Oligosaccharide derivative
    61.
    发明授权
    Oligosaccharide derivative 失效
    寡糖衍生物

    公开(公告)号:US07632930B2

    公开(公告)日:2009-12-15

    申请号:US12029337

    申请日:2008-02-11

    CPC分类号: C07H15/203 C07H17/02

    摘要: Compounds having the formula (I): wherein A represents a group such as a cyclic group, R1 and R2 represent groups such as alkyl groups or hydroxymethyl groups, and n represents 1 or 2, or pharmacologically acceptable salts thereof or pharmacologically acceptable esters thereof have superior activity and stability, and are useful for the treatment and/or prevention of diabetes mellitus, or the like.

    摘要翻译: 具有式(I)的化合物:其中A表示诸如环状基团的基团,R 1和R 2表示诸如烷基或​​羟甲基的基团,n表示1或2,或其药学上可接受的盐或其药理学上可接受的酯具有 优异的活性和稳定性,并且可用于治疗和/或预防糖尿病等。

    BENZYLPHENYL GLUCOPYRANOSIDE DERIVATIVE
    63.
    发明申请
    BENZYLPHENYL GLUCOPYRANOSIDE DERIVATIVE 审中-公开
    苯甲酰基吡咯烷酮衍生物

    公开(公告)号:US20090137499A1

    公开(公告)日:2009-05-28

    申请号:US12280510

    申请日:2007-08-03

    摘要: The present invention relates to a benzylphenyl glucopyranoside derivative having an excellent inhibitory effect on human SGLT1 and/or SGLT2 activity. There is provided a compound or a pharmacologically acceptable salt thereof represented by the following general formula (I): wherein R1 represents a hydrogen atom, an amino group, a hydroxy C1-C6 alkyl group, etc.; R2 represents a hydrogen atom, etc.; R3 represents a C1-C6 alkyl group, a hydroxy C1-C6 alkyl group, etc.; R4 represents a hydrogen atom, a C2-C7 acyl group, etc.; R5, R6, R7, and R8 are the same or different and each represents a hydrogen atom or a C1-C6 alkyl group, provided that R5, R6, R7 and R8 are not hydrogen atoms at the same time; n is 0 to 4; and X is CH or N.

    摘要翻译: 本发明涉及对人SGLT1和/或SGLT2活性具有优异抑制作用的苄基苯基吡喃葡萄糖苷衍生物。 提供由以下通式(I)表示的化合物或其药理学上可接受的盐:其中R1表示氢原子,氨基,羟基C1-C6烷基等; R2表示氢原子等; R3表示C1-C6烷基,羟基C1-C6烷基等; R4表示氢原子,C2-C7酰基等; R5,R6,R7和R8相同或不同,各自表示氢原子或C1-C6烷基,条件是R5,R6,R7和R8不同时为氢原子; n为0〜4; X为CH或N.

    Oligosaccharide Derivative
    64.
    发明申请
    Oligosaccharide Derivative 失效
    寡糖衍生物

    公开(公告)号:US20080194495A1

    公开(公告)日:2008-08-14

    申请号:US12029337

    申请日:2008-02-11

    IPC分类号: A61K31/702 C07H15/02 A61P3/10

    CPC分类号: C07H15/203 C07H17/02

    摘要: Compounds having the formula (I): wherein A represents a group such as a cyclic group, R1 and R2 represent groups such as alkyl groups or hydroxymethyl groups, and n represents 1 or 2, or pharmacologically acceptable salts thereof or pharmacologically acceptable esters thereof have superior activity and stability, and are useful for the treatment and/or prevention of diabetes mellitus, or the like.

    摘要翻译: 具有式(I)的化合物:其中A表示诸如环状基团的基团,R 1和R 2表示例如烷基或羟甲基的基团,n 代表1或2,或其药学上可接受的盐或其药理学上可接受的酯具有优异的活性和稳定性,并且可用于治疗和/或预防糖尿病等。

    Air shower apparatus
    65.
    发明授权

    公开(公告)号:US07052389B2

    公开(公告)日:2006-05-30

    申请号:US11075794

    申请日:2005-03-10

    IPC分类号: F24F7/07

    摘要: An air shower for removing a particle from an object by blowing air to the object which includes at least one first outlet for discharging the air from the at least one first outlet toward at least a portion of the object so that a flow axis of the air flowing out of the at least one first outlet is swung frequently and alternately in a first swingable direction, and at least one second outlet for discharging the air from the at least one second outlet so that a flow axis of the air flowing out of the at least one second outlet is swung frequently and alternately in a second swingable direction which is different from the first swingable direction. The first swingable direction and the second swingable direction extend so as to be non-parallel to one another and to intersect one another.

    Air shower apparatus
    66.
    发明申请
    Air shower apparatus 有权
    空气淋浴器

    公开(公告)号:US20050159100A1

    公开(公告)日:2005-07-21

    申请号:US11075794

    申请日:2005-03-10

    摘要: An air shower for removing a particle from an object by blowing air to the object which includes at least one first outlet for discharging the air from the at least one first outlet toward at least a portion of the object so that a flow axis of the air flowing out of the at least one first outlet is swung frequently and alternately in a first swingable direction, and at least one second outlet for discharging the air from the at least one second outlet so that a flow axis of the air flowing out of the at least one second outlet is swung frequently and alternately in a second swingable direction which is different from the first swingable direction. The first swingable direction and the second swingable direction extend so as to be non-parallel to one another and to intersect one another.

    摘要翻译: 一种用于通过向所述物体吹送空气来从物体除去颗粒的空气淋浴器,所述空气淋浴器包括至少一个用于将空气从所述至少一个第一出口排出到所述物体的至少一部分的第一出口,使得所述空气的流动轴线 从至少一个第一出口流出的频率在第一可摆动方向上频繁地和交替地摆动,以及至少一个第二出口,用于从至少一个第二出口排出空气,使得空气的流动轴流出 在与第一可摆动方向不同的第二可摆动方向上频繁地和交替地摆动至少一个第二出口。 第一可摆动方向和第二可摆动方向彼此不平行并且彼此相交。

    On board refueling vapor recovery system and fuel vapor passage using for the same
    67.
    发明授权
    On board refueling vapor recovery system and fuel vapor passage using for the same 有权
    船上加油蒸汽回收系统和燃油蒸汽通道使用相同

    公开(公告)号:US06851458B2

    公开(公告)日:2005-02-08

    申请号:US10219933

    申请日:2002-08-16

    摘要: An on board refueling vapor recovery system includes a first fuel vapor passage for connecting a fuel tank with a canister, a second fuel vapor passage for connecting an inlet portion of a fuel filler pipe with the fuel vapor passage (a tank main body) and a check valve in the second fuel vapor passage. The check valve is integrated with a first quick connector of a resin hose (a resin tube) which constitutes the second fuel vapor passage. Therefore, the number of man hours required for assembling the on board refueling vapor recovery system can be reduced. In addition, the space required for installing any of the on board refueling vapor recovery system can also be reduced. Furthermore, the amount of released fuel evaporative emissions or fuel evaporative emissions can be reduced.

    摘要翻译: 船上加油蒸汽回收系统包括用于将燃料箱与罐连接的第一燃料蒸汽通道,用于将燃料加注管的入口部分与燃料蒸汽通道(罐主体)连接的第二燃料蒸汽通道和 在第二燃料蒸气通道中的止回阀。 止回阀与构成第二燃料蒸气通道的树脂软管(树脂管)的第一快速连接器一体化。 因此,可以减少组装船上加油蒸气回收系统所需的人工小时数。 此外,也可以减少安装任何车载加油蒸气回收系统所需的空间。 此外,可以减少释放的燃料蒸发排放量或燃料蒸发排放量。

    Neuraminic acid derivatives, their preparation and their medical use
    68.
    发明授权
    Neuraminic acid derivatives, their preparation and their medical use 有权
    神经氨酸衍生物,其制备及其用途

    公开(公告)号:US06451766B1

    公开(公告)日:2002-09-17

    申请号:US09969851

    申请日:2001-10-03

    IPC分类号: C07D31500

    CPC分类号: C07D309/28 Y10S530/807

    摘要: Compounds of formula (I) or their salts or esters: [wherein R1 is alkyl or haloalkyl; R2 and R3 each represents hydrogen or aliphatic acyl; X is hydroxy, halogen, alkoxy, or a group of formula RaO—, where Ra is aliphatic acyl; Y is a group of formula RbRcN— or RbRcN—O—, where Rb and Rc each is hydrogen or alkyl; and Z is oxygen or sulfur] have excellent sialidase inhibitory activity and are therefore useful for the treatment and prevention of influenza and other viral diseases where the replication of the virus is susceptible to sialidase inhibitors.

    摘要翻译: 式(I)化合物或其盐或酯:[其中R1是烷基或卤代烷基; R2和R3各自表示氢或脂族酰基; X是羟基,卤素,烷氧基或式RaO-基团,其中Ra是脂族酰基; Y是式RbRcN-或RbRcN-O-的基团,其中Rb和Rc各自为氢或烷基; 和Z是氧或硫]具有优异的唾液酸酶抑制活性,因此可用于治疗和预防病毒复制对唾液酸酶抑制剂敏感的流行性感冒和其他病毒性疾病。

    Optical scanning device
    70.
    发明授权
    Optical scanning device 有权
    光学扫描装置

    公开(公告)号:US09122059B2

    公开(公告)日:2015-09-01

    申请号:US13824137

    申请日:2011-11-24

    摘要: Optical scanning device 1 according to the present invention includes: main movable portion 10; a pair of torsionally deformable main torsion beams 21 and 22 arranged opposite to each other at both ends of main movable portion 10 and swingably supporting main movable portion 10; and main driving unit 30 that drives main movable portion 10 to oscillate. Main movable portion 10 includes mirror unit 11 having reflection surface 11a for reflecting light, and a pair of permanent magnets 12 and 13 arranged opposite to each other to sandwich mirror unit 11, each permanent magnet extending along oscillation axis X-X of main movable portion 10. Main driving unit 30 includes yoke unit 31, 32, and 33 arranged along oscillation axis X-X of main movable portion 10 to surround permanent magnets 12 and 13, and coil 34 wound on yoke unit 31, 32, and 33 and configured to be energized to magnetize yoke unit 31, 32, and 33, thereby generating magnetic fields to be applied on permanent magnets 12 and 13.

    摘要翻译: 根据本发明的光学扫描装置1包括:主可动部10; 一对在主可动部10的两端彼此相对设置并且可摆动地支撑主可动部10的可扭转主扭力梁21和22; 以及驱动主可动部10振动的主驱动部30。 主可动部分10包括具有用于反射光的反射表面11a的反射镜单元11和彼此相对布置以夹持反射镜单元11的一对永磁体12和13,每个永磁体沿着主可动部分10的振动轴线XX延伸。 主驱动单元30包括沿着主可动部分10的摆动轴线XX布置以围绕永磁体12和13的轭单元31,32和33,以及缠绕在轭单元31,32和33上的线圈34, 磁化轭单元31,32和33,从而产生施加在永磁体12和13上的磁场。