摘要:
As a result of studies on compounds having a selective inhibitory activity against 17βHSD type 5, the present inventors have confirmed that a {1-[(indol-2-yl)carbonyl]piperidyl}alkanol derivative has a potent selective inhibitory activity against 17βHSD type 5. The invention has been completed based on these findings. The compound of the present invention can be used as an agent for treating and/or an agent for preventing diseases associated with 17βHSD type 5, such as benign prostatic hyperplasia and prostate cancer, without accompanying adverse effects due to a decrease in testosterone.
摘要:
The present invention relates to an amorphous, vitreous phosphorus-potassium fertilizer obtained by melting raw materials containing phosphorus pentoxide (P2O5), potassium oxide (K2O), providers of SiO2 and silicates, and providers of MgO and CaO. The fertilizer of the present invention is produced by a process of melting the raw materials, followed by quenching, enabling the formation of a vitreous and amorphous material containing phases of phosphorus and of potassium, which are soluble in a weak acid.
摘要翻译:本发明涉及通过将含有五氧化二磷(P 2 O 5),氧化钾(K 2 O),SiO 2和硅酸盐的提供者以及MgO和CaO的提供者的原料熔化而获得的无定形磷酸钾钾肥。 本发明的肥料是通过熔化原料,然后淬火的方法生产的,能够形成含有磷和钾的玻璃状和无定形物质,它们可溶于弱酸。
摘要:
A inkjet printer including a plurality of heads installed in a staggered arrangement, and a relay board for receiving image data, a control signal conforming to each head, and a timing signal for determining timed intervals to emit ink particles from the control unit of the inkjet printer, and for sending the received image data, control signal and timing signal to the aforementioned plurality of respective drive signal generating circuits.
摘要:
An automatic exposure (AE) sensor includes a line-selecting circuit for line selection between horizontal lines and vertical lines, in addition to components of a typical AE sensor. The line-selecting circuit temporally filters a SYNC pulse for notifying a subsequent circuit about a pulse timing of an imaging signal to select a line to be read out and to cause the subsequent circuit to change an active pixel region. The number of selected lines is determined by an external input. The active pixel region is reduced when the AE sensor is incorporated in a device having a low performance CPU, thereby reducing load on the CPU. The active pixel region is increased when the AE sensor is incorporated in a device having a high performance CPU, thereby effectively using the CPU performance to achieve higher density control.
摘要:
In a high-voltage transformer, an insulating ring is placed on and along the inner surface of the core housing, and gaps are formed between the tips of the flange-like plates of the coil bobbin and the inner side of the insulating ring. With such a construction, the gaps and the insulating ring are provided between the coil bobbin and the inner wall of the core housing, so that the flange-like plates of the coil bobbin do not come in contact with the inner surface of cylindrical wall of the core housing. Therefore, a surface distance of the coil bobbin ranges to a contact surface of the coil bobbin where it comes in contact with the front wall of the core housing. The surface distance is elongated. The voltage drop by the creepage discharge does no occur.
摘要:
A regenerative pump includes a casing which a recessed fluid flow passage interconnecting a suction port and a discharge port is formed in an arcuate shape. An impeller is provided rotatably with respect to the casing and formed with a plurality of vane members which face the recessed fluid flow passage. A recessed damping portion is formed in a terminal end portion of the recessed fluid flow passage on a discharge port side thereof to begin at a position corresponding to the discharge port and extend along a rotating direction of the impeller. The recessed damping portion has a depth which is smaller than that of a main depth of the recessed fluid flow passage and substantially constant.
摘要:
A wire harness is constructed by bundling a plurality of electric wires in which conductors are surrounded with insulating coatings respectively. The electric wires are constructed of aluminum electric wires in which the conductors consist of aluminum or aluminum alloy and copper electric wires in which the conductors consist of copper or copper alloy. A plurality of the aluminum electric wires is disposed so as to surround the copper electric wires having a lower shape retention property than the aluminum electric wires. The bundles electric wires include bent portions formed by bending or curving the bundled electric wires respectively.
摘要:
The present invention relates to a new cyclic peptide compound or a salt thereof, which has anti-hepatitis C virus activities based on inhibitory activity against the RNA replication of hepatitis C virus replicon, to a process for preparation thereof comprising a rearrangement reaction under a mild acidic condition and the following amino acid changing reactions etc., to a pharmaceutical composition comprising the same, and to a method for prophylactic and/or therapeutic treatment of hepatitis C in a human being or an animal.
摘要:
The present invention relates to a new cyclic peptide compound or a salt thereof, which has anti-hepatitis C virus activities based on inhibitory activity against the RNA replication of hepatitis C virus replicon, to a process for preparation thereof comprising a rearrangement reaction under a mild acidic condition and the following amino acid changing reactions etc., to a pharmaceutical composition comprising the same, and to a method for prophylactic and/or therapeutic treatment of hepatitis C in a human being or an animal.
摘要:
The present invention relates to a novel compound or a salt thereof, which is useful as a CRTH2 antagonist, especially as a medicament for disorder that participates eosinophil, for example, allergic disorder such as asthma, allergic rhinitis, allergic dermatitis, conjunctival inflammation, hives, eosinophilic bronchitis, food allergy, inflammation of the nasal sinuses, multiple sclerosis, angiitis, or chronic obstructive pulmonary disease (COPD) and the like.