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">1.发明公开PHARMAZEUTISCHE ZUSAMMENSETZUNG UND DEREN VERWENDUNG SOWIE ANWENDUNGSREGIME DIESER PHARMAZEUTISCHEN ZUSAMMENSETZUNG ZUR BEDARFSWEISEN ( ON-DEMAND") KONTRAZEPTION 审中-公开药物组合物及其使用和本制度药物组合物，买家方式的应用（ON-DEMAND“）避孕
公开(公告)号：EP2999469A1
公开(公告)日：2016-03-30
申请号：EP14724746.4
申请日：2014-05-16
发明人： LINDENTHAL, Bernhard , BRÄUER, Nico , SERNO, Peter , ROTGERI, Andrea , FUHRMANN, Ulrike , BUCHMANN, Bernd , MENGEL, Anne , RÖHN, Ulrike , TER LAAK, Antonius
IPC分类号： A61K31/416 , A61K31/4439 , A61K31/505 , A61K31/5415 , A61P15/18
CPC分类号： A61K31/454 , A61K31/18 , A61K31/192 , A61K31/196 , A61K31/365 , A61K31/405 , A61K31/407 , A61K31/416 , A61K31/42 , A61K31/444 , A61K31/4545 , A61K31/5377 , A61K31/5415 , A61K31/542 , A61K31/635 , A61K2300/00
摘要： The invention relates to a pharmaceutical composition for an on-demand non-hormonal contraception and to a method for producing said pharmaceutical composition. The composition contains 2H-indazoles as novel EP2 receptor antagonists in combination with COX inhibitors. The invention further relates to a method for the female-controlled on-demand non-hormonal contraception, wherein a pharmaceutical composition which contains EP2 receptor antagonists in combination with COX inhibitors is taken on-demand prior to an expected sexual intercourse.
摘要翻译： 本发明涉及一种用于按需以及制备该药用组合物处理非激素避孕的药物组合物。 后者包括2H-吲唑与COX抑制剂的组合新颖EP2受体拮抗剂。 本发明进一步更提供用于非激素女性控制点播避孕其中包括EP2受体拮抗剂与COX抑制剂的组合的药物组合物采取之前预期性交需求的方法。
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公开(公告)号：EP3580211A1
公开(公告)日：2019-12-18
申请号：EP18703958.1
申请日：2018-02-02
发明人： GUTCHER, Ilona , RÖHN, Ulrike , SCHMEES, Norbert , ZORN, Ludwig , RÖSE, Lars , BADER, Benjamin , KOBER, Christina , CARRETERO, Rafael , STÖCKIGT, Detlef , IRLBACHER, Horst , PLATTEN, Michael
IPC分类号： C07D401/14 , C07D405/14 , C07D401/04 , C07D403/04 , C07D237/04 , C07D237/24 , C07D409/04 , C07D413/04 , C07D417/04 , C07D417/14 , A61K31/501 , A61P35/00
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公开(公告)号：EP3049390A1
公开(公告)日：2016-08-03
申请号：EP14771910.8
申请日：2014-09-24
发明人： RÖHN, Ulrike , ELLERMANN, Manuel , STRASSBURGER, Julia , WENDT, Astrid , RÖHRIG, Susanne , WEBSTER, Robert, Alan , SCHMIDT, Martina, Victoria , TERSTEEGEN, Adrian , BEYER, Kristin , SCHÄFER, Martina , BUCHMÜLLER, Anja , GERDES, Christoph , SPERZEL, Michael , SANDMANN, Steffen , HEITMEIER, Stefan , HILLISCH, Alexander , ACKERSTAFF, Jens , TERJUNG, Carsten
IPC分类号： C07D209/42 , A61P7/02 , A61K31/16 , C07D231/56 , C07D235/08 , C07D235/26 , C07D249/08 , C07D249/10 , C07D257/04 , C07D263/58 , C07D401/12 , C07D401/14 , C07D403/12 , C07D413/12 , C07D417/12
CPC分类号： C07D401/12 , C07D209/42 , C07D231/56 , C07D235/08 , C07D235/26 , C07D249/04 , C07D249/08 , C07D249/10 , C07D257/04 , C07D263/58 , C07D401/14 , C07D403/12 , C07D413/12 , C07D417/12 , C07D451/04 , C07D487/04
摘要： The invention relates to substituted phenylalanine derivatives and to methods for the production thereof, in addition to the use of said derivatives for producing drugs for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and/or perioperative heavy blood loss.
摘要翻译： 除了使用所述衍生物生产用于治疗和/或预防疾病，特别是心血管疾病和/或围手术期严重失血的药物之外，本发明涉及取代的苯丙氨酸衍生物和其制备方法。
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公开(公告)号：EP3713926A1
公开(公告)日：2020-09-30
申请号：EP18800216.6
申请日：2018-11-16
发明人： LEFRANC, Julien , SCHMEES, Norbert , RÖHN, Ulrike , ZORN, Ludwig , GÜNTHER, Judith , GUTCHER, Ilona , RÖSE, Lars , BADER, Benjamin , STÖCKIGT, Detlef , PLATTEN, Michael
IPC分类号： C07D401/04 , C07D403/04 , C07D409/04 , C07D413/04 , A61K31/506 , A61P35/00
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公开(公告)号：EP3049410A1
公开(公告)日：2016-08-03
申请号：EP14772148.4
申请日：2014-09-24
发明人： RÖHN, Ulrike , ELLERMANN, Manuel , STRASSBURGER, Julia , WENDT, Astrid , RÖHRIG, Susanne , WEBSTER, Robert Alan , SCHMIDT, Martina Victoria , TERSTEEGEN, Adrian , BEYER, Kristin , SCHÄFER, Martina , BUCHMÜLLER, Anja , GERDES, Christoph , SPERZEL, Michael , SANDMANN, Steffen , HEITMEIER, Stefan , HILLISCH, Alexander , ACKERSTAFF, Jens , TERJUNG, Carsten
IPC分类号： C07D413/12 , C07D257/04 , C07D401/12 , A61K31/41 , A61K31/454 , A61K31/496 , A61P7/00 , A61P9/00
CPC分类号： C07D257/04 , C07D249/08 , C07D401/12 , C07D405/12 , C07D413/12
摘要： The invention relates to substituted phenylalanine derivatives and to methods for the production thereof, in addition to the use of said derivatives for producing medicaments for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and/or perioperative heavy blood loss.
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公开(公告)号：EP3049408A1
公开(公告)日：2016-08-03
申请号：EP14772147.6
申请日：2014-09-24
发明人： RÖHN, Ulrike , ELLERMANN, Manuel , STRASSBURGER, Julia , WENDT, Astrid , RÖHRIG, Susanne , WEBSTER, Robert Alan , SCHMIDT, Martina Victoria , TERSTEEGEN, Adrian , BEYER, Kristin , SCHÄFER, Martina , BUCHMÜLLER, Anja , GERDES, Christoph , SPERZEL, Michael , SANDMANN, Steffen , HEITMEIER, Stefan , HILLISCH, Alexander , ACKERSTAFF, Jens , TERJUNG, Carsten
IPC分类号： C07D403/12 , C07D231/56 , C07D401/12 , C07D235/26 , C07D405/12 , C07D249/10 , C07D257/04 , A61P7/02
CPC分类号： C07D405/12 , C07D231/56 , C07D235/26 , C07D249/08 , C07D249/10 , C07D257/04 , C07D401/12 , C07D403/12
摘要： The invention relates to substituted phenylalanine derivatives and to methods for the production thereof, in addition to the use of said derivatives for producing drugs for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and/or perioperative heavy blood loss.
摘要翻译： 本发明涉及取代的苯丙氨酸衍生物及其制备方法，以及其用于生产用于治疗和/或预防特别是心血管疾病和/或严重围手术期失血的疾病的药物的用途。
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公开(公告)号：EP2376463A1
公开(公告)日：2011-10-19
申请号：EP09767957.5
申请日：2009-11-28
发明人： HASSFELD, Jorma , RÖHN, Ulrike , FRIEBE, Matthias , LEHMANN, Lutz , HEINRICH, Tobias , KRAUSE, Sabine , BROCKSCHNIEDER, Damian , DYRKS,Thomas , THIELE, Andrea , BÖMER, Ulf , MÖNNING, Ursula , BERGER, Markus , SIEGEL, Stephan
IPC分类号： C07D277/82 , C07D417/12 , A61K31/428 , A61P25/28
CPC分类号： C07D277/82 , C07D417/12
摘要： This invention relates to compounds of formula I (benzothiazoles) suitable for labelling or already labelled by
18 F, methods of preparing such a compound, compositions comprising such compounds, kits comprising such compounds or compositions and uses of such compounds, compositions or kits for diagnostic imaging.-
公开(公告)号：EP3580211B1
公开(公告)日：2020-12-02
申请号：EP18703958.1
申请日：2018-02-02
发明人： GUTCHER, Ilona , RÖHN, Ulrike , SCHMEES, Norbert , ZORN, Ludwig , RÖSE, Lars , BADER, Benjamin , KOBER, Christina , CARRETERO, Rafael , STÖCKIGT, Detlef , IRLBACHER, Horst , PLATTEN, Michael
IPC分类号： C07D401/14 , C07D405/14 , C07D401/04 , C07D403/04 , C07D237/04 , C07D237/24 , C07D409/04 , C07D413/04 , C07D417/04 , C07D417/14 , A61K31/501 , A61P35/00
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公开(公告)号：EP3049407A1
公开(公告)日：2016-08-03
申请号：EP14771920.7
申请日：2014-09-24
发明人： RÖHN, Ulrike , ELLERMANN, Manuel , STRASSBURGER, Julia , WENDT, Astrid , RÖHRIG, Susanne , WEBSTER, Robert Alan , SCHMIDT, Martina Victoria , TERSTEEGEN, Adrian , BEYER, Kristin , SCHÄFER, Martina , BUCHMÜLLER, Anja , GERDES, Christoph , SPERZEL, Michael , SANDMANN, Steffen , HEITMEIER, Stefan , HILLISCH, Alexander , ACKERSTAFF, Jens , TERJUNG, Carsten
IPC分类号： C07D403/12 , C07D413/12 , C07D471/04 , C07D401/12 , A61K31/41 , A61K31/437 , A61K31/4725 , A61P7/00 , A61P9/00
CPC分类号： C07D403/12 , C07D401/12 , C07D413/12 , C07D471/04
摘要： The invention relates to substituted phenylalanine derivatives and to methods for the production thereof, in addition to the use of said derivatives for producing medicaments for the treatment and/or prophylaxis of diseases, in particular cardiovascular diseases and/or perioperative heavy blood loss.
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10.发明公开SUBSTITUIERTE PHENYLALANIN-DERIVATE UND IHRE VERWENDUNG ZUR BEHANDLUNG VON THROMBOTISCHEN / THROMBOEMBOLISCHEN ERKRANKUNGEN 审中-公开取代的苯丙氨酸衍生物及其血栓/血栓栓塞性疾病的治疗
公开(公告)号：EP3049406A1
公开(公告)日：2016-08-03
申请号：EP14771915.7
申请日：2014-09-24
发明人： RÖHN, Ulrike , ELLERMANN, Manuel , STRASSBURGER, Julia , WENDT, Astrid , RÖHRIG, Susanne , WEBSTER, Robert Alan , SCHMIDT, Martina Victoria , TERSTEEGEN, Adrian , BEYER, Kristin , SCHÄFER, Martina , BUCHMÜLLER, Anja , GERDES, Christoph , SPERZEL, Michael , SANDMANN, Steffen , HEITMEIER, Stefan , HILLISCH, Alexander , ACKERSTAFF, Jens , TERJUNG, Carsten
IPC分类号： C07D403/12 , C07D231/56 , C07D401/12 , C07D235/26 , C07D413/12 , C07D249/10 , C07D257/04 , C07D271/07 , A61K31/41 , A61K31/416 , A61K31/4184 , A61K31/4196 , A61K31/4245 , A61K31/454 , A61K31/496
CPC分类号： C07D257/04 , C07B2200/07 , C07D231/56 , C07D235/26 , C07D237/32 , C07D249/08 , C07D249/10 , C07D271/07 , C07D401/12 , C07D403/12 , C07D413/12
摘要： The invention relates to substituted phenylalanine derivatives of formula (I), in which R
1 stands for a group of formula (II) or formula (III), R
2 stands for hydrogen, fluorine, chlorine, methyl, or methoxy, R
3 stands for hydrogen, fluorine, chlorine, C
1 -C
4 alkyl, methoxy, or trifluoromethyl, and R
4 stands for amino, cyano, C
1 -C
3 alkoxy, C
1 -C
3 alkylamino, C
1 -C
3 alkoxycarbonyl, C
1 -C
3 alkylcarbonylamino, C
1 -C
3 alkysulfonyl, -S(O)
2 NR
10 R
11 , or 5- to 7-membered heterocyclyl bonded by means of a nitrogen atom. The invention further relates to the use thereof to produce drugs for treating and/or preventing illnesses, in particular cardiovascular diseases and/or perioperative heavy blood loss.摘要翻译： 本发明涉及substituiertem苯丙氨酸衍生物和用于制备方法，以及它们的其用途对于生产药物用于治疗和/或预防疾病，爱的特别心血管病症和/或严重围手术期失血。 TRG416065
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