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116 条记录 (耗时 0.037 秒)

    Microbicidal and growth regulating compositions
    1.
    发明授权
    Microbicidal and growth regulating compositions 失效
    杀菌和生长调节组合物

    公开(公告)号：US4940481A

    公开(公告)日：1990-07-10

    申请号：US468522

    申请日：1983-02-22

    申请人： Urs Muller ,  Hans Tobler ,  Hermann Rempfler ,  Alfred Meyer

    发明人： Urs Muller ,  Hans Tobler ,  Hermann Rempfler ,  Alfred Meyer

    IPC分类号： A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

    CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

    摘要： The invention relates to azolylpropane derivatives of the general formula I ##STR1## wherein R.sub.1 is an azolyl group,R.sub.2 and R.sub.3, each independently of the other, is hydrogen, alkyl, alkenyl, alkynyl, aralkyl, cyanoalkyl or alkoxycarbonylalkyl, and one of R.sub.2 and R.sub.3 always has a meaning other than hydrogen,R.sub.4 is C.sub.3 -C.sub.8 cycloalkyl, unsubstituted or substituted by alkyl; unsubstituted or substituted phenyl; or is C.sub.1 -C.sub.10 alkyl, unsubstituted or substituted by phenyl or substituted phenyl,R.sub.5 is an unsubstituted or a mono- or polysubstituted radical selected from the group consisting of C.sub.1 -C.sub.8 alky, C.sub.3 -C.sub.8 cycloalkyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, phenyl, naphthyl, biphenyl, benzylphenyl, benzyloxyphenyl, phenoxyphenyl and aralkyl,R.sub.6 is hydrogen, alkyl or alkyl substituted by cyano, alkoxy or alkoxycarbonyl, or is an unsubstituted or substituted radical selected from the group consisting of alkylcarbonyl, phenylcarbonyl, carbamoyl, aralkyl, alkoxycarbonyl, alkylsulfonyl, phenylsulfonyl or sulfamoyl, andX is oxygen or sulfur,including the acid addition salts, quaternary azolium salts and metal complexes thereof.The invention further discloses methods of preparing these compounds as well as agrochemical compositions which contain one of said compounds as active component. The invention relates further to a method of controlling phytopathogenic microorganisms and/or of regulating plant growth with the compounds of formula I.

    摘要翻译： 本发明涉及通式Ⅰ（I）的吡唑基丙烷衍生物，其中R 1是唑基，R 2和R 3各自独立地是氢，烷基，烯基，炔基，芳烷基，氰基烷基或烷氧羰基烷基，和 R2和R3中的一个总是具有除氢之外的含义，R4是未被取代或被烷基取代的C3-C8环烷基; 未取代或取代的苯基; 或未被取代或被苯基或取代的苯基取代的C1-C10烷基，R5是未取代的或选自C1-C8烷基，C3-C8环烷基，C3-C6链烯基，C3-C6炔基，苯基， 萘基，联苯基，苄基苯基，苄氧基苯基，苯氧基苯基和芳烷基，R6是氢，被氰基，烷氧基或烷氧基羰基取代的烷基或烷基，或是选自烷基羰基，苯基羰基，氨基甲酰基，芳烷基，烷氧基羰基， 烷基磺酰基，苯基磺酰基或氨磺酰基，X是氧或硫，包括酸加成盐，季氮鎓盐及其金属络合物。 本发明还公开了制备这些化合物的方法以及含有所述化合物之一作为活性组分的农用化学组合物。 本发明还涉及用式I化合物控制植物病原微生物和/或调节植物生长的方法。

    Microbicidal and growth-regulating compositions
    2.
    发明授权
    Microbicidal and growth-regulating compositions 失效
    杀菌和生长调节组合物

    公开(公告)号：US4758670A

    公开(公告)日：1988-07-19

    申请号：US567998

    申请日：1984-01-04

    申请人： Urs Muller ,  Hermann Rempfler ,  Hans Tobler

    发明人： Urs Muller ,  Hermann Rempfler ,  Hans Tobler

    IPC分类号： A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D405/06 ,  C07D521/00 ,  A01N43/64

    CPC分类号： C07D231/12 ,  A01N43/50 ,  A01N43/653 ,  C07D233/56 ,  C07D249/08

    摘要： Fluoroazolylpropane derivatives of the formula I ##STR1## are described, in which Az is imidazolyl or triazolyl, R.sup.1 is hydrogen, alkyl or aralkyl which is unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, nitro, cyano, carboxyl or alkoxycarbonyl, R.sup.2 is C.sub.1 -C.sub.10 -alkyl which is unsubstituted or substituted by alkoxy, aralkoxy or phenyl, it being possible for the aromatic nuclei of aralkoxy and phenyl in turn to be unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.3 is hydrogen, alkyl, alkylcarbonyl or aralkyl which is unsubstituted or substituted by halogen, alkoxy, alkyl, halogenoalkyl, cyano, carboxyl or alkoxycarbonyl, R.sup.5 is an unsubstituted or monosubstituted or polysubstituted radical selected from the series comprising C.sub.1 -C.sub.8 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, phenyl, naphthyl, biphenyl, benzylphenyl, benzyloxyphenyl, phenoxyphenyl and aralkyl, and X is oxygen or sulfur; including the acid addition salts, quaternary azolium salts and metal complexes.Methods of preparing these products are also disclosed, as are agrochemical compositions containing one of these compounds as the active substance. A process for controlling phytopathogenic microorganisms and/or for regulating plant growth by means of these substances is also described.

    摘要翻译： 描述了式I的氟唑基丙烷衍生物，其中Az是咪唑基或三唑基，R1是氢，未被取代或被卤素，烷基，烷氧基，卤代烷基，硝基，氰基，羧基或烷氧基羰基取代的烷基或芳烷基，R2 是未被取代或被烷氧基，芳烷氧基或苯基取代的C 1 -C 10 - 烷基，芳烷氧基和苯基的芳族核可能是未被取代的或被卤素，烷基，烷氧基，卤代烷基，氰基，羧基或烷氧基羰基 R 3是未取代的或被卤素，烷氧基，烷基，卤代烷基，氰基，羧基或烷氧基羰基取代的烷基，烷基，烷基羰基或芳烷基，R 5是未取代的或单取代的或多取代的基团，其选自包括C 1 -C 8烷基， C 3 -C 8 - 环烷基，C 3 -C 6 - 烯基，C 3 -C 6炔基，苯基，萘基，联苯基，苄基苯基，苄氧基苯基，苯氧基苯基和芳烷基，X是氧或硫; 包括酸加成盐，季铵盐和金属络合物。 还公开了制备这些产物的方法，以及含有这些化合物之一作为活性物质的农药组合物。 还描述了通过这些物质控制植物病原微生物和/或调节植物生长的方法。

    5-acylaminopyrimidines
    4.
    发明授权
    5-acylaminopyrimidines 失效
    5-酰氨基嘧啶

    公开(公告)号：US4718934A

    公开(公告)日：1988-01-12

    申请号：US853308

    申请日：1986-04-17

    申请人： Helmut Zondler ,  Hans Tobler ,  Urs Muller

    发明人： Helmut Zondler ,  Hans Tobler ,  Urs Muller

    IPC分类号： A01N43/54 ,  C07D239/42 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D239/50

    CPC分类号： C07D239/42 ,  A01N43/54 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12

    摘要： The invention relates to novel 5-acylaminopyrimidines of the general formula I ##STR1## wherein R.sub.1 is lower alkyl, lower alkoxy, lower alkoxy-lower alkyl, thioalkyl or halogen; phenyl or phenoxy, each unsubstituted or substituted by halogen, halo-lower alkyl, carbalkoxy-lower alkyl, halo-lower alkoxy, lower alkoxy, phenoxy, halophenoxy, halo-lower alkylthio, cyano or nitro; lower alkenyl or lower alkynyl, or unsubstituted or substituted cycloalkylR.sub.2 is lower alkyl which is unsubstituted or substituted by halogen, cyano or lower alkoxy; phenyl or phenyl-lower alkyl, each unsubstituted or substituted; pyridyl, thienyl or furyl, in which the nucleus is unsubstituted or substituted, or is pyranyl, dihydropyranyl, C.sub.3 -C.sub.7 cycloalkyl or C.sub.3 -C.sub.7 alkenyl, andR.sub.3 is hydrogen or C.sub.1 -C.sub.8 alkyl and R.sub.2 and R.sub.3, together with the carbon atom to which they are attached, may form a cycloalkyl radical, which compounds are effective as plant growth regulators. The invention relates further to compositions which contain at least one of these compounds as active ingredient, and to the use thereof, as well as to the corresponding novel 5-aminopyrimidines and, as intermediates, to the novel azomethines from which they are obtained.

    摘要翻译： 本发明涉及通式Ⅰ（I）的新的5-酰氨基嘧啶，其中R1是低级烷基，低级烷氧基，低级烷氧基 - 低级烷基，硫代烷基或卤素; 苯基或苯氧基，各自未被取代或被卤素，卤代低级烷基，烷氧基 - 低级烷基，卤代低级烷氧基，低级烷氧基，苯氧基，卤代苯氧基，卤代低级烷硫基，氰基或硝基取代。 低级烯基或低级炔基，或未取代或取代的环烷基R2是未被取代或被卤素，氰基或低级烷氧基取代的低级烷基; 苯基或苯基 - 低级烷基，各自未取代或取代; 吡啶基，噻吩基或呋喃基，其中核是未取代或取代的，或是吡喃基，二氢吡喃基，C 3 -C 7环烷基或C 3 -C 7链烯基，R 3是氢或C 1 -C 8烷基，R 2和R 3与它们的碳原子一起 可以形成环烷基，该化合物作为植物生长调节剂是有效的。 本发明进一步涉及含有这些化合物中的至少一种作为活性成分的组合物及其用途，以及相应的新的5-氨基嘧啶以及作为中间体获得的新的偶氮甲碱的组合物。

    Fluorinated azolyl ethanol growth regulators and microbicides
    5.
    发明授权
    Fluorinated azolyl ethanol growth regulators and microbicides 失效
    氟化唑类乙醇生长调节剂和杀菌剂

    公开(公告)号：US4610716A

    公开(公告)日：1986-09-09

    申请号：US558140

    申请日：1983-12-05

    申请人： Elmar Sturm ,  Urs Muller ,  Hans Tobler

    发明人： Elmar Sturm ,  Urs Muller ,  Hans Tobler

    IPC分类号： A01N43/50 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

    CPC分类号： C07D303/22 ,  A01N43/50 ,  A01N43/653 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08

    摘要： The compounds described are those of the general formula I ##STR1## in which R.sub.1 is an azolyl group; R.sub.2 is C.sub.1 -C.sub.12 -alkyl; R.sub.3 is hydrogen, C.sub.1 -C.sub.12 -alkyl, C.sub.2 -C.sub.4 -alkenyl or C.sub.2 -C.sub.4 -alkinyl, or benzyl which is unsubstituted or substituted by C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -haloalkyl, halogen and/or cyano; R.sub.4 is hydrogen, fluorine or C.sub.1 -C.sub.6 -alkyl; R.sub.5 is an unsubstituted or substituted radical chosen from the series comprising phenyl, naphthyl, biphenyl, benzylphenyl and benzyloxyphenyl, the substituents being chosen from the series comprising halogen, cyano, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -alkylthio, C.sub.1 -C.sub.6 -haloalkoxy, C.sub.1 -C.sub.3 -haloalkylthio, nitro and/or thiocyano; and X is oxygen or sulfur; including the acid addition salts, quaternary azolium salts and metal complexes.Methods for the preparation of these products are also disclosed, as well as agrochemical compositions containing one of these compounds as the active substance. A method of controlling phytopathogenic microorganisms and/or of regulating plant growth with the aid of these substances is furthermore described.

    摘要翻译： 所述的化合物是通式Ⅰ的化合物（Ⅰ），其中R1是唑基; R2是C1-C12-烷基; R3是氢，C1-C12-烷基，C2-C4-烯基或C2-C4-炔基，或未被取代或被C1-C6-烷基，C1-C6-烷氧基，C1-C6-卤代烷基，卤素和 /或氰基; R4是氢，氟或C1-C6-烷基; R5是选自包括苯基，萘基，联苯基，苄基苯基和苄氧基苯基的系列的未取代或取代的基团，所述取代基选自卤素，氰基，C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基C 1 -C 6 - 卤代烷基 ，C 1 -C 6 - 烷硫基，C 1 -C 6卤代烷氧基，C 1 -C 3卤代烷硫基，硝基和/或氰基氰基; X为氧或硫; 包括酸加成盐，季铵盐和金属络合物。 还公开了制备这些产品的方法，以及含有这些化合物之一作为活性物质的农药组合物。 进一步描述了借助于这些物质控制植物病原微生物和/或调节植物生长的方法。

    Heterocyclic amide derivatives useful as microbiocides
    8.
    发明授权
    Heterocyclic amide derivatives useful as microbiocides 有权
    用作杀微生物剂的杂环酰胺衍生物

    公开(公告)号：US08183416B2

    公开(公告)日：2012-05-22

    申请号：US12765929

    申请日：2010-04-23

    申请人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    发明人： Hans Tobler ,  Harald Walter ,  Josef Ehrenfreund ,  Camilla Corsi

    IPC分类号： C07C205/06

    CPC分类号： C07C205/06 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  C07C205/11 ,  C07C205/12 ,  C07C205/37 ,  C07C205/45 ,  C07C211/61 ,  C07C2603/66 ,  C07D207/34 ,  C07D207/46 ,  C07D213/89 ,  C07D231/14 ,  C07D249/04 ,  C07D263/34 ,  C07D277/56 ,  C07D327/06

    摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R6, R7 and R8; R1 is hydrogen, C1-4 alkyl, C1-4 haloalkyl, C1-4alkoxy, C1-4haloalkoxy, CH2C≡CR9, CH2CR10═CHR11, CH═C═CH2 or COR12; R2 and R3 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl or C1-4 haloalkoxy; R4 and R5 are each independently selected from halo, cyano and nitro; or one of R4 and R5 is hydrogen and the other is selected from halo, cyano and nitro; R6, R7 and R8 are each, independently, hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4haloalkoxy(C1-4)alkyl or C1-4haloalkoxy, provided that at least one of R6, R7 and R8 is not hydrogen; R9, R10 and R11 are each, independently, hydrogen, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 alkoxy(C1-4)alkyl; and R12 is hydrogen, C1-6 alkyl, C1-6haloalkyl, C1-4 alkoxy(C1-4)alkyl, C1-4 alkylthio(C1-4)-alkyl, C1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被R6基团取代 ，R7和R8; R 1是氢，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基，C 1-4卤代烷氧基，CH 2C≡CR9，CH 2 CR 10 = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R4和R5各自独立地选自卤素，氰基和硝基; 或者R 4和R 5中的一个是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4卤代烷氧基（C 1-4）烷基或C 1 -4卤代烷氧基，条件是R 6，R 7和R 8中的至少一个不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4烷氧基（C 1-4）烷基; 并且R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷氧基（C 1-4）烷基，C 1-4烷硫基（C 1-4） - 烷基，C 1-4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或 用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

    Process for the production of carboxanilides
    10.
    发明授权
    Process for the production of carboxanilides 有权
    生产甲酰苯胺的方法

    公开(公告)号：US07820830B2

    公开(公告)日：2010-10-26

    申请号：US12093619

    申请日：2006-11-13

    申请人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    发明人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    IPC分类号： C07D231/14

    CPC分类号： C07D231/14

    摘要： The present invention relates to a novel process for the preparation of a compound of general formula (I): wherein R1 is H or C1-4 alkyl and R2 is difluoromethyl or trifluoromethyl, which comprises reacting a compound of general formula (II): wherein R1 has the meaning given above and X is chloro or bromo, with a compound of general formula (III): wherein R2 has the meaning given above, in the presence of a base, a palladium catalyst and a ferrocenyl biphoshine ligand of the Josiphos type, the reaction being carried out in an ether solvent at a reflux temperature of at least 100° C.

    摘要翻译： 本发明涉及一种制备通式（I）化合物的新方法：其中R1是H或C1-4烷基，R2是二氟甲基或三氟甲基，其包括使通式（II）的化合物：其中 R1具有上面给出的含义，X是氯或溴，与通式（III）的化合物：其中R 2具有上面给出的含义，在碱存在下，钯催化剂和Josiphos型的二茂铁基二膦配体 ，反应在乙醚溶剂中在至少100℃的回流温度下进行。