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    Pryidine-2,3-dicarboxylic acid diamide derivatives and herbicides comprising said derivatives as active ingredient
    2.
    发明授权
    Pryidine-2,3-dicarboxylic acid diamide derivatives and herbicides comprising said derivatives as active ingredient 失效
    包含所述衍生物的Pryidine-2,3-二羧酸二酰胺衍生物和除草剂作为活性成分

    公开(公告)号：US5843868A

    公开(公告)日：1998-12-01

    申请号：US825642

    申请日：1997-04-01

    申请人： Masanori Tonishi ,  Takeshi Katsuhira ,  Takashi Ohtsuka ,  Yuzo Miura

    发明人： Masanori Tonishi ,  Takeshi Katsuhira ,  Takashi Ohtsuka ,  Yuzo Miura

    IPC分类号： A01N43/40 ,  A01N43/42 ,  C07D213/82 ,  C07D213/89 ,  C07D405/12 ,  C07D213/30

    CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/42 ,  C07D213/89 ,  C07D405/12

    摘要： The present invention provides a pyridine-2,3-dicarboxylic acid diamide derivatives represented by the following formula (I) and herbicides containing them as an active ingredient. ##STR1## �wherein R.sub.1 represents one to three substituents such as H, halogen, cyano, nitro, (halo)alkyl, (halo)alkoxy, (halo)alkylthio, (C.sub.3-6)cycloalkyl, alkenyl, alkynyl, substituted phenyl, substituted phenoxy, etc. and R.sub.1 may represent alkylene or alkenylene together with an adjacent carbon atom; R.sub.2 represents H, halogen, cyano, nitro, (halo)alkyl or (halo)alkoxy; R.sub.3 represents H or alkyl; R.sub.4 and R.sub.5 each represent H, (halo)alkyl, cycloalkyl, substituted cycloalkylalkyl, etc.; and n represents an integer of 0 or 1!. The present compounds exhibit excellent effect for controlling paddy field weeds and the like.

    摘要翻译： 本发明提供由下式（I）表示的吡啶-2,3-二羧酸二酰胺衍生物和含有它们作为有效成分的除草剂。 （I）[其中R 1表示一至三个取代基如H，卤素，氰基，硝基，（卤代）烷基，（卤代）烷氧基，（卤代）烷硫基，（C 3-6）环烷基，烯基，炔基， 取代的苯基，取代的苯氧基等，R 1可以与相邻的碳原子一起代表亚烷基或亚烯基; R 2表示H，卤素，氰基，硝基，（卤代）烷基或（卤代）烷氧基; R3表示H或烷基; R4和R5各自表示H，（卤素）烷基，环烷基，取代的环烷基烷基等; n表示0或1的整数]。 本发明化合物对于控制水田杂草等具有优异的效果。

    Fused-heterocycle dicarboxylic acid diamide derivatives or salts thereof, herbicide and usage thereof
    3.
    发明授权
    Fused-heterocycle dicarboxylic acid diamide derivatives or salts thereof, herbicide and usage thereof 失效
    熔融 - 杂环二羧酸二酰胺衍生物或其盐，除草剂及其用途

    公开(公告)号：US06444617B1

    公开(公告)日：2002-09-03

    申请号：US09744579

    申请日：2001-01-26

    申请人： Hideo Takaishi ,  Takeshi Katsuhira ,  Hiroshi Yamaguchi ,  Youichi Kawabata ,  Hiroto Harayama ,  Yoshiki Oda ,  Masahiko Murai

    发明人： Hideo Takaishi ,  Takeshi Katsuhira ,  Hiroshi Yamaguchi ,  Youichi Kawabata ,  Hiroto Harayama ,  Yoshiki Oda ,  Masahiko Murai

    IPC分类号： A01N4356

    CPC分类号： C07D215/54 ,  A01N43/42 ,  A01N43/60 ,  A01N43/90

    摘要： A fused heterocyclic dicarboxylic acid diamide derivative represented by formula (I): wherein R1 is H, (C1-C6) alkyl; R2 and R3 are H, (halo) (C1-C6) alkyl, (C3-C8) cycloalkyl, substituted amino (C1-C6) alkyl, (substituted) phenyl (C1-C6) alkyl, (substituted) phenyl (C1-C6) alkoxy or the like or R2 and R3, taken conjointly, represent a (substituted) 5- or 6-membered heterocycle having at least one of O, S and N; X is H, halogen, NO2, CN, (C1-C6) alkyl, (substituted) phenyl, (substituted) phenoxy or the like; is or the like wherein Y, R4 and R9 are H, halogen, NO2, CN, (C1-C6) alkyl or the like, and A, B, D, E, F, G, J and K are O, S, N, sulfinyl or the like; and a herbicide containing said derivative as active ingredient.

    摘要翻译： 由式（I）表示的稠合杂环二羧酸二酰胺衍生物：其中R 1是H，（C 1 -C 6）烷基; （C 1 -C 6）烷基，（取代的）苯基（C 1 -C 6）烷基，（取代的）苯基（C 1 -C 6）烷基，（取代的） C6）烷氧基等或R2和R3一起表示具有O，S和N中的至少一个的（取代的）5元或6元杂环; X是H，卤素，NO 2，CN，（C 1 -C 6）烷基，（取代的）苯基，（取代的）苯氧基等;其中Y，R 4和R 9是H，卤素，NO 2，CN，（C 1 -C 6）烷基等，A，B，D，E，F，G，J和K是O，S，N，亚磺酰基等; 和含有所述衍生物作为活性成分的除草剂。

    Processes for producing pyrazoloacridone derivative and synthetic intermediate thereof
    5.
    发明申请
    Processes for producing pyrazoloacridone derivative and synthetic intermediate thereof 审中-公开
    吡唑并吖啶酮衍生物及其合成中间体的制备方法

    公开(公告)号：US20060217554A1

    公开(公告)日：2006-09-28

    申请号：US10551816

    申请日：2004-04-23

    申请人： Nobuaki Tsubakihara ,  Takeshi Katsuhira ,  Masahiko Kinugawa ,  Nobuyuki Kato

    发明人： Nobuaki Tsubakihara ,  Takeshi Katsuhira ,  Masahiko Kinugawa ,  Nobuyuki Kato

    IPC分类号： C07D471/04

    CPC分类号： C07D471/06 ,  C07D231/56

    摘要： (wherein R represents lower alkyl; R1 represents a hydrogen atom, —CH2X or —OC(═O)R3; and R2 represents a hydrogen atom, nitro, halogen, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkoxy, substituted or unsubstituted lower alkylthio or substituted or unsubstituted aryl) The present invention provides a simple industrial process for producing pyrazoloacridone derivatives having an antitumor activity, 1-(2-carboxyphenyl)indazole derivatives, which are useful as synthetic intermediates thereof, or the like; and the like. For example, the present invention provides a process for producing a 1-(2-carboxyphenyl)indazole derivative represented by general formula (IV) which comprises steps of reacting a compound represented by above general formula (I) with a compound represented by above general formula (II) in the presence of a base to produce a compound represented by above general formula (III); and hydrolyzing a cyano group of the resulting compound represented by general formula (III).

    摘要翻译： （其中R表示低级烷基; R 1表示氢原子，-CH 2 X或-OC（-O）R 3）;和 R 2表示氢原子，硝基，卤素，取代或未取代的低级烷基，取代或未取代的低级烷氧基，取代或未取代的低级烷硫基或取代或未取代的芳基）本发明提供了简单的工业方法 制备具有抗肿瘤活性的吡唑并吖啶酮衍生物，可用作其合成中间体的1-（2-羧基苯基）吲唑衍生物等; 等等。 例如，本发明提供一种制备由通式（IV）表示的1-（2-羧基苯基）吲唑衍生物的方法，该方法包括以下步骤：使由上述通式（I）表示的化合物与上述通式 式（II）的化合物在碱存在下反应制备由上述通式（III）表示的化合物; 并水解由通式（III）表示的所得化合物的氰基。