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    Process for producing L-allysine acetals
    31.
    发明授权
    Process for producing L-allysine acetals 失效
    生产L-赖氨酸乙缩醛的方法

    公开(公告)号：US06174707B1

    公开(公告)日：2001-01-16

    申请号：US09202901

    申请日：1999-03-04

    Applicant: Naoaki Taoka ,  Takehiko Matsumoto ,  Kenji Inoue

    Inventor： Naoaki Taoka ,  Takehiko Matsumoto ,  Kenji Inoue

    IPC: G01N3853

    CPC classification number: C12P7/40 ,  C12P13/04 ,  C12P41/006

    Abstract: The present invention has for its object to provide a method for producing an L-allysine acetal which involves a fewer steps and is efficient. This invention relates to method for producing an L-allysine acetal which comprises; converting a D,L-allysine acetal of the following general formula (1) (wherein R1 and R2 are the same or different, and each of them represents an alkyl group having 1 to 8 carbon atoms, or they combinedly form a ring and represent an alkylene group having 2 to 8 carbon atoms) to a mixture of a 2-oxo-6,6-dialkoxyhexanoic acid of the following general formula (2) (wherein R1 and R2 are as defined above) and an L-allysine acetal of the following general formula (3) (wherein R1 and R2 are as defined above) by reacting in the presence of an enzyme capable of stereoselective oxidative deamination of D-amino acids and; isolating said L-allysine acetal after said converting.

    Abstract translation: 本发明的目的是提供一种生产L-赖氨酸缩醛的方法，该方法涉及较少的步骤并且是有效的。本发明涉及L-赖氨酸缩醛的制备方法，其包括：将D，L-烯丙基乙缩醛 的下述通式（1）（其中，R 1和R 2相同或不同，它们各自表示碳原子数1〜8的烷基，或者它们组合形成环，表示碳原子数2〜8的亚烷基 原子）与下述通式（2）的2-氧代-6,6-二烷氧基己酸（其中R 1和R 2如上定义）和下列通式（3）的L-烯丙基缩醛的混合物 其中R1和R2如上所定义）通过在能够进行D-氨基酸的立体选择性氧化脱氨作用的酶存在下反应;和在所述转化后分离所述L-赖氨酸缩醛。

    Shoe press belt and manufacturing method therefor
    32.
    发明授权
    Shoe press belt and manufacturing method therefor 失效
    鞋带及其制造方法

    公开(公告)号：US5968318A

    公开(公告)日：1999-10-19

    申请号：US94829

    申请日：1998-06-15

    Applicant: Yasuo Hasegawa ,  Kenji Inoue

    Inventor： Yasuo Hasegawa ,  Kenji Inoue

    IPC: D21F3/00 ,  D21F3/02 ,  D21F7/08 ,  B05D3/12

    CPC classification number: D21F3/0227 ,  D21F3/0236 ,  Y10S162/901

    Abstract: A shoe press belt for the shoe press of a paper making machine includes first and second resin layers and a base layer. Resin is coated and cured on the polished surface of a cylindrical mandrel to form the first resin layer endlessly. An inner layer of the base layer is formed by spirally winding a relatively narrower belt shaped mesh with warp threads running in the major direction of the belt and weft threads running perpendicular thereto, with the weft threads against the outer surface of the first resin layer, and without overlapping the end edges of the belt-shaped mesh. An outer layer of the base layer is formed by inserting the mandrel, with the first resin layer and the belt-shaped mesh layer applied, into a tubular mesh, and pulling the ends of the tubular mesh apart, so as to reduce its diameter and press it radially against the belt-shaped mesh layer. A second resin layer is then applied over the base layer and impregnates the base layer down to the outer surface of the first resin layer, so that the base layer is included within the second resin layer when the second resin layer is cured.

    Abstract translation: 用于造纸机的靴式压榨机的靴形压榨带包括第一和第二树脂层和基底层。 树脂在圆柱形心轴的抛光表面上被涂覆和固化，从而形成第一树脂层。 基层的内层通过螺旋卷绕相对较窄的带状网，通过沿着主带方向延伸的经线和垂直于其的纬纱螺旋卷绕，纬纱相对于第一树脂层的外表面， 并且不重叠带状网的端边缘。 基层的外层通过将第一树脂层和带状网层施加到管状网中并将管状网的端部分开来将芯棒插入，从而减小其直径和 将其径向按压在带状网格层上。 然后将第二树脂层施加在基层上，并将基底层浸渍到第一树脂层的外表面，使得当第二树脂层固化时，基层包含在第二树脂层内。

    Processes for producing .alpha.-halo ketones, .alpha.-halohydrins and epoxides
    33.
    发明授权
    Processes for producing .alpha.-halo ketones, .alpha.-halohydrins and epoxides 失效
    制备α-卤代酮，α-卤代醇和环氧化物的方法

    公开(公告)号：US5929284A

    公开(公告)日：1999-07-27

    申请号：US722102

    申请日：1996-12-18

    Applicant: Akira Nishiyama ,  Tadashi Sugawa ,  Hajime Manabe ,  Kenji Inoue ,  Noritaka Yoshida

    Inventor： Akira Nishiyama ,  Tadashi Sugawa ,  Hajime Manabe ,  Kenji Inoue ,  Noritaka Yoshida

    IPC: C07C29/143 ,  C07C45/48 ,  C07C269/06 ,  C07C319/20 ,  C07C323/43 ,  C07D303/36 ,  C07C45/00

    CPC classification number: C07D303/36 ,  C07C269/06 ,  C07C29/143 ,  C07C319/20 ,  C07C45/48

    Abstract: Processes for efficiently producing .alpha.-halo ketones, .alpha.-halohydrins and epoxides on an industrial scale. The prosesses include one for producing an .alpha.-halo ketone of general formula (3) by decarboxylating a product of reaction between a carboxilic acid derivative of general formula (1) and a metal enolate prepared from an .alpha.-haloacetic acid of general formula (2) or an acceptable salt thereof, one for producing an by reducing the .alpha.-halo ketone (3), and one for producing an epoxide (13) by treating the .alpha.-halohydrin (11) with a base to effect ring closure. The above prosesses are particularly suitable for producing optically active .alpha.-halo ketones, .alpha.-halohydrins and epoxides from the corresponding .alpha.-amino acid derivatives. ##STR1##

    Abstract translation: PCT No.PCT / JP96 / 00212 Sec。 371日期：1996年12月18日 102（e）1996年12月18日日期PCT 1996年2月2日PCT PCT。 第WO96 / 23756号公报 日期1996年8月8日工业规模高效生产α-卤代酮，α-卤代醇和环氧化物的方法。 前药包括通过使通式（1）的羧酸衍生物与由通式（2）的α-卤代乙酸制备的金属烯醇化物脱羧的方法来制备通式（3）的α-卤代酮， ）或其可接受的盐，其中通过用碱来还原α-卤代酮（3）和通过用碱处理α-卤代醇（11）来制备环氧化物（13）来制备，以实现闭环。 上述产品特别适用于从相应的α-氨基酸衍生物制备光学活性的α-卤代酮，α-卤代醇和环氧化物。

    Battery terminal with core wire end cover
    34.
    发明授权
    Battery terminal with core wire end cover 失效
    带芯线端盖的电池端子

    公开(公告)号：US5893781A

    公开(公告)日：1999-04-13

    申请号：US843386

    申请日：1997-04-15

    Applicant: Hideki Matsunaga ,  Kenji Inoue

    Inventor： Hideki Matsunaga ,  Kenji Inoue

    IPC: H01R4/38 ,  H01R4/70 ,  H01R11/12 ,  H01R11/28 ,  H01R4/42

    CPC classification number: H01R11/284 ,  Y10S439/948

    Abstract: A fastening member 30 of a battery terminal 10 has a core wire covering member 32 formed by bending a pair of protecting members 32a which extend from the root portion of a wire barrel 31. The core wire covering member 32 is between the connecting portion 20 and the usual wire barrel portion 31, and is approximately rectangular when seen in cross-section. A clamp bolt 50 and nut 51 are tightened by means of a spanner or the like, thereby attaching the battery terminal 10 to a battery post P. The covering member 32 ensures that the end of the core wire or loose strands of the core wire do not interfere with the tightening operation or become caught on the operator's hand or on a tool. The wire covering members 33, 34 may include inspection apertures 33c, 34b.

    Abstract translation: 电池端子10的紧固构件30具有通过弯曲从线筒31的根部延伸的一对保护构件32a而形成的芯线覆盖构件32.芯线覆盖构件32位于连接部20和 通常的线筒部分31，并且在横截面看时是大致矩形的。 夹紧螺栓50和螺母51通过扳手等紧固，从而将电池端子10连接到电池柱P.盖构件32确保芯线的末端或芯线的松散线做 不会干扰拧紧操作或被抓在操作者的手上或工具上。 电线覆盖部件33,34可以包括检查孔33c，34b。

    Method of producing 3-amino-2-hydroxy-1-propanol derivatives
    37.
    发明授权
    Method of producing 3-amino-2-hydroxy-1-propanol derivatives 失效
    3-氨基-2-羟基-1-丙醇衍生物的制备方法

    公开(公告)号：US5744630A

    公开(公告)日：1998-04-28

    申请号：US436344

    申请日：1995-07-18

    Applicant: Kenji Inoue ,  Hiroshi Awaji ,  Satomi Takahashi

    Inventor： Kenji Inoue ,  Hiroshi Awaji ,  Satomi Takahashi

    IPC: C07C271/16 ,  C07D263/24 ,  C07D263/20

    CPC classification number: C07D263/24 ,  C07C271/16 ,  Y02P20/55

    Abstract: The present invention has for its object to provide an efficient and economical method for producing an 3-amino-2-hydroxy-1-propanol derivative and an oxazolidinone derivative derived therefrom, both of which are of use as intermediates for the production of drugs including HIV protease inhibitors. The invention relates to a method for producing an 3-amino-2-hydroxy-1-propanol derivative of general formula (2) ##STR1## (wherein R.sup.1 represents alkyl, aralkyl or aryl; R.sup.2 and R.sup.3 independently represent hydrogen or an amino-protecting group, provided, however, that both R.sup.2 and R.sup.3 are not concurrently hydrogen) and an oxazolidinone derivative derived therefrom.

    Abstract translation: PCT No.PCT / JP94 / 01540 Sec。 371 1995年7月18日第 102（e）日期1995年7月18日PCT 1994年9月20日PCT PCT。 公开号WO95 / 08530 1995年3月30日发明内容本发明的目的是提供一种生产3-氨基-2-羟基-1-丙醇衍生物和衍生自其的恶唑烷酮衍生物的有效且经济的方法，它们均用作 生产药物包括HIV蛋白酶抑制剂。 本发明涉及制备通式（2）的3-氨基-2-羟基-1-丙醇衍生物的方法（2）（其中R1代表烷基，芳烷基或芳基; R2和R3独立地表示氢或 氨基保护基，但是R2和R3不同时为氢）和衍生自其的恶唑烷酮衍生物。

    Connector housing locking mechanism
    39.
    发明授权
    Connector housing locking mechanism 失效
    连接器外壳锁定机构

    公开(公告)号：US5711684A

    公开(公告)日：1998-01-27

    申请号：US589539

    申请日：1996-01-22

    Applicant: Kenji Inoue ,  Hiroyuki Hayashi

    Inventor： Kenji Inoue ,  Hiroyuki Hayashi

    IPC: H01R13/639 ,  H01R13/52 ,  H01R13/627

    CPC classification number: H01R13/6272 ,  H01R13/5205 ,  H01R13/5219

    Abstract: A female connector housing 11 has a locking arm 30 integrally moulded thereon, the locking arm 30 having a fitting projection 31. A male connector housing 21 has a fitting hole 24 formed on hood member 22 thereof. Two slots 34 are formed on either side of the fitting projection 31 so as to extend along the longitudinal direction of the locking arm 30. The locking arm 30 is thus partitioned into a fitting arm member 35 which includes the fitting projection 31, and two supporting arm members 36 which are formed on both sides thereof. The foot members 36a of the supporting arm members 36 are thicker than the foot member 35a of the fitting arm member 35, and thus the engagement load of the arm 30 is large, but the projection 35a is nevertheless relatively easy to disengage.

    Abstract translation: 阴连接器壳体11具有一体地模制在其上的锁定臂30，锁定臂30具有配合突起31.阳连接器壳体21具有形成在其罩部件22上的配合孔24。 两个槽34形成在嵌合突起31的两侧，以沿着锁定臂30的纵向方向延伸。因此，锁定臂30被分隔成包括配合突起31的配合臂构件35和两个支撑 臂部件36形成在其两侧。 支撑臂构件36的脚构件36a比装配臂构件35的脚构件35a厚，因此臂30的接合负荷大，但突起35a相对容易脱离。

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