N-p-propargyloxyphenethyl-thioacetic acid amides
    1.
    发明授权
    N-p-propargyloxyphenethyl-thioacetic acid amides 失效
    N-对 - 丙酰氧基苯乙基 - 硫代乙酰胺

    公开(公告)号:US07105545B2

    公开(公告)日:2006-09-12

    申请号:US10472577

    申请日:2002-04-02

    摘要: The invention relates to N-propargyloxy-phenethyl thioacetic acid amide derivatives of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5, R6, R7 and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is hydroxy, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenysulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl, optionally substituted alkynylsulfonyl or a group —O—CO—R11, —O—CO—O—R11 or —O—CO—CO—O—R11 wherein R11 is hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted heteroaryl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi

    摘要翻译: 本发明涉及通式(I)的N-炔丙氧基 - 苯乙基硫代乙酰胺衍生物,其包括其旋光异构体和这些异构体的混合物,其中R 1是氢,烷基,环烷基或任选取代的 芳基,R 2和R 3各自独立地是氢或烷基,R 4是烷基,烯基或炔基,R 5, R 6,R 7,R 8和R 8各自独立地为氢或烷基,R 9为 氢,任选取代的烷基,任选取代的烯基或任选取代的炔基,R 10是任选取代的芳基或任选取代的杂芳基,Z是羟基,任选取代的芳氧基,任选取代的烷氧基,任选取代的炔氧基,任选地 取代的芳硫基,任选取代的烷硫基,任选取代的炔硫基,任选取代的烷基亚磺酰基,任选取代的烯基亚磺酰基,任选的 取代的炔基亚磺酰基,任选取代的烷基磺酰基,任选取代的链烯基磺酰基,任选取代的炔基磺酰基或基团-O-CO-R 11,-O-CO-OR 11或-O- 其中R 11是氢,任选取代的烷基,任选取代的环烷基,任选取代的芳基或任选取代的杂芳基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止由植物病原微生物特别是真菌侵染植物

    Phenyl-propargylether derivatives
    2.
    发明授权
    Phenyl-propargylether derivatives 有权
    苯基 - 炔丙基醚衍生物

    公开(公告)号:US06683211B1

    公开(公告)日:2004-01-27

    申请号:US10276476

    申请日:2002-11-15

    IPC分类号: C07C23305

    摘要: The invention relates to phenyl-propargylether derivatives of the general formula I including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5, R6, R7, and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

    摘要翻译: 本发明涉及通式I的苯基 - 炔丙基醚衍生物,包括其光学异构体和这些异构体的混合物,其中R 1是氢,烷基,环烷基或任选取代的芳基,R 2和R 3各自独立地是氢或烷基,R 4是烷基, 或炔基,R 5,R 6,R 7和R 8各自独立地为氢或烷基,R 9为氢,任选取代的烷基,任选取代的烯基或任选取代的炔基,R 10为任选取代的芳基或任选取代的杂芳基,且Z为卤素, 芳氧基,任选取代的烷氧基,任选取代的烯氧基,任选取代的炔氧基,任选取代的芳硫基,任选取代的烷硫基,任选取代的烯硫基; 任选取代的炔基硫基,任选取代的烷基亚磺酰基,任选取代的烯基亚磺酰基,任选取代的炔基亚磺酰基,任选取代的烷基磺酰基,任选取代的链烯基磺酰基或任选取代的炔基磺酰基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止植物病原微生物特别是真菌侵染植物。