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公开(公告)号:US20050215435A1
公开(公告)日:2005-09-29
申请号:US10503762
申请日:2003-01-30
申请人: Markus Menges , Michael Puhl , Costin Rentzea , Albrecht Harreus , Christoph Bussche-Hunnefeld , Andreas Gypser , Anja Schwogler , Matthias Witschel , Cyrill Zagar , Klaus Grossmann , Helmut Schiffer , Franz Rohl
发明人: Markus Menges , Michael Puhl , Costin Rentzea , Albrecht Harreus , Christoph Bussche-Hunnefeld , Andreas Gypser , Anja Schwogler , Matthias Witschel , Cyrill Zagar , Klaus Grossmann , Helmut Schiffer , Franz Rohl
IPC分类号: C07C233/87 , A01N37/46 , C07C231/02 , C07C235/52 , C07C317/44 , A01N37/18
CPC分类号: A01N37/46
摘要: Phenylalanine derivatives of the formula I where the radicals are as defined in the description, and the use of these compounds as herbicides and/or for regulating plant growth is described.
摘要翻译: 其中基团如说明书中所定义的式I的苯丙氨酸衍生物以及这些化合物作为除草剂和/或用于调节植物生长的用途被描述。
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2.Tryptophan aminotransferase, indole-3-pyruvate decarboxylase and indole-3-acetaldehyde oxidase as novel targets for herbicides 审中-公开
标题翻译: 色氨酸氨基转移酶,吲哚-3-丙酮酸脱羧酶和吲哚-3-乙醛氧化酶作为除草剂的新靶标公开(公告)号:US20050159312A1
公开(公告)日:2005-07-21
申请号:US10508837
申请日:2003-03-19
申请人: Klaus Grossmann , Helmut Schiffer , Matthias Witschel , Cyril Zagar , Costin Rentzea , Markus Menges
发明人: Klaus Grossmann , Helmut Schiffer , Matthias Witschel , Cyril Zagar , Costin Rentzea , Markus Menges
IPC分类号: C12Q1/52 , A01N37/46 , A61P43/00 , C12Q1/02 , C12Q1/26 , C12Q1/48 , C12Q1/527 , A01N25/00 , C07C237/20
摘要: The present invention relates to tryptophan aminotransferase, indole-3-pyruvate decarboxylase and indole-3-acetaldehyde oxidase as novel targets for herbicides, to test methods for identifying herbicidally active inhibitors of one or more of the abovementioned enzymes, to the herbicidally active inhibitors identified by means of this method, and to methods for controlling undesired vegetation based on the inhibitors according to the invention.
摘要翻译: 本发明涉及色氨酸氨基转移酶,吲哚-3-丙酮酸脱羧酶和吲哚-3-乙醛氧化酶作为除草剂的新靶标,以测定鉴定出的一种或多种上述酶的除草活性抑制剂的方法 通过该方法,以及基于根据本发明的抑制剂来控制不希望的植物的方法。
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公开(公告)号:US06387849B1
公开(公告)日:2002-05-14
申请号:US09381474
申请日:1999-09-21
申请人: Olaf Menke , Gerhard Hamprecht , Markus Menges , Robert Reinhard , Peter Schäfer , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
发明人: Olaf Menke , Gerhard Hamprecht , Markus Menges , Robert Reinhard , Peter Schäfer , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
IPC分类号: C07D23954
CPC分类号: C07D239/54 , A01N43/54 , C07C251/48 , C07C265/12 , C07D239/56
摘要: Novel hydroximic acid derivatives I and salts thereof, where X=O, S; Y=O, S; R1=H, C1-C4-alkyl, NH2, C1-C4-alkylamino or di(C1-C4-alkyl)amino; R2=C1-C3-haloalkyl; R3=H, halogen, C1-C4-alkyl; R4=H, halogen; R5=CN, halogen; R6=C1-C6-alkyl, C2-C6-alkenyl, C3-C6-alkynyl or phenyl-C1-C6-alkyl, where the phenyl ring of this group may be unsubstituted or may carry 1-3 substituents; R7=a C1-C6-alkyl, C2-C6-alkenyl, C3-C6-alkynyl or phenyl-C1-C6-alkyl, where these 4 groups may be unsubstituted or may carry 1 to 2 substituents; Use: As herbicides; for the desiccation/defoliation of plants.
摘要翻译: 其中X = O,S; Y = O,S; R1 = H,C1-C4-烷基,NH2,C1-C4-烷基氨基或二(C1-C4-烷基)氨基的新型氢亚甲酸衍生物I和盐; R2 = C1-C3-卤代烷基; R3 = H,卤素,C1-C4-烷基; R4 = H,卤素; R5 = CN,卤素; R6 = C1-C6-烷基,C2-C6-烯基,C3-C6-炔基或 苯基-C 1 -C 6烷基,其中该基团的苯环可以是未取代的或可以带有1-3个取代基; R 7 = C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 3 -C 6炔基或苯基-C 1 C 1-6 - 烷基,其中这4个基团可以是未取代的或可以携带1至2个取代基;用途:作为除草剂; 用于植物的干燥/脱叶。
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公开(公告)号:US06191280B1
公开(公告)日:2001-02-20
申请号:US09423961
申请日:1999-11-17
申请人: Gerhard Hamprecht , Markus Menges , Olaf Menke , Robert Reinhard , Peter Schäfer , Cyrill Zagar
发明人: Gerhard Hamprecht , Markus Menges , Olaf Menke , Robert Reinhard , Peter Schäfer , Cyrill Zagar
IPC分类号: C07D21332
CPC分类号: C07D213/70 , C07B45/06 , C07D213/71
摘要: A process for preparing thiopyridines of the formula I where the substituents are as defined in the description.
摘要翻译: 制备式I的硫代吡啶的方法,其中取代基如说明书中所定义。
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公开(公告)号:US6150303A
公开(公告)日:2000-11-21
申请号:US463246
申请日:2000-01-21
申请人: Olaf Menke , Markus Menges , Gerhard Hamprecht , Robert Reinhard , Peter Schafer , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
发明人: Olaf Menke , Markus Menges , Gerhard Hamprecht , Robert Reinhard , Peter Schafer , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
IPC分类号: A01N43/80 , C07D261/04 , A01N43/72
CPC分类号: C07D261/04
摘要: Substituted 3-phenylisoxazolines I, and their salts and enol ethers, are described as herbicides ##STR1## where X.dbd.--O--, --S--, --N(R.sup.9)--;R.sup.1 .dbd.CN, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylsulfonyl;R.sup.2 .dbd.H or unsubstituted or substituted C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkyl)carbonyl, C.sub.1 -C.sub.6 -alkylsulfonyl, C.sub.2 -C.sub.6 -alkenyl, (C.sub.2 -C.sub.6 -alkenyl)carbonyl, C.sub.2 -C.sub.6 -alkynyl, (C.sub.2 -C.sub.6 -alkynyl)carbonyl;R.sup.3 .dbd.H, halogen;R.sup.4 .dbd.CN, halogen, C.sub.1 -C.sub.3 -haloalkyl;R.sup.5 .dbd.H, CN, halogen, C.sub.1 -C.sub.3 -haloalkyl;R.sup.6 .dbd.H, CN, halogen, C.sub.1 -C.sub.3 -haloalkyl or unsubstituted or substituted C.sub.1 -C.sub.6 -alkoxy;R.sup.7 .dbd.CN, halogen;R.sup.8 in position .alpha., R.sup.7 in this case being in position .beta., or in position .beta., R.sup.7 in this case being in position .alpha., is1) H, OH, SH, CN, NO.sub.2, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -haloalkoxy, C.sub.1 -C.sub.6 -haloalkylthio, C.sub.1 -C.sub.6 -alkylthio-(C.sub.1 -C.sub.6 -alkyl)carbonyl, (C.sub.1 -C.sub.6 -alkyl)iminooxycarbonyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxyamino-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkylamino-C.sub.1 -C.sub.6 -alkyl,2) unsubstituted or substituted C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio, C.sub.3 -C.sub.6 -cycloalkoxy, C.sub.3 -C.sub.6 -cycloalkylthio, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkenylthio, C.sub.2 -C.sub.6 -alkynyloxy, C.sub.2 -C.sub.6 -alkynylthio, (C.sub.1 -C.sub.6 -alkyl)carbonyloxy, (C.sub.1 -C.sub.6 -alkyl)carbonylthio, (C.sub.1 -C.sub.6 -alkoxy)carboxyloxy, (C.sub.2 -C.sub.6 -alkenyl)carbonyloxy, (C.sub.2 -C.sub.6 -alkenyl)carbonylthio, (C.sub.2 -C.sub.6 -alkynyl)carbonyloxy, (C.sub.2 -C.sub.6 -alkynyl)carbonylthio, C.sub.1 -C.sub.6 -alkylsulfonyloxy or C.sub.1 -C.sub.6 -alkylsulfonyl,3) 29 further radicals;R.sup.9 .dbd.H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkyl, (C.sub.1 -C.sub.6 -alkoxy)carbonyl-C.sub.1 -C.sub.6 -alkyl, (C.sub.3 -C.sub.6 -alkenyloxy)carbonyl-C.sub.1 -C.sub.6 -alkyl, unsubstituted or substituted phenyl or phenyl-C.sub.1 -C.sub.6 -alkyl.
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公开(公告)号:US06448205B1
公开(公告)日:2002-09-10
申请号:US09242463
申请日:1999-02-17
申请人: Peter Schäfer , Michael Rack , Gerhard Hamprecht , Helmut Walter , Karl-Otto Westphalen , Ulf Misslitz , Markus Menges , Cyrill Zagar , Olaf Menke
发明人: Peter Schäfer , Michael Rack , Gerhard Hamprecht , Helmut Walter , Karl-Otto Westphalen , Ulf Misslitz , Markus Menges , Cyrill Zagar , Olaf Menke
IPC分类号: A01N4340
CPC分类号: C07D405/10 , A01N43/40 , C07D213/71 , C07D405/12 , C07D409/10 , C07D411/10
摘要: Substituted 2-phenylpyridines of formula I where R1 to R5 are described herein, their use as herbicides and for the desiccation and/or defoliation of plants.
摘要翻译: 式I中的取代的2-苯基吡啶,其中R 1至R 5在本文中描述,其用作除草剂和用于植物的干燥和/或脱叶的用途。
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公开(公告)号:US06432880B1
公开(公告)日:2002-08-13
申请号:US09869840
申请日:2001-07-05
申请人: Olaf Menke , Markus Menges , Ingo Sagasser , Gerhard Hamprecht , Robert Reinhard , Cyrill Zagar , Karl-Otto Westphalen , Martina Otten , Helmut Walter
发明人: Olaf Menke , Markus Menges , Ingo Sagasser , Gerhard Hamprecht , Robert Reinhard , Cyrill Zagar , Karl-Otto Westphalen , Martina Otten , Helmut Walter
IPC分类号: A01N4340
CPC分类号: A01N43/40
摘要: 2-Phenylpyridines I an their salts, wherein R1 to R17, X1-X3 are as defined in the specification. The compounds are useful as herbicides, desiccants and defoliants.
摘要翻译: 2-苯基吡啶盐酸盐,其中R1至R17,X1-X3如说明书中所定义。 该化合物可用作除草剂,干燥剂和脱叶剂。
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8.1-sulfonyl-3-phenylpyrazoles and their use as herbicides and for desiccating or defoliating plants 失效
标题翻译: 1-磺酰基-3-苯基吡唑及其作为除草剂的用途,用于干燥或脱叶植物公开(公告)号:US6054413A
公开(公告)日:2000-04-25
申请号:US254923
申请日:1999-03-17
申请人: Cyrill Zagar , Gerhard Hamprecht , Markus Menges , Olaf Menke , Peter Schafer , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
发明人: Cyrill Zagar , Gerhard Hamprecht , Markus Menges , Olaf Menke , Peter Schafer , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
IPC分类号: A01N43/56 , C07D231/12 , C07D231/18 , C07D231/24 , C07D401/12 , C07D403/12 , C07D405/12 , A01N43/84 , C07D231/14 , C07D413/12
CPC分类号: C07D231/18 , A01N43/56 , C07D231/24
摘要: The present invention relates to novel 1-sulfonyl-3-phenylpyrazoles of the formula I ##STR1## and agriculturally useful salts of I. Furthermore, the invention relates tothe use of the compounds I as herbicides and/or for the desiccation and/or defoliation of plants,herbidical compositions and compositions for the desiccation and/or defoliation of plants which comprise the compounds I as active ingredients,
摘要翻译: PCT No.PCT / EP97 / 04911 Sec。 371日期1999年3月17日 102(e)1999年3月17日PCT 1997年9月9日PCT公布。 公开号WO98 / 12182 日期:1998年3月26日本发明涉及式I的新型1-磺酰基-3-苯基吡唑和I的农业上有用的盐。此外,本发明涉及化合物I作为除草剂和/或用于干燥和/ /或用于将化合物I作为活性成分的植物的干燥和/或脱叶的植物脱叶,草药组合物和组合物,
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公开(公告)号:US06383986B1
公开(公告)日:2002-05-07
申请号:US09462583
申请日:2000-01-11
申请人: Markus Menges , Gerhard Hamprecht , Olaf Menke , Robert Reinhard , Peter Schäfer , Cyrill Zagar , Karl-Otto Westphalen , Martina Otten , Helmut Walter
发明人: Markus Menges , Gerhard Hamprecht , Olaf Menke , Robert Reinhard , Peter Schäfer , Cyrill Zagar , Karl-Otto Westphalen , Martina Otten , Helmut Walter
IPC分类号: A01N4340
CPC分类号: C07D401/04 , A01N43/78 , C07D413/04 , C07D417/04
摘要: 2-(Benzaryl)pyridines I and salts thereof where n=zero, 1; R1=H, CN, NO2, NH2, OH, SH, SO2—OH, SO2—Cl, SO2—NH2, halogen, optionally halogenated alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; R2, R3=H, halogen; R4=CN, OH, halogen, alkoxy or optionally substituted benzyloxy; X=—Y—C(ZR5)═N— where the nitrogen is attached to &agr; or &bgr; and Y=—O—, —S—, —N(R6)—; Z=a chemical bond, —O—, —S—, —S(O)—, —SO2—, —N(R7)—; R5, R6, R7=H, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, phenyl or 3- to 7-membered heterocyclyl; or R5=H, CN, SH, NH2, halogen, —CH2—CH(halogen)-R8, —CH═CH—R8 or —CH═C(halogen)-R8 (R8=COOH, alkoxycarbonyl, alkylthiocarbonyl, CONH2, alkylaminocarbonyl or dialkylaminocarbonyl), when Z=a chemical bond; or R5+R7=1,3-propylene, tetramethylene, pentamethylene or ethyleneoxyethylene. Use: as herbicides, desiccants or defoliants.
摘要翻译: 2-(苯甲基)吡啶I及其盐,其中n = 0,1; R 1 = H,CN,NO 2,NH 2,OH,SH,SO 2 -OH,SO 2 -Cl,SO 2 -NH 2,卤素,任选卤代烷基,烷氧基,烷硫基 ,烷基亚磺酰基,烷基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; R2,R3 = H,卤素; R4 = CN,OH,卤素,烷氧基或任选取代的苄氧基; X = -YC(ZR5)= N-,其中氮连接到α或β 且Y = -O - , - S - , - N(R 6) - ; Z =化学键,-O - , - S - , - S(O) - , - SO 2 - , - N(R 7) R5,R6,R7 = H,任选取代的烷基,烯基,炔基,环烷基,苯基或3-至7-元杂环基; 或R 5 = H,CN,SH,NH 2,卤素,-CH 2 -CH(卤素)-R 8,-CH = CH-R 8或-CH = C(卤素)-R 8(R 8 = COOH,烷氧基羰基,烷硫基羰基,CONH 2,烷基氨基羰基 或二烷基氨基羰基),当Z =化学键时; 或R 5 + R 7 = 1,3-丙烯,四亚甲基,五亚甲基或亚乙基氧乙烯。使用:作为除草剂,干燥剂或脱叶剂。
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10.Substituted 2-benz(o)ylpyridines, their preparation and their use as herbicides 失效
标题翻译: 取代的2-苯并(o)吡啶,其制备及其作为除草剂的用途公开(公告)号:US06337305B1
公开(公告)日:2002-01-08
申请号:US09381033
申请日:1999-09-15
申请人: Peter Schäfer , Gerhard Hamprecht , Markus Menges , Olaf Menke , Michael Rack , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
发明人: Peter Schäfer , Gerhard Hamprecht , Markus Menges , Olaf Menke , Michael Rack , Cyrill Zagar , Karl-Otto Westphalen , Ulf Misslitz , Helmut Walter
IPC分类号: C07D21330
CPC分类号: C07D213/61 , A01N43/40
摘要: Substituted 2-benz(o)ylpyridines I and salts thereof where n=0, 1; X=CO, CH2, CH(C1-C4-alkyl), CH—OH, CH—CN, CH-halogen, C(halogen)2, CH—CONH2, CH—CO—O(C1-C4-alkyl), CH—O(C1-C4-alkyl), C(CN)(C1-C4-alkyl); R1=halogen, C1-C4-haloalkyl, C1-C4-alkylthio, C1-C4-alkylsulfinyl, C1-C4-alkylsulfonyl; R2=H, halogen; R3=H, NO2, OH, halogen, C1-C4-alkoxy; R4=H, NO2, OH, halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy; R5=H, NO2, CN, halogen, C1-C8-alkyl, C3-C8-alkenyl, C3-C8-alkynyl, C3-C8-cycloalkyl, C1-C8-haloalkyl, C2-C8-haloalkenyl, C2-C8-haloalkinyl, C1-C4-alkoxy-C1-C4-alkyl, C2-C4-alkenyloxy-C1-C4-alkyl, C2-C4-alkynyloxy-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfonyl-C1-C4-alkyl, cyano-C1-C8-alkyl, cyano-C2-C8-alkenyl, cyano-C3-C8-alkynyl, unsubstituted or substituted OH, SH, SO—H, —SO2—H, COOH or NH—COOH, —SO2Cl, —N(R9,R10), —NH—SO2—(C1-C8-alkyl), —N[—SO2—(C1-C8-alkyl)]2, —N(C1-C8-alkyl)[—SO2—(C1-C8-alkyl)], —SO2—N(R9,R10), —O—CO—NH—R9, unsubstituted or substituted CHO, —O—CHO or —NH—CHO, —NH—CO—NH—R9, —O—CS—NH2, —O—CS—N(C1-C8-alkyl)2, —CO—N(R9,R10), —CS—N(R9,R10), —CO—NH—SO2—(C1-C4-alkyl).
摘要翻译: 取代的2-苯并(o)吡啶I和其中n = 0,1; X = CO,CH 2,CH(C 1 -C 4 - 烷基),CH-OH,CH-CN,CH-卤素,C(卤素) CH-CONH 2,CH-CO-O(C 1 -C 4 - 烷基),CH-O(C 1 -C 4 - 烷基),C(CN)(C 1 -C 4 - 烷基); R 1 =卤素,C 1 -C 4卤代烷基, C 1 -C 4烷硫基,C 1 -C 4烷基亚磺酰基,C 1 -C 4烷基磺酰基; R 2 = H,卤素; R 3 = H,NO 2,OH,卤素,C 1 -C 4 - 烷氧基; R 4 = H,NO 2,OH,卤素, C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基; R 5 = H,NO 2,CN,卤素,C 1 -C 8烷基,C 3 -C 8 - 烯基,C 3 -C 8炔基,C 3 -C 8 - 环烷基,C 1 -C 8 - 卤代烷基,C 2 -C 8 - 卤代烯基,C 2 -C 8 - 卤代炔基,C 1 -C 4 - 烷氧基-C 1 -C 4烷基,C 2 -C 4 - 烯氧基-C 1 -C 4烷基,C 2 -C 4 - C 1 -C 4烷基,C 1 -C 4烷硫基-C 1 -C 4烷基,C 1 -C 4烷基亚磺酰基-C 1 -C 4烷基,C 1 -C 4烷基磺酰基-C 1 -C 4 - 烷基,氰基-C 1 -C 8烷基, 氰基-C 2 -C 8 - 烯基,氰基-C 3 -C 8 - 炔基,未取代或取代的OH,SH,SO-H,-SO 2 -H,COOH或NH-COOH,-SO 2 Cl,-N(R 9,R 10) NH-SO 2 - (C 1 -C 8 - 烷基),-N [-SO 2 - (C 1 -C 8 - 烷基)] 2,-N(C 1 -C 8 - 烷基) -SO 2 -N(R 9,R 10),-O-CO-NH-R 9,未取代的 取代的CHO,-O-CHO或-NH-CHO,-NH-CO-NH-R9,-O-CS-NH2,-O-CS-N(C1-
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