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    Antimycotically active substituted 2-aminothiazoles
    1.
    发明授权
    Antimycotically active substituted 2-aminothiazoles 失效
    抗微生物活性取代的2-氨基丁酸

    公开(公告)号：US5104879A

    公开(公告)日：1992-04-14

    申请号：US596626

    申请日：1990-10-11

    申请人： Joachim Ippen ,  Bernd Baasner ,  Klaus Schaller ,  Miklos von Bittera

    发明人： Joachim Ippen ,  Bernd Baasner ,  Klaus Schaller ,  Miklos von Bittera

    IPC分类号： A61K31/505 ,  A61P31/04 ,  C07C45/00 ,  C07C45/63 ,  C07C49/80 ,  C07C49/84 ,  C07D417/12 ,  C07D417/14

    CPC分类号： C07D417/12 ,  C07C45/004 ,  C07C45/63 ,  C07C49/80 ,  C07C49/84 ,  C07D417/14

    摘要： Antimicotically active 2-aminothiazoles have been found having the formula ##STR1## in which R.sup.1 represents hydrogen or alkyl andR.sup.2 represents optionally substituted cyclohexyl or phenyl which is substituted by halogen, alkyl, halogenoalkyl, halogenoalkoxy, dioxyhalogenoalkyl or halogenoalkylthio,and their physiologically tolerable acid addition salts,with the exception of the compounds 4-(4-chlorophenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]thiazole and 4-(2,4-dichlorophenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]-thiazole and 4-(4-chloro-2-methylphenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]-thiazole and with the exception of the physiologically tolerable acid addition salts of these compoundshave been found.

    摘要翻译： 已经发现具有式“IMAGE”的反活性2-氨基噻唑，其中R1代表氢或烷基，R2代表任选取代的环己基或被卤素，烷基，卤代烷基，卤代烷氧基，二卤基烷基或卤代烷硫基取代的苯基，以及它们的生理可耐受酸 加成盐，除4-（4-氯苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基]噻唑和4-（2,4-二氯苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基] - 噻唑和4-（4-氯-2-甲基苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基] - 噻唑，除了这些化合物的生理可耐受酸加成盐之外。

    Pesticidal 3-aryl-pyrrolidine-2,4-diones
    8.
    发明授权
    Pesticidal 3-aryl-pyrrolidine-2,4-diones 失效
    杀虫剂3-芳基 - 吡咯烷-2,4-二酮

    公开(公告)号：US5186737A

    公开(公告)日：1993-02-16

    申请号：US678479

    申请日：1991-04-01

    申请人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hageman ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    发明人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hageman ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    IPC分类号： A01N43/36 ,  A01N47/06 ,  C07D207/38 ,  C07D405/12

    CPC分类号： C07D405/12 ,  A01N43/36 ,  A01N47/06 ,  C07D207/38

    摘要： Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally subsituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译： 式（I）的杀虫，杀螨，除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基，卤素或烷氧基，Y代表氢，烷基，卤素，烷氧基或卤代烷基，Z 表示烷基，卤素或烷氧基，n表示0-3的数，R表示氢或表示基团-CO-R1或-CO-O-R2，其中R1表示烷基，烯基，烷氧基烷基，烷硫基烷基，聚烷氧基烷基或环烷基 任何取代的苯基，取代的杂芳基，取代的苯氧基烷基或取代的噻唑烷基，或代表任意取代的苯基，任选取代的苯基烷基，取代的杂芳基， 取代的苯氧基烷基和取代的硫代氧基烷基，R 2表示烷基，链烯基，烷氧基烷基，聚烷氧基烷基或任选取代的苯基或环烷基，各w 任选被卤素取代的基团，A代表烷基，烯基，炔基，烷氧基烷基，聚烷氧基烷基，烷硫基烷基或环烷基，任选被杂原子中断，每个基团任选被卤素取代，或表示任选取代的芳基烷基 卤素，烷基，卤代烷基，烷氧基或硝基，B和C *彼此独立地表示氢，烷基或烷氧基烷基。

    Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas
    9.
    发明授权
    Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas 失效
    3-芳基 - 吡咯烷-2,4-二酮的杀虫互变异构体

    公开(公告)号：US5045560A

    公开(公告)日：1991-09-03

    申请号：US460208

    申请日：1990-01-02

    申请人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hagemann ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    发明人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hagemann ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    IPC分类号： A01N43/36 ,  A01N47/06 ,  C07D207/38 ,  C07D405/12

    CPC分类号： C07D405/12 ,  A01N43/36 ,  A01N47/06 ,  C07D207/38

    摘要： Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally substituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译： 式（I）的杀虫，杀螨，除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基，卤素或烷氧基，Y代表氢，烷基，卤素，烷氧基或卤代烷基，Z 表示烷基，卤素或烷氧基，n表示0-3的数，R表示氢或表示基团-CO-R1或-CO-O-R2，其中R1表示烷基，烯基，烷氧基烷基，烷硫基烷基，聚烷氧基烷基或环烷基 任何取代的苯基，取代的杂芳基，取代的苯氧基烷基或取代的噻唑烷基，或代表任意取代的苯基，任选取代的苯基烷基，取代的杂芳基， 取代的苯氧基烷基和取代的硫代氧基烷基，R 2表示烷基，链烯基，烷氧基烷基，聚烷氧基烷基或任选取代的苯基或环烷基，各w 任选被卤素取代的基团，A代表烷基，链烯基，炔基，烷氧基烷基，聚烷氧基烷基，烷硫基烷基或环烷基，任选被杂原子间隔，每个基团任选被卤素取代，或表示任选取代的芳基烷基 卤素，烷基，卤代烷基，烷氧基或硝基，B和C *彼此独立地表示氢，烷基或烷氧基烷基。

    Fluorine-containing acetophenones optionally halogenated on the CH.sub.3 -group and their precurser fluorine-containing benzonitriles
    10.
    发明授权
    Fluorine-containing acetophenones optionally halogenated on the CH.sub.3 -group and their precurser fluorine-containing benzonitriles 失效
    任选在CH3-基上卤化的含氟苯乙酮及其前体含氟苯腈

    公开(公告)号：US5142092A

    公开(公告)日：1992-08-25

    申请号：US739738

    申请日：1991-07-30

    申请人： Ernst Kysela ,  Bernd Baasner ,  Klaus Schaller

    发明人： Ernst Kysela ,  Bernd Baasner ,  Klaus Schaller

    IPC分类号： C07C45/00 ,  C07C45/63 ,  C07C49/80 ,  C07C49/807 ,  C07C49/84 ,  C07C255/50 ,  C07C255/54

    CPC分类号： C07C45/63 ,  C07C255/50 ,  C07C255/54 ,  C07C45/004 ,  C07C49/80 ,  C07C49/807 ,  C07C49/84

    摘要： Fluorine-containing acetophenones, optionally halogenated on the CH.sub.3 group, of the formula ##STR1## in which X represents hydrogen, chlorine or bromine and the radicals R.sub.1 to R.sub.5 have the following meaning,a) R.sub.1 and R.sub.4 denote fluorine, R.sub.2 and R.sub.5 denote chlorine and R.sub.3 denotes CF.sub.3, orb) R.sub.1, R.sub.3 and R.sub.4 denote fluorine and R.sub.2 and R.sub.5 denote hydrogen, orc) R.sub.1, R.sub.4 and R.sub.5 denote hydrogen, R.sub.2 denotes chlorine and R.sub.3 denotes CF.sub.3, ord) R.sub.1, R.sub.4 and R.sub.5 denote hydrogen, R.sub.2 denotes chlorine and R.sub.3 denotes OCF.sub.3, ore) R.sub.1, R.sub.4 and R.sub.5 denote hydrogen and R.sub.2 and R.sub.3 denote CF.sub.3, orf) R.sub.1 denotes chlorine, R.sub.2 denotes CF.sub.3 and R.sub.3, R.sub.4 and R.sub.5 denote hydrogen, org) R.sub.1 denotes chlorine, R.sub.2, R.sub.3 and R.sub.4 denote hydrogen and R.sub.5 denotes CF.sub.3, orh) R.sub.1 denotes chlorine, R.sub.2, R.sub.4 and R.sub.5 denote hydrogen and R.sub.3 denotes CF.sub.3and a process for their preparation from the corresponding fluorinated benzonitriles or benzyl halides by reaction with an organomagnesium compound capable of introducing methyl groups and subsequent hydrolysis, if appropriate followed by a chlorination or bromination.

    摘要翻译： 其中X表示氢，氯或溴，R 1至R 5基团的式（I）中任选卤代的含氟苯乙酮具有下列含义：a）R 1和R 4表示氟，R 2 或R 3表示CF 3，或b）R 1，R 3和R 4表示氟，R 2和R 5表示氢，或c）R 1，R 4和R 5表示氢，R 2表示氯，R 3表示CF 3，或d） R4和R5表示氢，R2表示氯，R3表示OCF3，或e）R1，R4和R5表示氢，R2和R3表示CF3，或f）R1表示氯，R2表示CF3和R3，R4和R5表示氢， 或g）R 1表示氯，R 2，R 3和R 4表示氢，R 5表示CF 3，或h）R 1表示氯，R 2，R 4和R 5表示氢，R 3表示CF 3，以及由相应的氟化苯腈或苄基 通过与能够引入甲基的有机镁化合物反应并随后h进行卤化反应 如果合适，然后进行氯解或溴化。