NOVEL IMIDAZOLE DERIVATIVES
    64.
    发明申请
    NOVEL IMIDAZOLE DERIVATIVES 审中-公开
    新咪唑衍生物

    公开(公告)号:US20110311649A1

    公开(公告)日:2011-12-22

    申请号:US12739852

    申请日:2008-10-24

    Abstract: The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, hydroxyl, C1-C4alkoxy, OR6, C1-C4haloalkoxy or cyano; R5 is halogen; R6 is hydrogen, C3-C7 cycloalkyl, C3-C10 alkylcycloalkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 haloalkenyl, C3-C7 cycloalkenyl, C2-C6 alkynyl, C2-C6 haloalkynyl or C2-C6 alkyloxyalkyl; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.

    Abstract translation: 本发明涉及式(I)的新咪唑衍生物作为具有杀微生物活性,特别是杀真菌活性的活性成分:其中R1是卤素,C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢,卤素,C1-C4烷基,C1-C4卤代烷基,羟基,C1-C4烷氧基,OR6,C1-C4卤代烷氧基或氰基; R5是卤素; R6是氢,C3-C7环烷基,C3-C10烷基环烷基,C1-C6卤代烷基,C2-C6烯基,C2-C6卤代烯基,C3-C7环烯基,C2-C6炔基,C2-C6卤代炔基或C2-C6烷氧基烷基; X是N或C(R); 且R为氢,卤素,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C(R)时,R 2不能是任选取代的芳基。

    NOVEL PYRIDAZINE DERIVATIVES
    65.
    发明申请
    NOVEL PYRIDAZINE DERIVATIVES 审中-公开
    新的吡咯烷酮衍生物

    公开(公告)号:US20100113457A1

    公开(公告)日:2010-05-06

    申请号:US12447025

    申请日:2007-10-23

    CPC classification number: C07D237/12 A01N43/58 C07D237/14 C07D237/24

    Abstract: The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is halogen, nitro, cyano, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, C1-C4alkylthio or C1-C4haloalkylthio; R3 is an optionally substituted aryl; R4 is fluoro, cyano, C1-C6haloalkyl, C3-C6cycloalkyl, C1-C6haloalkoxy, C1-C6alkylthio or C1-C6haloalkylthio; and n is a whole number from 1 to 4; or an agrochemically usable salt form thereof.

    Abstract translation: 本发明涉及具有杀微生物活性,特别是杀真菌活性的活性成分的式(I)的新哒嗪衍生物,其中R1是氢,C1-C6烷基,C1-C6卤代烷基或C3-C6环烷基; R 2是卤素,硝基,氰基,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 4烷硫基或C 1 -C 4卤代烷硫基; R3是任选取代的芳基; R 4是氟,氰基,C 1 -C 6卤代烷基,C 3 -C 6环烷基,C 1 -C 6卤代烷氧基,C 1 -C 6烷硫基或C 1 -C 6卤代烷硫基; n为1〜4的整数; 或其农业化学上可用的盐形式。

    Pesticidally active ketone and oxime derivatives
    67.
    发明授权
    Pesticidally active ketone and oxime derivatives 失效
    杀虫活性酮和肟衍生物

    公开(公告)号:US07569727B2

    公开(公告)日:2009-08-04

    申请号:US12098594

    申请日:2008-04-07

    Abstract: Compounds of formula wherein A0, A1 and A2 are each independently of the others a bond or a C1-C6alkylene bridge; A3 is a C1-C6alkylene bridge which is unsubstituted or substituted by from one to six identical or different substituents selected from halogen and C3-C8cycloalkyl; Y is, for example, O, S, SO or SO2; M is O or NOR6, X1 and X2 are each independently of the other fluorine, chlorine or bromine; R1, R2 and R3 are, for example, H, halogen, OH, SH, CN, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkylcarbonyl, C2-C6alkenyl, C2-C6haloalkenyl or C2-C6alkynyl; Q is, for example, O, S, SO or SO2; W is, for example, O, S, SO, SO2, —C(═O)—O— or —O—C(═O)—; T is, for example, a bond, O, S, SO, SO2, —C(═O)—O— or —O—C(═O)—; D is CH or N; R4 is, for example, H, halogen, OH, SH, CN, nitro, C1-C6alkyl or C1-C6haloalkyl; R5 is, for example, C1-C12alkyl, C3-C8cycloalkyl or —N(R7)2; R7 is H, C1-C6alkyl, C1-C3haloalkyl, C1-C6alkylcarbonyl, C1-C3haloalkylcarbonyl, C1-C6alkoxycarbonyl, C3-C8cycloalkyl, C3-C8 cycloalkylcarbonyl or formyl; k is 0, 1, 2, 3 or 4; m is 1 or 2; and q is 0, 1 or 2; and, where applicable, their possible E/Z isomers, E/Z isomeric mixtures and/or tautomers, in each case in free form or in salt form, a process for the preparation of those compounds and their use, pesticidal compositions in which the active ingredient has been selected from those compounds and agrochemically acceptable salts thereof, and a process for the preparation of those compositions and their use, to plant propagation material treated with those compositions, and a method of controlling pests.

    Abstract translation: 下式化合物其中A0,A1和A2各自独立地为键或C1-C6亚烷基桥; A3是C1-C6亚烷基桥,其未被取代或被1-6个相同或不同的选自卤素和C 3 -C 8环烷基的取代基取代; Y是例如O,S,SO或SO 2; M为O或NOR6,X1和X2各自独立地为氟,氯或溴; R1,R2和R3是例如H,卤素,OH,SH,CN,硝基,C1-C6烷基,C1-C6卤代烷基,C1-C6烷基羰基,C2-C6链烯基,C2-C6卤代烯基或C2-C6炔基; Q是例如O,S,SO或SO 2; W是例如O,S,SO,SO 2,-C(-O)-O-或-O-C(-O) - ; T是例如键O,S,SO,SO 2,-C(-O)-O-或-O-C(-O) - ; D是CH或N; R4是例如H,卤素,OH,SH,CN,硝基,C1-C6烷基或C1-C6卤代烷基; R5是例如C1-C12烷基,C3-C8环烷基或-N(R7)2; R 7是H,C 1 -C 6烷基,C 1 -C 3卤代烷基,C 1 -C 6烷基羰基,C 1 -C 3卤代烷基羰基,C 1 -C 6烷氧基羰基,C 3 -C 8环烷基,C 3 -C 8环烷基羰基或甲酰基; k为0,1,2,3或4; m为1或2; q为0,1或2; 在适用情况下,它们可能的E / Z异构体,E / Z异构体混合物和/或互变异构体,在每种情况下为游离形式或盐形式,制备这些化合物及其用途的方法,其中 已经从这些化合物和农业化学上可接受的盐中选择活性成分,以及这些组合物的制备方法及其用途,用这些组合物处理的繁殖材料以及控制害虫的方法。

    Pesticidal Heterocyclic Dihaloallyl Compounds
    69.
    发明申请
    Pesticidal Heterocyclic Dihaloallyl Compounds 失效
    杀虫杂环二卤代烯化合物

    公开(公告)号:US20070299064A1

    公开(公告)日:2007-12-27

    申请号:US10597005

    申请日:2005-01-07

    Abstract: The invention relates to compounds of formula wherein Het, A1, A2, A3, A4, D, W, T, Q, Y, X1, X2, R1, R2, R3, R4, k and m are as defined hereinabove, and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, to a process for the preparation of and to the use of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, to pesticidal compositions in which the active ingredient has been selected from those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in agrochemically usable salt form, to a process for the preparation of and to the use of those compositions, to plant propagation material treated with those compositions, to a method of controlling pests, to intermediates and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, for the preparation of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, and to a process for the preparation of and to the use of those intermediates and, where applicable, possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof.

    Abstract translation: 本发明涉及下式的化合物,其中Het,A 1,A 2,A 3,A 4, D,W,T,Q,Y,X 1,X 2,R 1,R 2, R 3,R 4,k和m如上所定义,并且在适用的情况下,可能的E / Z异构体,E / Z异构体和/或互变异构体的混合物 在各种情况下以游离形式或盐形式,涉及制备和使用这些化合物,E / Z异构体,E / Z异构体和/或互变异构体的混合物的方法,其中所述化合物 活性成分选自这些化合物,E / Z异构体,E / Z异构体和/或互变异构体的混合物,在每种情况下以游离形式或以农业化学上可用的盐形式,用于制备和/ 这些组合物,用这些组合物处理的繁殖材料,控制害虫的方法,中间体以及可能的E / Z异构体的E / Z异构体的混合物 其各自为游离形式或盐形式,用于制备这些化合物,E / Z异构体,E / Z异构体和/或互变异构体的混合物,以及制备和/或 使用这些中间体,并且在适用的情况下可能使用E / Z异构体,E / Z异构体和/或其互变异构体的混合物。

    4-(3,3-Dihalo-Allyloxy) Phenoxy Alkyl Derivatives

    公开(公告)号:US20070142445A1

    公开(公告)日:2007-06-21

    申请号:US11675149

    申请日:2007-02-15

    Abstract: Compounds of formula wherein A1, A2 and A3 are each independently of the others a bond or a C1-C6alkylene bridge; A4 is a C1-C6alkylene bridge; D is CH or N; W is, for example, O, NR7 or S; T is, for example, a bond, O, NH or NR7; Q is O, NR7, S, SO or SO2; Y is O, NR7, S, SO or SO2; X1 and X2 are each independently of the other fluorine, chlorine or bromine; R1, R2 and R3 are, for example, H, halogen, CN, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkylcarbonyl or C2-C6alkenyl; R4 is, for example, H, halogen, CN, nitro or C1-C6alkyl; R5 and R6 are, for example, H, CN, OH, C1-C6alkyl, C3-C8cycloalkyl, C3-C8cycloalkyl-C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; R7 is H, C1-C6alkyl, C1-C6alkoxyalkyl or C1-C6alkylcarbonyl; k, when D is nitrogen, is 1, 2 or 3; or, when D is CH, is 1, 2, 3 or 4; and m is 1 or 2; and, where applicable, their possible E/Z isomers, E/Z isomeric mixtures and/or tautomers, in each case in free form or in salt form, a process for the preparation of those compounds and their use, pesticidal compositions in which the active ingredient has been selected from those compounds or an agrochemically acceptable salt thereof, a process for the preparation of those compositions and their use, plant propagation material treated with those compositions, and a method of controlling pests.

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