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    Aminopropylaminobleomycin derivatives and process for preparation thereof
    41.
    发明授权
    Aminopropylaminobleomycin derivatives and process for preparation thereof 失效
    氨丙基氨基甜菜碱素衍生物及其制备方法

    公开(公告)号：US4537880A

    公开(公告)日：1985-08-27

    申请号：US635096

    申请日：1984-07-27

    Applicant: Hamao Umezawa ,  Akio Fujii ,  Yasuhiko Muraoka ,  Tokuji Nakatani ,  Takeyo Fukuoka ,  Katsutoshi Takahashi

    Inventor： Hamao Umezawa ,  Akio Fujii ,  Yasuhiko Muraoka ,  Tokuji Nakatani ,  Takeyo Fukuoka ,  Katsutoshi Takahashi

    IPC: C07H15/26 ,  A61K31/70 ,  A61K31/7028 ,  A61P35/00 ,  C07K9/00 ,  A61K37/00 ,  C07C103/52

    CPC classification number: C07K9/003 ,  Y10S930/19 ,  Y10S930/27

    Abstract: An aminopropylaminobleomycin represented by the following formula or a salt thereof, which is minimized in side effects such as pulmonary toxicity:[BX]--NH--(CH.sub.2).sub.3 --A--(CH.sub.2).sub.3 --Bwherein[BX] represents the acyl group of bleomycinic acid whose formula differs from that of bleomycin acid by the removal of the hydroxyl group from the carboxyl group of said acid;A represents a group of the general formula ##STR1## wherein R.sub.1 is a lower alkyl or benzyl,R.sub.2 is a lower alkyl or benzyl,R is a lower alkylene, andn is 0 or 1; andB represents a group of the formula ##STR2## wherein (i) R.sub.3 is hydrogen and R.sub.4 is(a) benzyl substituted by one or more halogen atoms, provided that the benzyl is substituted by two halogen atoms when R.sub.1 is lower alkyl,(b) benzyl substituted by cyano, two or more alkoxy groups or two or more benzyloxy groups,(c) lower alkyl substituted by cycloalkyl or anthranyl,(d) phenylethyl substituted by one or more halogen atoms, or(e) diphenylethyl; or(ii) both R.sub.3 and R.sub.4 are benzyl which may be substituted by one or more(a) benzyloxy groups,(b) ring substituted benzyloxy groups in which the ring substituents may be one or more halogen atoms, lower alkoxy groups or benzyloxy groups, or(c) cycloalkylmethoxy groups;and a process for the preparation thereof.

    Abstract translation: 由下式表示的氨丙基氨基伯基霉素或其盐，其在副作用如肺毒性方面最小化：[BX] -NH-（CH2）3-A-（CH2）3-B其中[BX]表示酰基 通过从所述酸的羧基除去羟基，其公式不同于博来霉素酸的博来霉素酸; A表示通式为其中R 1为低级烷基或苄基的基团，R 2为低级烷基或苄基，R为低级亚烷基，n为0或1; 并且B代表下式的基团：其中（i）R3是氢，R4是（a）被一个或多个卤素原子取代的苄基，条件是当R 1是低级烷基时，苄基被两个卤原子取代，（ （c）由氰基，两个或更多个烷氧基或两个或更多个苄氧基取代的苄基，（c）被环烷基或蒽基取代的低级烷基，（d）被一个或多个卤素原子取代的苯基乙基，或（e）二苯基乙基; 或（ii）R 3和R 4均为可被一个或多个（a）苄氧基取代的苄基，（b）环取代的苄氧基，其中环取代基可以是一个或多个卤素原子，低级烷氧基或苄氧基 ，或（c）环烷基甲氧基; 及其制备方法。

    Motor-driven compressor
    43.
    发明授权
    Motor-driven compressor 有权
    电动压缩机

    公开(公告)号：US09246320B2

    公开(公告)日：2016-01-26

    申请号：US13251425

    申请日：2011-10-03

    Applicant: Tetsuya Yamada ,  Ken Suitou ,  Shingo Enami ,  Akio Fujii

    Inventor： Tetsuya Yamada ,  Ken Suitou ,  Shingo Enami ,  Akio Fujii

    IPC: H02G15/013 ,  F04B35/04 ,  F04B39/12 ,  F04C23/00 ,  F04C18/02

    CPC classification number: H02G15/013 ,  F04B35/04 ,  F04B39/12 ,  F04B39/121 ,  F04C18/0215 ,  F04C23/008 ,  F04C2240/803

    Abstract: A motor-driven compressor includes a shell, an electric motor, a first conductor electrically connected to an external power source, a second conductor electrically connected to the electric motor, a connector connecting the first conductor and the second conductor and a connector case. The connector case has a first case member, a second case member, a first and a second seal members interposed between the first and the second case members, a hole through which the first conductor is inserted and a third seal member sealing between the first conductor and the connector case. A first main seal of the first seal member and a second main seal of the second seal member cooperate to form a cylindrical seal portion for sealing the second conductor that is inserted through the cylindrical seal portion when the first and the second seal members are joined.

    Abstract translation: 电动压缩机包括外壳，电动马达，电连接到外部电源的第一导体，电连接到电动机的第二导体，连接第一导体和第二导体的连接器以及连接器壳体。 连接器壳体具有第一壳体构件，第二壳体构件，插入在第一和第二壳体构件之间的第一和第二密封构件，插入第一导体的孔和密封在第一导体之间的第三密封构件 和连接器盒。 第一密封构件的第一主密封件和第二密封构件的第二主密封件协作以形成圆柱形密封部分，用于在第一和第二密封构件接合时密封插入通过圆柱形密封部分的第二导体。

    IMAGING APPARATUS
    44.
    发明申请
    IMAGING APPARATUS 有权
    成像设备

    公开(公告)号：US20120321274A1

    公开(公告)日：2012-12-20

    申请号：US13598004

    申请日：2012-08-29

    Applicant: Akio Fujii

    Inventor： Akio Fujii

    IPC: H04N5/77

    CPC classification number: H04N1/333 ,  H04N1/212 ,  H04N5/23245 ,  H04N5/772 ,  H04N5/781 ,  H04N5/85 ,  H04N5/907 ,  H04N9/7921 ,  H04N9/8042 ,  H04N9/8047 ,  H04N19/115 ,  H04N19/124 ,  H04N19/152 ,  H04N19/154 ,  H04N19/60 ,  H04N19/61 ,  H04N2201/212 ,  H04N2201/33357

    Abstract: An imaging apparatus includes a signal processing unit that generates moving image data and still image data using image data output from an imaging unit, a moving image coding unit that encodes the moving image data, a still image coding unit that encodes the still image data, a recording unit that records the coded moving and still image data on a recording medium, a setting unit that sets a data rate of the coded moving image data, and a control unit that controls the moving and still image coding units. The control unit controls the moving image coding unit based on the set data rate to adjust the data rate of the moving image data and the still image coding unit based on the set data rate and a recording data rate of the recording medium to adjust an amount of the still image data.

    Abstract translation: 一种成像装置，包括：信号处理单元，其使用从成像单元输出的图像数据生成运动图像数据和静止图像数据;运动图像编码单元，对运动图像数据进行编码;静止图像编码单元，对静止图像数据进行编码; 记录单元，其将编码的移动和静止图像数据记录在记录介质上，设置单元，其设置编码的运动图像数据的数据速率;以及控制单元，其控制移动和静止图像编码单元。 控制单元基于设定的数据速率来控制运动图像编码单元，以基于设定的数据速率和记录介质的记录数据速率来调整运动图像数据和静止图像编码单元的数据速率，以调整量 的静止图像数据。

    Product package and prize for crane claw arcade game
    45.
    发明授权
    Product package and prize for crane claw arcade game 有权
    产品包装和起重机爪游戏机奖

    公开(公告)号：US08011509B1

    公开(公告)日：2011-09-06

    申请号：US12752682

    申请日：2010-04-01

    Applicant: Yoshitaka Sakamaki ,  Akio Fujii ,  Darin Pilcher ,  Jim Wulfers

    Inventor： Yoshitaka Sakamaki ,  Akio Fujii ,  Darin Pilcher ,  Jim Wulfers

    IPC: A63F11/00

    CPC classification number: G07F17/3297 ,  G07F17/32

    Abstract: A package for storing a prize associated with a crane claw arcade game includes a sidewall, a first and second end panels, a cavity, at least one first side aperture, and optionally at least one second side aperture. The sidewall includes a plurality of side panels, wherein each includes opposing first and second side edges and opposing first and second end edges. The cavity is adapted to store the prize associated with the crane claw arcade game. The first side aperture is defined by a first side panel of the plurality of side panels, and the optional second side aperture is defined by a second side panel of the plurality of side panels. The first and second side apertures are adapted to receive a finger of a claw of the crane claw arcade game to facilitate retrieval of the package from a housing of the arcade game.

    Abstract translation: 用于存储与起重机爪拱形游戏机相关联的奖品的包装包括侧壁，第一和第二端板，空腔，至少一个第一侧孔和可选地至少一个第二侧孔。 侧壁包括多个侧板，其中每个包括相对的第一和第二侧边缘以及相对的第一和第二端边缘。 该腔适于存储与起重机爪游戏机相关联的奖品。 第一侧孔由多个侧板的第一侧板限定，并且可选的第二侧孔由多个侧板的第二侧板限定。 第一和第二侧孔适于接收起重机爪拱形游戏的爪的手指，以便于从街机游戏的外壳取回包装。

    MOTOR-DRIVEN COMPRESSOR
    47.
    发明申请
    MOTOR-DRIVEN COMPRESSOR 有权
    电机驱动压缩机

    公开(公告)号：US20110058973A1

    公开(公告)日：2011-03-10

    申请号：US12877249

    申请日：2010-09-08

    Applicant: Tetsuya YAMADA ,  Shingo Enami ,  Akio Fujii ,  Junya Yano ,  Ken Suitou

    Inventor： Tetsuya YAMADA ,  Shingo Enami ,  Akio Fujii ,  Junya Yano ,  Ken Suitou

    IPC: F04C15/00 ,  F04C2/02

    CPC classification number: F04C23/008 ,  F04C18/0215 ,  F04C2240/30 ,  F04C2240/803 ,  H01R13/405 ,  H01R13/533 ,  H02G3/22 ,  H02K5/12 ,  H02K5/225

    Abstract: A motor-driven compressor includes a compression mechanism, an electric motor, a compressor housing, a conductive member, a terminal base, an insulating member, a connection terminal, a wire assembly, a terminal housing, first and second holes formed through the terminal housing and first and second seal members. The conductive member extends from the inside to the outside of the compressor housing and connected electrically to the connection terminal at a terminal connection. The wire assembly has a core wire connecting electrically between the connecting terminal and the electric motor, and an insulator covering the core wire. The terminal housing disposed in the compressor housing covers the terminal connection. The wire assembly has an insulating tube covering the insulator, wherein both ends of the insulating tube are opened for communicating with the inside and the outside of the terminal housing through a clearance formed between the insulating tube and the insulator.

    Abstract translation: 电动压缩机包括压缩机构，电动机，压缩机壳体，导电构件，端子座，绝缘构件，连接端子，线组件，端子壳体，通过端子形成的第一和第二孔 外壳和第一和第二密封件。 导电构件从压缩机壳体的内部延伸到外部并且在端子连接处电连接到连接端子。 线组件具有在连接端子和电动机之间电连接的芯线，以及覆盖芯线的绝缘体。 设置在压缩机壳体中的端子壳体覆盖端子连接。 电线组件具有覆盖绝缘体的绝缘管，其中绝缘管的两端被打开以通过形成在绝缘管和绝缘体之间的间隙与端子壳体的内部和外部连通。

    2'-HYDROXY-PROTECTED RIBONUCLEOSIDE DERIVATIVE AND PRODUCTION METHOD THEREOF
    48.
    发明申请
    2'-HYDROXY-PROTECTED RIBONUCLEOSIDE DERIVATIVE AND PRODUCTION METHOD THEREOF 失效
    2'-羟基保护的核糖核苷衍生物及其生产方法

    公开(公告)号：US20110009609A1

    公开(公告)日：2011-01-13

    申请号：US12919295

    申请日：2009-02-26

    Applicant: Hirofumi Maeda ,  Akio Fujii ,  Masaru Mitsuda

    Inventor： Hirofumi Maeda ,  Akio Fujii ,  Masaru Mitsuda

    IPC: C07H19/22 ,  C07H19/00

    CPC classification number: C07H19/067 ,  C07H19/167

    Abstract: The present invention relates to a method for producing a 2′-hydroxy-protected nucleoside derivative by reacting a ribonucleoside with an acylating reagent in the presence of a metal complex consisting of a copper compound and an optically active ligand. By the method according to the present invention, a 2′-hydroxy-protected ribonucleoside derivative, which is an important intermediate for producing an oligonucleoside, can be easily produced with good regioselectivity from a nucleoside derivative of which 2′,3′-hydroxy groups are not protected.

    Abstract translation: 本发明涉及通过在由铜化合物和光学活性配体组成的金属络合物的存在下使核糖核苷与酰化剂反应来制备2'-羟基保护的核苷衍生物的方法。 通过本发明的方法，可以容易地制备作为制备寡核苷酸的重要中间体的2'-羟基保护的核糖核苷衍生物，其从2'，3'-羟基的核苷衍生物具有良好的区域选择性 没有保护。

    METHOD FOR PRODUCING OPTICALLY ACTIVE HYDROXYCARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF
    49.
    发明申请
    METHOD FOR PRODUCING OPTICALLY ACTIVE HYDROXYCARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF 失效
    生产光学活性羟基羧酸衍生物或其盐的方法

    公开(公告)号：US20100191011A1

    公开(公告)日：2010-07-29

    申请号：US12376803

    申请日：2007-08-08

    Applicant: Susumu Amano ,  Akio Fujii ,  Shohei Yamamoto ,  Masaru Mitsuda

    Inventor： Susumu Amano ,  Akio Fujii ,  Shohei Yamamoto ,  Masaru Mitsuda

    IPC: C07C51/347

    CPC classification number: C07B53/00 ,  C07B2200/07 ,  C07C51/00 ,  C07C51/367 ,  C07C201/12 ,  C07C59/48 ,  C07C205/56

    Abstract: The present invention has its object to provide a method for producing an optically active hydroxycarboxylic acid derivative which is an intermediate important for production of medicines, agrochemicals, chemical products, and so on. The production method of the present invention comprises: carrying out a hydrogen-transfer reduction of a ketocarboxylic acid or a salt thereof by the reaction of an optically active diamine complex to produce an optically active hydroxycarboxylic acid derivative. According to the present invention, it is possible to safely and efficiently produce an industrially-useful optically active hydroxycarboxylic acid derivative.

    Abstract translation: 本发明的目的在于提供一种光学活性羟基羧酸衍生物的制造方法，该方法是制备药物，农药，化学品等的重要中间体。 本发明的制造方法包括：通过光学活性二胺配合物的反应进行酮羧酸或其盐的氢转移还原反应，生成光学活性羟基羧酸衍生物。 根据本发明，可以安全有效地制备工业上有用的光学活性羟基羧酸衍生物。

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