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公开(公告)号：WO2008130321A3
公开(公告)日：2008-10-30
申请号：PCT/SE2008/050460
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , KERS, Inger , MACSARI, Istvan , NYLÖF, Martin , ROTTICCI, Didier
Inventor： BESIDSKI, Yevgeni , KERS, Inger , MACSARI, Istvan , NYLÖF, Martin , ROTTICCI, Didier
IPC: C07D405/12 , A61K31/341 , A61K31/353 , A61K31/357 , A61K31/4155 , A61K31/4192 , A61K31/428 , A61K31/4418 , A61K31/4709 , A61K31/4725 , A61K31/495 , A61P29/00 , C07D213/82 , C07D249/06 , C07D295/135 , C07D307/68 , C07D311/20 , C07D417/12
Abstract: The present invention relates to new compounds. The present invention relates to new compounds, to pharmaceutical composition containing said compounds and to the use of said compounds in therapy. The present invention further relates to processes for the preparation of said compounds and to new intermediates useful in the preparation thereof.
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公开(公告)号：WO2008130319A2
公开(公告)日：2008-10-30
申请号：PCT/SE2008050458
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI YEVGENI , CLAESSON ALF , CSJERNYIK GABOR , GRAVENFORS YLVA , KERS INGER , SKOGHOLM KARIN , SOHN DANIEL
Inventor： BESIDSKI YEVGENI , CLAESSON ALF , CSJERNYIK GABOR , GRAVENFORS YLVA , KERS INGER , SKOGHOLM KARIN , SOHN DANIEL
IPC: C07D405/12 , C07C235/54 , C07C309/65 , C07D211/46 , C07D217/04
CPC classification number: C07C309/65 , C07C235/54 , C07C2602/10 , C07D211/46 , C07D217/04 , C07D405/12
Abstract: The present invention relates to new compounds and to pharmaceutical composition containing said compounds and to the use of said compounds in therapy. The present invention further relates to processes for the preparation of said compounds and to new intermediates useful in the preparation thereof.
Abstract translation: 本发明涉及新化合物和含有所述化合物的药物组合物和所述化合物在治疗中的用途。 本发明还涉及制备所述化合物的方法和可用于其制备的新中间体。
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3.发明申请NOVEL BENZIMIDAZOLE DERIVATIVES AS VANILLOID RECEPTOR 1 (VRL) INHIBITORS 审中-公开新型苯并咪唑衍生物作为VANILLOID受体1（VRL）抑制剂
公开(公告)号：WO2007073303A3
公开(公告)日：2007-08-30
申请号：PCT/SE2006001467
申请日：2006-12-21
Applicant: ASTRAZENECA AB , BESIDSKI YEVGENI , GRIFFIN ANDREW , LABRECQUE DENIS , JOHNSTONE SHAWN , JONES PAUL , KERS INGER , NYLOEF MARTIN , SKOGHOLM KARIN
Inventor： BESIDSKI YEVGENI , GRIFFIN ANDREW , LABRECQUE DENIS , JOHNSTONE SHAWN , JONES PAUL , KERS INGER , NYLOEF MARTIN , SKOGHOLM KARIN
IPC: C07D235/08 , A61K31/4184 , A61K31/4439 , A61P1/04 , A61P11/06 , A61P17/06 , A61P19/02 , A61P29/00 , A61P35/00 , C07D401/12 , C07D405/12 , C07D409/12
CPC classification number: C07D401/12 , C07D235/08 , C07D405/12 , C07D409/12
Abstract: The present invention relates to new compounds (I) or salts, solvates or solvated salts thereof, processes for their preparation and to new intermediates used in the preparation thereof, pharmaceutical compositions containing said compounds and to the use of said compounds in therapy.
Abstract translation: 本发明涉及新化合物（I）或其盐，溶剂合物或溶剂化盐，其制备方法及其制备中使用的新中间体，含有所述化合物的药物组合物和所述化合物在治疗中的用途。
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4.发明申请NOVEL N- (8-HETEROARYLTETRAHYDRONAPHTALENE-2YL) OR N- (5- HETEROARYLCHROMANE-3-YL) CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN 审中-公开用于治疗疼痛的新型N-（8-羟基乙基四氢呋喃-2-基）或N-（5-异喹啉-3-基）羧酰胺衍生物
公开(公告)号：WO2008130320A3
公开(公告)日：2008-12-18
申请号：PCT/SE2008050459
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI YEVGENI , KERS INGER , NYLOEF MARTIN , SANDBERG LARS , SKOGHOLM KARIN
Inventor： BESIDSKI YEVGENI , KERS INGER , NYLOEF MARTIN , SANDBERG LARS , SKOGHOLM KARIN
IPC: C07D405/14 , A61K31/415 , A61K31/4192 , A61K31/42 , A61K31/4418 , A61K31/4433 , A61K31/4439 , A61K31/455 , A61K31/506 , A61P29/00 , C07D213/75 , C07D231/12 , C07D261/08 , C07D401/12 , C07D403/12 , C07D405/04 , C07D413/12
CPC classification number: C07D405/14
Abstract: The present invention relates to new compounds of formula (I) and to pharmaceutical composition containing said compounds and to the use of said compounds in therapy. The present invention further relates to processes for the preparation of said compounds and to new intermediates useful in the preparation thereof.
Abstract translation: 本发明涉及新的式（I）化合物和含有所述化合物的药物组合物和所述化合物在治疗中的用途。 本发明还涉及制备所述化合物的方法和可用于其制备的新中间体。
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公开(公告)号：WO2008130320A2
公开(公告)日：2008-10-30
申请号：PCT/SE2008/050459
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , SANDBERG, Lars , SKOGHOLM, Karin
Inventor： BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , SANDBERG, Lars , SKOGHOLM, Karin
IPC: C07D405/14 , A61K31/415 , A61K31/4192 , A61K31/42 , A61K31/4418
CPC classification number: C07D405/14
Abstract: The present invention relates to new compounds of formula (I) and to pharmaceutical composition containing said compounds and to the use of said compounds in therapy. The present invention further relates to processes for the preparation of said compounds and to new intermediates useful in the preparation thereof.
Abstract translation: 本发明涉及新的式（I）化合物和含有所述化合物的药物组合物和所述化合物在治疗中的用途。 本发明还涉及制备所述化合物的方法和可用于其制备的新中间体。
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Patent Agency Ranking
公开(公告)号：WO2004100865A2
公开(公告)日：2004-11-25
申请号：PCT/SE2004/000738
申请日：2004-05-13
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , ROTTICCI, Didier , SLAITAS, Andis , SVENSSON, Mats
Inventor： BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , ROTTICCI, Didier , SLAITAS, Andis , SVENSSON, Mats
IPC: A61K
CPC classification number: C07D209/08 , C07C215/16 , C07C229/56 , C07C233/15 , C07C233/47 , C07C311/16 , C07C317/14 , C07C317/36 , C07D235/06 , C07D235/08 , C07D401/12 , C07D403/04 , C07D405/12 , C07D417/12
Abstract: The present invention relates to new compounds of formula (I) wherein R 1 to R 9 are as defined as in formula I, or salts, solvates or solvated salts thereof, processes for their preparation and to new intermediates used in the preparation thereof, pharmaceutical formulations containing said compounds and to the use of said compounds in therapy.
Abstract translation: 本发明涉及新的式（I）化合物，其中R 1至R 9如式I中所定义，或其盐，溶剂合物或溶剂化盐，其制备方法和用于 其制备方法，含有所述化合物的药物制剂和所述化合物在治疗中的用途。
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公开(公告)号：WO2012039657A1
公开(公告)日：2012-03-29
申请号：PCT/SE2010/051021
申请日：2010-09-22
Applicant: ASTRAZENECA AB , AURELL, Carl-Johan , BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin
Inventor： AURELL, Carl-Johan , BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin
IPC: C07D405/14 , A61K31/497 , A61P29/00
CPC classification number: C07D405/14 , C07D311/62 , C07D405/04 , C07F5/025
Abstract: The present invention relates to the compound N-[(3S)-5-(5-methoxypyrazin-2-yl)-3,4- dihydro-2H-chromen-3-yl]-6-[(2,2,2-trifluoroethoxy)methyl]pyridine-3-carboxamide, or a pharmaceutical composition comprising said compound and to the use of said compounds in therapy.
Abstract translation: 本发明涉及化合物N - [（3S）-5-（5-甲氧基吡嗪-2-基）-3,4-二氢-2H-色烯-3-基] -6 - [（2,2,2 - 三氟乙氧基）甲基]吡啶-3-甲酰胺，或包含所述化合物的药物组合物和所述化合物在治疗中的用途。
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8.发明申请
公开(公告)号：WO2008130319A3
公开(公告)日：2008-10-30
申请号：PCT/SE2008/050458
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , CLAESSON, Alf , CSJERNYIK, Gabor , GRAVENFORS, Ylva , KERS, Inger , SKOGHOLM, Karin , SOHN, Daniel
Inventor： BESIDSKI, Yevgeni , CLAESSON, Alf , CSJERNYIK, Gabor , GRAVENFORS, Ylva , KERS, Inger , SKOGHOLM, Karin , SOHN, Daniel
IPC: C07D405/12 , C07C235/54 , C07C309/65 , C07D211/46 , C07D217/04 , C07D249/06 , C07D263/34 , C07D265/30 , C07D295/088 , C07D295/135 , C07D295/155 , C07D295/192 , C07D311/74 , C07D401/12 , C07D413/12
Abstract: The present invention relates to new compounds and to pharmaceutical composition containing said compounds and to the use of said compounds in therapy. The present invention further relates to processes for the preparation of said compounds and to new intermediates useful in the preparation thereof.
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公开(公告)号：WO2006033620A1
公开(公告)日：2006-03-30
申请号：PCT/SE2005/001364
申请日：2005-09-19
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , SLAITAS, Andis
Inventor： BESIDSKI, Yevgeni , KERS, Inger , NYLÖF, Martin , SLAITAS, Andis
IPC: C07D401/04 , A61K31/4184 , A61K31/4439 , A61P29/00 , C07D235/06 , C07D405/12
CPC classification number: C07D235/08 , C07D401/04 , C07D403/12 , C07D405/12
Abstract: The present invention relates to new compounds (I) or salts, solvates or solvated salts thereof, processes for their preparation and to new intermediates used in the preparation thereof, pharmaceutical compositions containing said compounds and to the use of said compounds in therapy.
Abstract translation: 本发明涉及新化合物（I）或其盐，溶剂合物或溶剂化盐，其制备方法及其制备中使用的新中间体，含有所述化合物的药物组合物和所述化合物在治疗中的用途。
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10.发明申请
公开(公告)号：WO2008130322A1
公开(公告)日：2008-10-30
申请号：PCT/SE2008/050461
申请日：2008-04-22
Applicant: ASTRAZENECA AB , BESIDSKI, Yevgeni , GRAVENFORS, Ylva , KERS, Inger , NYLÖF, Martin , ROTTICCI, Didier
Inventor： BESIDSKI, Yevgeni , GRAVENFORS, Ylva , KERS, Inger , NYLÖF, Martin , ROTTICCI, Didier
IPC: C07D405/12 , A61K31/353 , A61K31/381 , A61K31/4025 , A61K31/4155 , A61K31/4178 , A61K31/422 , A61K31/4433 , A61K31/506 , A61P29/00 , C07D311/04 , C07D409/12 , C07D413/12 , C07D413/14
CPC classification number: C07D413/12 , C07D311/58 , C07D405/12 , C07D409/12 , C07D413/14
Abstract: The present invention relates to new compounds and pharmaceutically-acceptable salts thereof,and to new intermediates used in the preparation thereof, pharmaceutical compositions containing said compounds and to the use of said compounds in therapy.
Abstract translation: 本发明涉及新化合物及其药学上可接受的盐，以及其制备中使用的新中间体，含有所述化合物的药物组合物和所述化合物在治疗中的用途。
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