Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives
    1.
    发明授权
    Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives 失效
    杀虫剂1,2,3,4-四氢-5-硝基 - 嘧啶衍生物

    公开(公告)号:US4902689A

    公开(公告)日:1990-02-20

    申请号:US271551

    申请日:1988-11-15

    摘要: Insecticidal 1,2,3,4-tetrahydro-5-nitropyrimidines of the formula ##STR1## in which R.sup.1 stands for hydrogen or for optionally substituted radicals from the group consisting of benzyl, picolyl (pyridylmethyl) and phenoxyalkyl,n stands for the number 0 or 1 andR.sup.2 stands for the --A--R.sup.3 group, in whichA stands for a direct bond or for the --(CH.sub.2).sub.m -- or --(CH.sub.2).sub.x --Y--(CH.sub.2).sub.z -- groupings, wherem stands for the numbers 1 to 4,x and z stand for the numbers 0, 1 or 2, it being possible for x and z to be identical or different, andY stands for oxygen, sulphur or for the --NH-- or ##STR2## groupings, whereR.sup.4 stands for optionally alkoxycarbonyl-substituted C.sub.1 -C.sub.4 -alkyl, cyano, hydroxyl or for phenyl, andR.sup.3 stands for halogeno-C.sub.1 -C.sub.4 -alkyl or for an optionally substituted radical selected from the group consisting of phenyl, naphthyl, anthryl, phenanthryl, pyridyl, furyl, thienyl, piperidyl and 1,3-benzodioxolyl, with certain exceptions,and salts thereof.

    摘要翻译: 式(I)的杀虫剂1,2,3,4-四氢-5-硝基嘧啶,其中R1代表氢或任选取代的基团,由苄基,吡啶甲基(吡啶基甲基)和苯氧基烷基组成的组中,n表示 对于数字0或1,并且R 2表示-A-R 3基团,其中A表示直接键或 - 表示 - (CH 2)m - 或 - (CH 2)x Y-(CH 2)z - 基团,其中m 代表数字1至4,x和z表示数字0,1或2,x和z可以相同或不同,Y表示氧,硫或-NH-或

    1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives
    3.
    发明授权
    1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives 失效
    1,2,3,6-四氢-5-硝基 - 嘧啶衍生物

    公开(公告)号:US4831036A

    公开(公告)日:1989-05-16

    申请号:US52102

    申请日:1987-05-18

    CPC分类号: C07D487/04 A01N43/90

    摘要: New 1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives of the formula ##STR1## in which n represents the numbers 0, 1 or 2,R.sup.1 represents hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, aralkyl and hetarylalkyl, andR.sup.2 represents dialkylamino, alkoxy, alkenyloxy, aralkoxy or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl and hetarylalkyl,and their acid addition salts have been found.It has furthermore been found that these 1,2,3,6-tetrahydro-5-nitor-pyrimidine derivatives have unexpectedly high activity as insecticides, nematicides and ectoparasiticides.

    摘要翻译: 新的具有式“IMAGE”的1,2,3,6-四氢-5-硝基 - 嘧啶衍生物,其中n表示数字0,1或2,R 1表示氢或任选取代的基团,其包含烷基,烯基, 烷基,芳烷基和杂芳基烷基,并且R2表示二烷基氨基,烷氧基,烯氧基,芳烷氧基或任选被取代的基团,包括烷基,烯基,炔基,环烷基,芳烷基和杂芳基烷基,及其酸加成盐。 此外已经发现,这些1,2,3,6-四氢-5-硝基 - 嘧啶衍生物作为杀虫剂,杀线虫剂和外寄生虫杀螨剂具有出人意料的高活性。

    Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives
    4.
    发明授权
    Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives 失效
    杀虫剂1,2,3,4-四氢-5-硝基 - 嘧啶衍生物

    公开(公告)号:US4895850A

    公开(公告)日:1990-01-23

    申请号:US271555

    申请日:1988-11-15

    IPC分类号: A01N43/90 C07D487/04

    CPC分类号: C07D487/04

    摘要: Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives of the formula ##STR1## in which n is 0 or 1,A is a direct bond, --(CH.sub.2).sub.m -- or --(CH.sub.2).sub.x --Y--(CH.sub.2).sub.z,m is a number from 1 to 4,x and z each independently is 0, 1 or 2,Y is oxygen, sulphur, --NH-- or ##STR2## R.sup.2 is optionally alkoxycarbonyl-substituted C.sub.1 -C.sub.4 -alkyl, or cyano, hydroxyl or phenyl, andR.sup.1 is halogeno-C.sub.1 -C.sub.4 -alkyl or an optionally substituted radical from the group consisting of phenyl, naphthyl, anthryl, phenanthryl, pyridyl, furyl, thienyl, piperidyl and 1,3-benzodioxolyl,and their acid addition salts.

    摘要翻译: 式(I)的杀虫剂1,2,3,4-四氢-5-硝基 - 嘧啶衍生物,其中n为0或1,A为直接键, - (CH 2)m - 或 - (CH 2 )xY-(CH 2)z,m为1至4的数,x和z各自独立地为0,1或2,Y为氧,硫,-NH-或R 2为烷氧基羰基取代的C1- C 1 -C 4烷基或氰基,羟基或苯基,R 1为卤代-C 1 -C 4 - 烷基或任选取代的苯基,萘基,蒽基,菲基,吡啶基,呋喃基,噻吩基,哌啶基和1,3 - 苯并二恶唑基和它们的酸加成盐。

    Microcapsule suspensions
    6.
    发明授权
    Microcapsule suspensions 失效
    微胶囊悬浮液

    公开(公告)号:US06730635B2

    公开(公告)日:2004-05-04

    申请号:US10221464

    申请日:2002-09-12

    IPC分类号: A01N2528

    摘要: The invention relates to microcapsule suspensions containing (A) a particulate disperse phase of microcapsules comprising: (1) sleeves that are reaction products of mixtures of toluylene diisocyanate and 4,4′-methylenebis-(cyclohexyl isocyanate) with at least one diamine and/or polyamine, and (2) a capsule filling comprising: (i) at least one solid insecticidally and/or herbicidally active compound, (ii) at least one liquid aliphatic hydrocarbon having a boiling point above 160° C., (iii) at least one oil-soluble polymeric dispersing agent, and (iv) optional agrochemically active compounds that are liquid at room temperature, and (B) a liquid aqueous phase comprising water, optional additives, and optional agrochemically active compounds in non-encapsulated form that are solid at room temperature.

    摘要翻译: 本发明涉及包含(A)微胶囊的颗粒分散相的微胶囊悬浮液,其包含:(1)作为甲苯二异氰酸酯和4,4'-亚甲基双(环己基异氰酸酯)与至少一种二胺和/ 或多胺,和(2)胶囊填充物,其包含:(i)至少一种固体杀虫剂和/或除草活性化合物,(ii)至少一种沸点高于160℃的液体脂族烃,(iii) 至少一种油溶性聚合物分散剂,和(iv)在室温下为液体的任选的农用化学活性化合物,和(B)包含水,任选的添加剂和非封装形式的任选的农业化学活性化合物的液体水相, 在室温下固体。

    Microcapsule formulations
    8.
    发明申请
    Microcapsule formulations 有权
    微胶囊制剂

    公开(公告)号:US20050221991A1

    公开(公告)日:2005-10-06

    申请号:US10515590

    申请日:2003-05-16

    CPC分类号: A01N25/28 Y10S514/963

    摘要: The invention relates to novel microcapsule formulations of (A) a particulate disperse phase of microcapsules comprising (1) a polyurea and/or polyurethane coating with average layer thicknesses of between 5 and 20 nm, and (2) a capsule filling comprising at least one penetrant and, optionally, additives, and (B) a suspension comprising (1) at least one solid agrochemical active compound, (2) additives, (3) water, and (4) optionally, one or more agrochemical active compounds that are liquid at room temperature. The invention further relates to a process for the preparation of these microcapsule formulations and to their use for applying agrochemical active compounds.

    摘要翻译: 本发明涉及(A)微胶囊的颗粒分散相的新型微胶囊制剂,其包含(1)平均层厚度为5至20nm的聚脲和/或聚氨酯涂层,和(2)胶囊填充物,其包含至少一种 渗透剂和任选的添加剂,和(B)悬浮液,其包含(1)至少一种固体农业化学活性化合物,(2)添加剂,(3)水和(4)任选的一种或多种液体的农药活性化合物 在室温下。 本发明还涉及制备这些微胶囊制剂的方法及其用于施用农药活性化合物的用途。