摘要:
Succinoylamino hydroxyethylamino sulfonyl urea derivatives of the formula: wherein R1-R6, R7, R7′, R8, R30-R34, X′, Y, Y′, t, x, and n are as defined herein, are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
摘要翻译:下式的琥珀酰氨基羟基氨基磺酰脲衍生物:其中R 1,R 6,R 7,R 7, R 8,R 30,R 34,X',Y,Y',t,x和n如本文所定义, 作为逆转录病毒蛋白酶抑制剂是有效的,特别是作为HIV蛋白酶的抑制剂。
摘要:
A method and apparatus for providing a real-time multimedia fishing tournament weigh-in data distribution system over the Internet. The system includes a data detection module for detecting components of real-time multimedia fishing tournament data. A client module residing at a tournament site obtains and distributes multimedia fishing tournament data received from the data detection module to a server module via the Internet. The server module in turn processes and streams the processed real-time multimedia fishing tournament data to one or more users coupled to the Internet.
摘要:
A synthesis is described for intermediates which are readily amenable to the large scale preparation of hydroxyethylurea-based chiral HIV protease inhibitors. The method includes forming a diastereoselective epoxide from a chiral alpha amino aldehyde.
摘要:
A process for the coupled production of alkyl tert-butyl ethers and butene oligomers from a mixture containing isobutane and n-butane. The isobutane is converted to the alkyl tert-butyl ether and the n-butane is converted to the oligomers. The ratio of the two reaction products may be controlled by setting the ratio of n-butane to isobutane appropriately by isomerization.
摘要:
A process and apparatus for measurement of nonuniformity of mass of a gyro rotor having a single bearing. The gyro rotor, which is mounted in a radially fixed and spherically yielding pivot, is rotated to a predetermined speed. The static imbalance of the rotating rotor is then determined by measuring the magnitude and angular position of excursion of the rotating rotor. A force couple acting on the gyro rotor and drift of mass of the gyro rotor are determined by sensing movement of a surface of the rotating rotor at two different times. Preferably, the determination of static imbalance, force couple, and drift are obtained in a single course of measurement. After the preceding have been measured, the components of a mass balancing operation for correcting the measured nonuniformities are determined.
摘要:
A print paste for printing textiles of polyester, cellulose acetate, cellulose triacetate and mixtures of the same with other fibers which is based on a disperse dye, thickener, ethanolamide of a carboxylic acid and water and which is characterized by a content of at least one phenol which has been oxyethylated twice to six times. The paste yields prints having excellent color strength and levelness.
摘要:
A spinal fixation device including two plates and a coupling element for coupling the plates in a fixed manner about adjacent spinous processes of the spine. Each plate is preferably equipped with integral spikes on the inwardly facing surfaces for pressing into the spinal processes and thereby augmenting the purchase between the plates and the spinous processes. Each plate contains a central aperture through which the coupling element passes in order to couple the plates together.
摘要:
A surgical fixation system having an improved mechanism to prevent the back out of screws employed in securing a surgical fixation plate to an intended orthopedic location.
摘要:
A spinal fixation apparatus comprising an upper and lower endplate. Depending distally in a longitudinal direction from the upper endplate is an inner sleeve that fits inside an outer sleeve that depends distally in a longitudinal direction from the lower endplate. The inner sleeve includes grooves located on its outer surface. A finger cage including resilient fingers fits around the outer sleeve. The fingers have ends that include male grooves. The ends of the fingers fit into apertures located in the outer sleeve. The apparatus further includes a locking mechanism that pushes the tips of the fingers through the apertures of the outer sleeve such that they mesh with the grooves of the inner sleeve. When the locking mechanism is unlocked the tips of the fingers disengage from the grooves of the inner sleeve, and the inner sleeve slide axially within the outer cage, adjusting the height of the device.
摘要:
N-heterocyclic moiety containing hydroxyethylamino compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.