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公开(公告)号:US07105545B2
公开(公告)日:2006-09-12
申请号:US10472577
申请日:2002-04-02
CPC分类号: C07C327/44 , A01N37/36 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/30 , A01N43/32 , A01N43/40 , A01N43/54
摘要: The invention relates to N-propargyloxy-phenethyl thioacetic acid amide derivatives of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5, R6, R7 and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is hydroxy, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenysulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl, optionally substituted alkynylsulfonyl or a group —O—CO—R11, —O—CO—O—R11 or —O—CO—CO—O—R11 wherein R11 is hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted heteroaryl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi
摘要翻译: 本发明涉及通式(I)的N-炔丙氧基 - 苯乙基硫代乙酰胺衍生物,其包括其旋光异构体和这些异构体的混合物,其中R 1是氢,烷基,环烷基或任选取代的 芳基,R 2和R 3各自独立地是氢或烷基,R 4是烷基,烯基或炔基,R 5, R 6,R 7,R 8和R 8各自独立地为氢或烷基,R 9为 氢,任选取代的烷基,任选取代的烯基或任选取代的炔基,R 10是任选取代的芳基或任选取代的杂芳基,Z是羟基,任选取代的芳氧基,任选取代的烷氧基,任选取代的炔氧基,任选地 取代的芳硫基,任选取代的烷硫基,任选取代的炔硫基,任选取代的烷基亚磺酰基,任选取代的烯基亚磺酰基,任选的 取代的炔基亚磺酰基,任选取代的烷基磺酰基,任选取代的链烯基磺酰基,任选取代的炔基磺酰基或基团-O-CO-R 11,-O-CO-OR 11或-O- 其中R 11是氢,任选取代的烷基,任选取代的环烷基,任选取代的芳基或任选取代的杂芳基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止由植物病原微生物特别是真菌侵染植物
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公开(公告)号:US06683211B1
公开(公告)日:2004-01-27
申请号:US10276476
申请日:2002-11-15
IPC分类号: C07C23305
CPC分类号: C07D239/26 , A01N37/36 , C07C233/22 , C07C235/34 , C07C323/60 , C07C323/62 , C07C2602/10 , C07D213/56 , C07D307/79 , C07D317/60 , C07D319/18 , C07D333/24 , C07D333/28
摘要: The invention relates to phenyl-propargylether derivatives of the general formula I including the optical isomers thereof and mixtures of such isomers, wherein R1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R2 and R3 are each independently hydrogen or alkyl, R4 is alkyl, alkenyl or alkynyl, R5, R6, R7, and R8 are each independently hydrogen or alkyl, R9 is hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkynyl, R10 is optionally substituted aryl or optionally substituted heteroaryl, and Z is halogen, optionally substituted aryloxy, optionally substituted alkoxy, optionally substituted alkenyloxy, optionally substituted alkynyloxy, optionally substituted arylthio, optionally substituted alkylthio, optionally substituted alkenylthio; optionally substituted alkynylthio, optionally substituted alkylsulfinyl, optionally substituted alkenylsulfinyl, optionally substituted alkynylsulfinyl, optionally substituted alkylsulfonyl, optionally substituted alkenylsulfonyl or optionally substituted alkynylsulfonyl. These compounds possess useful plant protecting properties and may advantageously be employed in agricultural practice for controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
摘要翻译: 本发明涉及通式I的苯基 - 炔丙基醚衍生物,包括其光学异构体和这些异构体的混合物,其中R 1是氢,烷基,环烷基或任选取代的芳基,R 2和R 3各自独立地是氢或烷基,R 4是烷基, 或炔基,R 5,R 6,R 7和R 8各自独立地为氢或烷基,R 9为氢,任选取代的烷基,任选取代的烯基或任选取代的炔基,R 10为任选取代的芳基或任选取代的杂芳基,且Z为卤素, 芳氧基,任选取代的烷氧基,任选取代的烯氧基,任选取代的炔氧基,任选取代的芳硫基,任选取代的烷硫基,任选取代的烯硫基; 任选取代的炔基硫基,任选取代的烷基亚磺酰基,任选取代的烯基亚磺酰基,任选取代的炔基亚磺酰基,任选取代的烷基磺酰基,任选取代的链烯基磺酰基或任选取代的炔基磺酰基。 这些化合物具有有用的植物保护性质,并且可有利地用于农业实践中以控制或防止植物病原微生物特别是真菌侵染植物。
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公开(公告)号:US20130324553A1
公开(公告)日:2013-12-05
申请号:US13984449
申请日:2012-02-08
IPC分类号: A01N43/56 , C07D231/12 , A01N43/60 , C07D401/06
CPC分类号: A01N43/56 , A01N43/58 , A01N43/60 , C07D231/12 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/14 , C07D417/14
摘要: The present invention provides compounds of formula (I): wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译: 本发明提供式(I)化合物:其中取代基如权利要求1中所定义,可用作活性成分,其具有杀微生物活性,特别是杀真菌活性。
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公开(公告)号:US20130317064A1
公开(公告)日:2013-11-28
申请号:US13984459
申请日:2012-02-08
IPC分类号: A01N43/78 , C07D417/14
CPC分类号: A01N43/78 , C07D413/04 , C07D413/14 , C07D417/14
摘要: The present invention provides compounds of formula I: wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译: 本发明提供了式I化合物:其中取代基如权利要求1所定义,可用作具有杀微生物活性,特别是杀真菌活性的活性成分。
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公开(公告)号:US08748432B2
公开(公告)日:2014-06-10
申请号:US13984449
申请日:2012-02-08
IPC分类号: A61K31/497 , A61K31/4523 , C07D403/14 , C07D401/14
CPC分类号: A01N43/56 , A01N43/58 , A01N43/60 , C07D231/12 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/14 , C07D409/14 , C07D417/14
摘要: The present invention provides compounds of formula (I): wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译: 本发明提供式(I)化合物:其中取代基如权利要求1中所定义,可用作活性成分,其具有杀微生物活性,特别是杀真菌活性。
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公开(公告)号:US08748431B2
公开(公告)日:2014-06-10
申请号:US13989797
申请日:2011-11-25
申请人: Sarah Sulzer-Mosse , Clemens Lamberth , Mathias Stephan Respondek , Laura Quaranta , Fredrik Cederbaum , Guillaume Berthon
发明人: Sarah Sulzer-Mosse , Clemens Lamberth , Mathias Stephan Respondek , Laura Quaranta , Fredrik Cederbaum , Guillaume Berthon
IPC分类号: A61K31/497 , A61K31/4523 , A61K31/4427 , A61K31/41 , A61K31/42 , C07D401/14 , C07D241/36 , C07D413/14 , C07D285/06 , C07D261/06
CPC分类号: A01N43/82 , A01N43/60 , A01N43/80 , C07D401/14 , C07D413/14 , C07D417/14 , C07D513/04
摘要: Compounds of the formula I Formula (I) wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译: 其中取代基如权利要求1中所定义的式I化学式(I)的化合物可用作具有杀微生物活性,特别是杀真菌活性的活性成分。
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公开(公告)号:US20130324544A1
公开(公告)日:2013-12-05
申请号:US13989797
申请日:2011-11-25
申请人: Sarah Sulzer-Mosse , Clemens Lamberth , Mathias Stephan Respondek , Laura Quaranta , Fredrik Cederbaum , Guillaume Berthon
发明人: Sarah Sulzer-Mosse , Clemens Lamberth , Mathias Stephan Respondek , Laura Quaranta , Fredrik Cederbaum , Guillaume Berthon
CPC分类号: A01N43/82 , A01N43/60 , A01N43/80 , C07D401/14 , C07D413/14 , C07D417/14 , C07D513/04
摘要: Compounds of the formula I Formula (I) wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译: 其中取代基如权利要求1中所定义的式I化学式(I)的化合物可用作具有杀微生物活性,特别是杀真菌活性的活性成分。
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公开(公告)号:US20100022475A1
公开(公告)日:2010-01-28
申请号:US11722232
申请日:2005-12-20
申请人: Kurt Nebel , Sebastian Volker Wendeborn , Clemens Lamberth , Patrick Jelf Crowley , Fredrik Cederbaum
发明人: Kurt Nebel , Sebastian Volker Wendeborn , Clemens Lamberth , Patrick Jelf Crowley , Fredrik Cederbaum
CPC分类号: C07D487/04 , A01N55/00 , C07F7/0812
摘要: The present invention relates to novel triazolopyrimidine derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity(I): wherein the substituents are as defined in claim 1. Characterizing feature is the cyclic silyl group.
摘要翻译: 本发明涉及式I的新型三唑并嘧啶衍生物作为具有杀微生物活性,特别是杀真菌活性(I)的活性成分:其中取代基如权利要求1所定义。其特征在于环状甲硅烷基。
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公开(公告)号:US09174987B2
公开(公告)日:2015-11-03
申请号:US13234793
申请日:2011-09-16
申请人: David John Hughes , Paul Anthony Worthington , Charles Adam Russell , Eric Daniel Clarke , James Edward Peace , Mark Richard Ashton , Thomas Stephen Coulter , Richard Spurring Roberts , Louis-Pierre Molleyres , Fredrik Cederbaum , Jerome Cassayre , Peter Maienfisch
发明人: David John Hughes , Paul Anthony Worthington , Charles Adam Russell , Eric Daniel Clarke , James Edward Peace , Mark Richard Ashton , Thomas Stephen Coulter , Richard Spurring Roberts , Louis-Pierre Molleyres , Fredrik Cederbaum , Jerome Cassayre , Peter Maienfisch
IPC分类号: A01N43/90 , A01N47/38 , C07D471/10 , A01P5/00 , A01P7/02 , A01P7/04 , A01P9/00 , A01N47/34 , C07D211/70 , C07D211/76 , C07D491/10
CPC分类号: A01N43/90 , A01N47/34 , A01N47/38 , C07B2200/11 , C07D211/70 , C07D211/76 , C07D471/10 , C07D491/10
摘要: Insecticidal, acaricidal, nematicidal or molluscicidal compounds of formula (I) wherein Y is a single bond, C═O, C═S or S(O)q where q is 0, 1 or 2; and R1, R2, R3, R4, R8, R9 are R10 are as defined in the claims or salts or N-oxides thereof, processes for preparing them and compositions containing them.
摘要翻译: 其中Y是单键,C = O,C = S或S(O)q,其中q是0,1或2的式(I)的杀虫,杀螨,杀线虫或杀软体动物化合物; 且R 1,R 2,R 3,R 4,R 8,R 9为R 10如权利要求中所定义或其盐或N-氧化物,制备方法和含有它们的组合物。
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公开(公告)号:US08546569B2
公开(公告)日:2013-10-01
申请号:US13371002
申请日:2012-02-10
申请人: Peter Maienfisch , Louis-Pierre Molleyres , Jerome Cassayre , Fredrik Cederbaum , Camilla Corsi , Thomas Pitterna
发明人: Peter Maienfisch , Louis-Pierre Molleyres , Jerome Cassayre , Fredrik Cederbaum , Camilla Corsi , Thomas Pitterna
IPC分类号: C07D241/04 , C07D295/00 , C07D401/00 , C07D403/00 , C07D405/00 , C07D409/00 , C07D411/00 , C07D413/00 , C07D417/00 , C07D419/00
CPC分类号: C07D211/34 , A01N43/40 , C07D211/52 , C07D401/04 , C07D401/12 , C07D401/14
摘要: The use of a compound of formula I Y is a single bond, C═O, C═S or S(O)m where m is 0, 1 or 2; the ring is a 6 membered aromatic ring or is a 5 or 6 membered heteroaromatic ring; Z and Z′ are provided that both are not N; R1, R2, R3, R3a, R4, R8 and Ra are specified organic groups and n and p are independently 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.
摘要翻译: 式I Y化合物的使用是单键,C = O,C = S或S(O)m,其中m为0,1或2; 该环为6元芳族环,或为5或6元杂芳环; Z和Z'都不是N; R1,R2,R3,R3a,R4,R8和Ra是指定的有机基团,n和p独立地为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。
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