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    NOVEL MICROBICIDES
    1.
    发明申请
    NOVEL MICROBICIDES 审中-公开
    新型微生物

    公开(公告)号：US20130281467A1

    公开(公告)日：2013-10-24

    申请号：US13881648

    申请日：2011-10-28

    申请人： Stephan Trah ,  Laura Quaranta ,  Clemens Lamberth ,  Martin Pouliot

    发明人： Stephan Trah ,  Laura Quaranta ,  Clemens Lamberth ,  Martin Pouliot

    IPC分类号： A01N43/54 ,  A01N43/90

    CPC分类号： A01N43/54 ,  A01N43/90 ,  C07D401/04 ,  C07D491/04 ,  C07D491/10

    摘要： Compounds of formula (I), wherein G represents together with the two carbon atoms of the pyrimidine ring to which it is attached, a 5- to 7-membered aliphatic carbocyclic or heterocyclic ring system which contain 0 to 2 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur; and wherein said 5- to 7-membered aliphatic carbocyclic or heterocyclic ring system can be mono-, di- or trisubstituted by substituents selected from the group consisting of halogen, keto, C1-C6alkyl, C1-C6alkoxy, C1-C6alkyloximino and C1-C6alkylendioxy; and wherein the other substituents R1, R2, R3, R4, R5 and R6 are as defined in claim 1, and their use as microbicides.

    摘要翻译： 式（I）化合物，其中G代表与其连接的嘧啶环的两个碳原子一起，含有0至2个选自以下的杂原子的5-至7-元脂族碳环或杂环系： 的氮，氧和硫; 并且其中所述5-至7-元脂族碳环或杂环系统可以被选自卤素，酮，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6烷氧基肟基和C 1 -C 6烷氧基的取代基单，二或三取代， C6烷基二氧基; 并且其中其它取代基R 1，R 2，R 3，R 4，R 5和R 6如权利要求1中所定义，及其作为杀微生物剂的用途。

    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER
    5.
    发明申请
    PYRIDAZINE DERIVATIVES USEFUL AS FUNGICIDES AND FOR THE TREATMENT OF CANCER 审中-公开
    用作杀真菌剂和治疗癌症的吡咯烷酮衍生物

    公开(公告)号：US20100273804A1

    公开(公告)日：2010-10-28

    申请号：US12809604

    申请日：2008-12-19

    申请人： Clemens Lamberth ,  Stephan Trah ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    发明人： Clemens Lamberth ,  Stephan Trah ,  Raphael Dumeunier ,  Sebastian Volker Wendeborn

    IPC分类号： A61K31/501 ,  A01N43/58 ,  C07D403/04 ,  C07D237/08 ,  A01P3/00 ,  A61K31/50 ,  A61P35/00

    CPC分类号： C07D237/12 ,  A01N43/58 ,  C07D237/14

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: formula (I) wherein R1 is C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is hydrogen or an optionally substituted alkyl, aryl or heteroaryl; R3 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; R4 is hydrogen, C1-C6alkyl or C1-C6haloalkyl; or R3 and R4 together can be part of a carbocyclic or heterocyclic 3- to 8-membered ring; R5 is optionally substituted aryl or heteroaryl; and R6 is hydroxy, halogen, C1-C6alkoxy, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的作为活性成分的式（I）的新哒嗪衍生物：式（I）其中R 1是C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; R 2是氢或任选取代的烷基，芳基或杂芳基; R3是氢，C1-C6烷基或C1-C6卤代烷基; R4是氢，C1-C6烷基或C1-C6卤代烷基; 或者R 3和R 4一起可以是碳环或杂环的3至8元环的一部分; R5是任选取代的芳基或杂芳基; R 6为羟基，卤素，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; 或其农业化学上可用的盐形式。

    PYRIDAZINE DERIVATIVES
    7.
    发明申请
    PYRIDAZINE DERIVATIVES 审中-公开
    吡啶衍生物

    公开(公告)号：US20100144674A1

    公开(公告)日：2010-06-10

    申请号：US12447028

    申请日：2007-10-23

    申请人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Wendeborn

    IPC分类号： A01N57/00 ,  C07D237/02 ,  A01N43/58 ,  A01N43/54 ,  A01N43/84 ,  A01P3/00 ,  A01P15/00

    CPC分类号： C07D237/14 ,  A01N43/58 ,  C07D237/08 ,  C07D237/12 ,  C07D307/60 ,  C07D307/79 ,  C07D401/04 ,  C07D401/12 ,  C07D403/04 ,  C07D405/04 ,  C07D405/12 ,  C07D407/04 ,  C07D409/04 ,  C07D409/12 ,  C07D413/04 ,  C07D417/04

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C8haloalkyl or C3-C6cycloalkyl; R2 is cycloalkyl, cycloalkylalkyl, halocycloalkyl, cycloalkoxy, halocycloalkoxy, cycloalkylalkoxy, halocycloalkylalkoxy, alkoxyalkyl, cycloalkoxyalkoxyalkyl, haloalkoxyalkyl, trialkylsilyl, alkylthioalkyl, haloalkylthioalkyl, cycloalkylthio, halocycloalkylthio, cycloalkylalkylthio, halocycloalkylalkylthio, alkylsulfinylalkyl, alkylsulfonylalkyl, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, C2-C6alkenyl, C2-C6alkynyl, optionally substituted arylsulfonyl, optionally substituted aryloxy, optionally optionally substituted heteroaryloxy, optionally substituted arylthio, optionally substituted heteroarylthio; or R2 together with an adjacent carbon atom forms an optionally substituted fused ring; R3 is an optionally substituted aryl; R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C8alkoxy, C1-C6haloalkoxy, hydroxy or cyano; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C8卤代烷基或C3-C6环烷基; R 2是环烷基，环烷基烷基，卤代环烷基，环烷氧基，卤代环烷氧基，环烷基烷氧基，卤代环烷基烷氧基，烷氧基烷基，环烷氧基烷氧基烷基，卤代烷氧基烷基，三烷基甲硅烷基，烷硫基烷基，卤代烷硫基烷基，环烷硫基，卤代环烷硫基，环烷基烷硫基，卤代环烷基烷硫基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷基亚磺酰基，卤代烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基， C 6链烯基，C 2 -C 6炔基，任选取代的芳基磺酰基，任选取代的芳氧基，任选任选取代的杂芳氧基，任选取代的芳硫基，任选取代的杂芳硫基; 或R 2与相邻的碳原子一起形成任选取代的稠环; R3是任选取代的芳基; R4是氢，卤素，C1-C6烷基，C1-C6卤代烷基，C1-C8烷氧基，C1-C6卤代烷氧基，羟基或氰基; n为1〜4的整数; 或其农业化学上可用的盐形式。

    PYRIDAZINE FUNGICIDES
    8.
    发明申请
    PYRIDAZINE FUNGICIDES 失效
    吡咯烷类杀真菌剂

    公开(公告)号：US20110112108A1

    公开(公告)日：2011-05-12

    申请号：US12863377

    申请日：2009-01-14

    申请人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wenderborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Raphael Dumeunier ,  Sebastian Volker Wenderborn

    IPC分类号： A61K31/501 ,  C07D401/04 ,  A01N43/48 ,  A61P35/00 ,  A01P3/00

    CPC分类号： C07D401/04

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is methyl, ethyl or isopropyl; R2 is chloro, fluoro, hydroxy or C1-C2alkoxy; R3 is H, chloro, fluoro, methoxy or C1-C3alkyl; R4 is chloro, fluoro or bromo; and R3 is H, fluoro or methoxy; or an agrochemically usable salt form thereof; with the proviso that when R1 is methyl, R2 is chloro and R3 is H, then R4 or R5 is different from fluoro.

    摘要翻译： 本发明涉及式（I）的新的哒嗪衍生物作为具有杀微生物活性的活性成分，特别是杀真菌活性：其中R1是甲基，乙基或异丙基; R2是氯，氟，羟基或C1-C2烷氧基; R3是H，氯，氟，甲氧基或C1-C3烷基; R4是氯，氟或溴; 且R 3为H，氟或甲氧基; 或其农业化学可用的盐形式; 条件是当R 1为甲基时，R 2为氯且R 3为H，则R 4或R 5不同于氟。

    NOVEL PYRIDAZINE DERIVATIVES
    9.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号：US20100029668A1

    公开(公告)日：2010-02-04

    申请号：US12374052

    申请日：2007-07-16

    申请人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    发明人： Stephan Trah ,  Clemens Lamberth ,  Sebastian Volker Wendeborn

    IPC分类号： A01N43/58 ,  C07D405/04 ,  A01P3/00

    CPC分类号： C07D401/14 ,  A01N43/58 ,  C07D403/14 ,  C07D405/14 ,  C07D407/14 ,  C07D409/14 ,  C07D417/14

    摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted heteroaryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.

    摘要翻译： 本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的杂芳基; R4是氢，卤素，C1-C6烷基，C1-C6卤代烷基，C1-C6烷氧基，C1-C6卤代烷氧基，羟基或氰基; 或其农业化学上可用的盐形式。