号:US13817491

    申请日:2012-02-22

    申请人: Tadashi Morita

    发明人: Tadashi Morita

    IPC分类号: H04B1/16

    摘要: The purpose of the present invention is to shorten a time required to perform Auto Gain Control (AGC) processing in a wireless device that can be applied to a plurality of wireless systems. On the basis of a first gain adjusted by means of a gain control unit (450-1), an initial gain setting unit (460) sets, for a variable gain unit (432-2), an initial gain (converted second initial gain) at the start of gain adjustment. Then, a gain control unit (450-2) sets the initial gain to a second gain at the time of starting the gain adjustment, and adjusts the second gain on the basis of IQ signals of a system, the IQ signals having the level adjusted by means of the variable gain unit (432-2).

    摘要翻译: 本发明的目的是缩短在可应用于多个无线系统的无线设备中执行自动增益控制(AGC)处理所需的时间。 基于通过增益控制单元(450-1)调整的第一增益,初始增益设置单元(460)针对可变增益单元(432-2)设置初始增益(转换后的第二初始增益 )在增益调整开始时。 然后,增益控制单元(450-2)在开始增益调整时将初始增益设置为第二增益,并且基于系统的IQ信号来调整第二增益,具有调整了电平的IQ信号 借助于可变增益单元(432-2)。

    TIME DIVISION RECEIVER AND TIME DIVISION RECEIVING METHOD
    8.
    发明申请
    TIME DIVISION RECEIVER AND TIME DIVISION RECEIVING METHOD 有权
    时间接收者和时间接收方法

    公开(公告)号:US20130136118A1

    公开(公告)日:2013-05-30

    申请号:US13814338

    申请日:2011-12-14

    申请人: Tadashi Morita

    发明人: Tadashi Morita

    IPC分类号: H04J3/00

    CPC分类号: H04J3/00 H04B1/163

    摘要: Provided are a time division receiver and a time division receiving method capable of mitigating leaks between branches for a time division multiplexed signal for which a plurality of branches have been time-division multiplexed even when processing using a single high-frequency circuit. In a time division receiver (100A), mixers (120-1 and 120-2) down-convert a time division multiplexed signal for which a plurality of branch signals have been time-division multiplexed. Time division separation units (130-1 and 130-2) separate the time division multiplexed signal which has been down-converted at the mixers (120-1 and 120-2) into branches, respectively. A residual charge initialization unit (160) initializes charges that are residual when a first branch signal passes for parasitic capacitances that occur in channels between the mixers (120-1 and 120-2) and the time division separation units (130-1 and 130-2) to the residual charges before passing of a second branch signal.

    摘要翻译: 提供了一种时分接收机和时分接收方法,即使在使用单个高频电路进行处理时,也能够减轻多个分支已被时分复用的时分复用信号的分支之间的泄漏。 在时分接收机(100A)中,对多个分支信号进行时分复用的时分复用信号进行下变频的混频器(120-1,120-2)。 分时分离单元(130-1和130-2)分别将已经在混频器(120-1和120-2)下变频的时分复用信号分离成分支。 剩余电荷初始化单元(160)初始化第一分支信号通过的混合器(120-1和120-2)与时分分离单元(130-1和130)之间的通道中发生的寄生电容时残留的电荷 -2)到通过第二分支信号之前的剩余电荷。

    Sampling mixer, quadrature demodulator, and wireless device
    9.
    发明授权
    Sampling mixer, quadrature demodulator, and wireless device 有权
    采样混频器,正交解调器和无线设备

    公开(公告)号:US08340617B2

    公开(公告)日:2012-12-25

    申请号:US12745240

    申请日:2008-12-10

    IPC分类号: H04B1/26

    摘要: There are provided a sampling mixer, quadrature demodulator, and a wireless device capable of suppressing receiving sensitivity degradation caused by alias components or second-order distortion components. In the sampling mixer (101), a sampling switch (5) and another sampling switch (36) sample a reception signal based on a local signal with a predetermined frequency. A control signal generator (15) generates a control signal for controlling a filter operation. An in-phase mixer (2) and a reverse-phase mixer (3) perform, based on the control signal, filter processing on the sample signal obtained by the sampling switch (5). A delay controller (117) controls the phase difference between the local signal and the control signal according to a reception-desired frequency.

    摘要翻译: 提供了能够抑制由别名分量或二阶失真分量引起的接收灵敏度劣化的采样混频器,正交解调器和无线装置。 在采样混频器(101)中,采样开关(5)和另一采样开关(36)基于具有预定频率的本地信号对接收信号进行采样。 控制信号发生器(15)产生用于控制滤波器操作的控制信号。 同相混合器(2)和反相混合器(3)根据控制信号执行由采样开关(5)获得的采样信号的滤波处理。 延迟控制器(117)根据接收期望频率来控制本地信号和控制信号之间的相位差。

    COMMUNICATION SYSTEM, COMMUNICATION METHOD, AND DATA PROCESSING APPARATUS
    10.
    发明申请
    COMMUNICATION SYSTEM, COMMUNICATION METHOD, AND DATA PROCESSING APPARATUS 有权
    通信系统,通信方法和数据处理设备

    公开(公告)号:US20120231735A1

    公开(公告)日:2012-09-13

    申请号:US13476673

    申请日:2012-05-21

    IPC分类号: H04B5/00

    摘要: A communication system and communication method enable various types of near field communication. NFC communication apparatuses have two features in that each can perform communication in two communication modes and that each can perform data transmission at a plurality of transfer rates. The two communication modes consist of a passive mode and an active mode. In the passive mode, between the NFC communication apparatuses, for example, a first NFC communication apparatus transmits data to a second NFC communication apparatus by modulating electromagnetic waves generated by itself, while the second NFC communication apparatus transmits data to the first NFC communication apparatus by performing load modulation on the electromagnetic waves generated by the first NFC communication apparatus. Alternatively, in the active mode, either of the NFC communication apparatuses transmits data by modulating electromagnetic waves generated by itself. The present innovation can be applied to, for example, an IC card system, etc.

    摘要翻译: 通信系统和通信方法能够进行各种类型的近场通信。 NFC通信设备具有两个特征,每个功能可以以两种通信模式执行通信,并且每个都可以以多个传输速率执行数据传输。 两种通信模式由被动模式和活动模式组成。 在被动模式中,NFC通信装置之间,例如第一NFC通信装置,通过调制由其自身产生的电磁波,向第二NFC通信装置发送数据,而第二NFC通信装置通过以下方式向第一NFC通信装置发送数据 对由第一NFC通信设备产生的电磁波执行负载调制。 或者,在活动模式中,NFC通信装置中的任一个通过调制由其自身产生的电磁波来发送数据。 本发明可以应用于例如IC卡系统等。