公开(公告)号：WO2011141414A1

公开(公告)日：2011-11-17

申请号：PCT/EP2011/057403

申请日：2011-05-09

Applicant: BAYER CROPSCIENCE AG ,  ARAKI, Koichi ,  MIHARA, Jun ,  SASAKI, Norio ,  BRUECHNER, Peter ,  DOMON, Kei ,  JANSEN, Johannes-Rudolf ,  LUI, Norbert

Inventor： ARAKI, Koichi ,  MIHARA, Jun ,  SASAKI, Norio ,  BRUECHNER, Peter ,  DOMON, Kei ,  JANSEN, Johannes-Rudolf ,  LUI, Norbert

IPC: C07D207/22 ,  C07C57/62 ,  C07C69/653 ,  A01N43/36

CPC classification number: C07D207/22 ,  C07C51/353 ,  C07C69/65 ,  C07C2601/14 ,  C07C57/62

Abstract: The present invention relates to a process for the manufacturing of 5-substituted 3-aryl-3-(trifluoro-methyl)-3,4-dihydro-2H-pyrroles of formula (I) which comprises the following steps: (i) reacting a compound of formula (II) with a isonitrile compound of formula (III) in the presence of a metal catalyst to obtain compounds of formula (IV) (ii) isomerizing compounds of formula (IV) to obtain compounds of formula (V) and (iii) reacting the dihydropyrrole compound of formula (V) under acidic conditions, to obtain compounds of formula (I), wherein X, n, Z, Y, and T are as defined in the description.

Abstract translation: 本发明涉及制备式（I）的5-取代的3-芳基-3-（三氟甲基）-3,4-二氢-2H-吡咯的方法，该方法包括以下步骤：（i）使 式（II）的化合物与式（III）的异腈化合物在金属催化剂的存在下反应，得到式（IV）的化合物（ⅱ）使式（Ⅳ）化合物异构化得到式（Ⅴ）和 （ⅲ）在酸性条件下使式（Ⅴ）的二氢吡咯化合物反应，得到其中X，n，Z，Y和T如说明书中所定义的式（Ⅰ）化合物。

公开(公告)号：WO2008122375A3

公开(公告)日：2009-01-15

申请号：PCT/EP2008002474

申请日：2008-03-28

Applicant: BAYER CROPSCIENCE AG ,  MIHARA JUN ,  MURATA TETSUYA ,  YAMAZAKI DAIEI ,  YONETA YASUSHI ,  SHIBUYA KATSUHIKO ,  SHIMOJO EIICHI ,  GOERGENS ULRICH ,  TURBERG ANDREAS ,  BACH THOMAS

Inventor： MIHARA JUN ,  MURATA TETSUYA ,  YAMAZAKI DAIEI ,  YONETA YASUSHI ,  SHIBUYA KATSUHIKO ,  SHIMOJO EIICHI ,  GOERGENS ULRICH ,  TURBERG ANDREAS ,  BACH THOMAS

IPC: C07D261/04 ,  A01N43/80 ,  C07D413/10 ,  C07D413/12

CPC classification number: C07D261/04 ,  C07D413/10 ,  C07D413/12

Abstract: The present invention relates to novel aryl isoxazoline derivatives having excellent insecticidal activity as insecticides and represented by the formula ( I ): and their use as insecticides and acarizides.

Abstract translation: 本发明涉及作为杀虫剂具有优良杀虫活性且由式（I）表示的新型芳基异恶唑啉衍生物及其作为杀虫剂和螨类的用途。

公开(公告)号：WO2008128711A1

公开(公告)日：2008-10-30

申请号：PCT/EP2008/003105

申请日：2008-04-14

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  GÖRGENS, Ulrich

Inventor： MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  GÖRGENS, Ulrich

IPC: C07C205/06 ,  C07D207/04 ,  C07D401/04 ,  C07D401/12 ,  C07D403/10 ,  C07D401/14 ,  A01N43/36 ,  A01N43/40

CPC classification number: C07D401/14 ,  A01N43/36 ,  A01N43/40 ,  C07C205/11 ,  C07D207/04 ,  C07D207/06 ,  C07D211/18 ,  C07D401/04 ,  C07D401/12 ,  C07D403/10

Abstract: The present invention provides novel aryl pyrrolidines having an excellent insecticidal action as insecticides. Aryl pyrrolidines represented by the formula (I) and use thereof as insecticide.

Abstract translation: 本发明提供作为杀虫剂具有优异杀虫作用的新型芳基吡咯烷。 由式（I）表示的芳基吡咯烷酮及其作为杀虫剂的用途。

公开(公告)号：WO2005026139A1

公开(公告)日：2005-03-24

申请号：PCT/EP2004/009931

申请日：2004-09-07

Applicant: BAYER CROPSCIENCE AG ,  WATANABE, Yukiyoshi ,  MIHARA, Jun ,  YAMAZAKI, Daiei ,  OTSU, Yuichi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  SHIRAKURA, Shinichi ,  NAKAMURA, Shin

Inventor： WATANABE, Yukiyoshi ,  MIHARA, Jun ,  YAMAZAKI, Daiei ,  OTSU, Yuichi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  SHIRAKURA, Shinichi ,  NAKAMURA, Shin

IPC: C07D285/08

CPC classification number: C07D285/08 ,  A01N43/82 ,  C07D417/04

Abstract: The invention relates to a compound of the formula (I) wherein R represents hydrogen, halogen, alkyl, cycloalkyl, alkoxyalkyl, alkylthioalkyl, haloalkyl, alkoxy, alkylthio, represents optionally substituted phenyl or benzyl, or represents optionally substituted heteroaryl containing at least one heteroatom selected from N, O and S, m represents 3, 4, 5, 6, 7, 8, 9 or 10, and n represents 0, 1 or 2, a process for preparing said compound, compositions comprising said compound and its use for combating pests.

Abstract translation: 本发明涉及式（I）化合物，其中R代表氢，卤素，烷基，环烷基，烷氧基烷基，烷硫基烷基，卤代烷基，烷氧基，烷硫基，代表任意取代的苯基或苄基，或代表任选取代的杂芳基，含有至少一个杂原子 选自N，O和S，m表示3,4,5,6,7,8,9或10，n表示0,1或2，制备所述化合物的方法，包含所述化合物的组合物及其用于 防治害虫

公开(公告)号：WO2010043315A1

公开(公告)日：2010-04-22

申请号：PCT/EP2009/007095

申请日：2009-10-05

Applicant: BAYER CROPSCIENCE AG ,  GÖRGENS, Ulrich ,  MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  ARAKI, Koichi ,  SASAKI, Norio ,  DOMON, Kei ,  HATAZAWA, Mamoru ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko

Inventor： GÖRGENS, Ulrich ,  MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  ARAKI, Koichi ,  SASAKI, Norio ,  DOMON, Kei ,  HATAZAWA, Mamoru ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko

IPC: C07D207/08 ,  C07D401/04 ,  C07D401/12 ,  C07D401/14 ,  C07D403/04 ,  C07D403/12 ,  C07D403/14 ,  C07D405/12 ,  C07D405/14 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/04 ,  C07D417/14 ,  A01N43/36

CPC classification number: A01N43/84 ,  A01N43/36 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/713 ,  A01N43/76 ,  A01N43/78 ,  C07D207/08 ,  C07D207/09 ,  C07D401/04 ,  C07D401/12 ,  C07D401/14 ,  C07D403/04 ,  C07D403/12 ,  C07D403/14 ,  C07D405/12 ,  C07D405/14 ,  C07D409/12 ,  C07D409/14 ,  C07D413/12 ,  C07D417/04 ,  C07D417/14

Abstract: The invention is directed to arylpyrrolidines compounds which exhibit excellent insecticidal efficacy and which may be used as in the agrochemical field or in the vield of veterinary medicine. The compounds are represented by formula (I):wherein the respective substituents are defined in the specification.

Abstract translation: 本发明涉及显示出优异杀虫功效的芳基吡咯烷酮化合物，其可以在农业化学领域或兽医药领域中使用。 化合物由式（I）表示：其中各个取代基在说明书中定义。

公开(公告)号：WO2010015355A2

公开(公告)日：2010-02-11

申请号：PCT/EP2009/005506

申请日：2009-07-30

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  MURATA, Tetsuya ,  DOMON, Kei ,  WATANABE, Yukiyoshi ,  YONETA, Yasushi ,  MORI, Takuma ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  GÖRGENS, Ulrich

Inventor： MIHARA, Jun ,  MURATA, Tetsuya ,  DOMON, Kei ,  WATANABE, Yukiyoshi ,  YONETA, Yasushi ,  MORI, Takuma ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  GÖRGENS, Ulrich

IPC: C07C237/42

CPC classification number: C07C237/42 ,  A01N37/18 ,  A01N43/40 ,  A01N43/50 ,  A01N43/52 ,  A01N43/56 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/78 ,  A01N43/84 ,  A01N55/00 ,  C07D213/82 ,  C07D241/24 ,  C07D285/06 ,  C07D401/12

Abstract: The present invention relates to novel Acylaminobenzamide derivatives represented by the following formula (I) and use thereof as pesticides: wherein V represents an aromatic ring group of V1 to V5 described in the detailed description, Q represents an aromatic ring group of Q1 to Q7 described in the detailed description, G 1 and G 2 represent O or S, R 1 represents hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, phenyl or a heterocyclic group and R 2 and R 3 represent hydrogen, alkyl, haloalkyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl or haloalkoxycarbonyl.

Abstract translation: 本发明涉及由下式（I）表示的新型酰氨基苯甲酰胺衍生物及其作为农药的用途：其中V表示详细描述中描述的V1至V5的芳环基团，Q表示所述的Q1至Q7的芳族环基团 在详细描述中，G1和G2表示O或S，R1表示氢，烷基，卤代烷基，烷氧基，卤代烷氧基，苯基或杂环基，R2和R3表示氢，烷基，卤代烷基，烷基羰基，卤代烷基羰基，烷氧基羰基或卤代烷氧基羰基。

公开(公告)号：WO2009097992A1

公开(公告)日：2009-08-13

申请号：PCT/EP2009/000559

申请日：2009-01-29

Applicant: BAYER CROPSCIENCE AG ,  GÖRGENS, Ulrich ,  YONETA, Yasushi ,  MURATA, Tetsuya ,  MIHARA, Jun ,  DOMON, Kei ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki

Inventor： GÖRGENS, Ulrich ,  YONETA, Yasushi ,  MURATA, Tetsuya ,  MIHARA, Jun ,  DOMON, Kei ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki

IPC: C07D207/20 ,  C07D249/10 ,  C07D403/10 ,  A01N43/36 ,  C07F7/10

CPC classification number: A01N43/36 ,  A01N43/50 ,  A01N43/56 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  C07D207/20 ,  C07D249/10 ,  C07D403/10 ,  C07F7/0812 ,  C07F7/0818

Abstract: The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as insecticides.

Abstract translation: 本发明涉及具有优异杀虫活性并因此可用作杀虫剂的式（I）的新型芳基吡咯啉化合物。

公开(公告)号：WO2008019760A1

公开(公告)日：2008-02-21

申请号：PCT/EP2007/006798

申请日：2007-08-01

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi

Inventor： MIHARA, Jun ,  MURATA, Tetsuya ,  YAMAZAKI, Daiei ,  YONETA, Yasushi ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi

IPC: C07D413/10 ,  C07D413/14 ,  A01N43/80

CPC classification number: C07D413/10 ,  A01N43/80 ,  C07D413/14

Abstract: Novel isoxazolines of the formula (I) wherein A represents C or N; R represents haloalkyl; X represents halogen or haloalkyl; 1 represents 0, 1 or 2; Y represents halogen, alkyl, alkoxy, haloalkyl, cyano, nitro, amino, acylamino, alkoxycarbonylamino, haloalkoxycarbonyl-amino or alkylsulfonylamino; m represents 0, 1 or 2; and G represents any one selected from heterocyclic groups described in the specification; and a use thereof as insecticides and for controlling animal parasites.

Abstract translation: 式（I）的新型异恶唑啉，其中A表示C或N; R代表卤代烷基; X表示卤素或卤代烷基; 1表示0,1或2; Y表示卤素，烷基，烷氧基，卤代烷基，氰基，硝基，氨基，酰氨基，烷氧基羰基氨基，卤代烷氧基羰基 - 氨基或烷基磺酰基氨基; m表示0,1或2; G表示选自说明书中记载的杂环基的任意一种; 以及其作为杀虫剂和控制动物寄生虫的用途。

公开(公告)号：WO2005000824A1

公开(公告)日：2005-01-06

申请号：PCT/EP2004/006367

申请日：2004-06-14

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT ,  YANAGI, Akihiko ,  YAMAGUCHI, Yoshihiro ,  NARABU, Shinichi ,  SHIRAKURA, Shinichi ,  NAKAMURA, Shin ,  MIHARA, Jun

Inventor： YANAGI, Akihiko ,  YAMAGUCHI, Yoshihiro ,  NARABU, Shinichi ,  SHIRAKURA, Shinichi ,  NAKAMURA, Shin ,  MIHARA, Jun

IPC: C07D277/18

CPC classification number: C07D207/273 ,  A01N43/36 ,  A01N43/76 ,  A01N43/78 ,  C07D263/28 ,  C07D277/18

Abstract: Novel azolidine derivatives of the formula (I) wherein R 1 represents halogen, alkyl, alkoxy, haloalkyl, haloalkoxy, haloalkylthio or haloalkylene-dioxy, m represents 0, 1, 2, 3, 4 or 5, the R 1 substituents are identical or different each other, when m represents 2, 3, 4 or 5, R 2 represents alkyl, X represents alkylidene, oxygen atom or sulfur atom, and A represents one of the groups described in the specification and their use as herbicides.

Abstract translation: 式（I）的新型唑烷衍生物，其中R 1表示卤素，烷基，烷氧基，卤代烷基，卤代烷氧基，卤代烷硫基或卤代亚烷基 - 二氧基，m表示0,1,2,3,4或5，R 1， 取代基相同或不同，当m表示2,3,4或5时，R 2表示烷基，X表示亚烷基，氧原子或硫原子，A表示说明书中描述的基团之一及其用途 作为除草剂。

公开(公告)号：WO2011080211A1

公开(公告)日：2011-07-07

申请号：PCT/EP2010/070629

申请日：2010-12-23

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  HATAZAWA, Mamoru ,  YAMAZAKI, Daiei ,  SASAKI, Norio ,  MURATA, Tetsuya ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

Inventor： MIHARA, Jun ,  HATAZAWA, Mamoru ,  YAMAZAKI, Daiei ,  SASAKI, Norio ,  MURATA, Tetsuya ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

IPC: C07D207/04 ,  C07D401/04 ,  A61K31/4439 ,  A61K31/402 ,  A01N43/36 ,  A01N43/40

CPC classification number: C07D401/04 ,  C07D207/08

Abstract: The present invention relates to novel pesticidal arylpyrrolidine compounds (arylpyrrolidines) having the general formula (I) wherein A, X 1 , X 2 , X 3 , X 4 , R 1 , R 2 , R 3 , R 4 , and G are as defined in the application and their use as pesticide, in particular for combating animal pests which occur in the agricultural and / or the veterinary field, as well as to a preparation methods for preparing such compounds.

Abstract translation: 本发明涉及具有通式（I）的新型农药芳基吡咯烷化合物（芳基吡咯烷），其中A，X 1，X 2，X 3，X 4，R 1，R 2，R 3，R 4和G如本申请中所定义， 杀虫剂，特别是用于对抗在农业和/或兽医领域中发生的动物害虫，以及制备这种化合物的制备方法。