公开(公告)号：WO2011080211A1

公开(公告)日：2011-07-07

申请号：PCT/EP2010/070629

申请日：2010-12-23

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  HATAZAWA, Mamoru ,  YAMAZAKI, Daiei ,  SASAKI, Norio ,  MURATA, Tetsuya ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

Inventor： MIHARA, Jun ,  HATAZAWA, Mamoru ,  YAMAZAKI, Daiei ,  SASAKI, Norio ,  MURATA, Tetsuya ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

IPC: C07D207/04 ,  C07D401/04 ,  A61K31/4439 ,  A61K31/402 ,  A01N43/36 ,  A01N43/40

CPC classification number: C07D401/04 ,  C07D207/08

Abstract: The present invention relates to novel pesticidal arylpyrrolidine compounds (arylpyrrolidines) having the general formula (I) wherein A, X 1 , X 2 , X 3 , X 4 , R 1 , R 2 , R 3 , R 4 , and G are as defined in the application and their use as pesticide, in particular for combating animal pests which occur in the agricultural and / or the veterinary field, as well as to a preparation methods for preparing such compounds.

Abstract translation: 本发明涉及具有通式（I）的新型农药芳基吡咯烷化合物（芳基吡咯烷），其中A，X 1，X 2，X 3，X 4，R 1，R 2，R 3，R 4和G如本申请中所定义， 杀虫剂，特别是用于对抗在农业和/或兽医领域中发生的动物害虫，以及制备这种化合物的制备方法。

公开(公告)号：WO2011018170A2

公开(公告)日：2011-02-17

申请号：PCT/EP2010/004739

申请日：2010-08-03

Applicant: BAYER CROPSCIENCE AG ,  MIHARA, Jun ,  ARAKI , Koichi ,  MORI , Takuma ,  MURATA , Tetsuya ,  YONETA, Yasushi ,  WATANABE , Yukiyoshi ,  SHIMOJO , Eiichi ,  ICHIHARA , Teruyuki ,  ATAKA , Masashi ,  SHIBUYA , Katsuhiko ,  GÖRGENS, Ulrich

Inventor： MIHARA, Jun ,  ARAKI , Koichi ,  MORI , Takuma ,  MURATA , Tetsuya ,  YONETA, Yasushi ,  WATANABE , Yukiyoshi ,  SHIMOJO , Eiichi ,  ICHIHARA , Teruyuki ,  ATAKA , Masashi ,  SHIBUYA , Katsuhiko ,  GÖRGENS, Ulrich

IPC: C07C233/66

CPC classification number: C07C233/66 ,  A01N37/42 ,  A01N37/44 ,  A01N37/48 ,  A01N37/50 ,  A01N43/40 ,  A01N43/56 ,  C07C235/84 ,  C07C237/40 ,  C07C237/42 ,  C07C237/48 ,  C07C251/44 ,  C07C251/48 ,  C07C255/19 ,  C07C255/57 ,  C07C271/22 ,  C07C275/24 ,  C07C309/66 ,  C07C311/06 ,  C07C323/60 ,  C07C2601/02 ,  C07C2601/04 ,  C07C2601/08 ,  C07C2601/10 ,  C07C2601/14 ,  C07C2602/08 ,  C07C2602/10 ,  C07D209/48 ,  C07D213/61 ,  C07D213/81 ,  C07D213/82 ,  C07D213/84 ,  C07D213/85 ,  C07D231/12 ,  C07D231/16 ,  C07D249/08 ,  C07D249/18 ,  C07D249/20 ,  C07D257/04 ,  C07D295/155 ,  C07D401/12

Abstract: The object of the present invention is to provide novel carboxamides which exhibit an excellent pesticidal activity as pesticides. Disclosed are the carboxamides represented by the following Formula (I) wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite controling agents.

Abstract translation: 本发明的目的是提供作为杀虫剂表现出优异杀虫活性的新型羧酰胺。 公开了由下列式（I）表示的羧酰胺，其中每个取代基如说明书中所定义，及其作为杀虫剂和动物寄生虫控制剂的用途。

公开(公告)号：WO2010015355A3

公开(公告)日：2010-12-16

申请号：PCT/EP2009005506

申请日：2009-07-30

Applicant: BAYER CROPSCIENCE AG ,  MIHARA JUN ,  MURATA TETSUYA ,  DOMON KEI ,  WATANABE YUKIYOSHI ,  YONETA YASUSHI ,  MORI TAKUMA ,  SHIMOJO EIICHI ,  SHIBUYA KATSUHIKO ,  ICHIHARA TERUYUKI ,  ATAKA MASASHI ,  GOERGENS ULRICH

Inventor： MIHARA JUN ,  MURATA TETSUYA ,  DOMON KEI ,  WATANABE YUKIYOSHI ,  YONETA YASUSHI ,  MORI TAKUMA ,  SHIMOJO EIICHI ,  SHIBUYA KATSUHIKO ,  ICHIHARA TERUYUKI ,  ATAKA MASASHI ,  GOERGENS ULRICH

IPC: C07C237/42 ,  A01N47/20

CPC classification number: C07C237/42 ,  A01N37/18 ,  A01N43/40 ,  A01N43/50 ,  A01N43/52 ,  A01N43/56 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/78 ,  A01N43/84 ,  A01N55/00 ,  C07D213/82 ,  C07D241/24 ,  C07D285/06 ,  C07D401/12

Abstract: The present invention relates to novel Acylaminobenzamide derivatives represented by the following formula (I) and use thereof as pesticides: wherein V represents an aromatic ring group of V1 to V5 described in the detailed description, Q represents an aromatic ring group of Q1 to Q7 described in the detailed description, G1 and G2 represent O or S, R1 represents hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, phenyl or a heterocyclic group and R2 and R3 represent hydrogen, alkyl, haloalkyl, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl or haloalkoxycarbonyl.

Abstract translation: 本发明涉及由下式（I）表示的新型酰氨基苯甲酰胺衍生物及其作为农药的用途：其中V表示详细描述中描述的V1至V5的芳环基团，Q表示所述的Q1至Q7的芳族环基团 在详细描述中，G1和G2表示O或S，R1表示氢，烷基，卤代烷基，烷氧基，卤代烷氧基，苯基或杂环基，R2和R3表示氢，烷基，卤代烷基，烷基羰基，卤代烷基羰基，烷氧基羰基或卤代烷氧基羰基。

公开(公告)号：WO2010133336A1

公开(公告)日：2010-11-25

申请号：PCT/EP2010/003019

申请日：2010-05-18

Applicant: BAYER CROPSCIENCE AG ,  MURATA, Tetsuya ,  YONETA, Yasushi ,  KISHIKAWA, Hidetoshi ,  MIHARA, Jun ,  YAMAZAKI, Daiei ,  HATAZAWA, Mamoru ,  SASAKI, Norio ,  DOMON, Kei ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  SHIBUYA, Katsuhiko ,  ATAKA, Masashi ,  GÖRGENS, Ulrich

Inventor： MURATA, Tetsuya ,  YONETA, Yasushi ,  KISHIKAWA, Hidetoshi ,  MIHARA, Jun ,  YAMAZAKI, Daiei ,  HATAZAWA, Mamoru ,  SASAKI, Norio ,  DOMON, Kei ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  SHIBUYA, Katsuhiko ,  ATAKA, Masashi ,  GÖRGENS, Ulrich

IPC: C07D207/20 ,  C07D401/04 ,  C07D401/14 ,  C07D403/10 ,  C07D403/14 ,  A01N43/36

CPC classification number: A01N43/40 ,  A01N43/36 ,  A01N43/50 ,  A01N43/56 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  C07D207/20 ,  C07D401/04 ,  C07D401/14 ,  C07D403/04 ,  C07D403/10 ,  C07D403/14 ,  C07D405/14

Abstract: The invention relates to novel arylpyrroline compounds of formula (I) which have excellent insecticidal activity and which can thus be used as an insecticide.

Abstract translation: 本发明涉及具有优异杀虫活性并因此可用作杀虫剂的式（I）的新型芳基吡咯啉化合物。

公开(公告)号：WO2010078899A3

公开(公告)日：2010-07-15

申请号：PCT/EP2009/008736

申请日：2009-12-08

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT ,  JESCHKE, Peter ,  VELTEN, Robert ,  NAUEN, Ralf ,  DAUCK, Hartwig ,  HAAS, Matthias ,  PITTA, Leonardo ,  SHIMOJO, Eiichi

Inventor： JESCHKE, Peter ,  VELTEN, Robert ,  NAUEN, Ralf ,  DAUCK, Hartwig ,  HAAS, Matthias ,  PITTA, Leonardo ,  SHIMOJO, Eiichi

IPC: A01N43/08 ,  A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/78 ,  A01P7/02 ,  A01P7/04

Abstract: Verfahren zur Bekämpfung tierischer Schädlinge, die gegenüber einer oder mehreren Klassen von Insektiziden resistent sind, wobei die tierischen Schädlinge und/oder deren Lebensraum mit Enaminocarbonylverbindungen der Formel (I), worin R 1 und A die in der Beschreibung angegebenen Bedeutungen haben, behandelt werden.

公开(公告)号：WO2009112275A1

公开(公告)日：2009-09-17

申请号：PCT/EP2009/001841

申请日：2009-03-13

Applicant: BAYER CROPSCIENCE AG ,  MURATA, Tetsuya ,  YONETA, Yasushi ,  MIHARA, Jun ,  DOMON, Kei ,  HATAZAWA, Mamoru ,  ARAKI, Koichi ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki ,  GÖRGENS, Ulrich ,  VOERSTE, Arnd ,  BECKER, Angela ,  FRANKEN, Eva-Maria ,  MÜLLER, Klaus-Helmut

Inventor： MURATA, Tetsuya ,  YONETA, Yasushi ,  MIHARA, Jun ,  DOMON, Kei ,  HATAZAWA, Mamoru ,  ARAKI, Koichi ,  SHIMOJO, Eiichi ,  SHIBUYA, Katsuhiko ,  ICHIHARA, Teruyuki ,  GÖRGENS, Ulrich ,  VOERSTE, Arnd ,  BECKER, Angela ,  FRANKEN, Eva-Maria ,  MÜLLER, Klaus-Helmut

IPC: C07D207/20 ,  C07D413/04 ,  C07D261/04 ,  A01N43/80

CPC classification number: C07D413/04 ,  A01N43/36 ,  A01N43/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/707 ,  A01N43/80 ,  C07D207/20 ,  C07D261/04

Abstract: Condensed-ring aryl compounds of formula (I) and use of the same as a agrochemical for controlling noxious organisms wherein (X) m Q, A, R 1 , (Y) n and the grouping -W 1 -W 2 -W 3 -W 4 - are as defined herein.

Abstract translation: 式（I）的缩环芳基化合物及其用作农药用于控制有毒生物，其中（X）mQ，A，R1，（Y）n和组-W1-W2-W3-W4-分别为 本文定义。

公开(公告)号：WO2007051560A1

公开(公告)日：2007-05-10

申请号：PCT/EP2006/010315

申请日：2006-10-26

Applicant: BAYER CROPSCIENCE AG ,  YANAGI, Akihiko ,  WATANABE, Yukiyoshi ,  MIHARA, Jun ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  EMOTO, Akira

Inventor： YANAGI, Akihiko ,  WATANABE, Yukiyoshi ,  MIHARA, Jun ,  SHIBUYA, Katsuhiko ,  SHIMOJO, Eiichi ,  EMOTO, Akira

IPC: C07D277/56 ,  A01N43/78

CPC classification number: A01N43/78 ,  C07D277/56

Abstract: 2-Acylaminothiazole-4-carboxamides of the formula (I) and application thereof as an insecticide. Formula (I), wherein R 1 represents phenyl which may be optionally substituted, or a 5- or 6-membered heterocyclic group containing at least one hetero atom selected from a group consisting of N, 0 and S which may be optionally substituted, R 2 represents halogen, C 1-6 alkyl or C 1-6 haloalkyl, R 3 represents C 1-6 haloalkyl, C 1-6 haloalkoxy, C 1-6 haloalkylthio, C 1-6 haloalkylsulf inyl or C 1-6 haloalkylsufonyl, R 4 represents halogen, C 1-6 alkyl or C 1-6 haloalkyl, and X represents hydrogen, halogen, C 1-6 alkyl or C 1-6 haloalkyl, and the use of the new compounds as insecticides.

Abstract translation: 式（I）的2-酰基氨基噻唑-4-甲酰胺及其作为杀虫剂的应用。 式（I）其中R 1表示可任意取代的苯基，或含有至少一个选自N，O和S的杂原子的5或6元杂环基 其可任选被取代，R 2表示卤素，C 1-6烷基或C 1-6 - 卤代烷基，R 3， / SUP表示C 1-6卤代烷基，C 1-6卤代烷氧基，C 1-6卤代烷硫基，C 1-6 卤代烷基亚磺酰基或C 1-6卤代烷基磺酰基，R 4表示卤素，C 1-6烷基或C 1〜 -6个卤代烷基，X表示氢，卤素，C 1-6烷基或C 1-6 - 卤代烷基，并且使用新化合物作为杀虫剂 。

公开(公告)号：WO2003097604A1

公开(公告)日：2003-11-27

申请号：PCT/EP2003/004714

申请日：2003-05-06

Applicant: BAYER CROPSCIENCE GMBH ,  ARAKI, Koichi ,  MURATA, Tetsuya ,  GUNJIMA, Koshi ,  NAKAKURA, Norihiko ,  SHIMOJO, Eiichi ,  ARNOLD, Christian ,  HEMPEL, Waltraud ,  JANS, Daniela ,  MALSAM, Olga ,  WAIBEL, Jutta, Maria

Inventor： ARAKI, Koichi ,  MURATA, Tetsuya ,  GUNJIMA, Koshi ,  NAKAKURA, Norihiko ,  SHIMOJO, Eiichi ,  ARNOLD, Christian ,  HEMPEL, Waltraud ,  JANS, Daniela ,  MALSAM, Olga ,  WAIBEL, Jutta, Maria

IPC: C07D213/82

CPC classification number: C07D213/82 ,  A01N43/40 ,  C07D401/06 ,  C07D413/06

Abstract: The invention relates to a 3-pyridylcarboxamide derivative of formula (I). Wherein the various symbols are as defined in the description, compositions thereof, their use for the control of pests, and to processes for their preparation.

Abstract translation: 本发明涉及式（I）的3-吡啶基羧酰胺衍生物。 其中各种符号如描述中所定义，其组成，其用于控制​​害虫的用途及其制备方法。

公开(公告)号：WO2011128299A1

公开(公告)日：2011-10-20

申请号：PCT/EP2011/055639

申请日：2011-04-11

Applicant: Bayer CropScience AG ,  MORADI, Ahmed Wahed ,  MUELLER, Thomas Norbert ,  MURATA, Tesuya ,  HATAZAWA, Mamoru ,  BRUECHNER, Peter ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GOERGENS, Ulrich

Inventor： MORADI, Ahmed Wahed ,  MUELLER, Thomas Norbert ,  MURATA, Tesuya ,  HATAZAWA, Mamoru ,  BRUECHNER, Peter ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GOERGENS, Ulrich

IPC: C07D207/18 ,  C07D249/08 ,  C07C233/31 ,  C07C233/33 ,  A01N37/18 ,  A01N43/653

CPC classification number: A01N37/18 ,  A01N43/653 ,  C07C201/12 ,  C07C205/45 ,  C07C225/16 ,  C07C231/12 ,  C07C233/31 ,  C07C233/32 ,  C07C233/61 ,  C07C235/14 ,  C07C253/30 ,  C07C255/56 ,  C07C271/24 ,  C07C317/44 ,  C07C323/60 ,  C07C2601/02 ,  C07C2602/10 ,  C07D207/18 ,  C07D207/20 ,  C07D249/08

Abstract: The invention is directed to method for the preparation of pyrrolines of the general formula (I) by catalytic hydration of a nitroketone of the general formula (II) employing a transition metal catalyst and gaseous hydrogen at an elevated pressure in a solvent, optionally in the presence of at least one additive selected among Lewis acids, Brønstedt acids, organic sulfur-containing compounds, organic or inorganic bases, and water scavengers, wherein in formulae (I) and (II) B 1 , B 2 , B 3 , B 4 , X, R, and T are as defined in the specification, and to a nitroketone of formula (II) to be used as intermediate in the process according to the invention and as pesticidal agent.

Abstract translation: 本发明涉及通过使用过渡金属催化剂和气态氢在溶剂中在升高的压力下催化水合通式（II）的硝基酮来制备通式（I）的吡咯烷的方法，任选地在 存在选自路易斯酸，布朗斯台德酸，有机含硫化合物，有机或无机碱和除水剂中的至少一种添加剂，其中式（I）和（II）B1，B2，B3，B4，X，R 和T如说明书中所定义，并且与在本发明的方法中用作中间体的式（II）的硝基酮和作为杀虫剂一起使用。

公开(公告)号：WO2011051455A1

公开(公告)日：2011-05-05

申请号：PCT/EP2010/066480

申请日：2010-10-29

Applicant: BAYER CROPSCIENCE AG ,  MURATA, Tetsuya ,  HATAZAWA, Mamoru ,  BRÜCHNER, Peter ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

Inventor： MURATA, Tetsuya ,  HATAZAWA, Mamoru ,  BRÜCHNER, Peter ,  SHIMOJO, Eiichi ,  ICHIHARA, Teruyuki ,  ATAKA, Masashi ,  SHIBUYA, Katsuhiko ,  GÖRGENS, Ulrich

IPC: C07D263/12 ,  C07D291/04 ,  A01N33/06

CPC classification number: C07D263/12 ,  C07D291/04

Abstract: The present invention relates to novel pesticidal azolidine derivatives as well as to oxazolidinone derivatives and their use as pesticides for combating animal parasites which occur in the agrochemical field and in the field of veterinary medicine, respectively. Formula (I) wherein X, m, R', Q, G, U, 1, A 1 to A 4 and R are as defined herein.

Abstract translation: 本发明涉及新型杀虫唑烷衍生物以及恶唑烷酮衍生物及其作为农药用于防治农药领域和兽医领域中的动物寄生虫的用途。 式（I）其中X，m，R'，Q，G，U，1，A1至A4和R如本文所定义。