Piperdine Compound and Process for Preparing the Same
    1.
    发明申请
    Piperdine Compound and Process for Preparing the Same 审中-公开
    哌啶化合物及其制备方法

    公开(公告)号:US20070244158A1

    公开(公告)日:2007-10-18

    申请号:US11660046

    申请日:2005-09-16

    摘要: The present invention is to provide a piperidine compound represented by the formula [I]: wherein Ring A is an optionally substituted benzene ring, Ring B is an optionally substituted benzene ring, R1 is hydrogen atom or a substituent for amino group, R2 is hydrogen atom, an optionally substituted hydroxyl group, an optionally substituted amino group, an optionally substituted alkyl group, a substituted carbonyl group or a halogen atom, Z is oxygen atom or —N(R3)—, R3 is hydrogen atom or an optionally substituted alkyl group, R4a and R4b may be the same or different, and each is hydrogen atom or an optionally substituted alkyl group, or may be bonded to each other at the both ends to form an alkylene group, or a pharmaceutically acceptable salt thereof, which has an excellent tachykinin receptor antagonistic action.

    摘要翻译: 本发明提供由式[I]表示的哌啶化合物:其中环A是任选取代的苯环,环B是任选取代的苯环,R 1是氢原子或 氨基的取代基R 2是氢原子,任选取代的羟基,任选取代的氨基,任选取代的烷基,取代的羰基或卤素原子,Z是氧原子或 -N(R 3) - ,R 3是氢原子或任选取代的烷基,R 4a和R 4b, / SUP>可以相同或不同,并且各自为氢原子或任选取代的烷基,或者可以在两端彼此键合形成亚烷基或其药学上可接受的盐,其具有优异的 速激肽受体拮抗作用。

    Piperidine compound and process for preparing the same
    2.
    发明授权
    Piperidine compound and process for preparing the same 失效
    哌啶化合物及其制备方法

    公开(公告)号:US07390905B2

    公开(公告)日:2008-06-24

    申请号:US10581045

    申请日:2004-11-26

    IPC分类号: C07D211/30 C07D211/32

    摘要: The present invention relates to a piperidine compound represented by the formula [I]: wherein Ring A represents an optionally substituted benzene ring, Ring B represents an optionally substituted benzene ring, R1 represents an optionally substituted hydoxyl group, a substituted thiol group, a substituted sulfonyl group, etc., or a group represented by the formula: R11 represents a substituted carbonyl group or a substituted sulfonyl group, R12 represents hydrogen atom or an optionally substituted alkyl group, R2 represents hydrogen atom, etc., Z represent oxygen atom or a group represented by —N(R3)—, R3 represents an optionally substituted alkyl group, etc., R4a represents an optionally substituted alkyl group, R4b represents an optionally substituted alkyl group, or a pharmaceutically acceptable salt thereof, having an excellent tachykinin receptor antagonistic action.

    摘要翻译: 本发明涉及由式[I]表示的哌啶化合物:其中环A表示任选取代的苯环,环B表示任选取代的苯环,R 1表示任选取代的羟基 取代的硫醇基,取代的磺酰基等,或由下式表示的基团:R 11表示取代的羰基或取代的磺酰基,R 12 >表示氢原子或任选取代的烷基,R 2表示氢原子等,Z表示氧原子或由-N(R 3 O 3) - 表示的基团, R 3表示任选取代的烷基等,R 4a表示任选取代的烷基,R 4b表示任选取代的烷基 基团或其药学上可接受的盐,具有优异的速激肽受体拮抗作用。

    Piperidine compound and process for preparing the same
    3.
    发明申请
    Piperidine compound and process for preparing the same 失效
    哌啶化合物及其制备方法

    公开(公告)号:US20070112029A1

    公开(公告)日:2007-05-17

    申请号:US10581045

    申请日:2004-11-26

    IPC分类号: A61K31/445 C07D211/56

    摘要: Disclosed are a novel piperidine compound represented by the general formula [I] below which has an excellent tachykinin receptor antagonizing activity and pharmacologically acceptable salts thereof. [I] In the formula, ring A represents an optionally substituted benzene ring; ring B represents an optionally substituted benzene ring; R1 represents an optionally substituted hydroxyl group, a thiol group having a substituent, a sulfonyl group having a substituent, or a group represented by the following formula [II]: wherein R11 represents a carbonyl group having a substituent or a sulfonyl group having a substituent and R12 represents a hydrogen atom or an optionally substituted alkyl group; R2 represents a hydrogen atom or the like; Z represents an oxygen atom or a group represented by —N(R3)— wherein R3 represents an optionally substituted alkyl group or the like; R4a represents an optionally substituted alkyl group; and R4b represents an optionally substituted alkyl group.

    摘要翻译: 公开了由下述通式[I]表示的新型哌啶化合物,其具有优异的速激肽受体拮抗活性及其药理学上可接受的盐。 式中,环A表示任选取代的苯环; 环B表示任选取代的苯环; R 1表示任选取代的羟基,具有取代基的硫醇基,具有取代基的磺酰基或由下式[II]表示的基团:其中R 11, SUP>表示具有取代基的羰基或具有取代基的磺酰基,R 12表示氢原子或任选取代的烷基; R 2表示氢原子等; Z表示氧原子或由-N(R 3 O 3)表示的基团,其中R 3表示任选取代的烷基等; R 4a表示任选取代的烷基; R 4b表示任选取代的烷基。

    THIOMORPHOLINE COMPOUND AND PROCESS FOR PREPARING THE SAME
    5.
    发明申请
    THIOMORPHOLINE COMPOUND AND PROCESS FOR PREPARING THE SAME 审中-公开
    吡咯啉化合物及其制备方法

    公开(公告)号:US20090281095A1

    公开(公告)日:2009-11-12

    申请号:US12065537

    申请日:2006-09-01

    IPC分类号: A61K31/541 C07D417/04

    CPC分类号: C07D211/58

    摘要: The present invention discloses a thiomorpholine compound represented by the formula [I]: wherein Ring A represents an optionally substituted benzene ring; Ring B represents an optionally substituted benzene ring; R1 represents hydrogen atom, an optionally substituted hydroxyl group, an optionally substituted amino group, an optionally substituted alkyl group, a substituted carbonyl group or a halogen atom; R2 represents hydrogen atom or an optionally substituted alkyl group; and R3a and R3b may be the same or different from each other, and each represent hydrogen atom or an optionally substituted alkyl group, or combined to each other at the both ends thereof to form an alkylene group, and n is an integer of 1 or 2, or a pharmaceutically acceptable salt thereof.

    摘要翻译: 本发明公开了式[I]表示的硫代吗啉化合物:其中环A表示任选取代的苯环; 环B表示任选取代的苯环; R1表示氢原子,任选取代的羟基,任选取代的氨基,任选取代的烷基,取代的羰基或卤素原子; R2表示氢原子或任选取代的烷基; 并且R 3a和R 3b可以相同或不同,并且各自表示氢原子或任选取代的烷基,或者在其两端彼此结合形成亚烷基,n为1的整数或 2,或其药学上可接受的盐。

    PROTECTIVE FILM FOR AUTOMOTIVE WHEEL
    6.
    发明申请
    PROTECTIVE FILM FOR AUTOMOTIVE WHEEL 审中-公开
    汽车保护膜

    公开(公告)号:US20120040178A1

    公开(公告)日:2012-02-16

    申请号:US13266710

    申请日:2010-04-22

    摘要: Provided is a protective film for an automotive wheel having excellent performances, which can sufficiently prevent scratching of the wheel surface and staining, and also the generation of rust at a disc brake inside the wheel during a period until delivery of an automobile; and can be easily peeled. The protective film for an automotive wheel of the present invention is a protective film for an automotive wheel, including a base layer and a pressure-sensitive adhesive layer, wherein the pressure-sensitive adhesive layer of the protective film is bonded onto the back surface of the base layer of the protective film, and an adhesive force to the back surface after storage at 50° C. for 24 hours in an state of being bonded is from 0.1 to 2 N/20 mm at any peeling speed of 0.3 m/minute, 10 m/minute and 30 m/minute.

    摘要翻译: 本发明提供一种具有优异性能的汽车轮保护膜,其能够充分防止车轮表面的划伤和污染,并且在汽车的交付期间内的车轮内的盘式制动器的生锈; 并且可以容易地剥离。 本发明的汽车用轮用保护膜是用于汽车轮的保护膜,包括基层和压敏粘合剂层,其中保护膜的粘合剂层粘合到 保护膜的基层和在接合状态下在50℃下保存24小时后的背面的粘合力为0.1〜2N / 20mm,剥离速度为0.3m /分钟 ,10米/分钟和30米/分钟。

    Film for protecting mother glass for flat panel display and use thereof
    7.
    发明申请
    Film for protecting mother glass for flat panel display and use thereof 审中-公开
    用于保护用于平板显示器的母玻璃的膜和其用途

    公开(公告)号:US20050253277A1

    公开(公告)日:2005-11-17

    申请号:US11109568

    申请日:2005-04-19

    摘要: An object of the present invention is to provide a surface protecting film which dramatically improves an efficiency of transporting and storing a mother glass, has better peelability from an adherend when peeled without polluting a mother glass surface, and gives reinforcing effect by adopting a pressure-sensitive adhesive protecting film, and use thereof. This invention relates to a film for protecting a mother glass for a flat panel display having a pressure-sensitive adhesive layer on one side of a film substrate, wherein a surface roughness Ra of the pressure-sensitive adhesive layer is 0.2 μm or smaller, and a surface roughness Rz is 1.0 μm or smaller, and wherein the pressure-sensitive adhesive layer comprises a crosslinked copolymer containing a (meth)acrylic acid ester monomer and a vinyl-based monomer having a functional group as a component, and a glass transition temperature of the copolymer obtained by a Fox's equation is −25 to −10° C.

    摘要翻译: 本发明的目的是提供一种显着提高母玻璃的输送和储存效率的表面保护膜,在不污染母玻璃表面的情况下剥离时与被粘物的剥离性更好,并且通过采用压敏粘合剂, 敏感性保护膜及其用途。 本发明涉及一种用于保护用于平板显示器的母玻璃的膜,该平板显示器在膜基底的一侧具有压敏粘合剂层,其中压敏粘合剂层的表面粗糙度Ra为0.2μm或更小,以及 表面粗糙度Rz为1.0μm以下,并且其中粘合剂层包含含有(甲基)丙烯酸酯单体和具有官能团的乙烯基类单体作为组分的交联共聚物,玻璃化转变温度 通过Fox's方程得到的共聚物为-25〜-10℃

    Transport apparatus with differential force system
    9.
    发明授权
    Transport apparatus with differential force system 失效
    带有差速系统的运输设备

    公开(公告)号:US4262859A

    公开(公告)日:1981-04-21

    申请号:US49564

    申请日:1979-06-18

    申请人: Takeshi Yamanaka

    发明人: Takeshi Yamanaka

    IPC分类号: G11B15/295 G03B1/04 G11B15/32

    CPC分类号: G11B15/295

    摘要: Tape apparatus in which a length of pliant material is fed between supply and take-up rolls in edge driven relationship with a capstan. A static force provided, for example, by friction or a spring is utilized to maintain the take-up roll against the capstan with a greater force than the supply roll, and in the event of a reversal of tape direction, this force is immediately and automatically applied to the new take-up roll and removed from the new supply roll.

    摘要翻译: 带状装置,其中一根柔顺材料的长度以与主导管的边缘驱动关系供给在供应辊和卷取辊之间。 使用例如通过摩擦或弹簧提供的静力用于以比供给辊更大的力将卷取辊保持在主导轴上,并且在带方向反转的情况下,该力是立即和 自动应用于新的卷取辊,并从新的供应卷中取出。