Benzylamine analogues
    43.
    发明授权
    Benzylamine analogues 失效
    苄胺类似物

    公开(公告)号:US07504393B2

    公开(公告)日:2009-03-17

    申请号:US11583404

    申请日:2006-10-19

    摘要: A compound of the formula (I): wherein R1 is a C1-C6 alkyl group, an amino group, a (C1-C6 alkyl)amino group, a di(C1-C6 alkyl)amino group or a nitrogen-containing saturated heterocyclic group; R3 is a hydrogen atom or a C1-C6 alkyl group; Arom is an unsubstituted or substituted aryl group or an unsubstituted or substituted heteroaryl group; wherein the substituted aryl group is substituted at 1 to 5 positions and the substituted heteroaryl group is substituted at 1 to 3 positions; and wherein the substituents of the aryl group and of the heteroaryl group are independently selected from the group consisting of halogen atom, C1-C6 alkyl, halogeno C1-C6 alkyl, C1-C6 alkoxy, C1-C6 alkylthio, C1-C3 alkylenedioxy, C1-C7 alkanoyl, C2-C7 alkyloxycarbonyl, amino, C1-C7 alkanoylamino, hydroxyl, mercapto, cyano, nitro and carboxyl; A is a C1-C6 alkylene group; Ra together with R2 is a C2-C3 alkylene group containing a double bond; E is a single bond, an oxygen atom, a sulfur atom or a group of the formula: —NR4—, wherein R4 is a hydrogen atom or a C1-C7 alkanoyl group; X1 and X2 are the same or different and are an oxygen atom or a sulfur atom, or a pharmacologically acceptable salt or ester thereof.

    摘要翻译: 式(I)的化合物:其中R1是C1-C6烷基,氨基,(C1-C6烷基)氨基,二(C1-C6烷基)氨基或含氮饱和杂环 组; R3是氢原子或C1-C6烷基; Arom是未取代或取代的芳基或未取代或取代的杂芳基; 其中取代的芳基在1至5个位置被取代,取代的杂芳基在1至3个位置被取代; 并且其中芳基和杂芳基的取代基独立地选自卤素原子,C 1 -C 6烷基,卤代C 1 -C 6烷基,C 1 -C 6烷氧基,C 1 -C 6烷硫基,C 1 -C 3亚烷基二氧基, C 1 -C 7烷酰基,C 2 -C 7烷氧基羰基,氨基,C 1 -C 7烷酰氨基,羟基,巯基,氰基,硝基和羧基; A是C1-C6亚烷基; R a与R 2一起是含有双键的C 2 -C 3亚烷基; E是单键,氧原子,硫原子或式-NR4-基团,其中R4是氢原子或C1-C7烷酰基; X1和X2相同或不同,为氧原子或硫原子,或其药理学上可接受的盐或酯。

    Cylinder liner and cylinder block
    44.
    发明授权
    Cylinder liner and cylinder block 有权
    气缸套和气缸体

    公开(公告)号:US07273029B2

    公开(公告)日:2007-09-25

    申请号:US11330338

    申请日:2006-01-12

    IPC分类号: F02F1/00

    CPC分类号: F02F1/004 F02F1/18

    摘要: A cast iron cylinder liner of the present invention includes a plurality of grooves formed on an outer surface of the cylinder liner. Each of the grooves extends in a circumferential direction of the cylinder liner in a ring or spiral shape, and the grooves divide the outer surface of the cylinder liner into a plurality of ring or spiral sections. The outer surfaces of the ring sections have a uniform distance from the central axis of the cylinder liner over the entire area of the outer surfaces, and the grooves being arranged symmetrically with respect to the center of the cylinder liner in an axial direction thereof. Each of the grooves has a J-shaped longitudinal cross-section including a first inclination part and a groove bottom part. The first inclination part extends from the outer surface of one of the ring sections or of one turn of the spiral sections toward the center of the cylinder liner in an axial direction thereof. The groove bottom part has a longitudinal cross-section approximately in the form of a circular arc, and extends from the first inclination part in a direction away from the center of the cylinder liner in an axial direction thereof.

    摘要翻译: 本发明的铸铁气缸套包括形成在气缸套的外表面上的多个槽。 每个凹槽在气缸套的圆周方向上以环形或螺旋形状延伸,并且凹槽将气缸套的外表面分成多个环形或螺旋形部分。 环形部分的外表面在外表面的整个区域上与气缸套的中心轴线具有均匀的距离,并且凹槽相对于气缸套的中心在其轴向方向上对称地布置。 每个凹槽具有包括第一倾斜部分和凹槽底部部分的J形纵向横截面。 第一倾斜部分从环形部分中的一个的外表面或螺旋部分的一匝沿其轴向朝向气缸套的中心延伸。 槽底部具有大致呈圆弧形状的纵向截面,并且沿着其轴向方向从气缸套的中心沿远离中心的方向从第一倾斜部延伸。

    High-strength steel sheet suitable for deep drawing and process for
producing the same
    46.
    发明授权
    High-strength steel sheet suitable for deep drawing and process for producing the same 失效
    适用于深冲的高强度钢板及其制造方法

    公开(公告)号:US5618355A

    公开(公告)日:1997-04-08

    申请号:US556962

    申请日:1995-12-12

    摘要: A high-strength steel sheet suitable for deep drawing, characterized by comprising 0.04 to 0.25 mass % of C and 0.3 to 3.0 mass %, in total, of at least one of Si and Al, the steel sheet having multiple phases structure comprising ferrite as a main phase (a phase having the highest volume fraction), not less than 3 vol. % of austenite, and bainite and martensite; said steel satisfying a requirement that a value obtained by dividing volume fraction of Vg (vol. %) of austenite before working by the content of C (mass %) contained in the whole steel, Vg/C, is 40 to 140, a requirement that Vp (volume fraction of austenite at the time of plane strain tensile deformation)/Vs (volume fraction of austenite at the time of shrink flanging deformation) is not more than 0.8, and a requirement represented by the formula220

    摘要翻译: PCT No.PCT / JP95 / 00832 Sec。 371 1995年12月12日第 102(e)日期1995年12月12日PCT 1995年4月26日PCT PCT。 WO95 / 29268 PCT出版物 日期:1995年11月2日适用于深拉深的高强度钢板,其特征在于,含有0.04〜0.25质量%的C和0.3〜3.0质量%的Si和Al中的至少一种,所述钢板具有多个 包含铁素体作为主相(具有最高体积分数的相),不小于3体积%的相结构。 %的奥氏体,贝氏体和马氏体; 所述钢满足以下要求:通过将在整个钢中含有的C(质量%)的含量Vg / C,将工作前奥氏体的Vg(体积%)的体积分数除以40〜140, Vp(平面应变拉伸变形时的奥氏体的体积分数)/ Vs(收缩凸缘变形时的奥氏体的体积分率)为0.8以下,由式220表示的要求

    Radio receiver for locating the strongest signal carrying a selected
program
    47.
    发明授权
    Radio receiver for locating the strongest signal carrying a selected program 失效
    用于定位携带选定节目的最强信号的无线电接收机

    公开(公告)号:US5493711A

    公开(公告)日:1996-02-20

    申请号:US152840

    申请日:1993-11-15

    申请人: Kazuo Koyama

    发明人: Kazuo Koyama

    IPC分类号: H03J7/18 H04B1/06 H04B1/10

    摘要: A receiver has a random counter, which outputs a timer signal to a control circuit. A zero-cross point detection circuit generates a detection signal which is input to the control circuit. When the random counter outputs a timer signal and the zero-cross detection circuit detects a zero-cross point, a muting function is activated. Simultaneously, different frequencies are scanned for broadcasts containing the same program and having higher field strengths. If on re-checking zero-cross point detection, a zero-cross point is found or a predetermined interval has expired, then the muting function is deactivated. The frequency with the greater field strength is selected.

    摘要翻译: 接收机具有随机计数器,其将定时器信号输出到控制电路。 零交叉点检测电路产生输入到控制电路的检测信号。 当随机计数器输出定时器信号并且过零检测电路检测到零交叉点时,静音功能被激活。 同时,对包含相同程序并具有较高场强的广播扫描不同的频率。 如果重新检查过零点检测,则发现零交叉点或预定间隔已过期,则静音功能被停用。 选择具有较大场强的频率。

    Process for producing hot-rolled steel sheet having high r value
    49.
    发明授权
    Process for producing hot-rolled steel sheet having high r value 失效
    具有高,高值的热轧钢板的制造方法

    公开(公告)号:US4769088A

    公开(公告)日:1988-09-06

    申请号:US11824

    申请日:1987-02-06

    摘要: An r value of a hot-rolled steel sheet is enhanced by: a specific composition consisting of not more than 0.015 wt % of C, from 1.0 to 2.5 wt % of Mn, from 0.005 to 0.10 wt % of Al, from 0.01 to 0.06 wt % of Nb, from 0.01 to 0.1 wt % of Ti; and, controlled rolling, characterized by in the rough rolling, imparting, in a temperature range of from 980.degree. to 1100.degree. C., a heavy reduction of not less than 20% per pass to the steel sheet; completing a finishing rolling at from Ar.sub.3 to 930.degree. C. and maintaining a total reduction at a temperature of not more than Ar.sub.3 +150.degree. C. to not less than 90%; and, coiling at a temperature of from 600.degree. to 800.degree. C.

    摘要翻译: 通过以下方式提高热轧钢板的上下限值:由不大于0.015重量%的C,1.0〜2.5重量%的Mn,0.005〜0.10重量%的Al,0.01〜 0.06重量%的Nb,0.01〜0.1重量%的Ti; 并进行轧制,其特征在于粗轧,在980℃〜1100℃的温度范围内,每次通过钢板的重量减少20%以上; 完成从Ar3到930℃的精轧,并且在不高于Ar3 + 150℃的温度下保持总的还原至不低于90%; 并在600〜800℃的温度下卷取。

    Apparatus for packaging, weighing and labeling merchandise
    50.
    发明授权
    Apparatus for packaging, weighing and labeling merchandise 失效
    用于包装,称重和标签商品的设备

    公开(公告)号:US4578926A

    公开(公告)日:1986-04-01

    申请号:US584397

    申请日:1984-02-27

    摘要: Merchandise discharged from a packaging machine in a lateral posture can be reliably aligned into a longitudinal posture, and the merchandise can then be sent to a labeling machine with one side of each article in sliding contact with an article-aligning member at all times, irrespective of the size of tray used. This enables the omission of the operations of correcting the posture and position of articles by an operator, and the articles can always be labeled at correct portions thereof, said turn conveyor is so formed that the height of a start end thereof can be regulated to enable the turn conveyor, alignment conveyor, weighing machine and labeling machine to be connected to a packaging machine which has an article discharge section at a height different from that of the turn conveyor or an intermediate conveyor connected to the discharge section of the packaging machine.

    摘要翻译: 从侧面姿势的包装机排出的商品能够可靠地对准纵向姿势,然后可以将商品发送到贴标机,每个物品的一侧始终与物品对齐部件滑动接触,不管 的托盘使用大小。 这样可以省略由操作人员修正物品的姿势和位置的操作,并且物品可以总是在其正确的部分被标记,所述转动输送机被形成为可以调节其起始端的高度,以使得能够 转盘式输送机,定位输送机,称重机和贴标机连接到包装机上,该包装机具有与转盘输送机不同的高度的物品排出部分或连接到包装机的排出部分的中间输送机。