6-Piperazinyl-3,4-dihydroquinazolin-2(1H)-ones
    51.
    发明授权
    6-Piperazinyl-3,4-dihydroquinazolin-2(1H)-ones 有权
    6-哌嗪基-3,4-二氢喹唑啉-2(1H) - 酮

    公开(公告)号:US09205087B1

    公开(公告)日:2015-12-08

    申请号:US14848058

    申请日:2015-09-08

    Inventor: Nisar Ullah

    CPC classification number: A61K31/517 A01N43/54 C07D239/80 C07D401/12

    Abstract: A series of new 6-piperazinyl-3,4-dihydroquinazolin-2(1H)-ones have been synthesized. The compounds are structurally related to adoprazine, a potential atypical antipsychotics bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties. Buchwald-Hartwig coupling of suitably modified aryl bromides with tert-butyl piperazine-1-carboxylate afforded the advanced intermediate piperazinyl-3,4-dihydroquinazolin-2(1H)-one. The reductive amination of the latter with appropriately designed biarylaldehydes accomplished the synthesis of these compounds.

    Abstract translation: 已经合成了一系列新的6-哌嗪基-3,4-二氢喹唑啉-2(1H) - 酮。 这些化合物在结构上与具有强力D2受体拮抗剂和5-HT1A受体激动剂特性的潜在非典型抗精神病药的阿扑
    肼有关。 适当改性的芳基溴与哌嗪-1-羧酸叔丁酯的Buchwald-Hartwig偶联得到高级中间体哌嗪基-3,4-二氢喹唑啉-2(1H) - 酮。 后者与适当设计的二芳基醛的还原胺化完成了这些化合物的合成。

    METHOD FOR FORMING CHALCOGENIDE LAYERS
    53.
    发明申请
    METHOD FOR FORMING CHALCOGENIDE LAYERS 审中-公开
    形成混合层的方法

    公开(公告)号:US20150340525A1

    公开(公告)日:2015-11-26

    申请号:US14697344

    申请日:2015-04-27

    Inventor: Souhaib Oueslati

    Abstract: A method is provided for forming on a substrate a chalcogenide layer, the chalcogenide layer containing at least two metallic elements and containing Se. The method comprises depositing on the substrate a metallic layer containing the at least two metallic elements; and annealing the metallic layer in an environment comprising both a S-containing vapor such as H2S vapor and a Se-containing vapor such as H2Se vapor, thereby forming the chalcogenide layer. The annealing may for example be done at a temperature in the range between 450° C. and 550° C., resulting in a layer with good morphological quality and large grain size, the layer being free of S. A method of the various embodiments may for example be used for forming an absorber layer of a photovoltaic cell.

    Abstract translation: 提供了一种在衬底上形成硫族化物层的方法,硫族化物层含有至少两种金属元素并含有Se。 该方法包括在基底上沉积含有至少两种金属元素的金属层; 并且在包含含S蒸气如H 2 S蒸气和含Se蒸汽如H 2 Se蒸气的环境中退火金属层,从而形成硫族化物层。 退火可以例如在450℃至550℃的范围内的温度下进行,导致具有良好形态质量和较大晶粒尺寸的层,该层不含S。各种实施方案的方法 可以例如用于形成光伏电池的吸收层。

    Structured control instruction fetch unit
    55.
    发明授权
    Structured control instruction fetch unit 有权
    结构化控制指令提取单元

    公开(公告)号:US09170811B2

    公开(公告)日:2015-10-27

    申请号:US13737894

    申请日:2013-01-09

    Abstract: The structured control instruction fetch unit is a structured instruction stream controller that processes expand (XP), expand register indirect (XPR), loop (LOOP), and break (BRK) instructions for structured control. The fetch unit processes stop bits that mark the end of instruction blocks. Any instruction can be marked with a stop bit to indicate that it is the last one in an instruction block. All instructions are encoded with a predicate to reduce the use of control instructions and to simplify the control. A control stack guides instruction fetching by storing return addresses, loop block addresses, loop predicates, and loop counters. Control instructions and stop bits manage operation of the control stack. An instruction unit feeds execution units and includes a set-associative instruction cache, a control stack, an instruction buffer that decouples instruction fetching from execution, instruction decoders, and program counter (PC) control logic.

    Abstract translation: 结构化控制指令提取单元是结构化指令流控制器,其处理用于结构化控制的扩展(XP),扩展寄存器间接(XPR),循环(LOOP)和中断(BRK)指令。 提取单元处理停止标记指令块结束的位。 任何指令都可以用停止位来标记,表示它是指令块中的最后一个指令。 所有指令都用谓词进行编码,以减少控制指令的使用并简化控制。 控制堆栈通过存储返回地址,循环块地址,循环谓词和循环计数器来指导读取指令。 控制指令和停止位管理控制堆栈的操作。 指令单元馈送执行单元,并且包括集合关联指令高速缓存,控制堆栈,将执行指令取出分离的指令缓冲器,指令解码器和程序计数器(PC)控制逻辑。

    SYSTEM OF SUPPORT THRUST FROM WASTED EXHAUST
    56.
    发明申请
    SYSTEM OF SUPPORT THRUST FROM WASTED EXHAUST 有权
    支持系统从废气排除

    公开(公告)号:US20150300292A1

    公开(公告)日:2015-10-22

    申请号:US14789150

    申请日:2015-07-01

    Inventor: Omair M. ALHATIM

    CPC classification number: F02K1/30 F02K1/28 F02K1/46

    Abstract: Systems and methods for influencing thrust of a gas turbine engine are disclosed. A system includes a plurality of pipes positioned at an exhaust nozzle of the gas turbine engine. Each one of the plurality of pipes includes: an inlet inside the exhaust nozzle; an outlet inside the exhaust nozzle; and an intermediate portion outside the exhaust nozzle.

    Abstract translation: 公开了用于影响燃气涡轮发动机的推力的系统和方法。 系统包括位于燃气涡轮发动机的排气喷嘴处的多个管。 多个管中的每一个包括:排气喷嘴内的入口; 排气喷嘴内部的出口; 和排气喷嘴外侧的中间部。

    UML model integration and refactoring method
    58.
    发明授权
    UML model integration and refactoring method 有权
    UML模型集成和重构方法

    公开(公告)号:US09158503B2

    公开(公告)日:2015-10-13

    申请号:US14049112

    申请日:2013-10-08

    CPC classification number: G06F8/20 G06F8/72

    Abstract: The UML model integration and refactoring method steps include extending the metamodels, composing an integrated UML model derived from the extended metamodels, defining refactoring opportunities and transformation operations during the integrated UML composition, and applying a set of composite refactorings to remove an identified smell from the integrated UML model.

    Abstract translation: UML模型集成和重构方法步骤包括扩展元模型,构建从扩展元模型导出的集成UML模型,在集成UML组合期间定义重构机会和转换操作,以及应用一组复合重构以从 集成UML模型。

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