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公开(公告)号：US07193092B2
公开(公告)日：2007-03-20
申请号：US10643552
申请日：2003-08-19
申请人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
发明人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
IPC分类号： C07F7/08 , C07F7/18 , C07F9/6553
CPC分类号： C07D497/04 , C07B2200/07 , C07C209/52 , C07C231/18 , C07F9/65515 , C07C211/48 , C07C233/05
摘要： The present invention relates to chiral diphosphorus compounds and their transition metal complexes, to a process for preparing chiral diphosphorus compounds and their transition metal complexes and also to their use in asymmetric syntheses.
摘要翻译： 本发明涉及手性二磷化合物及其过渡金属络合物，涉及制备手性二磷化合物及其过渡金属配合物的方法，以及它们在不对称合成中的用途。
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公开(公告)号：US07057061B2
公开(公告)日：2006-06-06
申请号：US10256700
申请日：2002-09-27
申请人： Claus Dreisbach , Benjamin Meseguer , Thomas Prinz , Ulrich Scholz , Hans-Christian Militzer , Friederike Agel , Birgit Drieβen-Hölscher
发明人： Claus Dreisbach , Benjamin Meseguer , Thomas Prinz , Ulrich Scholz , Hans-Christian Militzer , Friederike Agel , Birgit Drieβen-Hölscher
IPC分类号： C07F9/655
CPC分类号： C07F9/65744 , B01J31/185 , B01J2231/4261 , B01J2231/643 , B01J2231/645 , B01J2531/822 , C07B53/00 , C07B2200/07 , C07C45/505 , C07C67/303 , C07C231/12 , C07C231/18 , C07F9/6571 , C07F9/657154 , C07F9/65719 , C07C69/34 , C07C233/47
摘要： The present invention relates to catalysts comprising chiral monophosphorus compounds and their use, the chiral monophosphorus compounds themselves and also their precursors.
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13.发明授权Method of preserving materials using 4-methylene-2-amino-cyclopentane-1-carboxylic acids 失效使用4-亚甲基-2-氨基 - 环戊烷-1-羧酸保存材料的方法
公开(公告)号：US5770622A
公开(公告)日：1998-06-23
申请号：US709073
申请日：1996-09-06
申请人： Joachim Mittendorf , Franz Kunisch , Michael Matzke , Hans-Christian Militzer , Rainer Endermann , Karl Georg Metzger , Klaus-Dieter Bremm , Manfred Plempel
发明人： Joachim Mittendorf , Franz Kunisch , Michael Matzke , Hans-Christian Militzer , Rainer Endermann , Karl Georg Metzger , Klaus-Dieter Bremm , Manfred Plempel
IPC分类号： C07C61/15 , C07C61/20 , C07C61/35 , C07C61/39 , C07C61/40 , C07C69/74 , C07C69/753 , C07C69/757 , C07C229/48 , C07C237/04 , C07C251/42 , C07C271/22 , C07C271/24 , C07C271/34 , C07C271/36 , C07D265/12 , C07D307/93 , A01N37/00
CPC分类号： C07C251/42 , C07C229/48 , C07C237/04 , C07C271/22 , C07C271/24 , C07C271/34 , C07C271/36 , C07C61/15 , C07C61/20 , C07C61/35 , C07C61/39 , C07C61/40 , C07C69/74 , C07C69/753 , C07C69/757 , C07D265/12 , C07D307/93 , C07C2101/08 , C07C2101/10 , C07C2103/18
摘要： The invention relates to cyclopentane- and -pentene-.beta.-amino acids, processes for their preparation and their use as medicaments, and to prevent contamination of materials such as wood and leather.
摘要翻译： 本发明涉及环戊烷和戊烯-β-氨基酸，其制备方法及其作为药物的用途，并且防止木材和皮革等材料的污染。
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公开(公告)号：US08653074B2
公开(公告)日：2014-02-18
申请号：US13291271
申请日：2011-11-08
申请人： Hans-Christian Militzer , Jörg Gries , Stefan Koep
发明人： Hans-Christian Militzer , Jörg Gries , Stefan Koep
IPC分类号： A61K31/5377 , C07D413/14
CPC分类号： C07D403/14 , A61K31/5377 , A61K45/06
摘要： The present application relates to sodium 1-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-(1H-1,2,3-triazol-1-yl)-1H-pyrazol-5-olate, to processes for its preparation, to its use for the treatment and/or prophylaxis of diseases and to its use for the preparation of medicaments for the treatment and/or prophylaxis of diseases, in particular cardiovascular and haematological diseases and kidney diseases, and for promoting wound healing.
摘要翻译： 本申请涉及1- [6-（吗啉-4-基）嘧啶-4-基] -4-（1H-1,2,3-三唑-1-基）-1H-吡唑-5-醇酸钠 ，其制备方法，其用于治疗和/或预防疾病及其用于制备用于治疗和/或预防疾病，特别是心血管和血液病和肾脏疾病的药物的用途，以及用于 促进伤口愈合。
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公开(公告)号：US08293899B2
公开(公告)日：2012-10-23
申请号：US10375344
申请日：2003-02-27
IPC分类号： C07D333/36 , C07D221/06 , C07D277/56 , C07D475/02 , C07D233/44
CPC分类号： C07D333/62 , C07D213/55 , C07D213/56 , C07D213/61 , C07D307/54 , C07D333/24 , C07D333/60
摘要： The present invention relates to a process for preparing stereoisomerically enriched 3-heteroaryl-3-hydroxycarboxylic esters by reducing 3-heteroaryl-3-oxocarboxylic esters in the presence of ruthenium-containing catalysts.
摘要翻译： 本发明涉及通过在含钌催化剂存在下还原3-杂芳基-3-氧代羧酸酯制备立体异构体富集的3-杂芳基-3-羟基羧酸酯的方法。
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16.发明授权Process for stereoselectively reducing 4-aryl-4-oxobutanoic acid derivatives 失效立体选择性还原4-芳基-4-氧代丁酸衍生物的方法公开(公告)号：US07329766B2
公开(公告)日：2008-02-12
申请号：US11153053
申请日：2005-06-15
IPC分类号： C07D409/00 , C07D307/02 , C07D407/00
CPC分类号： C07D307/33 , C07B2200/07 , C07C51/367 , C07C67/31 , C07D333/24 , C07D333/28 , C07D409/04 , C07C69/734 , C07C69/732 , C07C59/48
摘要： The present invention relates to a process for preparing stereoisomerically enriched 4-aryl-4-hydroxybutanoic acid derivatives by reducing 4-aryl-4-ketobutanoic acid derivatives in the presence of ruthenium-containing catalysts.
摘要翻译： 本发明涉及通过在含钌催化剂存在下还原4-芳基-4-酮丁酸衍生物制备立体异构体富集的4-芳基-4-羟基丁酸衍生物的方法。
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公开(公告)号：US20070155971A1
公开(公告)日：2007-07-05
申请号：US11707710
申请日：2007-02-16
申请人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
发明人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
IPC分类号： C07F15/00
CPC分类号： C07D497/04 , C07B2200/07 , C07C209/52 , C07C231/18 , C07F9/65515 , C07C211/48 , C07C233/05
摘要： The present invention relates to chiral diphosphorus compounds and their transition metal complexes, to a process for preparing chiral diphosphorus compounds and their transition metal complexes and also to their use in asymmetric syntheses.
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公开(公告)号：US20050154205A1
公开(公告)日：2005-07-14
申请号：US11076757
申请日：2005-03-10
IPC分类号： C07D233/10 , C07B61/00 , C07C1/32 , C07C2/88 , C07C15/14 , C07C17/263 , C07C22/08 , C07C41/30 , C07C45/68 , C07C49/84 , C07D233/04 , C07D233/54 , C07F15/00 , C07F15/04
CPC分类号： C07D233/56 , C07C1/321 , C07C2531/22 , C07D233/04 , C07F15/006 , C07F15/0086 , C07F15/04 , C07C15/14
摘要： The present invention relates to a process for preparing polyaryl compounds by coupling aryl halides or aryl sulphonates and reactive aryl compounds in the presence of novel transition metal complexes of N-heterocyclic carbenes which, just like the N-heterocyclic carbenes themselves and the salts from which they are derived, form part of the invention.
摘要翻译： 本发明涉及在N-杂环卡宾的新型过渡金属络合物存在下偶合芳基卤化物或芳基磺酸盐和反应性芳基化合物来制备聚芳基化合物的方法，其正如N-杂环卡宾本身及其盐 它们是衍生的，构成本发明的一部分。
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公开(公告)号：US20050080047A1
公开(公告)日：2005-04-14
申请号：US10643552
申请日：2003-08-19
申请人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
发明人： Benjamin Meseguer , Hans-Christian Militzer , Sergio Castillon , Carmen Claver , Yolanda Diaz , Mohamed Aghmiz , Ester Guiu , Ali Aghmiz , Anna Masdeu
IPC分类号： B01J31/24 , C07B53/00 , C07B61/00 , C07C67/303 , C07C69/34 , C07C209/52 , C07C211/48 , C07C231/12 , C07C231/18 , C07C233/05 , C07C233/47 , C07D497/04 , C07F7/18 , C07F9/655 , C07F9/6571 , C07F15/00 , C07F19/00 , A61K31/695 , A61K31/665 , C07F7/02
CPC分类号： C07D497/04 , C07B2200/07 , C07C209/52 , C07C231/18 , C07F9/65515 , C07C211/48 , C07C233/05
摘要： The present invention relates to chiral diphosphorus compounds and their transition metal complexes, to a process for preparing chiral diphosphorus compounds and their transition metal complexes and also to their use in asymmetric syntheses.
摘要翻译： 本发明涉及手性二磷化合物及其过渡金属络合物，涉及制备手性二磷化合物及其过渡金属络合物的方法，以及它们在不对称合成中的用途。
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20.发明申请Polyamino acid-catalyzed process for the enantioselective epoxidation of alpha,beta-unsaturated enones and alpha,beta-unsaturated sulfones 失效用于α，β-不饱和烯酮和α，β-不饱和砜的对映选择性环氧化的聚氨基酸催化方法公开(公告)号：US20050027131A1
公开(公告)日：2005-02-03
申请号：US10926458
申请日：2004-08-25
IPC分类号： C07D301/12 , C07B61/00 , C07D301/03 , C07D303/32 , C07D303/48 , C07D301/06
CPC分类号： C07D303/32 , C07B2200/07 , C07D303/48
摘要： The invention relates to a novel process that makes it possible to epoxidize α,β-unsaturated enones or α,β-unsaturated sulfones with high conversions and enantiomeric excesses in a two-phase system without addition of water in the presence of an organic solvent, a base, an oxidant, a diastereomer- and enantiomer-enriched homo-polyamino acid that has not been separately preactivated as catalyst, and a specific phase-transfer catalyst as cocatalyst.
摘要翻译： 本发明涉及一种新的方法，其可以在有机溶剂的存在下在不加水的情况下在两相体系中以高转化率和对映体过量进行环氧化的α，β-不饱和烯酮或α，β-不饱和砜， 没有单独预活化作为催化剂的碱，氧化剂，非对映异构体和对映体富集的均聚氨基酸，以及作为助催化剂的特定相转移催化剂。
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