N-Phenylsulfonyl-N'-pyrimidinylureas
    61.
    发明授权
    N-Phenylsulfonyl-N'-pyrimidinylureas 失效
    N-苯基磺酰基-N'-嘧啶基脲

    公开(公告)号:US4523944A

    公开(公告)日:1985-06-18

    申请号:US571985

    申请日:1984-01-19

    摘要: N-Phenylsulfonyl-N'-pyrimidinyl- and -triazinylureas of the general formula ##STR1## and the salts of these compounds with amines, with alkali or alkaline-earth metal bases or with quaternary ammonium bases, have good pre- and post-emergence selective, herbicidal and growth-regulating properties.The symbols in this formula are as follows:A is a C.sub.3 -C.sub.6 -alkynyl group,E is the methine group or nitrogen,X is oxygen, sulfur or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,m is the number one or two,R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl or C.sub.2 -C.sub.5 -alkenyl or a group --Y--R.sub.5,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.1 -C.sub.4 -haloalkyl, or a group --Y--R.sub.5, --COOR.sub.6, --NO.sub.2 or --CO--NR.sub.7 --R.sub.8,R.sub.3 and R.sub.4 independently of one another are each hydrogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -haloalkoxy, halogen or alkoxyalkyl having at most 4 carbon atoms,R.sub.5 and R.sub.6 are each C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl,R.sub.7 and R.sub.8 independently of one another are each hydrogen, C.sub.1 -C.sub.5 -alkyl, C.sub.2 -C.sub.5 -alkenyl or C.sub.2 -C.sub.6 -alkynyl, andY is oxygen, sulfur or a sulfinyl or sulfonyl bridge.

    摘要翻译: 具有通式(I)的N-苯基磺酰基-N'-嘧啶基 - 和 - 三嗪基脲和这些化合物与胺与碱金属或碱土金属碱或季铵碱的盐具有良好的前和后 芽后选择性,除草和生长调节性质。 该式中的符号如下:A是C 3 -C 6炔基,E是次甲基或氮,X是氧,硫或亚磺酰基或磺酰基桥,Z是氧或硫,m是第一个 或两个,R 1是氢,卤素,C 1 -C 5 - 烷基或C 2 -C 5 - 烯基或基团-Y-R 5,R 2是氢,卤素,C 1 -C 5 - 烷基,C 2 -C 5 - 烯基或C 1 -C 4 - 卤代烷基或基团-Y-R 5,-COOR 6,-NO 2或-CO-NR 7 -R 8,R 3和R 4彼此独立地为氢,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷基,C 1 -C 4卤代烷氧基,卤素或至多4个碳原子的烷氧基烷基,R 5和R 6各自为C 1 -C 5 - 烷基,C 2 -C 5 - 烯基或C 2 -C 6炔基,R 7和R 8 各自独立地为氢,C 1 -C 5 - 烷基,C 2 -C 5 - 烯基或C 2 -C 6 - 炔基,Y为氧,硫或亚磺酰基或磺酰基桥。

    N-Phenyl-substituted N-heterocyclic compounds, their preparation and use
in agents for regulating plant growth
    64.
    发明授权
    N-Phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth 失效
    N-苯基取代的N-杂环化合物,它们的制备和用于调节植物生长的试剂中

    公开(公告)号:US4208202A

    公开(公告)日:1980-06-17

    申请号:US896970

    申请日:1978-04-12

    CPC分类号: C07D213/64 A01N47/02

    摘要: The present invention relates to novel active compounds having a plant growth-inhibiting and herbicidal action and their preparation and to agents containing these active ingredients, and their use.The novel active compounds are saturated and unsaturated 4-membered to 7-membered ring nitrogen heterocyclic compounds which are substituted on the nitrogen atom by a phenyl radical which itself carries a trifluoromethanesulphonamido group --NH--SO.sub.2 --CF.sub.3 as a substituent. The phenyl radical can also carry other substituents and the heterocyclic structure can also be substituted. Oxo derivatives of the heterocyclic compound, in which the oxo group is preferably adjacent to the nitrogen atom, form a preferred sub-group of compounds.

    摘要翻译: 本发明涉及具有植物生长抑制和除草作用的新型活性化合物及其制备方法和含有这些活性成分的试剂及其用途。 新型活性化合物是在氮原子上被本身带有三氟甲磺酰氨基-NH-SO 2 -CF 3作为取代基的苯基取代的饱和和不饱和4元至7元环氮杂环化合物。 苯基也可以携带其它取代基,杂环结构也可以被取代。 其中氧代基​​优选与氮原子相邻的杂环化合物的氧代衍生物形成优选的化合物亚组。

    Herbicides
    66.
    发明授权
    Herbicides 失效
    除草剂

    公开(公告)号:US06204221B1

    公开(公告)日:2001-03-20

    申请号:US09297783

    申请日:1999-05-07

    IPC分类号: A01N4356

    摘要: Compounds of formula (I) in which A is ═N— or (a); W is a group (W1), (W2) or (W3); R11 is hydrogen, fluorine, chlorine, bromine or methyl; and R1 to R5, R13,n1 and n13 are as defined in claim 1, and the pyrazole N-oxydes, agrochemically tolerated salts and stereoisomers of these compounds of formula (I), have good pre- and post-emergent selective herbicidal properties. The preparation of these compounds and their use as herbidical active substances are described.

    摘要翻译: 其中A为= N-或(a)的式(I)化合物; W是组(W1),(W2)或(W3); R11是氢,氟,氯,溴或甲基; 并且R 1至R 5,R 13,n 1和n 13如权利要求1中所定义,并且这些式(I)化合物的吡唑N-氧化物,农业化学耐受的盐和立体异构体具有良好的芽前和芽后选择性除草性质。 描述了这些化合物的制备及其作为草药活性物质的用途。

    Process and a composition for immunizing plants against disease
    67.
    发明授权
    Process and a composition for immunizing plants against disease 失效
    用于免疫植物免疫疾病的方法和组合物

    公开(公告)号:US5523311A

    公开(公告)日:1996-06-04

    申请号:US405488

    申请日:1995-03-14

    摘要: A method and composition for the immunization of healthy useful plants against plant diseases containing as active ingredients compounds of formula ##STR1## in which: X is hydrogen, halogen, hydroxy, methyl, methoxy, HOOC or MOOC; Y is hydrogen, halogen, SO.sub.3 H, SO.sub.3 M, nitro, hydroxy or amino, M being the molar equivalent of an alkali metal or alkaline earth metal ion that is formed from a corresponding base or basic compound; and Z is cyano or --CO--A; A represents either --OH or --SH, the hydrogen atom of which may also be replaced by the molar equivalent of an inorganic or organic cationic residue, or wherein A represents any other organic residue which has a molecular weight of less than 900 and which may also contain one, or more than one, hetero atom, including the salts of the phytophysiologically tolerable 7-carboxylic acid or 7-thiocarboxylic acid with primary, secondary or tertiary amines or with inorganic bases.

    摘要翻译: 用于免疫针对植物疾病的健康有用植物的方法和组合物,其含有作为活性成分的式y-羟基,甲基,甲氧基,HOOC或MOOC的化合物; Y是氢,卤素,SO 3 H,SO 3 M,硝基,羟基或氨基,M是由相应的碱或碱化合物形成的碱金属或碱土金属离子的摩尔当量; 和Z是氰基或-CO-A; A表示-OH或-SH,其氢原子也可被无机或有机阳离子残基的摩尔当量代替,或其中A表示分子量小于900的任何其它有机残基, 还含有一个或多于一个杂原子,包括植物生理学上可耐受的7-羧酸或7-硫代羧酸与伯胺,仲胺或叔胺或与无机碱的盐。

    Pyridylsulfonylureas
    68.
    发明授权
    Pyridylsulfonylureas 失效
    吡啶磺酰脲

    公开(公告)号:US5407900A

    公开(公告)日:1995-04-18

    申请号:US096137

    申请日:1993-07-22

    CPC分类号: C07D521/00 A01N47/36

    摘要: (Cyclopropyl-triazinyl- and cyclopropyl-pyrimidinyl-)pyridylsulfonylureas of formula I ##STR1## wherein R and R.sub.1 are each independently of the other hydrogen or methyl;R.sub.2 is methyl, methoxy or ethoxy; andE is nitrogen or the methine group;and the salts of those compounds, have good selective herbicidal properties. The preparation of those compounds and the use thereof as herbicidal active ingredients are described.

    摘要翻译: (I)的(环丙基 - 三嗪基 - 和环丙基 - 嘧啶基)吡啶磺酰脲其中R和R 1各自独立地为氢或甲基; R2是甲基,甲氧基或乙氧基; E为氮或次甲基; 和这些化合物的盐具有良好的选择性除草性质。 描述了这些化合物的制备及其作为除草活性成分的用途。

    Pyridyl sulfonylurea herbicides
    69.
    发明授权
    Pyridyl sulfonylurea herbicides 失效
    吡啶基磺酰脲除草剂

    公开(公告)号:US5352654A

    公开(公告)日:1994-10-04

    申请号:US530690

    申请日:1990-05-30

    CPC分类号: C07D521/00 A01N47/36

    摘要: N-Pyridinesulfonyl-N'-pyrimidinyl- and -triazinylureas of the formula I ##STR1## in which R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 C.sub.4 haloalkoxy or CF.sub.3 ; R.sub.2 is hydrogen or C.sub.1 -C.sub.4 alkyl; A is C.sub.1 -C.sub.6 alkyl or C.sub.3 -C.sub.6 cycloalkyl, each of which is monosubstituted to trisubstituted by halogen, or is C.sub.1 -C.sub.4 alkyl or C.sub.3 -C.sub.6 cycloalkyl, each of which is substituted by C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkylsulfonyl, C.sub.1 -C.sub.4 alkylsulfinyl, C.sub.2 -C.sub.4 alkenyl, C.sub.5 -C.sub.6 cycloalkenyl, amino, C.sub.1 -C.sub.4 alkylamino, C.sub.1 -C.sub.4 dialkylamino or C.sub.2 -C.sub.4 alkynyl, it being possible for the C.sub.2 -C.sub.4 alkenyl radical and the C.sub.5 -C.sub.6 cycloalkenyl radical to be additionally monosubstituted to trisubstituted by halogen; or A is a 4- to 6-membered saturated heterocycle which contains a hetero atom selected from the group comprising O, N and SO.sub.2 ; or A is C.sub.1 -C.sub.4 alkyl which is substituted by a 4- to 6-membered saturated heterocycle which contains a hetero atom selected from the group comprising O, N and SO.sub.2 ; X is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkyl which is monosubstituted to trisubstituted by halogen, or is C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkoxy which is monosubstituted to trisubstituted by halogen; Y is halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkyl which is monosubstituted to trisubstituted by halogen, or is C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkoxy which is monosubstituted to trisubstituted by halogen, or is cyclopropyl, methylamino or dimethylamino; and E is nitrogen or the methine group, and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases have good selective herbicidal properties pre-emergence and post-emergence, and good growth-regulating properties.

    摘要翻译: 其中R 1是氢,卤素,C 1 -C 4烷基,C 1 -C 4烷氧基,C 1 -C 4烷硫基,C 1 -C 4卤代烷氧基或CF 3的式I的N-吡啶磺酰基-N'-嘧啶基 - 和 - 三嗪基脲; R2是氢或C1-C4烷基; A是C 1 -C 6烷基或C 3 -C 6环烷基,其各自被卤素单取代至三取代,或者是C 1 -C 4烷基或C 3 -C 6环烷基,其各自被C 1 -C 4烷氧基,C 1 -C 4烷硫基,C 1 -C 4烷基磺酰基, C 4烷基亚磺酰基,C 2 -C 4链烯基,C 5 -C 6环烯基,氨基,C 1 -C 4烷基氨基,C 1 -C 4二烷基氨基或C 2 -C 4炔基,C2-C4链烯基和C5-C6环烯基可另外被卤素单取代成三取代。 或A是含有选自O,N和SO 2的杂原子的4至6元饱和杂环; 或A是被含有选自O,N和SO 2的杂原子的4至6元饱和杂环取代的C 1 -C 4烷基; X是C 1 -C 3烷基,被卤素单取代至三取代的C 1 -C 3烷基,或是被卤素单取代至三取代的C 1 -C 3烷氧基或C 1 -C 3烷氧基; Y是卤素,C1-C3烷基,被卤素单取代至三取代的C1-C3烷基,或是C1-C3烷氧基,被卤素单取代至三取代的C1-C3烷氧基,或是环丙基,甲基氨基或二甲基氨基; 和E是氮或次甲基,这些化合物与胺,碱金属碱或碱土金属碱或季铵碱的盐在出苗前和出苗后具有良好的选择性除草特性,以及良好的生长调节性 。

    Compositions for protecting plants against disease
    70.
    发明授权
    Compositions for protecting plants against disease 失效
    用于保护植物免受疾病的组合物

    公开(公告)号:US5051436A

    公开(公告)日:1991-09-24

    申请号:US481422

    申请日:1990-02-16

    摘要: Novel N-acyl- and N-sulfonylbenzo-1,2,3-thiadiazole-7-carboxylic acid amides of formula ##STR1## in which X.sub.1 and X.sub.2 independently of one another are each hydrogen or together 1 to 3 halogen atoms; A is sulfonyl or carbonyl; Y is phenyl or phenyl substituted by C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 alkoxy, halogen, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkoxycarbonyl, C.sub.1 -C.sub.3 alkanoyloxymethyl, cyano and/or by nitro; R is hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.3 -C.sub.5 alkenyl or C.sub.3 -C.sub.5 alkynyl; and in which, furthermore, the group ##STR2## wherein A.sub.1 is methylene, carbonyl or sulfonyl; X.sub.3 is hydrogen, methyl or halogen; m is 2, 3 or 4; and n is zero, 1 or 2.The novel active ingredients have plant-protecting properties and are suitable especially for the preventive protection of plants against attack by phytopathogenic microorganisms such as fungi, bacteria and viruses.

    摘要翻译: 式(I)的新的N-酰基 - 和N-磺酰基苯并-1,2,3-噻二唑-7-羧酸酰胺,其中X 1和X 2彼此独立地各自为氢或一起为1-3个卤素原子 ; A是磺酰基或羰基; Y是苯基或被C 1 -C 2烷基,C 1 -C 2烷氧基,卤素,C 1 -C 2卤代烷基,C 1 -C 2烷氧基羰基,C 1 -C 3烷酰氧基甲基,氰基和/或硝基取代的苯基。 R是氢,C 1 -C 4烷基,C 1 -C 4卤代烷基,C 3 -C 5烯基或C 3 -C 5炔基; 此外,其中A1是亚甲基,羰基或磺酰基的组 X3是氢,甲基或卤素; m为2,3或4; 并且n为零,1或2.新型活性成分具有植物保护性质,特别适用于植物防止植物病原微生物如真菌,细菌和病毒侵袭的预防性保护。