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    2-analino pyrimidine compounds
    1.
    发明授权
    2-analino pyrimidine compounds 失效
    2-分析嘧啶化合物

    公开(公告)号：US5159078A

    公开(公告)日：1992-10-27

    申请号：US569319

    申请日：1990-08-17

    申请人： Hermann Rempfler ,  Dieter Durr ,  Rudolf C. Thummel

    发明人： Hermann Rempfler ,  Dieter Durr ,  Rudolf C. Thummel

    IPC分类号： A01N47/36 ,  A01N57/24 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D405/04 ,  C07D409/04 ,  C07F9/6512

    CPC分类号： C07D239/42 ,  A01N47/36 ,  A01N57/24 ,  C07D239/47 ,  C07D405/04 ,  C07D409/04 ,  C07F9/65127

    摘要： The present invention relates to novel N-phenyl-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions containing those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 are each, independently of the others, hydrogen; halogen; C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; nitro; cyano; C.sub.1 -C.sub.4 alkoxycarbonyl; C.sub.1 -C.sub.4 alkylcarbonyl; di-(C.sub.1 -C.sub.4 alkylamino)-carbonyl; mono-(C.sub.1 -C.sub.4 alkylamino)carbonyl; carbamoyl; C.sub.1 -C.sub.4 -haloalkyl-S(O).sub.n -; or -PO[O-(C.sub.1 -C.sub.4)-alkyl].sub.2 ;R.sup.4 is C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; phenyl that is unsubstituted or is substituted by up to three identical or different substituents from halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl and C.sub.1 -C.sub.4 alkoxy; 2-furanyl; 2-thienyl; 3-thienyl; C.sub.3 -C.sub.6 -cycloalkyl that is unsubstituted or is substituted by up to three identical or different C.sub.1 -C.sub.4 alkyl radicals; cyano; C.sub.2 -C.sub.4 haloalkenyl; C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkoxy; or halogen-C.sub.1 -C.sub.4 alkylthio;R.sup.5 is hydrogen; C.sub.1 -C.sub.3 alkyl; C.sub.1 -C.sub.3 haloalkyl; halogen; or C.sub.1 -C.sub.3 haloalkoxy; andn is 0, 1 or 2,with the proviso that when one of the radicals R.sup.1, R.sup.2 and R.sup.3 is nitro, that substituent may not be bonded in the 2- or 6-position of the phenyl ring.

    摘要翻译： 本发明涉及具有除草和植物生长调节活性的新型N-苯基-N-嘧啶-2-基脲，含有这些物质作为活性成分的农用化学组合物，用于控制杂草或用于调节 植物生长，以及制备新化合物的方法。 本发明还涉及新型中间体及其制备方法。 该化合物对应于式Ⅰ（I）其中R1，R2和R3各自独立地为氢; 卤素; C 1 -C 4烷基; C1-C4烷氧基; C 1 -C 4卤代烷基; C1-C4卤代烷氧基; C 1 -C 4烷基-S（O）n - ; 硝基 氰基; C1-C4烷氧基羰基; C1-C4烷基羰基; 二（C 1 -C 4烷基氨基） - 羰基; 单（C 1 -C 4烷基氨基）羰基; 氨基甲酰基; C 1 -C 4卤代烷基-S（O）n - ; 或-PO [O-（C 1 -C 4） - 烷基] 2; R4是C1-C6烷基; C1-C4烷氧基; C 1 -C 4烷基-S（O）n - ; C 1 -C 4卤代烷基; C1-C4卤代烷氧基; 未被取代或被卤素，C1-C4烷基，C1-C4卤代烷基和C1-C4烷氧基中最多三个相同或不同的取代基取代的苯基; 2-呋喃基; 2-噻吩基; 3-噻吩基; 未被取代或被至多三个相同或不同的C 1 -C 4烷基取代的C 3 -C 6环烷基; 氰基; C 2 -C 4卤代烯基; C 1 -C 4烷氧基-C 1 -C 4烷基; C1-C4烷氧基-C1-C4烷氧基; 或卤素-C 1 -C 4烷硫基; R5是氢; C1-C3烷基; C 1 -C 3卤代烷基; 卤素; 或C 1 -C 3卤代烷氧基; 并且n为0,1或2，条件是当基团R 1，R 2和R 3中的一个为硝基时，该取代基不能键合在苯环的2-或6-位。

    N-phenyl-N-pyrimidin-2-ylureas
    2.
    发明授权
    N-phenyl-N-pyrimidin-2-ylureas 失效
    N-苯基-N-嘧啶-2-基脲

    公开(公告)号：US4966622A

    公开(公告)日：1990-10-30

    申请号：US332193

    申请日：1989-04-03

    申请人： Hermann Rempfler ,  Dieter Durr ,  Rudolf C. Thummel

    发明人： Hermann Rempfler ,  Dieter Durr ,  Rudolf C. Thummel

    IPC分类号： A01N47/36 ,  A01N57/24 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D405/04 ,  C07D409/04 ,  C07F9/6512

    CPC分类号： C07D239/42 ,  A01N47/36 ,  A01N57/24 ,  C07D239/47 ,  C07D405/04 ,  C07D409/04 ,  C07F9/65127

    摘要： The present invention relates to novel N-phenyl-N-pyrimidin-2-ylureas having a herbicidal and plant growth-regulating activity, to agrochemical compositions containing those substances as active ingredients, to the use of the novel ureas for controlling weeds or for regulating plant growth, and to processes for the preparation of the novel compounds. The invention also relates to novel intermediates and to processes for the preparation thereof.The novel compounds correspond to formula I ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 are each, independently of the others, hydrogen; halogen; C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; nitro; cyano; C.sub.1 -C.sub.4 alkoxycarbonyl; C.sub.1 -C.sub.4 alkylcarbonyl; di-(C.sub.1 -C.sub.4 alkylamino)-carbonyl; mono-(C.sub.1 -C.sub.4 alkylamino)carbonyl; carbamoyl; C.sub.1 -C.sub.4 haloalkyl-S(O).sub.n -; or -PO[O-(C.sub.1 -C.sub.4)-alkyl].sub.2 ;R.sup.4 is C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.4 alkoxy; C.sub.1 -C.sub.4 alkyl-S(O).sub.n -; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.4 haloalkoxy; phenyl that is unsubstituted or is substituted by up to three identical or different substituents from halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl and C.sub.1 -C.sub.4 alkoxy; 2-furanyl; 2-thienyl; 3-thienyl; C.sub.3 -C.sub.6 -cycloalkyl that is unsubstituted or is substituted by up to three identical or different C.sub.1 -C.sub.4 alkyl radicals; cyano; C.sub.2 -C.sub.4 haloalkenyl; C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl; C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkoxy; or halogen-C.sub.1 -C.sub.4 alkylthio;R.sup.5 is hydrogen; C.sub.1 -C.sub.3 alkyl; C.sub.1 -C.sub.3 haloalkyl; halogen; or C.sub.1 -C.sub.3 haloalkoxy; andn is 0, 1 or 2,with the proviso that when one of the radicals R.sup.1, R.sup.2 and R.sup.3 is nitro, that substituent may not be bonded in the 2- or 6-position of the phenyl ring.

    摘要翻译： 本发明涉及具有除草和植物生长调节活性的新型N-苯基-N-嘧啶-2-基脲，含有这些物质作为活性成分的农用化学组合物，用于控制杂草或用于调节 植物生长，以及制备新化合物的方法。 本发明还涉及新型中间体及其制备方法。 该化合物对应于式Ⅰ（I）其中R1，R2和R3各自独立地为氢; 卤素; C 1 -C 4烷基; C1-C4烷氧基; C 1 -C 4卤代烷基; C1-C4卤代烷氧基; C 1 -C 4烷基-S（O）n - ; 硝基 氰基; C1-C4烷氧基羰基; C1-C4烷基羰基; 二（C 1 -C 4烷基氨基） - 羰基; 单（C 1 -C 4烷基氨基）羰基; 氨基甲酰基; C 1 -C 4卤代烷基-S（O）n - 或-PO [O-（C 1 -C 4） - 烷基] 2; R4是C1-C6烷基; C1-C4烷氧基; C 1 -C 4烷基-S（O）n - ; C 1 -C 4卤代烷基; C1-C4卤代烷氧基; 未被取代或被卤素，C1-C4烷基，C1-C4卤代烷基和C1-C4烷氧基中最多三个相同或不同的取代基取代的苯基; 2-呋喃基; 2-噻吩基; 3-噻吩基; 未被取代或被至多三个相同或不同的C 1 -C 4烷基取代的C 3 -C 6环烷基; 氰基; C 2 -C 4卤代烯基; C 1 -C 4烷氧基-C 1 -C 4烷基; C1-C4烷氧基-C1-C4烷氧基; 或卤素-C 1 -C 4烷硫基; R5是氢; C1-C3烷基; C 1 -C 3卤代烷基; 卤素; 或C 1 -C 3卤代烷氧基; 并且n为0,1或2，条件是当基团R 1，R 2和R 3中的一个为硝基时，该取代基不能键合在苯环的2-或6-位。

    1,2-dinitro-4-(3'-chloro-5'-trifluoromethyl)-2-pyridyloxy-benzene having herbicidal properties
    3.
    发明授权
    1,2-dinitro-4-(3'-chloro-5'-trifluoromethyl)-2-pyridyloxy-benzene having herbicidal properties 失效
    具有除草性的1,2-二硝基-4-（3'-氯-5'-三氟甲基）-2-吡啶氧基 - 苯

    公开(公告)号：US4610980A

    公开(公告)日：1986-09-09

    申请号：US592496

    申请日：1984-02-27

    申请人： Ludwig Maier ,  Hermann Rempfler ,  Dieter Durr

    发明人： Ludwig Maier ,  Hermann Rempfler ,  Dieter Durr

    IPC分类号： A01N57/24 ,  C07D213/64 ,  C07D213/643 ,  C07F9/58 ,  A01N43/40

    CPC分类号： C07D213/643 ,  A01N57/24 ,  C07F9/582

    摘要： The invention relates to novel 2-nitro-4- or -5-pyridyloxyphenylphosphonic acid derivatives of the formula ##STR1## wherein X is halogen or trifluoromethyl, Y is hydrogen or halogen, one of the two substituents A and E is a phosphonate group ##STR2## wherein R is C.sub.1 -C.sub.4 alkyl or hydrogen, and the other is a nitro group, including the metal salts thereof and the salts thereof with ammonium and organic nitrogen bases, and to the preparation and use thereof. These compounds may be used for controlling weeds, regulating plant growth, or as microbicides.

    摘要翻译： 本发明涉及下式的新的2-硝基-4-或5-吡啶氧基苯基膦酸衍生物，其中X是卤素或三氟甲基，Y是氢或卤素，两个取代基A和E之一是膦酸酯基， 其中R是C1-C4烷基或氢，另一个是硝基，包括其金属盐及其与铵和有机氮碱的盐，以及其制备和用途。 这些化合物可用于控制杂草，调节植物生长或作为杀微生物剂。

    1,2,4-triazolo[1,5-A]pyridi midin-2-ylsulfonyl-3-aminothiophene-2-carboxylic esters as antidotes for certain herbicides
    6.
    发明授权
    1,2,4-triazolo[1,5-A]pyridi midin-2-ylsulfonyl-3-aminothiophene-2-carboxylic esters as antidotes for certain herbicides 失效
    1,2,4-三唑并[1,5-A]哒啶-2-基磺酰基-3-氨基噻吩-2-羧酸酯作为某些除草剂的解毒剂

    公开(公告)号：US5041157A

    公开(公告)日：1991-08-20

    申请号：US461602

    申请日：1990-01-05

    申请人： Alfred Seiler ,  Hans-Dieter Schneider ,  Dieter Durr

    发明人： Alfred Seiler ,  Hans-Dieter Schneider ,  Dieter Durr

    IPC分类号： A01N25/32 ,  A01N37/22 ,  A01N37/24 ,  A01N43/90 ,  A01N47/36 ,  C07D487/04

    CPC分类号： C07D487/04 ,  A01N25/32

    摘要： The present invention relates to the novel use of antidotes of formula I ##STR1## wherein R.sup.1 is C.sub.1 -C.sub.6 alkyl or C.sub.3 -C.sub.6 cycloalkyl, and each of R.sup.2 and R.sup.3, independently of the other, is hydrogen, C.sub.1 -C.sub.3 alkyl, trifluoromethyl or cyclopropyl, with the proviso that only one of the symbols R.sup.2 and R.sup.3 may be hydrogen, for protecting cultivated plants from the phytotoxic action of herbicides. The invention relates also to novel compounds and the preparation thereof and to novel intermediates and the preparation thereof. The invention further relates to herbicidal composition that contain a combination of herbicide and antidote and to corresponding method of controlling weeds. Finally, the invention relates also to the seeds of cultivated plants protected by the treatment with the antidote.

    摘要翻译： 本发明涉及式Ⅰ的解毒剂（I）的新用途，其中R 1是C 1 -C 6烷基或C 3 -C 6环烷基，R 2和R 3各自独立地是氢，C 1 -C 3烷基，三氟甲基 或环丙基，条件是符号R2和R3中只有一个可以是氢，以保护栽培植物免受除草剂的植物毒性作用。 本发明还涉及新型化合物及其制备方法以及新型中间体及其制备方法。 本发明还涉及含有除草剂和解毒剂组合的除草组合物以及控制杂草的相应方法。 最后，本发明还涉及通过用解毒剂处理而保护的栽培植物的种子。

    Herbicidally active 2-substituted 5-penoxyphenylphosphonic acid derivatives
    8.
    发明授权
    Herbicidally active 2-substituted 5-penoxyphenylphosphonic acid derivatives 失效
    除草活性2-取代5-苯氧基苯基膦酸衍生物

    公开(公告)号：US4421548A

    公开(公告)日：1983-12-20

    申请号：US334861

    申请日：1981-12-28

    申请人： Ludwig Maier ,  Dieter Durr

    发明人： Ludwig Maier ,  Dieter Durr

    IPC分类号： A01N57/22 ,  A01N57/30 ,  A01N57/34 ,  C07F9/38 ,  C07F9/40 ,  C07F9/42 ,  C07F9/44 ,  A01N57/14

    CPC分类号： A01N57/22 ,  A01N57/30 ,  A01N57/34 ,  C07F9/3834 ,  C07F9/4021 ,  C07F9/42 ,  C07F9/4419

    摘要： The present invention relates to novel herbicidal and plant growth-inhibiting 2-substituted 5-phenoxyphenylphosphonic acid derivatives of the formula ##STR1## wherein each of R.sub.1 and R.sub.2 independently is hydroxyl, lower alkoxy, lower alkylthio, alkylamino, dialkylamino, chlorine, benzyloxy or benzylthio, X is halogen or a --CF.sub.3, --NO.sub.2, --CN, --CONH.sub.2 or --CSNH.sub.2 group, n is 0 to 3, and Y is --OH, halogen, NO.sub.2, --CN, NH.sub.2, --NHCO--R, --NHCOOR or --NH--SO.sub.2 --R, wherein R is an unsubstituted or halogenated lower alkyl radical. Preferred compounds are 2-nitro-5-(2'-chloro-4'-trifluoromethylphenoxy)-phenylphosphonic acid and the lower dialkyl esters thereof. The invention also relates to the production of the novel phosphonic acid derivatives, starting from a 3,4-dinitrodiphenyl ether and reacting it with a trialkylphosphite as first step. The invention further relates to herbicidal and plant growth-regulating compositions which contain one of the novel compounds as active component, and also to the use of these compounds and compositions for controlling weeds (also selectively), for inhibiting plant growth and desiccating parts of plants above the soil, as well as for totally destroying existing plant growth.

    摘要翻译： 本发明涉及新的除草和植物生长抑制的2-取代的5-取代的5-苯氧基苯基膦酸衍生物，其中R 1和R 2各自独立地是羟基，低级烷氧基，低级烷硫基，烷基氨基，二烷基氨基，氯 ，苄氧基或苄硫基，X为卤素或-CF 3，-NO 2，-CN，-CONH 2或-CSNH 2基，n为0至3，Y为-OH，卤素，NO 2，-CN，NH 2，-NHCO- R，-NHCOOR或-NH-SO 2 -R，其中R是未取代或卤代的低级烷基。 优选的化合物是2-硝基-5-（2'-氯-4'-三氟甲基苯氧基） - 苯基膦酸及其低级二烷基酯。 本发明还涉及从3,4-二硝基二苯醚开始并与其作为第一步与三烷基亚磷酸酯反应的新型膦酸衍生物的制备。 本发明还涉及含有新化合物之一作为活性成分的除草和植物生长调节组合物，以及这些化合物和组合物用于防治杂草（也可选择性）用于抑制植物生长和干燥植物部分的用途 在土壤之上，以及完全破坏现有的植​​物生长。

    Herbicidally active 2-substituted 5-phenoxyphenylphosphonic acid esters
    9.
    发明授权
    Herbicidally active 2-substituted 5-phenoxyphenylphosphonic acid esters 失效
    除草活性2-取代的5-苯氧基苯基膦酸酯

    公开(公告)号：US4391624A

    公开(公告)日：1983-07-05

    申请号：US269228

    申请日：1981-06-01

    申请人： Ludwig Maier ,  Dieter Durr

    发明人： Ludwig Maier ,  Dieter Durr

    IPC分类号： A01N57/22 ,  A01N57/30 ,  A01N57/34 ,  C07F9/38 ,  C07F9/40 ,  C07F9/42 ,  C07F9/44 ,  A01N57/18

    CPC分类号： A01N57/22 ,  A01N57/30 ,  A01N57/34 ,  C07F9/3834 ,  C07F9/4021 ,  C07F9/42 ,  C07F9/4419

    摘要： The present invention relates to novel herbicidal and plant growth-inhibiting 2-substituted 5-phenoxyphenylphosphonic acid derivatives of the formula ##STR1## wherein each of R.sub.1 and R.sub.2 independently is hydroxyl, lower alkoxy, lower alkylthio, alkylamino, dialkylamino, chlorine, benzyloxy or benzylthio, X is halogen or a --CF.sub.3, --NO.sub.2, --CN, --CONH.sub.2 or --CSNH.sub.2 group, n is 0 to 3, and Y is --OH, halogen, NO.sub.2, --CN, NH.sub.2, --NHCO--R, --NHCOOR or --NH--SO.sub.2 --R, wherein R is an unsubstituted or halogenated lower alkyl radical. Preferred compounds are 2-nitro-5-(2'-chloro-4'-trifluoromethylphenoxy)-phenylphosphonic acid and the lower dialkyl esters thereof. The invention also relates to the production of the novel phosphonic acid derivatives, starting from a 3,4-dinitrodiphenyl ether and reacting it with a trialkylphosphite as first step. The invention further relates to herbicidal and plant growth-regulating compositions which contain one of the novel compounds as active component, and also to the use of these compounds and compositions for controlling weeds (also selectively), for inhibiting plant growth and desiccating parts of plants above the soil, as well as for totally destroying existing plant growth.

    摘要翻译： 本发明涉及新的除草和植物生长抑制的2-取代的5-取代的5-苯氧基苯基膦酸衍生物，其中R 1和R 2各自独立地是羟基，低级烷氧基，低级烷硫基，烷基氨基，二烷基氨基，氯 ，苄氧基或苄硫基，X为卤素或-CF 3，-NO 2，-CN，-CONH 2或-CSNH 2基，n为0至3，Y为-OH，卤素，NO 2，-CN，NH 2，-NHCO- R，-NHCOOR或-NH-SO 2 -R，其中R是未取代或卤代的低级烷基。 优选的化合物是2-硝基-5-（2'-氯-4'-三氟甲基苯氧基） - 苯基膦酸及其低级二烷基酯。 本发明还涉及从3,4-二硝基二苯醚开始并与其作为第一步与三烷基亚磷酸酯反应的新型膦酸衍生物的制备。 本发明还涉及含有新化合物之一作为活性成分的除草和植物生长调节组合物，以及这些化合物和组合物用于防治杂草（也可选择性）用于抑制植物生长和干燥植物部分的用途 在土壤之上，以及完全破坏现有的植​​物生长。