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    Octacyclodepsipeptides having an endoparasiticidal action
    84.
    发明授权
    Octacyclodepsipeptides having an endoparasiticidal action 失效
    具有内寄生性杀伤作用的Octacyclodepsipeptide

    公开(公告)号：US06369028B1

    公开(公告)日：2002-04-09

    申请号：US08246029

    申请日：1994-05-19

    申请人： Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    发明人： Jürgen Scherkenbeck ,  Peter Jeschke ,  Hans-Georg Lerchen ,  Hermann Hagemann ,  Achim Harder ,  Norbert Mencke ,  Andrew Plant

    IPC分类号： A61K3800

    CPC分类号： C07D273/00 ,  C07C235/12 ,  C07C235/34

    摘要： The present invention relates to compounds of the general formula (I) in which R1, R2, R11 and R12 represent the same or different radicals selected from the group of C1-8-alkyl, C1-8-halogenoalkyl, C3-6-cycloalkyl, aralkyl or aryl, R3, R5, R7, R9, represent the same or different radicals selected from the group of hydrogen or straight-chain C1-5-alkyl or branched C4-7-alkyl which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl  carboxamide,  imidazolyl, indolyl, guanidino, —SH or C1-4-alkylthio, and furthermore represents aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, nitro or a —NR13R14 group in which R13 and R14 independently from each other represent hydrogen or alkyl or together with the adjoining nitrogen atom forms a 5, 6 or 7-membered ring which is optionally interrupted by O, S or N and which is optionally C1-4-alkyl substituted, R4, R6, R8, R10 represent the same or different radicals selected from the group of hydrogen, straight-chain C1-5-alkyl and represents isopropyl, sec.-butyl, t-butyl, C2-6-alkenyl, C3-7-cycloalkyl, which may optionally be substituted by hydroxyl, C1-4-alkoxy, carboxyl, carboxamide, imidazolyl, indolyl, guanidino, SH or C1-4-alkylthio and represent aryl, aralkyl or heteroarylmethyl which may be substituted by halogen, hydroxyl, C1-4-alkyl, C1-4-alkoxy, and stereoisomers thereof, to processes for their preparation and to their use as endoparasiticides.

    摘要翻译： 本发明涉及通式（I）的化合物，其中R 1，R 2，R 11和R 12表示相同或不同的选自C 1-8 - 烷基，C 1-8 - 卤代烷基，C 3-6 - 环烷基， 芳烷基或芳基，R 3，R 5，R 7，R 9表示相同或不同的选自氢或直链C 1-5烷基或支链C 4-7 - 烷基的基团，其可任选被羟基，C 1-4 烷氧基，羧基羧酰胺，咪唑基，吲哚基，胍基，-SH或C 1-4 - 烷硫基，此外表示可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基，硝基取代的芳基，芳烷基或杂芳基甲基 或-NR 13 R 14基团，其中R 13和R 14彼此独立地表示氢或烷基或与相邻的氮原子一起形成可选地被O，S或N中断的5,6或7-元环，并且其任选地为C1 R 4，R 6，R 8，R 10表示选自该基团的相同或不同的基团 的氢，直链C1-5 - 烷基，代表异丙基，仲丁基，叔丁基，C 2-6 - 烯基，C 3-7 - 环烷基，其可任选被羟基，C 1-4 - 烷氧基， 羧基，羧酰胺，咪唑基，吲哚基，胍基，SH或C 1-4 - 烷硫基，代表可被卤素，羟基，C 1-4 - 烷基，C 1-4 - 烷氧基及其立体异构体取代的芳基，芳烷基或杂芳基甲基， 其制备方法及其作为内寄生物杀虫剂的用途。

    Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas
    90.
    发明授权
    Pesticidal tautomers of 3-aryl-pyrrolidine-2,4-diones and use thereas 失效
    3-芳基 - 吡咯烷-2,4-二酮的杀虫互变异构体

    公开(公告)号：US5045560A

    公开(公告)日：1991-09-03

    申请号：US460208

    申请日：1990-01-02

    申请人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hagemann ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    发明人： Reiner Fischer ,  Bernd Baasner ,  Hermann Hagemann ,  Andreas Krebs ,  Albrecht Marhold ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Klaus Lurssen ,  Benedikt Becker ,  Klaus Schaller ,  Harry Strang

    IPC分类号： A01N43/36 ,  A01N47/06 ,  C07D207/38 ,  C07D405/12

    CPC分类号： C07D405/12 ,  A01N43/36 ,  A01N47/06 ,  C07D207/38

    摘要： Insecticidal, acaricidal, herbicidal and antimycotic 3-aryl-pyrrolidine-2,4-diones of the formula ##STR1## in which X represents alkyl, halogen or alkoxy,Y represents hydrogen, alkyl, halogen, alkoxy or halogenoalkyl,Z represents alkyl, halogen or alkoxy,n represents a number from 0-3,R represents hydrogen or represents the groups --CO--R.sup.1 or --CO--O--R.sup.2, in whichR.sup.1 represents alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl or cycloalkyl which can be interrupted by hetero atoms, each of which radicals is optionally substituted by halogen, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl or substituted hetaryloxyalkyl, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, andR.sup.2 represents alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl or optionally substituted phenyl or cycloalkyl, each of which radicals is optionally substituted by halogen,A represents alkyl, alkenyl, alkinyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl which is optionally interrupted by a hetero atom, each of which radicals is optionally substituted by halogen, or represents arylalkyl which is optionally substituted by halogen, alkyl, halogenoalkyl, alkoxy or nitro,B and C* independently of one another represent hydrogen, alkyl or alkoxyalkyl.

    摘要翻译： 式（I）的杀虫，杀螨，除草和抗真菌性3-芳基 - 吡咯烷-2,4-二酮其中X代表烷基，卤素或烷氧基，Y代表氢，烷基，卤素，烷氧基或卤代烷基，Z 表示烷基，卤素或烷氧基，n表示0-3的数，R表示氢或表示基团-CO-R1或-CO-O-R2，其中R1表示烷基，烯基，烷氧基烷基，烷硫基烷基，聚烷氧基烷基或环烷基 任何取代的苯基，取代的杂芳基，取代的苯氧基烷基或取代的噻唑烷基，或代表任意取代的苯基，任选取代的苯基烷基，取代的杂芳基， 取代的苯氧基烷基和取代的硫代氧基烷基，R 2表示烷基，链烯基，烷氧基烷基，聚烷氧基烷基或任选取代的苯基或环烷基，各w 任选被卤素取代的基团，A代表烷基，链烯基，炔基，烷氧基烷基，聚烷氧基烷基，烷硫基烷基或环烷基，任选被杂原子间隔，每个基团任选被卤素取代，或表示任选取代的芳基烷基 卤素，烷基，卤代烷基，烷氧基或硝基，B和C *彼此独立地表示氢，烷基或烷氧基烷基。