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    Pyrethroid Insecticide For Protecting Plants And Seed
    2.
    发明申请
    Pyrethroid Insecticide For Protecting Plants And Seed 审中-公开
    拟除虫菊酯杀虫剂用于保护植物和种子

    公开(公告)号：US20150230470A1

    公开(公告)日：2015-08-20

    申请号：US14429701

    申请日：2013-09-19

    申请人： BASF SE

    发明人： Bernd Wolf ,  Hans Theobald

    IPC分类号： A01N53/00 ,  C07C69/743

    CPC分类号： A01N53/00 ,  C07C69/743 ,  C07C2601/02

    摘要： The present invention relates to pyrethroid insecticides and the stereoisomers thereof and to compositions comprising the same. The invention also relates to the use of the insecticides or compositions comprising such insecticides for combating invertebrate pests. Furthermore, the invention relates to methods of applying such insecticides.

    摘要翻译： 本发明涉及拟除虫菊酯类杀虫剂及其立体异构体及其组合物。 本发明还涉及包含这种杀虫剂的杀虫剂或组合物用于防治无脊椎动物害虫的用途。 此外，本发明涉及应用这种杀虫剂的方法。

    Method for producing optically active 1-amino-2-vinylcyclopropanecarboxylic acid ester
    3.
    发明授权
    Method for producing optically active 1-amino-2-vinylcyclopropanecarboxylic acid ester 失效
    光学活性1-氨基-2-乙烯基环丙烷羧酸酯的制备方法

    公开(公告)号：US08742162B2

    公开(公告)日：2014-06-03

    申请号：US13388575

    申请日：2010-08-05

    申请人： Toshiaki Aikawa ,  Junichi Yasuoka ,  Tetsuya Ikemoto

    发明人： Toshiaki Aikawa ,  Junichi Yasuoka ,  Tetsuya Ikemoto

    IPC分类号： C07C67/30 ,  C07C67/317 ,  C07C69/743 ,  C07C69/747 ,  C07C67/48 ,  C07C67/62

    CPC分类号： C07B53/00 ,  C07C227/32

    摘要： 1-Amino-2-vinylcyclopropanecarboxylic acid ester, which is useful as a synthetic intermediate of pharmaceuticals, can be produced by a process of producing 1-amino-2-vinylcyclopropanecarboxylic acid ester represented by formula (4): including a step of hydrolysis of an optically active 1-N-(arylmethylene)amino-2-vinylcyclopropanecarboxylic acid ester represented by formula (3): which is obtained by reacting an N-(arylmethylene)glycine ester represented by formula (1): with a compound represented by formula (2): in the presence of a base and an optically active quaternary ammonium salt.

    摘要翻译： 可用作药物的合成中间体的1-氨基-2-乙烯基环丙烷羧酸酯可以通过制备由式（4）表示的1-氨基-2-乙烯基环丙烷羧酸酯的方法制备：包括水解 由式（3）表示的光学活性的1-N-（芳基亚甲基）氨基-2-乙烯基环丙烷羧酸酯：其由式（1）表示的N-（芳基亚甲基）甘氨酸酯与式 （2）：在碱和光学活性季铵盐的存在下。

    METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER
    5.
    发明申请
    METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER 审中-公开
    生产环糊精羧酸酯的方法

    公开(公告)号：US20120029227A1

    公开(公告)日：2012-02-02

    申请号：US13203916

    申请日：2010-03-12

    申请人： Jun Ohshita ,  Toru Uekawa

    发明人： Jun Ohshita ,  Toru Uekawa

    IPC分类号： C07C69/743

    CPC分类号： C07C253/30 ,  C07C2601/02 ,  C07C255/31

    摘要： A method for producing a cyclopropanecarboxylate represented by formula (III): wherein, R represents a chain hydrocarbon group having 1 to 10 carbon atoms optionally having at least one member selected from the group consisting of halogen atoms, acyl groups having 2 to 7 carbon atoms optionally having a substituent, alkoxy groups having 1 to 7 carbon atoms optionally having a substituent, alkylthio groups having 1 to 3 carbon atoms and phenyl groups optionally having a substituent, a cyclic hydrocarbon group having 3 to 10 carbon atoms or a hydrogen atom; comprising reacting a cyclopropanecarboxylate represented by formula (I): wherein, R represents the same meaning as described above; and 2-cyanopropionic acid in the presence of a base.

    摘要翻译： 一种由式（III）表示的环丙烷羧酸酯的制备方法：其中，R表示碳原子数1〜10的链状烃基，可以具有选自卤素原子，碳原子数2〜7的酰基中的至少1种 任选具有取代基，可以具有取代基的碳原子数1〜7的烷氧基，碳原子数1〜3的烷硫基和可以具有取代基的苯基，碳原子数3〜10的环状烃基或氢原子。 包括使由式（I）表示的环丙烷羧酸酯反应：其中，R表示与上述相同的含义; 和2-氰基丙酸在碱的存在下反应。

    Derivative of ester of carboxylic acid, and insecticide and insect proofing agent containing the same
    6.
    发明授权
    Derivative of ester of carboxylic acid, and insecticide and insect proofing agent containing the same 失效
    羧酸酯衍生物和含有其的杀虫剂和防虫剂

    公开(公告)号：US6107339A

    公开(公告)日：2000-08-22

    申请号：US722029

    申请日：1996-11-01

    申请人： Yoshio Katsuda ,  Koji Nakayama ,  Yoshihiro Minamite

    发明人： Yoshio Katsuda ,  Koji Nakayama ,  Yoshihiro Minamite

    IPC分类号： A01N53/00 ,  A01N53/06 ,  A01P7/04 ,  C07C67/08 ,  C07C69/743 ,  C07D307/45 ,  C07D317/54

    CPC分类号： C07D307/42 ,  A01N53/00 ,  C07C69/743 ,  C07D317/54

    摘要： The derivatives of esters of carboxylic acids represented by the general formula I: ##STR1## wherein: R.sub.1 is an alkyl group having a chain or branched chain of 1 to 4 carbon atoms; andR.sub.2 is a group represented by the following general formulae II, III or IV; ##STR2## wherein: R.sub.3 is a hydrogen atom or a methyl group;X is an oxygen atom or a methylidene group;R.sub.4 is an hydrogen atom or an ethynyl group;R.sub.5 and R.sub.6 are alike or differently selected from the group consisting of hydrogen, fluorine, chlorine atoms or methyl group;R.sub.7 is a hydrogen atom or a trifluoromethyl group;R.sub.8 is selected from the group consisting of propargyl, methoxymethyl or methylthio groups; orR.sub.7 and R.sub.8 may combine with each other to form a methylenedioxy chain; and the process for manufacturing the same, and the insecticides and the insect proofing agents containing the same as an active ingredient.The compounds represented by the general formula I are useful ingredients of insecticides and insect proofing agents which have both a fast-acting property and a lethal effect, and moreover, are highly safe to mammals; and therefore, insecticides and insect proofing agents containing the above compounds have a highly practical use.

    摘要翻译： PCT No.PCT / JP96 / 00254 Sec。 371日期：1996年11月1日 102（e）1996年11月1日PCT PCT 1996年2月7日PCT公布。 第WO96 / 24573号公报 日期：1996年8月15日由通式I表示的羧酸酯衍生物：其中：R1是具有1至4个碳原子的链或支链的烷基; R2是由下列通式II，III或IV表示的基团; 其中：R3是氢原子或甲基; X是氧原子或亚甲基; R4是氢原子或乙炔基; R 5和R 6相同或不同地选自氢，氟，氯原子或甲基; R7是氢原子或三氟甲基; R8选自炔丙基，甲氧基甲基或甲硫基; 或者R 7和R 8可以相互结合形成亚甲二氧基链; 及其制造方法，以及含有该活性成分的杀虫剂和防虫剂。 由通式I表示的化合物是具有快速作用性和致死作用的杀虫剂和防虫剂的有用成分，而且对哺乳动物是高度安全的; 因此，含有上述化合物的杀虫剂和防虫剂具有非常实用的用途。

    Process for the preparation of an oxirane, azirdine or cyclopropane
    7.
    发明授权
    Process for the preparation of an oxirane, azirdine or cyclopropane 失效
    制备环氧乙烷，氮杂环丁烷或环丙烷的方法

    公开(公告)号：US5703246A

    公开(公告)日：1997-12-30

    申请号：US617755

    申请日：1996-03-15

    申请人： Varinder Kumar Aggarwal ,  Hesham Nimer Hasan Abdel-Rahman ,  Hee Yoon Lee

    发明人： Varinder Kumar Aggarwal ,  Hesham Nimer Hasan Abdel-Rahman ,  Hee Yoon Lee

    IPC分类号： C07B37/10 ,  C07B41/00 ,  C07B43/00 ,  C07C2/86 ,  C07C13/04 ,  C07C13/28 ,  C07C45/68 ,  C07C49/293 ,  C07C69/743 ,  C07C69/753 ,  C07C211/16 ,  C07C303/30 ,  C07C303/34 ,  C07C303/40 ,  C07C315/04 ,  C07D203/02 ,  C07D203/22 ,  C07D203/24 ,  C07D301/02 ,  C07D303/04 ,  C07D303/08 ,  C07D303/16 ,  C07D303/40 ,  C07D303/46 ,  C07D407/04 ,  C07F9/564 ,  C07C203/00

    CPC分类号： C07D203/22 ,  C07C2/868 ,  C07D203/02 ,  C07D203/24 ,  C07D301/02 ,  C07D303/04 ,  C07D303/08 ,  C07D303/16 ,  C07D303/40 ,  C07D303/46 ,  C07D407/04 ,  C07F9/564 ,  C07C2101/02

    摘要： A process for the preparation of an oxirane, aziridine or cyclopropane of formula (I) wherein, X is oxygen, NR.sup.4 or CHR.sup.5 ; R.sup.1 is hydrogen, alkyl, aryl, heteroaromatic, heterocyclic or cycloalkyl; R.sup.2 is hydrogen, alkyl, aryl, heteroaromatic, CO.sub.2 R.sup.8, CHR.sup.14 NHR.sup.13, heterocyclic or cycloalkyl; or R.sup.1 and R.sup.2 join together to form a cycloalkyl ring; R.sup.3 is hydrogen, alkyl, aryl, heteroaromatic, CO.sub.2 R.sup.8, R.sup.8.sub.3 Sn, CONR.sup.8 R.sup.9 or trimethylsilyl; R.sup.4 and R.sup.5 are, independently, alkyl, cycloalkyl, aryl, heteroaromatic, SO.sub.2 R.sup.8, SO.sub.3 R.sup.8, COR.sup.8, CO.sub.2 R.sup.8, CONR.sup.8 R.sup.9 or CN, or R.sup.4 can also be P(O)(aryl).sub.2 ; R.sup.8 and R.sup.9 are independently alkyl, aryl or arylalkyl; R.sup.13 and R.sup.14 are independently hydrogen, alkyl or aryl; the process comprising reacting a mixture of a compound of formula (II), wherein R.sup.1, R.sup.2 and X are as defined above, and a sulphide of formula SR.sup.6 R.sup.7, wherein R.sup.6 and R.sup.7 are independently alkyl, aryl or heteroaomatic, or R.sup.6 and R.sup.7 join together to form a cycloalkyl ring which optionally includes an additional heteroatom, with either (i) a metallocarbon obtainable by reacting an alkylmetal with a methane derivative of formula CHR.sup.3 X'X", wherein R.sup.3 is as defined above, and X' and X" are independently, a leaving group, or (ii) a metallocarbon obtainable by reacting a compound of formula (III), (wherein R.sup.3 may not be hydrogen) with a suitable organometallic or inorganic reagent.

    摘要翻译： PCT No.PCT / GB94 / 02280第 371日期：1996年3月15日 102（e）1996年3月15日PCT 1994年10月19日PCT PCT。 公开号WO95 / 11230 日期：1995年04月27日制备式（I）的环氧乙烷，氮丙啶或环丙烷的方法，其中X是氧，NR 4或CHR 5; R 1是氢，烷基，芳基，杂芳族，杂环或环烷基; R2是氢，烷基，芳基，杂芳族，CO2R8，CHR14NHR13，杂环或环烷基; 或R 1和R 2连接在一起形成环烷基环; R3是氢，烷基，芳基，杂芳族，CO2R8，R83Sn，CONR8R9或三甲基甲硅烷基; R4和R5独立地是烷基，环烷基，芳基，杂芳族，SO2R8，SO3R8，COR8，CO2R8，CONR8R9或CN，或R4也可以是P（O）（芳基）2; R8和R9独立地是烷基，芳基或芳基烷基; R 13和R 14独立地是氢，烷基或芳基; 该方法包括使式（II）化合物（其中R 1，R 2和X如上所定义）和式SR 6 R 7的硫化物的混合物反应，其中R 6和R 7独立地为烷基，芳基或杂芳基，或R 6和R 7连接 一起形成任选地包括另外的杂原子的环烷基环，与（i）通过使烷基金属与式CHR 3 X'X“的甲烷衍生物反应得到的金属碳，其中R 3如上所定义，X'和X' 独立地是离去基团，或（ii）可通过使式（III）化合物（其中R 3可以不是氢）与合适的有机金属或无机试剂反应得到的金属碳。

    Vinylsulfone nor-pyrethric compounds
    9.
    发明授权
    Vinylsulfone nor-pyrethric compounds 失效
    乙烯基砜除虫菊酯化合物

    公开(公告)号：US5329017A

    公开(公告)日：1994-07-12

    申请号：US51177

    申请日：1993-04-22

    申请人： Didier Babin ,  Jean-Pierre Demoute ,  Jean Tessier

    发明人： Didier Babin ,  Jean-Pierre Demoute ,  Jean Tessier

    IPC分类号： C07C69/743 ,  C07D327/04

    CPC分类号： C07C69/743

    摘要： Novel all possible stereoisomers and mixtures thereof of vinylsulfone nor-pyrethric compounds of the formula ##STR1## wherein R.sub.a is selected from the group consisting of alkyl of 1 to 18 carbon atoms, alkenyl and alkynyl of 2 to 18 carbon atoms, cycloalkyl of 3 to 18 carbon atoms, cycloalkylalkyl of 4 to 18 carbon atoms and aryl of 6 to 14 carbon atoms unsubstituted or substituted with at least one functional group, n is 0, 1 or 2, R.sub.b is selected from the group consisting of alkyl of 1 to 18 carbon atoms, alkenyl and alkynyl of 2 to 18 carbon atoms, cycloalkyl of 3 to 18 carbon atoms, cycloalkylalkyl of 4 to 18 carbon atoms and aryl of 6 to 14 carbon atoms, all unsubstituted or unsubstituted with at least one functional group or R.sub.a and R.sub.b together with the C-S-C to which they are attached form ##STR2##

    摘要翻译： 其中R a选自1至18个碳原子的烷基，2至18个碳原子的烯基和炔基，3个环烷基的全部可能的立体异构体及其混合物， 至18个碳原子，4至18个碳原子的环烷基烷基和未被取代或被至少一个官能团取代的6至14个碳原子的芳基，n为0,1或2，Rb选自1至 2至18个碳原子的烯基和炔基，3至18个碳原子的环烷基，4至18个碳原子的环烷基烷基和6至14个碳原子的芳基，全部未取代或未取代，至少有一个官能团或Ra 和Rb与它们所连接的CSC一起形成