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    Process for the preparation of nitroguanidine derivatives
    53.
    发明授权
    Process for the preparation of nitroguanidine derivatives 失效
    制备硝基胍衍生物的方法

    公开(公告)号：US5245040A

    公开(公告)日：1993-09-14

    申请号：US777856

    申请日：1991-10-16

    申请人： Peter Maienfisch ,  Odd Kristiansen ,  Laurenz Gsell

    发明人： Peter Maienfisch ,  Odd Kristiansen ,  Laurenz Gsell

    IPC分类号： C07C277/00 ,  C07C279/32 ,  C07C279/36 ,  C07C323/44 ,  C07D213/36 ,  C07D213/40 ,  C07D213/61 ,  C07D213/89 ,  C07D233/64 ,  C07D239/26 ,  C07D251/08 ,  C07D261/08 ,  C07D263/32 ,  C07D265/06 ,  C07D265/30 ,  C07D265/32 ,  C07D271/04 ,  C07D271/06 ,  C07D271/08 ,  C07D273/00 ,  C07D273/04 ,  C07D277/20 ,  C07D277/32 ,  C07D279/06 ,  C07D279/12 ,  C07D285/00 ,  C07D285/18 ,  C07D285/34 ,  C07D307/52 ,  C07D333/20 ,  C07D401/06 ,  C07D401/14 ,  C07D417/06 ,  C07D471/04 ,  C07D498/04 ,  C07D513/04

    CPC分类号： C07D213/40 ,  C07C279/36 ,  C07D213/61 ,  C07D213/89 ,  C07D251/08 ,  C07D277/32 ,  C07D401/06 ,  C07D401/14 ,  C07D417/06

    摘要： A process for the preparation of 1,3-disubstituted 2-nitroguanidines of the formula I ##STR1## in which R.sub.1 is hydrogen or C.sub.1 -C.sub.4 alkyl, R.sub.2 is hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl or a radical --CH.sub.2 B; A is an unsubstituted or mono- to tetrasubstituted aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, which may contain one or two substituents from the group comprising C.sub.1 -C.sub.3 haloalkyl having 1 to 7 halogen atoms, cyclopropyl, halocyclopropyl having 1 to 3 halogen atoms, C.sub.2 -C.sub.3 alkenyl, C.sub.2 -C.sub.3 alkynyl, C.sub.2 -C.sub.3 haloalkenyl and C.sub.2 -C.sub.3 haloalkynyl having 1 to 4 halogen atoms, C.sub.1 -C.sub.3 haloalkoxy having 1 to 7 halogen atoms, C.sub.1 -C.sub.3 alkylthio, C.sub.1 -C.sub.3 haloalkylthio having 1 to 7 halogen atoms, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro and one to four substituents from the group comprising C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy and halogen; and B is optionally substituted phenyl or pyridyl, which comprises hydrolysing a compound of the formula II ##STR2## in which R.sub.3 is unsubstituted or substituted C.sub.1 -C.sub.10 alkyl, C.sub.3 -C.sub.6 cycloalkyl, phenyl or benzyl.The compounds of the formula I are suitable as intermediates for the preparation of pesticides.

    摘要翻译： 制备式I的1,3-二取代2-硝基胍的方法，其中R 1是氢或C 1 -C 4烷基，R 2是氢，C 1 -C 6烷基，C 3 -C 6环烷基或基团-CH 2 B ; A是未取代的或单取代或四取代的芳族或非芳族单环或双环杂环基团，其可以含有一个或两个取代基，该取代基包括具有1至7个卤素原子的C 1 -C 3卤代烷基，环丙基，具有1至3个卤素的卤代环丙基 C 1 -C 3烯基，C 2 -C 3炔基，C 2 -C 3卤代烯基和具有1至4个卤素原子的C 2 -C 3卤代炔基，具有1至7个卤素原子的C 1 -C 3卤代烷氧基，C 1 -C 3烷硫基，具有1至7个卤素原子的C 1 -C 3卤代烷硫基，烯丙氧基， 炔丙氧基，烯丙硫基，炔丙硫基，卤代烯丙氧基，卤代烯硫基，氰基和硝基，以及一至四个取代基，包括C 1 -C 3烷基，C 1 -C 3烷氧基和卤素; 并且B是任选取代的苯基或吡啶基，其包括水解其中R 3为未取代或取代的C 1 -C 10烷基，C 3 -C 6环烷基，苯基或苄基的式II化合物（II）。 式I的化合物适合作为制备农药的中间体。

    Anthelmintics
    54.
    发明授权
    Anthelmintics 失效
    ANTHELMINTICS

    公开(公告)号：US5081125A

    公开(公告)日：1992-01-14

    申请号：US586176

    申请日：1990-09-19

    申请人： Peter Maienfisch ,  Christor Hildenbrand ,  Jean-Claude Gehret

    发明人： Peter Maienfisch ,  Christor Hildenbrand ,  Jean-Claude Gehret

    IPC分类号： A23K1/16 ,  A61K31/44 ,  A61K31/4402 ,  A61K31/4418 ,  A61K31/505 ,  A61P33/00 ,  C07D213/64 ,  C07D213/643 ,  C07D213/70 ,  C07D213/84 ,  C07D213/85 ,  C07D239/34 ,  C07D239/38 ,  C07D239/56

    CPC分类号： C07D213/643 ,  C07D213/85 ,  C07D239/34 ,  C07D239/38

    摘要： Anthelmintically active compounds of formula I are described ##STR1## in which R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 thioalkyl, C.sub.1 -C.sub.2 haloalkyl, nitro, C.sub.1 -C.sub.2 alkoxy, or the group SO.sub.n R in which R is C.sub.1 -C.sub.2 alkyl or phenyl and n is 0, 1 or 2;R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.3 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.4 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.5 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.6 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.7 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, nitro, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.8 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.9 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.10 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio, C.sub.3 -C.sub.6 cycloalkyl or cyano;R.sub.11 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio or C.sub.3 -C.sub.6 cycloalkyl;R.sub.12 is hydrogen or halogen; and Y is .dbd.CH-- or .dbd.N-; including the physiologically tolerable acid additon salts thereof, and also the preparatin and use thereof and novel intermediates.

    摘要翻译： 式Ⅰ的驱虫活性化合物描述为其中R 1是氢，卤素，C 1 -C 2烷基，C 1 -C 2硫代烷基，C 1 -C 2卤代烷基，硝基，C 1 -C 2烷氧基或其中R是C 1 -C 2烷基的基团SO n R或 苯基，n为0,1或2; R 2是氢，卤素，C 1 -C 2烷基，C 1 -C 2卤代烷基，C 1 -C 2卤代烷氧基或C 1 -C 2烷氧基; R3是氢或C1-C2烷基; R4是氢或C1-C2烷基; R5是氢，卤素或C1-C5烷基; R6是氢，卤素或C1-C5烷基; R 7是氢，卤素，C 1 -C 2烷基，硝基，C 1 -C 2卤代烷基，C 1 -C 2卤代烷氧基或C 1 -C 2烷氧基; R 8是氢，卤素，C 1 -C 2烷基，C 1 -C 2卤代烷基，C 1 -C 2卤代烷氧基或C 1 -C 2烷氧基; R 9是氢，卤素，C 1 -C 2烷基，C 1 -C 2卤代烷基，C 1 -C 2卤代烷氧基或C 1 -C 2烷氧基; R 10是氢，卤素，C 1 -C 6烷基，C 1 -C 2卤代烷基，C 1 -C 2烷硫基，C 3 -C 6环烷基或氰基; R 11是氢，卤素，C 1 -C 6烷基，C 1 -C 2卤代烷基，C 1 -C 2烷硫基或C 3 -C 6环烷基; R 12是氢或卤素; 且Y为= CH-或= N-; 包括其生理上可耐受的酸加成盐，以及其制备及其用途和新型中间体。

    Composition for controlling parasites in productive livestock
    55.
    发明授权
    Composition for controlling parasites in productive livestock 失效
    用于控制生产性牲畜中的寄生虫的组成

    公开(公告)号：US4973711A

    公开(公告)日：1990-11-27

    申请号：US380844

    申请日：1989-07-13

    申请人： Peter Maienfisch

    发明人： Peter Maienfisch

    IPC分类号： C07D493/22 ,  A01N43/16 ,  A01N43/90 ,  A61K31/365 ,  A61P33/00 ,  C07H19/01

    CPC分类号： C07H19/01 ,  A01N43/90 ,  Y02P20/55

    摘要： Novel 13-spiro-2'-[tetrahydrofuran]-milbemycins of the formula I ##STR1## in which X represents one of the groups --CH(OR.sub.1)--, --C(.dbd.O)-- or --C(.dbd.N--OH)--;R.sub.1 represents hydrogen or a OH-protecting group;R.sub.2 represents methyl, ethyl, isopropyl or sec.-butyl or the group --C(CH.sub.3).dbd.CH--A in which A represents methyl, ethyl or isopropyl; andR.sub.3 represents hydrogen; C.sub.1 -C.sub.10 -alkyl; C.sub.1 -C.sub.10 -alkyl substituted by at least one substituent selected from the group consisting of halogen, C.sub.1 -C.sub.6 -alkoxy, C.sub.2 -C.sub.6 -alkoxyalkoxy, C.sub.3 -C.sub.9 -alkoxyalkoxyalkoxy, C.sub.1 -C.sub.6 -alkylthio, C.sub.3 -C.sub.7 -cycloalkyl, C.sub.1 -C.sub.3 -alkyl-substituted C.sub.3 -C.sub.7 -cycloalkyl, hydroxy, benzyloxy, C.sub.1 -C.sub.6 -acyl and C.sub.1 -C.sub.6 -acyloxy, it being possible for each of the above-mentioned radicals representing or containing an alkoxy group to be terminally substituted at a terminal alkoxy group by hydroxy, halogen, C.sub.1 -C.sub.6 -acyl or by C.sub.1 -C.sub.6 -acyloxy; C.sub.3 -C.sub.7 -cycloalkyl; C.sub.3 -C.sub.7 -cycloalkyl substituted by at least one substituent selected from the group consisting of halogen and C.sub.1 -C.sub.3 -alkyl; C.sub.3 -C.sub.7 -cycloalkenyl; C.sub.2 -C.sub.10 -alkenyl; C.sub.2 -C.sub.10 -alkynyl; a radical selected from the group consisting of C.sub.2 -C.sub.10 -alkenyl and C.sub.2 -C.sub.10 -alkynyl, which radical is substituted by halogen, C.sub.1 -C.sub.6 -alkoxy or by C.sub.1 -C.sub.6 -acyloxy; 1-adamantylmethyl; menthyl; carveyl; phenyl; benzyl; naphthyl; a radical selected from the group consisting of phenyl, benzyl and naphthyl, which radical is substituted by at least one substituent selected from the group consisting of halogen, C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 -haloalkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.3 -haloalkoxy, C.sub.1 -C.sub.3 -alkylthio, nitro and cyano; benzyl substituted by a phenoxy group; or a four- to six-membered heterocyclic radical that has from one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen and that is unsubstituted or is substituted by at least one substituent selected from the group consisting of halogen, C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 -haloalkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.3 -haloalkoxy, C.sub.1 -C.sub.3 -alkylthio, nitro and cyano, it being possible for the said heterocyclic radical also to be bonded via a C.sub.1 -C.sub.6 -alkylene bridge to the oxygen atom in the 5'-position of the tetrahydrofuran ring,their preparation and their use against parasites in productive livestock and against insect pests, are described.

    Pesticide
    57.
    发明授权
    Pesticide 有权
    农药

    公开(公告)号：US08673813B2

    公开(公告)日：2014-03-18

    申请号：US10801405

    申请日：2004-03-16

    申请人： Robert Senn ,  Peter Maienfisch ,  Peter Wyss

    发明人： Robert Senn ,  Peter Maienfisch ,  Peter Wyss

    IPC分类号： A01N25/26 ,  A01N43/02

    CPC分类号： A01N53/00 ,  A01N43/88 ,  A01N47/40 ,  A01N51/00 ,  A01N43/56 ,  A01N43/40 ,  A01N43/30 ,  A01N2300/00 ,  A01N57/12

    摘要： Composition for controlling insects and representatives of the order Acarina, which comprises a combination of variable amounts of one or more compounds of the formula in which A is an unsubstituted or, depending on the possibility of substitution on the ring system, mono- to tetrasubstituted, aromatic or non-aromatic monocyclic or bicyclic heterocyclic radical, in which the substituents of A can be chosen from the group consisting of C1-C3alkyl, C1-C3alkoxy, halogen, halo-C1-C3alkyl, cyclopropyl, halocyclopropyl, C2-C3alkenyl, C2-C3alkynyl, halo-C2-C3alkenyl, halo-C2-C3alkynyl, halo-C1-C3alkoxy, C1-C3alkylthio, Halo-C1-C3alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro; R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl; and X is N—NO2 or N—CN, in the free form or in salt form, if appropriate tautomers, in the free form or salt form, and one or more of the compounds (I) to (CLXXXIV) mentioned according to the invention and at least one auxiliary. A method of controlling pests, a process for the preparation of the composition, its use and plant propagation material treated with it, and the use of the compound of the formula (A) for the preparation of the composition, are described.

    摘要翻译： 用于控制昆虫的组合物和蜱螨纲的代表，其包含可变量的一种或多种下式的化合物的组合，其中A是未取代的，或者取决于在环系上取代的可能性为单 - 四取代的， 芳基或非芳族单环或双环杂环基，其中A的取代基可以选自C 1 -C 3烷基，C 1 -C 3烷氧基，卤素，卤代-C 1 -C 3烷基，环丙基，卤代环丙基，C 2 -C 3烯基，C 2 C 3炔基，卤代-C 2 -C 3烯基，卤代C 2 -C 3炔基，卤代-C 1 -C 3烷氧基，C 1 -C 3烷硫基，卤代-C 1 -C 3烷硫基，烯丙氧基，炔丙氧基，烯丙硫基，炔丙硫基，卤代烯氧基，卤代烯硫基，氰基和硝基。 R是氢，C 1 -C 6烷基，苯基-C 1 -C 4烷基，C 3 -C 6环烷基，C 2 -C 6烯基或C 2 -C 6炔基; 和X为游离形式或盐形式的N-NO 2或N-CN，如果适当的互变异构体，以游离形式或盐形式，以及根据本发明提及的一种或多种化合物（I）至（CLXXXIV） 发明和至少一种辅助剂。 描述了控制害虫的方法，用它制备组合物，其用途和植物繁殖材料的方法，以及使用式（A）化合物制备组合物。

    "> Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4
    60.
    发明申请
    Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4" Position Having Pesticidal Properties 有权
    在4'和4“位置具有农药性质的阿维菌素和阿维菌素单糖

    公开(公告)号：US20080194498A1

    公开(公告)日：2008-08-14

    申请号：US10568715

    申请日：2004-08-27

    申请人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

    发明人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

    IPC分类号： A01N43/90 ,  C07H17/08 ,  A01P17/00

    CPC分类号： A01N43/90 ,  C07H19/01

    摘要： Described is a compound of the formula (1) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.

    摘要翻译： 描述了式（1）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R 3是例如氢，未取代的或一至五取代的C 1 -C 12烷基，R 4是氢， 是例如一至五取代的C 1 -C 12烷基，未取代或单取代或五取代的C 3 -C 12烷基， 12环烷基; 或（2）X是S，其中R 3是例如氢，未取代的或一至五取代的C 1 -C 12 - 烷基和R 4是例如氢，未取代的或一至五取代的C 1 -C 12烷基; 或（3）X为0或S，其中R 3和R 4一起为例如三至七元亚烷基或四至七元亚烷基， 多元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 C 1 -C 12烷基，一至五取代C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。