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公开(公告)号：US20230373947A1
公开(公告)日：2023-11-23
申请号：US18229277
申请日：2023-08-02
Applicant: MITSUI CHEMICALS, INC.
Inventor： Kei Yoshida , Takeo Wakita , Hiroyuki Katsuta , Akiyoshi Kai , Yutaka Chiba , Kiyoshi Takahashi , Hiroko Kato , Nobuyuki Kawahara , Michikazu Nomura , Hidenori Daido , Junji Maki , Shinichi Banba
IPC: C07D333/38 , A01N37/44 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/16 , A01N43/30 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/78 , A01N43/80 , C07C237/42 , C07C317/40 , C07C323/42 , C07C327/48 , C07D207/416 , C07D213/64 , C07D213/73 , C07D213/81 , C07D213/82 , C07D213/89 , C07D215/52 , C07D231/14 , C07D231/16 , C07D239/30 , C07D241/24 , C07D263/34 , C07D275/03 , C07D277/56 , C07D307/24 , C07D307/68 , C07D307/84 , C07D309/08 , C07D309/28 , C07D317/62 , C07D333/68 , A01N43/40 , A01N37/22 , A01N43/60 , C07C237/48 , C07D207/34 , C07D239/28 , C07D261/18 , C07D307/85 , C07D317/46
CPC classification number: C07D333/38 , A01N37/44 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/16 , A01N43/30 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/78 , A01N43/80 , C07C237/42 , C07C317/40 , C07C323/42 , C07C327/48 , C07D207/416 , C07D213/64 , C07D213/73 , C07D213/81 , C07D213/82 , C07D213/89 , C07D215/52 , C07D231/14 , C07D231/16 , C07D239/30 , C07D241/24 , C07D263/34 , C07D275/03 , C07D277/56 , C07D307/24 , C07D307/68 , C07D307/84 , C07D309/08 , C07D309/28 , C07D317/62 , C07D333/68 , A01N43/40 , A01N37/22 , A01N43/60 , C07C237/48 , C07D207/34 , C07D239/28 , C07D261/18 , C07D307/85 , C07D317/46
Abstract: A compound represented by Formula (1):
The compound can be used as insecticides.-
2.发明授权公开(公告)号：US10005750B2
公开(公告)日：2018-06-26
申请号：US13823522
申请日：2011-10-06
Applicant: Michael F. Wempe , Hitoshi Endou
Inventor： Michael F. Wempe , Hitoshi Endou
IPC: C07D307/84 , C07D209/12 , C07D307/79 , C07D307/80
CPC classification number: C07D307/84 , C07D209/12 , C07D307/79 , C07D307/80
Abstract: A compound represented by the general Formula I: a pharmaceutically acceptable salt or ester thereof, a solvate thereof, a chelate thereof, a non-covalent complex thereof, a pro-drug thereof, a deuterated radio-labeled analog thereof, and mixtures of any of the foregoing, wherein: A-K are individually selected from carbon or nitrogen; X═—O, —NR1, or —S; R1-11 are individually selected from the group consisting of —H, C1-C6 alkyl, C6-C14 aryl, substituted C6-C14 aryl, C1-C14-alkoxy, halogen, hydroxyl, carboxy, cyano, C1-C6-alkanoyloxy, C1-C6-alkylthio, C1-C6-alkylsulfonyl, trifluoromethyl, hydroxy, C2-C6-alkoxycarbonyl, C2-C6-alkanoylamino, —O—R12, S—R12, —SO2—R12, —NHSO2R12 and —NHCO2R12, wherein R12 is phenyl, naphthyl, or phenyl or naphthly substituted with one to three groups selected from C1-C6-alkyl, C6-C10 aryl, C1-C6-alkoxy and halogen, and C4-C20 hydroxyheteroaryl wherein the heteroatoms are selected from the group consisting of sulfur, nitrogen, and oxygen.
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公开(公告)号：US20180009739A1
公开(公告)日：2018-01-11
申请号：US15547014
申请日：2016-01-28
Applicant: Jin-Quan YU , The Scripps Research Institute
Inventor： Jin-Quan Yu
IPC: C07C233/15 , C07D209/48 , C07B43/06 , C07C233/59 , C07C231/12 , C07D307/77 , C07D209/04
CPC classification number: C07C233/15 , C07B43/06 , C07C231/12 , C07C233/59 , C07C2602/10 , C07D209/04 , C07D209/42 , C07D209/48 , C07D307/77 , C07D307/84
Abstract: An alternative approach to formation of a C-C bond at a meta-position of an aromatic compound is disclosed that employs an ethylenically unsaturated bicyclic compound as a transient mediator to achieve meta-selective C-H activation with a simple and common ortho-directing group. The use of a pyridine-based ligand assists in relaying the palladium catalyst to the meta-position by the unsaturated bicyclic compound following initial ortho-C-H activation.
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4.发明申请公开(公告)号：US20180003702A1
公开(公告)日：2018-01-04
申请号：US15244135
申请日：2016-08-23
Applicant: SENOMYX, INC.
Inventor： Xiaodong LI , Lena LUUKKONEN , Hong XU
IPC: G01N33/543 , A23L27/00 , A23L27/20 , G01N33/566 , G01N33/50 , C07F9/655 , C07D405/12 , C07D317/68 , C07D307/84 , C07C275/34 , C07C275/30 , C07C235/54 , C07C233/65 , A61K47/24 , A61K47/22 , A61K8/55 , A61K8/49 , A23L2/56 , G01N33/74
CPC classification number: G01N33/543 , A23L2/56 , A23L27/202 , A23L27/203 , A23L27/2054 , A23L27/88 , A23V2002/00 , A61K8/4973 , A61K8/55 , A61K47/22 , A61K47/24 , C07C233/65 , C07C235/54 , C07C275/30 , C07C275/34 , C07D209/08 , C07D209/42 , C07D213/40 , C07D213/81 , C07D213/85 , C07D215/48 , C07D217/06 , C07D231/14 , C07D261/18 , C07D263/56 , C07D271/12 , C07D275/03 , C07D277/64 , C07D285/135 , C07D307/52 , C07D307/68 , C07D307/79 , C07D307/82 , C07D307/84 , C07D317/68 , C07D333/24 , C07D333/38 , C07D401/04 , C07D405/12 , C07D409/12 , C07D417/12 , C07F9/65517 , G01N33/5041 , G01N33/566 , G01N33/74 , G01N2333/726
Abstract: The invention relates to compounds that specifically bind a T1R1/T1R3 or T1R2/T1R3 receptor or fragments or sub-units thereof. The present invention also relates to the use of hetero-oligomeric and chimeric taste receptors comprising T1R1/T1R3 and T1R2/T1R3 in assays to identify compounds that respectively respond to umami taste stimuli and sweet taste stimuli. Further, the invention relates to the constitutive of cell lines that stably or transiently co-express a combination of T1R1 and T1R3; or T1R2 and T1R3; under constitutive or inducible conditions. The use of these cells lines in cell-based assays to identify umami and sweet taste modulatory compounds is also provided, particularly high throughput screening assays that detect receptor activity by use of fluorometric imaging.
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5.发明申请公开(公告)号：US20170101416A1
公开(公告)日：2017-04-13
申请号：US15312022
申请日：2015-05-19
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor： Tao WANG , Zhongxing Zhang , John F. Kadow
IPC: C07D491/048 , C07D405/10
CPC classification number: C07D491/048 , C07D307/84 , C07D405/10
Abstract: Compounds of Formula I, including their salts, as well as compositions and methods of using the compounds are set forth. The compounds have activity against hepatitis C virus (HCV) and may be useful in treating those infected with HCV: formula (I).
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Patent Agency Ranking
6.发明申请公开(公告)号：US20160038926A1
公开(公告)日：2016-02-11
申请号：US14654061
申请日：2013-12-20
Applicant: CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) , UNIVERSITÉ PAUL SABATIER TOULOUSE 3
Inventor： Montserrat GOMEZ , Emmanuelle TEUMA , Isabelle FAVIER , Faouzi CHAHDOURA
IPC: B01J35/00 , B01J31/06 , B01J31/28 , B01J23/44 , B01J23/46 , B01J23/72 , C07C41/20 , C07C45/62 , C07C67/303 , C07D209/08 , C07D211/62 , C07C209/60 , C07D295/135 , C07D295/096 , C07C319/18 , C07D307/79 , C07D307/89 , C07D401/06 , C07C45/64 , C07D249/04 , C07D403/14 , C07D307/84 , C07D493/04 , C07D405/06 , C07D493/14 , C07D493/18 , C07D211/94 , C07D401/04 , C07C5/03 , B01J31/02
CPC classification number: B01J35/0013 , B01J23/44 , B01J23/464 , B01J23/72 , B01J31/0202 , B01J31/0267 , B01J31/0271 , B01J31/06 , B01J31/24 , B01J31/2404 , B01J31/28 , B01J35/023 , B01J2231/34 , B01J2231/4211 , B01J2231/4216 , B01J2231/4227 , B01J2231/4261 , B01J2231/4266 , B01J2231/4283 , B01J2231/4294 , B01J2231/641 , B01J2231/645 , B01J2531/16 , B01J2531/822 , B01J2531/824 , B01J2531/90 , B01J2540/32 , B22F1/0022 , B22F1/0062 , B22F9/26 , B82Y30/00 , B82Y40/00 , C07B37/04 , C07C5/03 , C07C41/20 , C07C45/62 , C07C45/64 , C07C67/303 , C07C209/60 , C07C319/18 , C07C2531/02 , C07C2531/28 , C07C2601/14 , C07D209/08 , C07D211/62 , C07D211/94 , C07D249/04 , C07D295/096 , C07D295/135 , C07D307/79 , C07D307/84 , C07D307/89 , C07D401/04 , C07D401/06 , C07D403/14 , C07D405/06 , C07D493/04 , C07D493/14 , C07D493/18
Abstract: A catalytic system which is a suspension in glycerol of metal nanoparticles in at least one transition metal. The suspension also includes at least one compound stabilizing the metal nanoparticles, soluble in glycerol. The suspensions are obtained directly in glycerol. These are stable systems that can catalyse a reaction from an organic substrate, with high yields and activity, and excellent selectivity. Additionally, the use of the catalytic system for performing organic transformations such as hydrogenation or coupling reactions (formation of C—C, C—N, C—O, C—S . . . bonds), and for synthesizing polyfunctionnal molecules, in a single reactor, by multi-step, sequential or cascade reactions.
Abstract translation: 催化体系，其是在至少一种过渡金属中的金属纳米颗粒的甘油中的悬浮液。 悬浮液还包括至少一种稳定金属纳米颗粒的化合物，其可溶于甘油。 悬浮液直接在甘油中获得。 这些是可以以高产率和活性以及优异选择性催化有机底物的反应的稳定体系。 另外，使用用于进行有机转化如氢化或偶联反应（形成C-C，C-N，C-O，C-S键）的催化体系，并用于合成多官能分子 单反应器，通过多步，顺序或级联反应。
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公开(公告)号：US20150141395A1
公开(公告)日：2015-05-21
申请号：US14387883
申请日：2013-03-26
Applicant: Bristol-Myers Squibb Company
Inventor： Kap-Sun Yeung
IPC: C07D405/14
CPC classification number: C07D405/14 , A61K31/506 , A61K45/06 , C07D307/84
Abstract: The disclosure provides compounds of formula I, including their salts, as well as compositions and methods of using the compounds. The compounds have activity against hepatitis C virus (HCV) and may be useful in treating those infected with HCV.
Abstract translation: 本公开提供式I化合物，包括其盐，以及使用该化合物的组合物和方法。 该化合物具有抗丙型肝炎病毒（HCV）的活性，可用于治疗HCV感染者。
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公开(公告)号：US20150080588A1
公开(公告)日：2015-03-19
申请号：US14339918
申请日：2014-07-24
Applicant: JANSSEN PHARMACEUTICA NV
Inventor： Shawn Branum , Michael Reuman , Ronald K. Russell , Christopher A. Teleha
IPC: C07D309/10 , C07D307/937
CPC classification number: C07D309/10 , C07D307/84 , C07D307/937 , C07D405/14 , C07D413/06 , C07D413/14 , C07D471/04 , C07D487/08
Abstract: The present invention comprises processes for preparing compounds of Formula (I). wherein: R0, R1, R2, R3, R4, R5, and A are as defined in the specification.
Abstract translation: 本发明包括制备式（I）化合物的方法。 其中：R 0，R 1，R 2，R 3，R 4，R 5和A如说明书中所定义。
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9.发明申请AMIDE DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND USE THEREOF AS INSECTICIDE 有权酰胺衍生物，其制备方法及其作为杀虫剂的用途公开(公告)号：US20140206727A1
公开(公告)日：2014-07-24
申请号：US14220673
申请日：2014-03-20
Applicant: MITSUI CHEMICALS, INC.
Inventor： Kei Yoshida , Takeo Wakita , Hiroyuki Katsuta , Akiyoshi Kai , Yutaka Chiba , Kiyoshi Takahashi , Hiroko Kato , Nobuyuki Kawahara , Michikazu Nomura , Hidenori Daido , Junji Maki , Shinichi Banba
IPC: A01N43/40
CPC classification number: C07D333/38 , A01N37/22 , A01N37/44 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/16 , A01N43/30 , A01N43/40 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , C07C237/42 , C07C237/48 , C07C317/40 , C07C323/42 , C07C327/48 , C07D207/34 , C07D207/416 , C07D213/64 , C07D213/73 , C07D213/81 , C07D213/82 , C07D213/89 , C07D215/52 , C07D231/14 , C07D231/16 , C07D239/28 , C07D239/30 , C07D241/24 , C07D261/18 , C07D263/34 , C07D275/03 , C07D277/56 , C07D307/24 , C07D307/68 , C07D307/84 , C07D307/85 , C07D309/08 , C07D309/28 , C07D317/46 , C07D317/62 , C07D333/68
Abstract: A compound represented by Formula (1): The compound can be used as insecticides.
Abstract translation: 由式（1）表示的化合物：该化合物可以用作杀虫剂。
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公开(公告)号：US08722688B2
公开(公告)日：2014-05-13
申请号：US13798286
申请日：2013-03-13
Applicant: Bristol-Myers Squibb Company
Inventor： Kap-Sun Yeung , Kyle E. Parcella , John A. Bender , Brett R. Beno , Katharine A. Grant-Young , Ying Han , Piyasena Hewawasam , John F. Kadow , Andrew Nickel
IPC: A61K31/506
CPC classification number: A61K31/506 , A61K45/06 , C07D307/84 , C07D405/04 , C07D405/10 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/10 , C07D413/12 , C07D417/10 , C07D417/12 , C07D453/00 , C07D491/10
Abstract: The disclosure provides compounds of formula I, including their salts, as well as compositions and methods of using the compounds. The compounds have activity against hepatitis C virus (HCV) and may be useful in treating those infected with HCV.
Abstract translation: 本公开提供式I化合物，包括其盐，以及使用该化合物的组合物和方法。 该化合物具有抗丙型肝炎病毒（HCV）的活性，可用于治疗HCV感染者。
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