公开(公告)号：US4603130A

公开(公告)日：1986-07-29

申请号：US594298

申请日：1984-03-28

申请人： Ryuichi Iemura ,  Tsuneo Kawashima ,  Toshikazu Fukuda ,  Keizo Ito ,  Takashi Nose ,  Goro Tsukamoto

发明人： Ryuichi Iemura ,  Tsuneo Kawashima ,  Toshikazu Fukuda ,  Keizo Ito ,  Takashi Nose ,  Goro Tsukamoto

IPC分类号： A61K31/415 ,  A61K31/4184 ,  A61K31/55 ,  A61P43/00 ,  C07D235/14 ,  C07D403/06 ,  C07D403/04 ,  A61K31/495 ,  C07D241/02

CPC分类号： C07D235/14 ,  Y02P20/55

摘要： Novel benzimidazole derivatives of the formula: ##STR1## wherein R.sup.1 is a lower alkyl group, a lower alkenyl group or a lower alkynyl group, R.sup.2 is hydrogen atom, a lower alkyl group or a lower hydroxyalkyl group, and n is 2 or 3, or a pharmaceutically acceptable acid addition salt thereof, which have potent antihistaminic activity with less toxicity and hence are useful as an antihistaminics, and a process for the preparation of the compounds, and a pharmaceutical composition useful as antihistaminics containing the compound as an essential active ingredient.

摘要翻译： 下式的新型苯并咪唑衍生物：其中R1是低级烷基，低级烯基或低级炔基，R2是氢原子，低级烷基或低级羟烷基，n是2或3， 或其药学上可接受的酸加成盐，其具有有效的抗组胺活性，毒性低，因此可用作抗组胺剂，以及用于制备化合物的方法，以及用作抗组胺剂的药物组合物，其含有该化合物作为必需活性成分 。

公开(公告)号：US4430343A

公开(公告)日：1984-02-07

申请号：US436032

申请日：1982-10-22

申请人： Ryuichi Iemura ,  Tsuneo Kawashima ,  Toshikazu Fukuda ,  Keizo Ito ,  Takashi Nose ,  Goro Tsukamoto

发明人： Ryuichi Iemura ,  Tsuneo Kawashima ,  Toshikazu Fukuda ,  Keizo Ito ,  Takashi Nose ,  Goro Tsukamoto

IPC分类号： A61K31/415 ,  A61K31/4184 ,  A61K31/495 ,  A61K31/496 ,  A61K31/55 ,  A61P37/08 ,  A61P43/00 ,  C07D235/24 ,  C07D235/30 ,  C07D403/04 ,  C07D403/02

CPC分类号： C07D235/24 ,  C07D235/30 ,  C07D403/04 ,  Y02P20/55 ,  Y10S514/83 ,  Y10S514/861 ,  Y10S514/914

摘要： Novel benzimidazole derivatives of the formula: ##STR1## wherein R.sup.1 is an alkyl group having 1 to 3 carbon atoms, allyl group, propargyl group, or phenyl group; R.sup.2 is hydrogen atom or an alkyl group having 1 to 3 carbon atoms; and n is 2 or 3, or pharmaceutically acceptable acid addition salts thereof, which have excellent antihistaminic activities and are useful as antiallergics for various allergic diseases, and a process for the preparation thereof, and an antihistaminic composition containing the compound as an active ingredient.

摘要翻译： 具有下式的新型苯并咪唑衍生物：其中R 1是具有1至3个碳原子的烷基，烯丙基，炔丙基或苯基; R2是氢原子或碳原子数1〜3的烷基; 和n为2或3，或其药学上可接受的酸加成盐，其具有优异的抗组胺活性，并且可用作各种过敏性疾病的抗过敏药，及其制备方法，以及含有该化合物作为活性成分的抗组胺组合物。

公开(公告)号：US4192880A

公开(公告)日：1980-03-11

申请号：US949429

申请日：1978-10-10

申请人： Goro Tsukamoto ,  Koichiro Yoshino ,  Toshihiko Kohno ,  Masahiro Taguchi ,  Katsumi Dezawa ,  Hajime Kagaya ,  Keizo Ito ,  Takashi Nose

发明人： Goro Tsukamoto ,  Koichiro Yoshino ,  Toshihiko Kohno ,  Masahiro Taguchi ,  Katsumi Dezawa ,  Hajime Kagaya ,  Keizo Ito ,  Takashi Nose

IPC分类号： C07D235/18 ,  A61K31/415 ,  C07D235/08

CPC分类号： C07D235/18 ,  Y10S514/96

摘要： 2-Substituted benzimidazole compounds of the formula: ##STR1## wherein R.sub.1 is hydrogen, halogen, lower alkyl or lower alkoxy, and R.sub.2 is hydrogen or lower alkyl with the proviso that R.sub.1 and R.sub.2 do not stand for hydrogen simultaneously and, when R.sub.1 is hydrogen, R.sub.2 cannot mean a methyl group at 6th position on the pyridin-2-yl group or methyl an isobutyl group on the phenyl group; are useful as anti-inflammatory agents and/or analgesics.

摘要翻译： 2-取代的下式的苯并咪唑化合物：其中R 1是氢，卤素，低级烷基或低级烷氧基，R 2是氢或低级烷基，条件是R 1 并且R2不同时代表氢，当R1为氢时，R2不表示吡啶-2-基上第六位的甲基或苯基上的甲基异丁基; 可用作抗炎剂和/或止痛剂。

公开(公告)号：US4434162A

公开(公告)日：1984-02-28

申请号：US366415

申请日：1982-04-07

申请人： Goro Tsukamoto ,  Toshihiko Kohno ,  Koichiro Yoshino ,  Tominori Morita ,  Keizo Ito ,  Takashi Nose

发明人： Goro Tsukamoto ,  Toshihiko Kohno ,  Koichiro Yoshino ,  Tominori Morita ,  Keizo Ito ,  Takashi Nose

IPC分类号： C07F9/6541 ,  C07D277/66 ,  A61K31/425

CPC分类号： C07F9/6541 ,  Y10S514/929

摘要： A phosphonic acid ester of the formula ##STR1## exhibits calcium-antagonistic, coronary vasodilating and hypotensive activities. Pharmaceutical compositions containing the same are useful for the prophylaxis and treatment of circulatory organ diseases such as angina pectoris, hypertension and the like.

摘要翻译： 式“IMAGE”的膦酸酯显示钙拮抗，冠状血管扩张和降血压活性。 含有该组合物的药物组合物可用于预防和治疗诸如心绞痛，高血压等循环器官疾病。

公开(公告)号：US4188486A

公开(公告)日：1980-02-12

申请号：US856969

申请日：1977-12-02

申请人： Goro Tsukamoto ,  Koichiro Yoshino ,  Toshihiko Kohno ,  Masahiro Taguchi ,  Katsumi Dezawa ,  Hajime Kagaya ,  Keiso Ito ,  Takashi Nose

发明人： Goro Tsukamoto ,  Koichiro Yoshino ,  Toshihiko Kohno ,  Masahiro Taguchi ,  Katsumi Dezawa ,  Hajime Kagaya ,  Keiso Ito ,  Takashi Nose

IPC分类号： C07D235/18 ,  C07D401/02

CPC分类号： C07D235/18

摘要： 2-Substituted benzimidazole compounds of the formula: ##STR1## wherein R.sub.1 is hydrogen, halogen, lower alkyl or lower alkoxy, and R.sub.2 is hydrogen or lower alkyl with the proviso that R.sub.1 and R.sub.2 do not stand for hydrogen simultaneously and, when R.sub.1 is hydrogen, R.sub.2 cannot mean a methyl group at the 6th position on the pyridin-2-yl group or methyl an isobutyl group on the phenyl group; are useful as anti-inflammatory agents and/or analgesics.

摘要翻译： 2-取代的下式的苯并咪唑化合物：其中R 1是氢，卤素，低级烷基或低级烷氧基，R 2是氢或低级烷基，条件是R 1和R 2 不同时代表氢，当R1为氢时，R2不能指吡啶-2-基上第六位的甲基或苯基上的甲基异丁基; 可用作抗炎剂和/或止痛剂。

公开(公告)号：US4232010A

公开(公告)日：1980-11-04

申请号：US39311

申请日：1979-05-14

申请人： Goro Tsukamoto ,  Koichiro Yoshino ,  Tominori Morita ,  Takashi Nose ,  Mitsuo Okazaki

发明人： Goro Tsukamoto ,  Koichiro Yoshino ,  Tominori Morita ,  Takashi Nose ,  Mitsuo Okazaki

IPC分类号： C07D277/66 ,  C07D417/04 ,  C07F9/58 ,  C07F9/6541 ,  C07F9/6558 ,  A01N57/28 ,  C07F9/28 ,  C07D417/02

CPC分类号： C07D417/04 ,  C07D277/66 ,  C07F9/582 ,  C07F9/6541 ,  C07F9/65583

摘要： A phosphonic acid ester of the formula: ##STR1## and R is a lower alkyl, exhibits a calcium-antagonistic activity. Pharmaceutical compositions containing the same are useful in prophylaxis and treatment of ischemic heart diseases such as angina pectoris, myocardial, infarction, etc. and hypertension.

摘要翻译： 下式的膦酸酯：其中A是+ TR，并且R是低级烷基，表现出钙拮抗活性。 含有该组合物的药物组合物可用于预防和治疗心绞痛，心肌梗死等心肌梗塞等心肌缺血性心脏病和高血压。

公开(公告)号：US09049092B2

公开(公告)日：2015-06-02

申请号：US13431859

申请日：2012-03-27

申请人： Akio Sugiyama ,  Takashi Nose ,  Yoshihiko Hori ,  Hirobumi Furihata

发明人： Akio Sugiyama ,  Takashi Nose ,  Yoshihiko Hori ,  Hirobumi Furihata

IPC分类号： G06F3/038 ,  H04L25/49 ,  H04N7/01 ,  G06F13/00

CPC分类号： G09G3/2018 ,  G06F13/00 ,  G09G3/2096 ,  G09G5/008 ,  G09G5/18 ,  G09G2310/027 ,  G09G2310/08 ,  G09G2320/064 ,  G09G2330/06 ,  G09G2360/127 ,  G09G2360/16 ,  G09G2370/00 ,  H04L25/49 ,  H04L25/4908 ,  H04N7/01

摘要： A data transmission system for a display device, which is an mBnB encoding system encoding a signal of m (m is a natural number) bits into a signal of n (n is a natural number and n>m) bits on the basis of a certain translation table to be transmitted thereafter, the system including: an output driver of outputting a gray scale voltage in accordance with the data decoded at a receiver side, in which in the translation table, a bit pattern with a larger data change index from among 2n pieces of bit patterns of the n bits of the data is assigned to a bit pattern with a larger amplitude of the gray scale voltage from among 2m pieces of bit patterns of the m bits of the data.

摘要翻译： 一种用于显示装置的数据传输系统，其是将m（m是自然数）信号编码为n（n是自然数和n> m）位的信号的mBnB编码系统，其基于 该系统包括：输出驱动器，其根据在接收机侧解码的数据输出灰度级电压，其中在转换表中具有来自其中的更大的数据变化指数的位模式 从数据的m位的2m个位模式中，将数据的n位的2n个位模式分配给具有较大幅度的灰度级电压的位模式。

公开(公告)号：US08705135B2

公开(公告)日：2014-04-22

申请号：US11407055

申请日：2006-04-20

申请人： Hirobumi Furihata ,  Takashi Nose

发明人： Hirobumi Furihata ,  Takashi Nose

IPC分类号： G09G3/36 ,  H04N1/40

CPC分类号： G09G3/2007 ,  G09G3/3611 ,  G09G2320/0276 ,  G09G2320/0285 ,  G09G2320/0673 ,  G09G2330/021 ,  G09G2360/144

摘要： A display control apparatus according to an embodiment of the present invention includes: a grayscale converting circuit for converting input image data to output image data using a look-up table showing a correspondence between input image data of i bits and output image data of k bits larger than the i bits; and an LUT creating circuit for creating the look-up table based on γ data of 2k bits. The apparatus further includes a γ data storage circuit capable of storing the plural γ data in the LUT creating circuit.

摘要翻译： 根据本发明实施例的显示控制装置包括：灰度转换电路，用于使用查询表将输入图像数据转换为输出图像数据，该查找表示出i位的输入图像数据和k位的输出图像数据之间的对应关系 大于i位; 以及用于基于2k位的γ数据创建查找表的LUT创建电路。 该装置还包括能够在LUT生成电路中存储多个γ数据的γ数据存储电路。

公开(公告)号：US08566097B2

公开(公告)日：2013-10-22

申请号：US12791781

申请日：2010-06-01

申请人： Mikio Nakano ,  Takashi Nose ,  Ryo Taguchi ,  Kotaro Funakoshi ,  Naoto Iwahashi

发明人： Mikio Nakano ,  Takashi Nose ,  Ryo Taguchi ,  Kotaro Funakoshi ,  Naoto Iwahashi

IPC分类号： G10L15/00

CPC分类号： G10L15/063 ,  G10L15/187

摘要： A lexical acquisition apparatus includes: a phoneme recognition section 2 for preparing a phoneme sequence candidate from an inputted speech; a word matching section 3 for preparing a plurality of word sequences based on the phoneme sequence candidate; a discrimination section 4 for selecting, from among a plurality of word sequences, a word sequence having a high likelihood in a recognition result; an acquisition section 5 for acquiring a new word based on the word sequence selected by the discrimination section 4; a teaching word list 4A used to teach a name; and a probability model 4B of the teaching word and an unknown word, wherein the discrimination section 4 calculates, for each word sequence, a first evaluation value showing how much words in the word sequence correspond to teaching words in the list 4A and a second evaluation value showing a probability at which the words in the word sequence are adjacent to one another and selects a word sequence for which a sum of the first evaluation value and the second evaluation value is maximum, and wherein the acquisition section 5 acquires, as a new word, a word in the word sequence selected by the discrimination section that is not involved in the calculation of the first evaluation value.

摘要翻译： 词汇获取装置包括：音素识别部分2，用于从输入的语音中准备音素序列候选; 字符匹配部分3，用于基于音素序列候选来准备多个字序列; 鉴别部分4，用于从多个单词序列中选择识别结果中具有高可能性的单词序列; 获取部分5，用于基于由识别部分4选择的单词序列获取新单词; 用于教授名称的教学单词表4A; 以及教学词和未知词的概率模型4B，其中鉴别部分4针对每个单词序列计算第一评估值，其显示单词序列中多少单词​​对应于列表4A中的教学单词和第二评估 表示单词序列中的单词彼此相邻的概率的值，并且选择第一评价值和第二评价值的和为最大的单词序列，并且其中，获取单元5获取新的 字，由歧视部分选择的字序列中不涉及第一评估值的计算的单词。

公开(公告)号：US08493303B2

公开(公告)日：2013-07-23

申请号：US12213968

申请日：2008-06-26

申请人： Hirobumi Furihata ,  Takashi Nose

发明人： Hirobumi Furihata ,  Takashi Nose

IPC分类号： G09G3/36 ,  G09G3/28 ,  G09G5/02

CPC分类号： G09G3/3685 ,  G09G2310/027 ,  G09G2320/0673

摘要： A control driver for a liquid crystal display panel includes: an operation circuit, an LUT (Look-up Table), and a linear interpolation D/A converter. The operation circuit performs a certain operation on input image data to generate operation data, and outputs higher order bit data and lower order bit data of the operation data. The LUT includes a V-T (Voltage-Transmittance) characteristic of the liquid crystal display panel, and outputs first output data and second output data as display data based on the higher order bit data and the V-T characteristic. The linear interpolation D/A converter performs an linear interpolation operation and D/A conversion to generate output voltage supplied to the liquid crystal display panel in response to the first output data, the second output data and the lower order bit data.