Isoxazoline derivatives and herbicides containing the same as the active ingredient
    2.
    发明授权
    Isoxazoline derivatives and herbicides containing the same as the active ingredient 有权
    含有与活性成分相同的异恶唑啉衍生物和除草剂

    公开(公告)号:US06841519B1

    公开(公告)日:2005-01-11

    申请号:US10049039

    申请日:2000-08-09

    摘要: The isoxazoline derivative of the present invention is represented by the following general formula [I]: [wherein Q is a group represented by —S(O)n—(CR5R6)m- (wherein n is an integer of 0 to 2, m is an integer of 1 to 3, and R5 and R6 are a hydrogen atom, a cyano group, an alkoxycarbonyl group, if an alkyl group or the like); R1 and R2 are a hydrogen atom, all optionally substituted alkyl group, an alkoxycarbonyl group, an optionally substituted phenyl group or the like; R3 and R4 are a hydrogen atom, an optionally substituted alkyl group, a cycloalkyl group or the like; Y is a hydrogen atom, an alkoxycarbonyl group, a carboxyl group, an alkenyl group, an optionally substituted alkyl group or an optionally substituted phenyl group]. The herbicide of the present invention contains the above isoxazoline derivative as the active ingredient.

    摘要翻译: 本发明的异恶唑啉衍生物由以下通式[I]表示:[其中Q为-S(O)n - (CR 5 R 6)m - (其中n为0〜2的整数,m 为1〜3的整数,R5,R6为氢原子,氰基,烷氧基羰基,烷基等)。 R1和R2是氢原子,全部任选取代的烷基,烷氧基羰基,任意取代的苯基等; R3和R4是氢原子,任选取代的烷基,环烷基等; Y是氢原子,烷氧基羰基,羧基,烯基,任意取代的烷基或任意取代的苯基]。 本发明的除草剂含有上述异恶唑啉衍生物作为有效成分。

    Di- or tri-fluoromethanesulfonyl anilide derivatives, process for the preparation of them and herbicides containing them as the active ingredient
    3.
    发明授权
    Di- or tri-fluoromethanesulfonyl anilide derivatives, process for the preparation of them and herbicides containing them as the active ingredient 有权
    二 - 或三氟甲磺酰苯胺衍生物,其制备方法和含有它们作为活性成分的除草剂

    公开(公告)号:US06458748B1

    公开(公告)日:2002-10-01

    申请号:US09744209

    申请日:2001-01-22

    IPC分类号: C07D23952

    摘要: The present invention provides a novel compound which is effective for the removal of a wide variety of weeds including difficult-to-control weeds emerging in paddy field and which is safe to mammals; a process for production thereof; a herbicide containing the compound as an active ingredient; and novel raw material compounds used in said process. The present invention relates to a di- or trifluoromethanesulfonyl anilide derivative represented by the following general formula: (wherein R1 is a hydrogen atom, an alkyl group or an alkoxyalkyl group; and R2 is a hydrogen atom when R1 is a hydrogen atom or an alkyl group, and is a hydrogen atom or a fluorine atom when R1 is an alkoxyalkyl group), or a salt thereof, both of said derivative and said salt having a herbicidal activity.

    摘要翻译: 本发明提供了一种新颖的化合物,其有效去除各种杂草,包括难以控制的稻田中出现的杂草,对哺乳动物是安全的; 其生产方法; 含有该化合物作为活性成分的除草剂; 和所述方法中使用的新型原料化合物。本发明涉及由以下通式表示的二 - 或三氟甲磺酰苯胺衍生物:其中R1是氢原子,烷基或烷氧基烷基; R2是氢 当R 1为氢原子或烷基时为原子,当R 1为烷氧基烷基时为氢原子或氟原子)或其盐,所述衍生物和所述盐都具有除草活性。

    Indazolesulfonylurea derivative, its use and intermediate for its
production
    5.
    发明授权
    Indazolesulfonylurea derivative, its use and intermediate for its production 失效
    靛唑磺酰脲衍生物,其用途及其生产中间体

    公开(公告)号:US5670452A

    公开(公告)日:1997-09-23

    申请号:US630092

    申请日:1996-04-09

    摘要: The present invention provides an indazolesulfonylurea derivative represented by the general formula: ##STR1## wherein R.sup.1 is a hydrogen atom or an alkyl group, etc., R.sup.2 and R.sup.3 are the same or different and represent a hydrogen atom, a halogen atom, an alkyl group, the formula --COR.sup.4 (wherein R.sup.4 represents an alkoxy group, etc.), an alkoxy group, a haloalkoxy group or a cyano group, etc., X is an oxygen atom or a sulfur atom, Y is a hydrogen atom or an alkyl group, etc., A and B are the same or different and represent a halogen atom, an alkoxy group or an alkyl group, etc., and Z represents a nitrogen atom or a methine group, as well as a herbicide containing it as an active ingredient and an intermediate for its production. The compound of the present invention exhibits excellent herbicidal effects over a wide range from the preemergence stage to the growing stage of various weeds which are problematic in agricultural fields. Further, it is capable of controlling weeds germinating in paddy fields.

    摘要翻译: 本发明提供由通式如下的吲唑磺酰脲衍生物:其中R1是氢原子或烷基等,R2和R3相同或不同,代表氢原子,卤素原子 ,烷基,式-COR 4(其中R 4表示烷氧基等),烷氧基,卤代烷氧基或氰基等,X为氧原子或硫原子,Y为氢 原子或烷基等,A和B相同或不同,表示卤素原子,烷氧基或烷基等,Z表示氮原子或次甲基,除草剂 将其作为活性成分和其生产中间体。 本发明的化合物在农业领域有问题的各种杂草的出苗前期到生长期的广泛范围内表现出优异的除草效果。 此外,它能够控制稻田中发芽的杂草。

    Picolinic acid derivative, and herbicidal composition
    7.
    发明授权
    Picolinic acid derivative, and herbicidal composition 失效
    吡啶甲酸衍生物和除草组合物

    公开(公告)号:US5391537A

    公开(公告)日:1995-02-21

    申请号:US960844

    申请日:1992-10-14

    摘要: The present invention is to provide a novel picolinic acid derivative having the formula, ##STR1## (wherein R is a hydrogen atom, an alkyl group or others, R.sup.1 and R.sup.2 are the same or different, and are an alkyl group, an alkoxy group or others, X is a cyano group, a phenoxy group or others, Y is an oxygen atom or others, and n is 0 or 1) or a salt thereof; a method for preparing the same; and a herbicidal composition containing the same as an active ingredient.The picolinic acid derivative or the salt thereof of the present invention achieves an excellent herbicidal effect at a low dosage, and is effective for controlling the growth of various weeds in a wide range.The picolinic acid derivative or the salt thereof of the present invention can be applied to a paddy field, a cultivated field, a non-agricultural land and the like as a herbicidal composition.

    摘要翻译: 本发明提供具有下式的新颖的吡啶甲酸衍生物:其中R为氢原子,烷基或其它,R1和R2相同或不同,为烷基,烷氧基 或其它,X为氰基,苯氧基等,Y为氧原子等,n为0或1)或其盐; 其制备方法; 和含有该活性成分的除草组合物。 本发明的吡啶甲酸衍生物或其盐在低剂量下具有优异的除草效果,对于广泛控制各种杂草的生长是有效的。 本发明的吡啶甲酸衍生物或其盐可以作为除草组合物施用于稻田,栽培田,非农田等。

    Benzofuran-7-yl uracil derivatives and herbicides
    9.
    发明授权
    Benzofuran-7-yl uracil derivatives and herbicides 有权
    苯并呋喃-7-基尿嘧啶衍生物和除草剂

    公开(公告)号:US6130187A

    公开(公告)日:2000-10-10

    申请号:US117539

    申请日:1998-08-05

    摘要: A benzofuran-7-yl uracil derivative represented by the general formula (1): ##STR1## (wherein each of X and Y is a hydrogen atom, a halogen atom or the like, R.sup.1 is a hydrogen atom, an alkyl group or the like, R.sup.2 is a haloalkyl group or the like, R.sup.3 is a hydrogen atom, a halogen atom or the like, each of R.sup.4 and R.sup.5 which are independent of each other, is a hydrogen atom, an alkyl group, a haloalkyl group, a halogen atom, a cyano group, a phenyl group, a benzyl group, a nitro group or the like), and a herbicide containing it as an active ingredient.The compound of the present invention represented by the general formula (1) exhibits excellent herbicidal effects against various weeds which cause trouble in upland fields, such as, broad leaved weeds, gramineous weeds and perennial or annual cyperaceous weeds, over a wide range from the pre-emergence to the growing stage. It can further control annual weeds and perennial weeds growing in paddy fields.

    摘要翻译: PCT No.PCT / JP97 / 00320 Sec。 371日期:1998年8月5日 102(e)1998年8月5日PCT PCT 1997年2月7日PCT公布。 公开号WO97 / 29105 PCT 日期1997年8月14日由通式(1)表示的苯并呋喃-7-基尿嘧啶衍生物:其中X和Y各自为氢原子,卤素原子等,R 1为氢原子,烷基 R 2为卤代烷基等,R 3为氢原子,卤素原子等,R 4和R 5各自独立地为氢原子,烷基,卤代烷基 卤素原子,氰基,苯基,苄基,硝基等)和含有它的除草剂作为有效成分。 由通式(1)表示的本发明化合物对各种杂草具有优异的除草效果,其在高纬地区如阔叶杂草,禾本科杂草和多年生或一年生的季节性杂草中引起麻烦,范围广泛 出生前到成长阶段。 可以进一步控制在稻田中种植的一年生杂草和多年生杂草。

    Indazolesulfonylurea derivative, its use and intermediate for its
production
    10.
    发明授权
    Indazolesulfonylurea derivative, its use and intermediate for its production 失效
    靛唑磺酰脲衍生物,其用途及其生产中间体

    公开(公告)号:US5763616A

    公开(公告)日:1998-06-09

    申请号:US779437

    申请日:1997-01-07

    摘要: The present invention provides an indazolesulfonylurea derivative represented by the general formula: ##STR1## �wherein R.sup.1 is a hydrogen atom or an alkyl group, etc., R.sup.2 and R.sup.3 are the same or different and represent a hydrogen atom, a halogen atom, an alkyl group, the formula --COR.sup.4 (wherein R.sup.4 represents an alkoxy group, etc.), an alkoxy group, a haloalkoxy group or a cyano group, etc., X is an oxygen atom or a sulfur atom, Y is a hydrogen atom or an alkyl group, etc., A and B are the same or different and represent a halogen atom, an alkoxy group or an alkyl group, etc., and Z represents a nitrogen atom or a methine group!, as well as a herbicide containing it as an active ingredient and an intermediate for its production. The compound of the present invention exhibits excellent herbicidal effects over a wide range from the preemergence stage to the growing stage of various weeds which are problematic in agricultural fields. Further, it is capable of controlling weeds germinating in paddy fields.

    摘要翻译: 本发明提供由以下通式表示的吲唑磺酰脲衍生物:其中R1是氢原子或烷基等,R2和R3相同或不同,代表氢原子,卤素 原子,烷基,式-COR 4(其中R 4表示烷氧基等),烷氧基,卤代烷氧基或氰基等,X为氧原子或硫原子,Y为 氢原子或烷基等,A和B相同或不同,表示卤素原子,烷氧基或烷基等,Z表示氮原子或次甲基],以及 含有它作为活性成分的除草剂和用于其生产的中间体。 本发明的化合物在农业领域有问题的各种杂草的出苗前期到生长期的广泛范围内表现出优异的除草效果。 此外,它能够控制稻田中发芽的杂草。