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1.
公开(公告)号:US4902689A
公开(公告)日:1990-02-20
申请号:US271551
申请日:1988-11-15
IPC分类号: A01N43/90 , C07D487/04 , C09B67/00
CPC分类号: C07D487/04 , A01N43/90 , C09B67/0094
摘要: Insecticidal 1,2,3,4-tetrahydro-5-nitropyrimidines of the formula ##STR1## in which R.sup.1 stands for hydrogen or for optionally substituted radicals from the group consisting of benzyl, picolyl (pyridylmethyl) and phenoxyalkyl,n stands for the number 0 or 1 andR.sup.2 stands for the --A--R.sup.3 group, in whichA stands for a direct bond or for the --(CH.sub.2).sub.m -- or --(CH.sub.2).sub.x --Y--(CH.sub.2).sub.z -- groupings, wherem stands for the numbers 1 to 4,x and z stand for the numbers 0, 1 or 2, it being possible for x and z to be identical or different, andY stands for oxygen, sulphur or for the --NH-- or ##STR2## groupings, whereR.sup.4 stands for optionally alkoxycarbonyl-substituted C.sub.1 -C.sub.4 -alkyl, cyano, hydroxyl or for phenyl, andR.sup.3 stands for halogeno-C.sub.1 -C.sub.4 -alkyl or for an optionally substituted radical selected from the group consisting of phenyl, naphthyl, anthryl, phenanthryl, pyridyl, furyl, thienyl, piperidyl and 1,3-benzodioxolyl, with certain exceptions,and salts thereof.
摘要翻译: 式(I)的杀虫剂1,2,3,4-四氢-5-硝基嘧啶,其中R1代表氢或任选取代的基团,由苄基,吡啶甲基(吡啶基甲基)和苯氧基烷基组成的组中,n表示 对于数字0或1,并且R 2表示-A-R 3基团,其中A表示直接键或 - 表示 - (CH 2)m - 或 - (CH 2)x Y-(CH 2)z - 基团,其中m 代表数字1至4,x和z表示数字0,1或2,x和z可以相同或不同,Y表示氧,硫或-NH-或
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公开(公告)号:US4968695A
公开(公告)日:1990-11-06
申请号:US192445
申请日:1988-05-11
IPC分类号: A01N57/16 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/832 , A01N43/86 , A01N47/16 , A01N47/22 , A01N47/38 , A01N57/32 , C07D239/26 , C07D239/30 , C07D277/28 , C07D277/32 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , C07F9/645 , C07F9/6506 , C07F9/6527 , C07F9/6536 , C07F9/6539 , C07F9/6558
CPC分类号: C07D401/06 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/86 , A01N47/16 , A01N47/22 , A01N47/38 , A01N57/32 , C07D413/06 , C07D417/06
摘要: Pest-combating agents, in particular as insecticides which substituted nitroalkenes of the formula ##STR1## in which m represents 0, 1 or 2,A represents alkanediyl,R.sup.1 represents an optionally substituted five-or six-membered heterocyclic grouping,R.sup.2 represents hydrogen or alkyl,R.sup.3 represents hydrogen or optionally substituted alkyl, alkenyl, alkinyl, benzyl, furyl, furylmethyl, thenyl, thienyl or pyridyl,R.sup.4 represents optionally substituted phenyl, pyrimidinyl, imidazolyl or triazolyl andX represents oxygen, sulphur or the grouping N--R.sup.5,whereinR.sup.5 represents hydrogen, optionally substituted alkyl, alkenyl, alkinyl, or benzyl, formyl, or optionally substituted alkylcarbonyl, cycloalkylcarbonyl, alkenylcarbonyl, phenylcarbonyl or naphthylcarbonyl.
摘要翻译: 杀虫剂,特别是作为杀虫剂,其取代式为“IMAGE”的硝基烯烃,其中m代表0,1或2,A代表烷二基,R 1代表任选取代的五元或六元杂环基,R 2表示氢或 烷基,R 3表示氢或任选取代的烷基,烯基,炔基,苄基,呋喃基,呋喃基甲基,噻吩基,噻吩基或吡啶基,R4表示任选取代的苯基,嘧啶基,咪唑基或三唑基,X表示氧,硫或分组N-R5, 其中R5表示氢,任选取代的烷基,烯基,炔基或苄基,甲酰基或任选取代的烷基羰基,环烷基羰基,烯基羰基,苯基羰基或萘基羰基。
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公开(公告)号:US4831036A
公开(公告)日:1989-05-16
申请号:US52102
申请日:1987-05-18
IPC分类号: C07D401/12 , A01N43/48 , A01N43/90 , C07D20060101 , C07D239/06 , C07D409/12 , C07D417/12 , C07D487/04 , C07D521/00
CPC分类号: C07D487/04 , A01N43/90
摘要: New 1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives of the formula ##STR1## in which n represents the numbers 0, 1 or 2,R.sup.1 represents hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, aralkyl and hetarylalkyl, andR.sup.2 represents dialkylamino, alkoxy, alkenyloxy, aralkoxy or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl and hetarylalkyl,and their acid addition salts have been found.It has furthermore been found that these 1,2,3,6-tetrahydro-5-nitor-pyrimidine derivatives have unexpectedly high activity as insecticides, nematicides and ectoparasiticides.
摘要翻译: 新的具有式“IMAGE”的1,2,3,6-四氢-5-硝基 - 嘧啶衍生物,其中n表示数字0,1或2,R 1表示氢或任选取代的基团,其包含烷基,烯基, 烷基,芳烷基和杂芳基烷基,并且R2表示二烷基氨基,烷氧基,烯氧基,芳烷氧基或任选被取代的基团,包括烷基,烯基,炔基,环烷基,芳烷基和杂芳基烷基,及其酸加成盐。 此外已经发现,这些1,2,3,6-四氢-5-硝基 - 嘧啶衍生物作为杀虫剂,杀线虫剂和外寄生虫杀螨剂具有出人意料的高活性。
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4.
公开(公告)号:US4895850A
公开(公告)日:1990-01-23
申请号:US271555
申请日:1988-11-15
申请人: Ernst Gesing , Hilmar Wolf , Benedikt Becker , Bernhard Homeyer
发明人: Ernst Gesing , Hilmar Wolf , Benedikt Becker , Bernhard Homeyer
IPC分类号: A01N43/90 , C07D487/04
CPC分类号: C07D487/04
摘要: Insecticidal 1,2,3,4-tetrahydro-5-nitro-pyrimidine derivatives of the formula ##STR1## in which n is 0 or 1,A is a direct bond, --(CH.sub.2).sub.m -- or --(CH.sub.2).sub.x --Y--(CH.sub.2).sub.z,m is a number from 1 to 4,x and z each independently is 0, 1 or 2,Y is oxygen, sulphur, --NH-- or ##STR2## R.sup.2 is optionally alkoxycarbonyl-substituted C.sub.1 -C.sub.4 -alkyl, or cyano, hydroxyl or phenyl, andR.sup.1 is halogeno-C.sub.1 -C.sub.4 -alkyl or an optionally substituted radical from the group consisting of phenyl, naphthyl, anthryl, phenanthryl, pyridyl, furyl, thienyl, piperidyl and 1,3-benzodioxolyl,and their acid addition salts.
摘要翻译: 式(I)的杀虫剂1,2,3,4-四氢-5-硝基 - 嘧啶衍生物,其中n为0或1,A为直接键, - (CH 2)m - 或 - (CH 2 )xY-(CH 2)z,m为1至4的数,x和z各自独立地为0,1或2,Y为氧,硫,-NH-或R 2为烷氧基羰基取代的C1- C 1 -C 4烷基或氰基,羟基或苯基,R 1为卤代-C 1 -C 4 - 烷基或任选取代的苯基,萘基,蒽基,菲基,吡啶基,呋喃基,噻吩基,哌啶基和1,3 - 苯并二恶唑基和它们的酸加成盐。
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公开(公告)号:US5236923A
公开(公告)日:1993-08-17
申请号:US798685
申请日:1991-11-26
IPC分类号: A01N43/54 , A01N43/76 , C07D239/26 , C07D239/28 , C07D239/30 , C07D239/34 , C07D239/38 , C07D239/46 , C07D239/52 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12
CPC分类号: C07D239/28 , A01N43/54 , C07D239/34 , C07D239/47 , C07D239/52 , C07D405/12 , C07D413/10
摘要: New substituted pyrimidylamide oximes of the general formula (I) ##STR1## in which R.sup.1, R.sup.2, R.sup.3, A and Ar have the meanings given in the description, new intermediates for their preparation, and their use for combating pests.The new compounds of the formula (I) can be prepared by analogous processes, for example by reacting suitable pyrimidylamide oximes with suitable alkylating agents. The starting compounds which are also new, namely the pyrimidylamide oximes of the formula (II) in which --A--Ar represents hydrogen, can be prepared from suitable cynaopyrimidines with hydroxylamine or its acid adducts.
摘要翻译: 其中R 1,R 2,R 3,A和Ar具有本说明书中给出的含义的新的通式(I)的取代的嘧啶酰胺肟其制备的新中间体及其在防治害虫中的用途。 式(I)的新化合物可以通过类似的方法制备,例如通过使合适的嘧啶酰胺肟与合适的烷基化剂反应来制备。 也可以由具有羟胺或其酸加合物的合适的炔丙嘧啶制备也是新的起始化合物,即其中-A-Ar表示氢的式(II)的嘧啶酰胺肟。
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公开(公告)号:US06730635B2
公开(公告)日:2004-05-04
申请号:US10221464
申请日:2002-09-12
IPC分类号: A01N2528
CPC分类号: B01J13/02 , A01N25/04 , A01N25/10 , A01N25/28 , A01N51/00 , Y10S514/963 , A01N2300/00
摘要: The invention relates to microcapsule suspensions containing (A) a particulate disperse phase of microcapsules comprising: (1) sleeves that are reaction products of mixtures of toluylene diisocyanate and 4,4′-methylenebis-(cyclohexyl isocyanate) with at least one diamine and/or polyamine, and (2) a capsule filling comprising: (i) at least one solid insecticidally and/or herbicidally active compound, (ii) at least one liquid aliphatic hydrocarbon having a boiling point above 160° C., (iii) at least one oil-soluble polymeric dispersing agent, and (iv) optional agrochemically active compounds that are liquid at room temperature, and (B) a liquid aqueous phase comprising water, optional additives, and optional agrochemically active compounds in non-encapsulated form that are solid at room temperature.
摘要翻译: 本发明涉及包含(A)微胶囊的颗粒分散相的微胶囊悬浮液,其包含:(1)作为甲苯二异氰酸酯和4,4'-亚甲基双(环己基异氰酸酯)与至少一种二胺和/ 或多胺,和(2)胶囊填充物,其包含:(i)至少一种固体杀虫剂和/或除草活性化合物,(ii)至少一种沸点高于160℃的液体脂族烃,(iii) 至少一种油溶性聚合物分散剂,和(iv)在室温下为液体的任选的农用化学活性化合物,和(B)包含水,任选的添加剂和非封装形式的任选的农业化学活性化合物的液体水相, 在室温下固体。
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公开(公告)号:US5256632A
公开(公告)日:1993-10-26
申请号:US900867
申请日:1992-06-18
IPC分类号: A01N43/74 , A01N43/80 , A01N43/82 , C07D261/18 , C07D263/34 , C07D271/06 , C07D271/10 , C07D275/02 , C07D275/03 , C07D277/56 , C07D285/12 , A01N43/48 , C07D271/04 , C07D413/02
CPC分类号: C07D263/34 , A01N43/74 , A01N43/80 , A01N43/82 , C07D261/18 , C07D271/06 , C07D271/10 , C07D275/03 , C07D277/56 , C07D285/12
摘要: Herbicidal sulphonylated carboxamides of the formulaR.sup.1 --CO--NH--SO.sub.2 --(A).sub.n --R.sup.2 (I)in whichn represents the numbers 0 or 1,A represents oxygen, iminio (NH) or methylene (CH.sub.2),R.sup.1 represents a five-membered heteroaryl radical which contains 1 or 2 nitrogen atoms and additionally one oxygen or sulphur atom in the ring and which is optionally substituted by halogen or by alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or phenyl which are in each case optionally substituted, andR.sup.2 represents aryl or heteroaryl which are in each case optionally substituted,or salts thereof, with the exclusion of the compound 2-dimethylamino-N-(4-methyl-phenylsulphonyl)-5-thiazole carboxamide.
摘要翻译: 式R 1 -CO-NH-SO 2 - (A)n -R 2(I)的除草磺酰化羧酰胺,其中n表示数字0或1,A表示氧,亚氨基(NH)或亚甲基(CH 2),R 1表示 在环中含有1或2个氮原子和另外一个氧或硫原子的五元杂芳基,其任选被卤素或烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基,二烷基氨基或苯基取代。 并且R 2代表任意取代的芳基或杂芳基,或其盐,除去化合物2-二甲基氨基-N-(4-甲基 - 苯基磺酰基)-5-噻唑甲酰胺。
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公开(公告)号:US20050221991A1
公开(公告)日:2005-10-06
申请号:US10515590
申请日:2003-05-16
申请人: Hilmar Wolf , Peter Baur , Manfred Zimmermann
发明人: Hilmar Wolf , Peter Baur , Manfred Zimmermann
IPC分类号: B01J13/16 , A01N25/04 , A01N25/10 , A01N25/28 , A01N43/653
CPC分类号: A01N25/28 , Y10S514/963
摘要: The invention relates to novel microcapsule formulations of (A) a particulate disperse phase of microcapsules comprising (1) a polyurea and/or polyurethane coating with average layer thicknesses of between 5 and 20 nm, and (2) a capsule filling comprising at least one penetrant and, optionally, additives, and (B) a suspension comprising (1) at least one solid agrochemical active compound, (2) additives, (3) water, and (4) optionally, one or more agrochemical active compounds that are liquid at room temperature. The invention further relates to a process for the preparation of these microcapsule formulations and to their use for applying agrochemical active compounds.
摘要翻译: 本发明涉及(A)微胶囊的颗粒分散相的新型微胶囊制剂,其包含(1)平均层厚度为5至20nm的聚脲和/或聚氨酯涂层,和(2)胶囊填充物,其包含至少一种 渗透剂和任选的添加剂,和(B)悬浮液,其包含(1)至少一种固体农业化学活性化合物,(2)添加剂,(3)水和(4)任选的一种或多种液体的农药活性化合物 在室温下。 本发明还涉及制备这些微胶囊制剂的方法及其用于施用农药活性化合物的用途。
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公开(公告)号:US06096751A
公开(公告)日:2000-08-01
申请号:US307278
申请日:1999-05-07
申请人: Bernd-Wieland Kruger , Hermann Uhr , Johannes Kanellakopulos , Ernst-Rudolf Gesing , Hilmar Wolf , Andreas Turberg , Norbert Mencke , Christoph Erdelen , Ulrike Wachendorff-Neumann , Jurgen Hartwig
发明人: Bernd-Wieland Kruger , Hermann Uhr , Johannes Kanellakopulos , Ernst-Rudolf Gesing , Hilmar Wolf , Andreas Turberg , Norbert Mencke , Christoph Erdelen , Ulrike Wachendorff-Neumann , Jurgen Hartwig
IPC分类号: A01N43/54 , A01N43/78 , A01N43/90 , A01N47/06 , A01N47/12 , A01N47/22 , C07D401/12 , C07D401/14 , C07D417/12 , C07D487/04 , C07D498/04 , C07D407/12 , A01N43/34
CPC分类号: C07D401/12 , A01N43/54 , A01N43/90 , A01N47/12 , C07D487/04
摘要: The present invention relates to new substituted 1, 2, 3, 4-tetrahydro-5-nitro-pyrimidines of the formula (I) ##STR1## wherein Het, R.sup.1, R.sup.2, R.sup.3 and A are as defined herein,to processes for their preparation, and to their use as pesticides and ectoparasiticides.
摘要翻译: 本发明涉及其中Het,R 1,R 2,R 3和A如本文所定义的式(I)的新的取代的1,2,3,4-四氢-5-硝基嘧啶,其制备方法和 用作杀虫剂和杀螨剂。
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公开(公告)号:US5869491A
公开(公告)日:1999-02-09
申请号:US676272
申请日:1996-07-12
申请人: Bernd-Wieland Kruger , Hermann Uhr , Johannes Kanellakopulos , Ernst-Rudolf Gesing , Hilmar Wolf , Andreas Turberg , Norbert Mencke , Christoph Erdelen , Ulrike Wachendorff-Neumann , Jurgen Hartwig
发明人: Bernd-Wieland Kruger , Hermann Uhr , Johannes Kanellakopulos , Ernst-Rudolf Gesing , Hilmar Wolf , Andreas Turberg , Norbert Mencke , Christoph Erdelen , Ulrike Wachendorff-Neumann , Jurgen Hartwig
IPC分类号: A01N43/54 , A01N43/78 , A01N43/90 , A01N47/06 , A01N47/12 , A01N47/22 , C07D401/12 , C07D401/14 , C07D417/12 , C07D487/04 , C07D498/04
CPC分类号: C07D401/12 , A01N43/54 , A01N43/90 , A01N47/12 , C07D487/04
摘要: The present invention relates to new substituted 1,2,3,4-tetrahydro-5-nitro-pyrimidines of the formula (I) ##STR1## to processes for their preperation, and to their use as pesticides and ectoparasiticides.
摘要翻译: PCT No.PCT / EP95 / 00058 Sec。 371日期1996年7月12日 102(e)日期1996年7月12日PCT提交1995年1月9日PCT公布。 公开号WO95 / 19977 日期:1995年7月27日本发明涉及式(I)的新的取代的1,2,3,4-四氢-5-硝基 - 嘧啶(Ⅰ),用于其制备方法及其作为 杀虫剂和杀螨剂。
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