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公开(公告)号:US20140221330A1
公开(公告)日:2014-08-07
申请号:US14234456
申请日:2012-07-26
申请人: Akihiro Morinaka , Kazunori Maebashi , Takashi Ida , Muneo Hikida , Mototsugu Yamada , Takao Abe
发明人: Akihiro Morinaka , Kazunori Maebashi , Takashi Ida , Muneo Hikida , Mototsugu Yamada , Takao Abe
IPC分类号: C07C69/593 , A61K45/06 , C07C69/612 , A61K31/216 , C07C69/618 , C07C69/732 , C07D309/06 , A61K31/351 , C07C69/608 , C07D213/55 , A61K31/4406 , C07D295/108 , A61K31/5375 , C07D211/46 , A61K31/45 , C07D233/64 , A61K31/4174 , C07D207/12 , A61K31/4015 , A61K31/225
CPC分类号: C07C69/593 , A61K31/194 , A61K31/216 , A61K31/225 , A61K31/351 , A61K31/40 , A61K31/4015 , A61K31/407 , A61K31/4164 , A61K31/4174 , A61K31/4406 , A61K31/45 , A61K31/5375 , A61K45/06 , C07C57/13 , C07C57/26 , C07C57/30 , C07C57/42 , C07C57/48 , C07C57/50 , C07C59/46 , C07C59/64 , C07C63/66 , C07C69/608 , C07C69/612 , C07C69/618 , C07C69/732 , C07C217/18 , C07C233/65 , C07C235/20 , C07C237/22 , C07C279/08 , C07D207/12 , C07D211/46 , C07D213/55 , C07D233/64 , C07D295/108 , C07D309/06 , Y02A50/473 , A61K2300/00
摘要: An objective of the present invention is to provide a novel NDM (New Delhi metallo-β-lactamase) inhibitor that functions as a drug for restoring the antibacterial activity of β-lactam antibiotics that have been inactivated as a result of decomposition by NDM. According to the present invention, there is provided an NDM inhibitor contains a compound represented by general formula (I):
摘要翻译: 本发明的目的是提供一种新型的NDM(新德里金属 - β-内酰胺酶)抑制剂,其作为恢复由NDM分解而灭活的β-内酰胺抗生素的抗菌活性的药物 。 根据本发明,提供了含有通式(I)表示的化合物的NDM抑制剂:
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公开(公告)号:US20120163720A1
公开(公告)日:2012-06-28
申请号:US13394283
申请日:2009-09-04
申请人: Kanako Saito , Toshimitsu Kaneko , Takashi Ida
发明人: Kanako Saito , Toshimitsu Kaneko , Takashi Ida
CPC分类号: H04N1/3935 , G06T3/40
摘要: A specifying unit specifies a pixel value at a pixel position of a reference image to a pixel of a sample enlarged image at a position relative to a pixel position of the reference image as an initial pixel value. A selecting unit selects a target pixel from pixels other than pixels having the pixel values specified therefor including the pixels having the initial pixel values are set in the sample enlarged image. An allocating unit configured to allocate the pixel value of the pixel at a similar region position of the reference image to the pixel value of the target value in the sample enlarged image when a searching unit searches the similar region position similar to a pixel value pattern including a set of already specified pixels in a spatial neighborhood of the target pixel from the reference image is provided.
摘要翻译: 指定单元将参考图像的像素位置处的像素值指定为相对于参考图像的像素位置的位置处的样本放大图像的像素作为初始像素值。 选择单元从具有由其指定的像素值的像素以外的像素中选择目标像素,包括在样本放大图像中设置具有初始像素值的像素。 分配单元,被配置为当搜索单元搜索类似于像素值图案的类似区域位置时,将参考图像的类似区域位置处的像素的像素值分配给样本放大图像中的目标值的像素值,包括 提供了来自参考图像的目标像素的空间邻域中已经指定的像素集合。
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公开(公告)号:US20070206860A1
公开(公告)日:2007-09-06
申请号:US11745547
申请日:2007-05-08
申请人: Takashi Ida , Yoko Sambonsugi , Osamu Hori
发明人: Takashi Ida , Yoko Sambonsugi , Osamu Hori
IPC分类号: G06K9/48
CPC分类号: G06K9/00234 , G06F16/5854 , G06K9/6204 , G06T7/11 , G06T7/13 , G06T7/194 , G06T9/20 , G06T2207/10016 , G06T2207/20021 , H04N19/20 , H04N19/593
摘要: An object extraction method comprising the steps of comparing each portion of first image data obtained by capturing an extraction object with another portion of the first image data or second image data, thereby generating shape data as an image representing a provisional region of the extraction object in the first image data, and matching a contour of the shape data to a contour of the extraction object by using the first image data and the provisionally generated shape data.
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公开(公告)号:US07215709B2
公开(公告)日:2007-05-08
申请号:US10971284
申请日:2004-10-25
IPC分类号: H04B1/66
摘要: An alpha-map encoding apparatus includes a first down-sampling circuit (21) for down-sampling an alpha-map signal which represents the shape of an object and the position in the frame of the object at a down-sampling ratio based on size conversion ratio information, an up-sampling circuit (23) for up-sampling the alpha-map signal at an up-sampling ratio based on size conversion ratio information given to restore the down-sampled alpha-map signal to an original size, and outputting a local decoded alpha-map signal, a motion estimation/compensation circuit (25) for generating a motion estimation/compensation signal on the basis of the previous decoded video signal and a motion vector signal, a second down-sampling circuit (26) for down-sampling the motion estimation/compensation signal at the down-sampling ratio, a binary image encoder for encoding the alpha-map signal down-sampled by the first down-sampling circuit to a binary image in accordance with the motion estimation/compensation signal down-sampled by the second down-sampling circuit, and outputting an encoded binary image signal, and a multiplexer for multiplexing and outputting the encoded binary image signal and the up-sampling ratio information.
摘要翻译: 阿尔法 - 地图编码装置包括:第一下采样电路(21),用于以基于尺寸的下采样比下降采样表示对象的形状和对象的帧中的位置的阿尔法 - 转换比信息,上采样电路(23),用于基于给定的大小转换比率信息以上取样比对上述阿尔法 - 映射信号进行上采样以将下采样的阿尔法 - 映射信号恢复到原始大小;以及 输出局部解码的阿尔法 - 映射信号,基于先前解码的视频信号和运动矢量信号产生运动估计/补偿信号的运动估计/补偿电路(25),第二下采样电路(26) 用于以下采样比对运动估计/补偿信号进行下采样的二进制图像编码器,用于根据运动估计/运算将由第一下采样电路下采样的阿尔法 - 映射信号编码为二进制图像 由第二下采样电路进行下采样的信号信号,并输出编码的二进制图像信号,以及多路复用器,用于复用并输出编码的二进制图像信号和上采样比信息。
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公开(公告)号:US20060104609A1
公开(公告)日:2006-05-18
申请号:US11268618
申请日:2005-11-08
申请人: Yoshihiro Ohmori , Koji Yamamoto , Takashi Ida
发明人: Yoshihiro Ohmori , Koji Yamamoto , Takashi Ida
IPC分类号: H04N5/783
摘要: According to an embodiment, a reproducing device including: a unit storing pictures; a controller for controlling reproduction of the pictures; a unit displaying the pictures under controlling; a unit allowing an audience to indicate a reproducing mode such as an unmagnified speed reproduction, a fast-forwarding or the like; a calculator calculating a feature quantity from the stored pictures; a unit determining a time-wise shortened reproducing mode for a scene on basis of the calculated feature quantity; and a unit presenting the reproducing mode for a scene of the pictures under reproduction to the audience on basis of the determining. When seemingly unimportant scene is or is to be reproduced, a reproducing mode such as fast-forwarding and skipping some or whole of the scene is recommended to the audience; whereby the audience can interactively accelerate or abbreviate reproduction of the pictures and/or sounds while checking the pictures and/or sounds.
摘要翻译: 根据实施例,一种再现装置,包括:存储图像的单元; 用于控制图像的再现的控制器; 显示控制下的图片的单元; 允许观众指示诸如未放大的速度再现,快进等的再现模式的单元; 从所存储的图像计算特征量的计算器; 基于所计算的特征量确定场景的时间上缩短的再现模式的单元; 以及基于该确定向观众呈现正在再现的图片的场景的再现模式的单元。 当看似不重要的场景被复制出来的时候,向观众推荐一些复制方式,如快进和跳过一些或全部场景; 由此观众可以在检查图片和/或声音的同时交互地加速或缩写图片和/或声音的再现。
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公开(公告)号:US06961471B2
公开(公告)日:2005-11-01
申请号:US10972538
申请日:2004-10-26
CPC分类号: G06T3/4023 , G06T3/40 , H04N19/20 , H04N19/29 , H04N19/59
摘要: A video encoding apparatus is provided with a resolution converting section, an encoding section, and a transmitting section. The resolution converting section enlarges or reduces a binary picture which represents the shape of an object. The encoding section encodes a binary picture reduced by the resolution converting section. The reduction ratio used by the resolution converting section is encoded, and the transmitting section transmits this encoded reduction ratio along with encoded data on the binary picture. The amount of encoded data produced from the encoding section is controlled by changing the enlargement/reduction ratio used by the resolution converting section.
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公开(公告)号:US20050084160A1
公开(公告)日:2005-04-21
申请号:US10972538
申请日:2004-10-26
CPC分类号: G06T3/4023 , G06T3/40 , H04N19/20 , H04N19/29 , H04N19/59
摘要: A video encoding apparatus is provided with a resolution converting section, an encoding section, and a transmitting section. The resolution converting section enlarges or reduces a binary picture which represents the shape of an object. The encoding section encodes a binary picture reduced by the resolution converting section. The reduction ratio used by the resolution converting section is encoded, and the transmitting section transmits this encoded reduction ratio along with encoded data on the binary picture. The amount of encoded data produced from the encoding section is controlled by changing the enlargement/reduction ratio used by the resolution converting section.
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公开(公告)号:US06754269B1
公开(公告)日:2004-06-22
申请号:US09634550
申请日:2000-08-08
IPC分类号: H04N712
摘要: An alpha-map encoding apparatus includes a first down-sampling circuit (21) for down-sampling an alpha-map signal which represents the shape of an object and the position in the frame of the object at a down-sampling ratio based on size conversion ratio information, an up-sampling circuit (23) for up-sampling the alpha-map signal at an up-sampling ratio based on size conversion ratio information given to restore the down-sampled alpha-map signal to an original size, and outputting a local decoded alpha-map signal, a motion estimation/compensation circuit (25) for generating a motion estimation/compensation signal on the basis of the previous decoded video signal and a motion vector signal, a second down-sampling circuit (26) for down-sampling the motion estimation/compensation signal at the down-sampling ratio, a binary image encoder for encoding the alpha-map signal down-sampled by the first down-sampling circuit to a binary image in accordance with the motion estimation/compensation signal down-sampled by the second down-sampling circuit, and outputting an encoded binary image signal, and a multiplexer for multiplexing and outputting the encoded binary image signal and the up-sampling ratio information.
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公开(公告)号:US06519285B2
公开(公告)日:2003-02-11
申请号:US09783549
申请日:2001-02-15
申请人: Noboru Yamaguchi , Toshiaki Watanabe , Takashi Ida
发明人: Noboru Yamaguchi , Toshiaki Watanabe , Takashi Ida
IPC分类号: H04N732
CPC分类号: G06T3/40 , G06T3/4084 , H04N19/124 , H04N19/129 , H04N19/132 , H04N19/146 , H04N19/152 , H04N19/159 , H04N19/176 , H04N19/18 , H04N19/187 , H04N19/196 , H04N19/30 , H04N19/36 , H04N19/46 , H04N19/48 , H04N19/61 , H04N19/619
摘要: An encoding apparatus includes an encoder for encoding an alpha-map signal for discriminating a background from an object of an input picture in motion compensation prediction (MV)+transform encoding which uses MV in a domain of each of N×N transform coefficients (n), a transform circuit for transforming Pf into n in accordance with the alpha-map signal, an inverse transform circuit for reconstructing Pf by inversely transforming n in accordance with the alpha-map signal, a selector for obtaining a motion compensation prediction value (p) in the mth layer (m=2 to M) by switching p in the mth layer and p in the (m−1)th layer for each n, the selector selecting p in the mth layer for n by which a quantized output (Q) in the (m−1)th layer is 0 and selecting p in the (m−1)th layer for n by which Q=1 or more, an adder for calculating a difference df between a prediction error signal in the mth layer and a dequantized output in the (m−1)th layer, and an encoder for encoding and outputting the quantized signal of df. This encoding apparatus realizes SNR scalability in M layers.
摘要翻译: 编码装置包括编码器,用于对运动补偿预测(MV)+变换编码中的每个N×N变换系数(n)的MV使用的MV进行编码,用于区分来自输入图像的对象的背景的阿尔法 - 用于根据阿尔法 - 映射信号将Pf变换为n的变换电路,用于通过根据阿尔法 - 映射信号逆变换n来重建Pf的逆变换电路,用于获得运动补偿预测值(p)的选择器 通过在第m层切换第m层(m = 2至M),并且对于每个n,在第(m-1)层中选择p,选择器选择在第m层中的n,其中量化输出(Q) 在第(m-1)层为0并且在第(m-1)层中选择p为Q = 1以上的n的加法器,用于计算第m层中的预测误差信号与 第(m-1)层中的去量化输出和用于编码和输出的编码器 df的量化信号。 该编码装置实现M层中的SNR可伸缩性。
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公开(公告)号:US06310056B1
公开(公告)日:2001-10-30
申请号:US09355272
申请日:1999-07-28
申请人: Yuko Kano , Kazuhiro Aihara , Yumiko Toyooka , Toshiro Sasaki , Hiromasa Takizawa , Kenichi Fushihara , Kazuko Kobayashi , Kunio Atsumi , Katsuyoshi Iwamatsu , Takashi Ida
发明人: Yuko Kano , Kazuhiro Aihara , Yumiko Toyooka , Toshiro Sasaki , Hiromasa Takizawa , Kenichi Fushihara , Kazuko Kobayashi , Kunio Atsumi , Katsuyoshi Iwamatsu , Takashi Ida
IPC分类号: A61K31429
CPC分类号: C07D519/00
摘要: The carbapenem derivatives represented by the following formula (I) is disclosed. These compounds have strong anti-bacterial activities against bacteria including methicillin resistant Staphylococcus aureus, penicillin resistant Streptococcus pneumoniae, Enterococci, influenza, and &bgr;-lactamase producing bacteria, and have high stabilities to DHP-1 wherein R1 represents hydrogen or methyl, either one of R2, R3, R4, or R5 represents the bond to the 2-position on the carbapenem ring, and the remaining three respectively represent hydrogen, halogen, nitro, cyano, alkyl, cycloalkyl, alkylthio, alkenyl, formyl, alkylcarbonyl, alkoxycarbonyl, aminosulfonyl, aryl carbonyl, aryl, carbamoyl, N-lower alkylcarbamoyl, N,N-di-lower alkylaminocarbonyl, lower alkoxyiminomethyl, or hydroxyiminomethyl, R6 is not present or represents alkyl, cycloalkyl, or alkenyl, and R is not present, or represents hydrogen or a group which may be metabolically hydrolyzed in the body, provided that when R6 is not present, R represents hydrogen or a group which may be metabolically hydrolyzed in the body, and when R6 is present, R is not present, and the compound forms an inner salt.
摘要翻译: 公开了由下式(I)表示的碳青霉烯衍生物。 这些化合物对包括耐甲氧西林金黄色葡萄球菌,青霉素耐药性肺炎链球菌,肠球菌,流感和β-内酰胺酶生产细菌在内的细菌具有很强的抗细菌活性,并且对于DHP-1具有高稳定性,其中R 1表示氢或甲基,R 2 ,R 3,R 4或R 5表示碳青霉烯环上2-位的键,其余3个分别表示氢,卤素,硝基,氰基,烷基,环烷基,烷硫基,烯基,甲酰基,烷基羰基,烷氧基羰基,氨基磺酰基, 芳基羰基,芳基,氨基甲酰基,N-低级烷基氨基甲酰基,N,N-二低级烷基氨基羰基,低级烷氧基亚氨基甲基或羟基亚氨基甲基,R6不存在或表示烷基,环烷基或烯基,R不存在,或表示氢或 可以在体内代谢水解的基团,条件是当R 6不存在时,R代表氢或可以代谢地水解的基团 e体,当R 6存在时,R不存在,且该化合物形成内盐。
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