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公开(公告)号:US5719146A
公开(公告)日:1998-02-17
申请号:US597780
申请日:1996-02-07
申请人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
IPC分类号: A01N43/64 , A01N43/653 , A01N43/72 , A01N43/80 , A01N43/832 , A01N43/836 , A01N43/84 , A01N43/88 , A01N47/40 , A01N51/00 , C07D401/06 , C07D401/14 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D419/06
CPC分类号: C07D401/06 , A01N47/40 , A01N51/00 , C07D401/14 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D419/06
摘要: Insecticidal heterocyclic compounds of the formula ##STR1## wherein A represents a five-membered or six-membered heteroaryl group containing one to three hetero atoms selected from the group consisting of S, O and N, said heteroaryl group being unsubstituted or substituted by a halogen atom or C.sub.1-4 alkyl group, Z represents a three-membered straight chain, each member being selected from the group consisting of CH.sub.2 --, O, S and N--R.sup.2 with at least one of said three members being O, S or N--R.sup.2, E represents CH.sub.2, O, S or N--R.sup.2, wherein R.sup.2 represents a hydrogen atom, a C.sub.1-4 alkyl group, a C.sub.1-4 alkoxy group or the group ##STR2## wherein R.sup.3 represents a hydrogen atom or halogen atom, X represents CH or N, Y represents a nitro group or cyano group, and R.sup.1 represents a hydrogen atom or methyl group.
摘要翻译: 式(I)的杀虫杂环化合物其中A表示含有1-3个选自S,O和N的杂原子的五元或六元杂芳基,所述杂芳基是未取代或取代的 通过卤原子或C 1-4烷基,Z表示三元直链,每个成员选自CH 2 - ,O,S和N-R 2,所述三个成员中的至少一个为O, S或N-R2,E表示CH 2,O,S或N-R 2,其中R 2表示氢原子,C 1-4烷基,C 1-4烷氧基或基团,其中R 3表示氢原子 或卤原子,X表示CH或N,Y表示硝基或氰基,R 1表示氢原子或甲基。
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公开(公告)号:US5622956A
公开(公告)日:1997-04-22
申请号:US461903
申请日:1995-06-05
申请人: Kozo Shiokawa , Shinichi Tsuboi , Shoko Sasaki , Koichi Moriya , Yumi Hattori , Katsuhiko Shibuya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Shoko Sasaki , Koichi Moriya , Yumi Hattori , Katsuhiko Shibuya
IPC分类号: A01N43/90 , A01N47/12 , A01N47/18 , C07D471/04 , C07D487/04 , C07D498/04 , C07D513/04 , A61K31/505
CPC分类号: C07D471/04 , A01N43/90 , A01N47/18 , C07D487/04 , C07D513/04
摘要: Nitro-substituted heterocyclic compounds of the formula (I) ##STR1## wherein R is hydrogen or alkyl,Z is an optionally substituted aryl or optionally substituted heterocyclic group containing at least one atom selected from N, O and S,A is optionally substituted ethylene or optionally substituted trimethylene, andB stands for 2 or 3 members of a heterocyclic ring which is formed, together with the adjacent C-atom and N-atom and at least one of said members may represent a hetero atom and may be optionally substituted, provided that when B stands for 3 members, two of which are carbon atoms and the other one is a nitrogen atom which is located in the middle of the three members, then at least one of said two carbon atoms must be substituted by a keto group. Such compounds being useful as insecticides.
摘要翻译: 式(I)的硝基取代的杂环化合物其中R是氢或烷基,Z是任选取代的芳基或含有至少一个选自N,O和S的原子的任选取代的杂环基,A是 任选取代的乙烯或任选取代的三亚甲基,B代表与相邻C原子和N-原子一起形成的杂环的2或3个成员,并且所述成员中的至少一个可以表示杂原子,并且可以是 任选取代,条件是当B代表3个成员时,其中两个是碳原子,另一个是位于三个成员中间的氮原子,则所述两个碳原子中的至少一个必须被 一个酮基。 这些化合物可用作杀虫剂。
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公开(公告)号:US5622914A
公开(公告)日:1997-04-22
申请号:US529963
申请日:1995-09-19
申请人: Yoshio Kurahashi , Koichi Moriya , Haruko Sawada , Haruhiko Sakuma , Ryo Watanabe , Asami Ito
发明人: Yoshio Kurahashi , Koichi Moriya , Haruko Sawada , Haruhiko Sakuma , Ryo Watanabe , Asami Ito
IPC分类号: A01N43/50 , A01N43/56 , C07D401/04 , C07D521/00 , C07F7/08 , A01N43/42 , C07D215/44
CPC分类号: C07D231/12 , A01N43/50 , A01N43/56 , C07D233/56 , C07D249/08 , C07D401/04 , C07F7/0812
摘要: Combatting fungi and bacteria with quinoline derivatives of the formula ##STR1## in which X is a nitrogen atom and Y is a CH-group orY is a nitrogen atom and X is a CH-group,R is hydrogen, halogen, acetyl or alkyl which is optionally substituted by one to three radicals independently selected from the group consisting of alkoxy, phenyl, hydroxy, halogen and cyano, orR is alkenyl which is optionally substituted by one to three radicals independently selected from the group consisting of halogen, cyano, alkoxy, phenyl and hydroxy, orR is alkynyl which is optionally substituted by one to three radicals independently selected from the group consisting of halogen, phenyl, trimethylsilyl, hydroxy, cyano, alkoxy, alkylamino, dialkylamino, alkylcarbonyl, tolyl, alkoxycarbonyl and alkylcarbonyloxy, orR is cycloalkyl which is optionally substituted by one to three radicals independently selected from the group consisting of halogen and cyano,A is hydrogen or halogen andB is halogen or halogenoalkyl,or an acid addition salt or metal salt complex thereof, and processes for their preparation. Most of these compounds are new.
摘要翻译: 用真菌和细菌与其中X是氮原子并且Y是CH-基团或Y是氮原子并且X是CH-基团的式(I)的喹啉衍生物反应,R是氢,卤素, 乙酰基或烷基,其任选地被一至三个独立地选自烷氧基,苯基,羟基,卤素和氰基的基团取代,或R是任选被一至三个独立地选自卤素 氰基,烷氧基,苯基和羟基,或R是任选被一至三个独立地选自卤素,苯基,三甲基甲硅烷基,羟基,氰基,烷氧基,烷基氨基,二烷基氨基,烷基羰基,甲苯基,烷氧基羰基 和烷基羰基氧基,或R是任选被一至三个独立地选自卤素和氰基的基团取代的环烷基,A是氢或卤素,B是卤素或 卤代烷基或其酸加成盐或金属盐络合物,及其制备方法。 这些化合物大部分是新的。
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公开(公告)号:US5461167A
公开(公告)日:1995-10-24
申请号:US067642
申请日:1993-05-25
申请人: Kozo Shiokawa , Shinichi Tsuboi , Shinzo Kagabu , Koichi Moriya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Shinzo Kagabu , Koichi Moriya
IPC分类号: A01N43/78 , A01N20060101 , A01N33/18 , A01N43/00 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/647 , A01N43/653 , A01N43/66 , A01N43/72 , A01N43/74 , A01N43/76 , A01N43/80 , A01N43/82 , A01N43/84 , A01N43/86 , A01N43/88 , A01N47/02 , A01N47/16 , A01N47/22 , A01N47/38 , A01N51/00 , A01N57/32 , C07D20060101 , C07D207/20 , C07D207/22 , C07D211/70 , C07D211/72 , C07D213/00 , C07D213/61 , C07D233/20 , C07D233/52 , C07D239/06 , C07D239/18 , C07D263/10 , C07D263/28 , C07D265/08 , C07D277/00 , C07D277/10 , C07D277/18 , C07D279/00 , C07D279/06 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D405/06 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/06 , C07D413/14 , C07D417/06 , C07D417/14 , C07D419/06 , C07F9/6558 , C07D277/20
CPC分类号: C07D239/06 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/653 , A01N43/74 , A01N43/80 , A01N43/82 , A01N43/86 , A01N47/02 , A01N47/16 , A01N47/22 , A01N47/38 , A01N51/00 , A01N57/32 , C07D207/20 , C07D207/22 , C07D211/70 , C07D211/72 , C07D233/20 , C07D233/52 , C07D239/18 , C07D263/10 , C07D263/28 , C07D265/08 , C07D277/10 , C07D277/18 , C07D279/06 , C07D401/06 , C07D401/14 , C07D403/06 , C07D405/06 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/06 , C07D413/14 , C07D417/06 , C07D417/14 , C07F9/65583
摘要: Novel insecticides of the formula ##STR1## in which n is 0 or 1,X is S, O, ##STR2## Y is N or ##STR3## Z is a 5- or 6-membered nitrogen-containing heterocyclic ring, and R to R.sup.9 variously represent hydrogen or specified organic radicals.
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公开(公告)号:US5314897A
公开(公告)日:1994-05-24
申请号:US90566
申请日:1993-07-12
申请人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
IPC分类号: C07D239/48 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/647 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/824 , A01N47/18 , C07D213/61 , C07D213/74 , C07D213/79 , C07D239/06 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/12 , C07D407/12 , C07D413/12 , C07D417/12
CPC分类号: C07D401/14 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/647 , A01N43/78 , A01N43/80 , A01N43/82 , A01N47/18 , C07D213/74 , C07D239/06 , C07D401/12 , C07D417/12
摘要: Insecticidal nitro-substituted heterocyclic compounds of the formula ##STR1## wherein R.sup.1 represents hydrogen, cyano or C.sub.1-4 alkyl,m represents 0 or 1,n represents 0 or 1,R.sup.2 represents hydrogen or C.sub.1-4 alkyl,R.sup.3 represents hydrogen, C.sub.1-6 alkyl optionally substituted substituted by cyano, halogen or C.sub.1-4 alkoxy, C.sub.3-4 alkenyl, C.sub.3-4 alkynyl, optionally substituted phenyl, optionally substituted benzyl or optionally substituted heterocyclic-methyl,T represents an optionally substituted two- or three-membered divalent or trivalent chain comprising hetero atoms and/or carbon atom, andA represents optionally substituted phenyl or an optionally substituted five- or six-membered heterocyclic radical comprising at least one hetero atom selected from the group consisting of N, O and S.
摘要翻译: 式(I)的杀虫硝基取代的杂环化合物,其中R1表示氢,氰基或C1-4烷基,m表示0或1,n表示0或1,R2表示氢或C1-4烷基,R3表示 氢,任选被氰基,卤素或C 1-4烷氧基取代的C 1-6烷基,C 3-4烯基,C 3-4炔基,任选取代的苯基,任选取代的苄基或任选取代的杂环甲基,T代表任选取代的二价基团, 或包含杂原子和/或碳原子的三元二价或三价链,并且A表示任选取代的苯基或任选取代的五元或六元杂环基,其包含至少一个选自N,O 和S.
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公开(公告)号:US5308855A
公开(公告)日:1994-05-03
申请号:US987513
申请日:1992-12-07
IPC分类号: A01N47/44 , A01N51/00 , C07D213/61 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , C07D417/14 , C07D521/00 , A61K31/44
CPC分类号: C07D231/12 , A01N47/44 , A01N51/00 , C07D233/56 , C07D249/08 , C07D401/06 , C07D417/06
摘要: Insecticidal guanidine derivatives of the formula ##STR1## wherein Z represents an optionally substituted five- or six-membered ring containing at least one ring hetero atom selected from the group consisting of oxygen, sulfur and nitrogen,R.sup.1 represents hydrogen atoms or a C.sub.1-4 alkyl group, R.sup.2 and R.sup.3 each independently represents hydrogen, C.sub.1-4 alkyl, C.sub.1-4 haloalkyl or optionally substituted phenyl,R.sup.4 and R.sup.5 each independently represents hydrogen, C.sub.1-4 alkyl, C.sub.3-4 alkenyl, C.sub.3-4 alkynyl, optionally substituted benzyl or a group of the formula Z-C(R.sup.1)H-,n represents the integer 2 or 3, andY represents nitro or cyano.
摘要翻译: 式y的杀虫胍衍生物取代的含有至少一个选自氧,硫和氮的环杂原子的五元或六元环,R 1表示氢原子或C 1-4烷基,R 2和R 3各自 独立地表示氢,C 1-4烷基,C 1-4卤代烷基或任选取代的苯基,R 4和R 5各自独立地表示氢,C 1-4烷基,C 3-4烯基,C 3-4炔基,任选取代的苄基或式 ZC(R1)H-,n表示整数2或3,Y表示硝基或氰基。
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公开(公告)号:US5117053A
公开(公告)日:1992-05-26
申请号:US755257
申请日:1991-09-05
申请人: Yoshio Kurahashi , Kozo Shiokawa , Shinzo Kagabu , Shinji Sakawa , Koichi Moriya
发明人: Yoshio Kurahashi , Kozo Shiokawa , Shinzo Kagabu , Shinji Sakawa , Koichi Moriya
摘要: Novel fungicidally active N-benzyl-cyclopropanecarboxamides of the formula ##STR1## wherein X=represents halogen,n=represents 1 or 2,R.sup.1 =represents hydrogen, halogen or lower alkyl,R.sup.2 =represents lower alkyl, halogen-substituted lower alkyl or hydrogen, andR.sup.3 =represents hydrogen or lower alkyl.The acid components thereof, other than when R.sup.1 is hydrogen or alkyl and R.sup.2 is hydrogen or alkyl, are also new.
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公开(公告)号:US5032589A
公开(公告)日:1991-07-16
申请号:US487004
申请日:1990-03-01
申请人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Koichi Moriya , Yumi Hattori , Ikuro Honda , Katsuhiko Shibuya
IPC分类号: A01N43/64 , A01N43/653 , A01N43/72 , A01N43/80 , A01N43/832 , A01N43/836 , A01N43/84 , A01N43/88 , A01N47/40 , A01N51/00 , C07D401/06 , C07D401/14 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D419/06
CPC分类号: C07D401/06 , A01N47/40 , A01N51/00 , C07D401/14 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D419/06
摘要: Insecticidal heterocyclic compounds of the formula ##STR1## wherein A represents a five-membered or six-membered heteroaryl group containing one to three hetero atoms selected from the group consisting of S, O and N, said heteroaryl group being unsubstituted or substituted by a halogen atom or C.sub.1-4 alkyl group, Z represents a three-membered straight chain, each member being selected from the group consisting of CH.sub.2 --, O, S and N--R.sup.2 with at least one of said three members being O, S or N--R.sup.2, E represents CH.sub.2, O, S or N--R.sup.2 wherein R.sup.2 represents a hydrogen atom, a C.sub.1-4 alkyl group, a C.sub.1-4 alkoxy group or the group ##STR2## wherein R.sup.3 represents a hydrogen atom or halogen atom, X represents CH or N, Y represents a nitro group or cyano group, and R.sup.1 represents a hydrogen atom or methyl group.
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公开(公告)号:US4882344A
公开(公告)日:1989-11-21
申请号:US243545
申请日:1988-09-13
申请人: Kozo Shiokawa , Shinichi Tsuboi , Shoko Sasaki , Koichi Moriya , Yumi Hattori , Katsuhiko Shibuya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Shoko Sasaki , Koichi Moriya , Yumi Hattori , Katsuhiko Shibuya
IPC分类号: A01N43/40 , A01N43/50 , A01N43/78 , A01N51/00 , C07D213/26 , C07D213/57 , C07D213/74 , C07D213/75 , C07D213/76 , C07D213/77 , C07D239/42 , C07D277/32 , C07D277/48 , C07D277/50 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , A61K31/44
CPC分类号: C07D213/75 , A01N43/50 , A01N51/00 , C07D213/77 , C07D239/42 , C07D277/32 , C07D277/48 , C07D277/50 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06
摘要: Novel insecticidally active heterocyclic compounds of the formula ##STR1## wherein W represents a substituted pyridyl group, or a 5- or 6-membered optionally substituted heterocyclic group containing at least two hetero atoms selected from oxygen, sulfur and nitrogen atoms,R represents a hydrogen atom or an alkyl group,Y represents .dbd.N-- or ##STR2## R' represents a hydrogen atom, an alkyl group, an aryl group, an acyl group, an alkoxycarbonyl group or a cyano group,Z represents a nitro group or a cyano group, andT represents 3 or 4 optionally substituted ring members of a 5- or 6-membered unsaturated heterocyclic ring which it forms together with the adjoining carbon atom and nitrogen atom, said 5- or 6-membered unsaturated heterocyclic ring containing 1 to 3 hetero atoms which are selected from oxygen, sulfur and nitrogen atoms and at least one of which is a nitrogen atom.
摘要翻译: 新颖的具有下式的杀虫活性杂环化合物,其中W代表取代的吡啶基,或含有至少两个选自氧,硫和氮原子的杂原子的5或6元任选取代的杂环基,R代表氢 原子或烷基,Y表示= N-或R'表示氢原子,烷基,芳基,酰基,烷氧基羰基或氰基,Z表示硝基或氰基 并且T表示与邻接的碳原子和氮原子一起形成的5或6元不饱和杂环的3或4个任选取代的环成员,所述5或6元不饱和杂环含有1至3个 杂原子,其选自氧,硫和氮原子,并且其中至少一个是氮原子。
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公开(公告)号:US4845106A
公开(公告)日:1989-07-04
申请号:US68991
申请日:1987-07-01
申请人: Kozo Shiokawa , Shinichi Tsuboi , Shinzo Kagabu , Koichi Moriya
发明人: Kozo Shiokawa , Shinichi Tsuboi , Shinzo Kagabu , Koichi Moriya
IPC分类号: A01N43/78 , A01N20060101 , A01N33/18 , A01N43/00 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/647 , A01N43/653 , A01N43/66 , A01N43/72 , A01N43/74 , A01N43/76 , A01N43/80 , A01N43/82 , A01N43/84 , A01N43/86 , A01N43/88 , A01N47/02 , A01N47/16 , A01N47/22 , A01N47/38 , A01N51/00 , A01N57/32 , C07D20060101 , C07D207/20 , C07D207/22 , C07D211/70 , C07D211/72 , C07D213/00 , C07D213/61 , C07D233/20 , C07D233/52 , C07D239/06 , C07D239/18 , C07D263/10 , C07D263/28 , C07D265/08 , C07D277/00 , C07D277/10 , C07D277/18 , C07D279/00 , C07D279/06 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D405/06 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/06 , C07D413/14 , C07D417/06 , C07D417/14 , C07D419/06 , C07F9/6558
CPC分类号: C07D239/06 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/653 , A01N43/74 , A01N43/80 , A01N43/82 , A01N43/86 , A01N47/02 , A01N47/16 , A01N47/22 , A01N47/38 , A01N51/00 , A01N57/32 , C07D207/20 , C07D207/22 , C07D211/70 , C07D211/72 , C07D233/20 , C07D233/52 , C07D239/18 , C07D263/10 , C07D263/28 , C07D265/08 , C07D277/10 , C07D277/18 , C07D279/06 , C07D401/06 , C07D401/14 , C07D403/06 , C07D405/06 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/06 , C07D413/14 , C07D417/06 , C07D417/14 , C07F9/65583
摘要: Novel insecticides of the formula ##STR1## in which n is 0 or 1,X is S, O, ##STR2## Y is N or ##STR3## Z is a 5- or 6-membered nitrogen-containing heterocyclic ring, and R to R.sup.9 variously represent hydrogen or specified organic radicals.
摘要翻译: 式中,n为0或1的新型杀虫剂,其中X为S,O,Y为N或Z为5或6元含氮杂环,R为 R9各自表示氢或特定的有机基团。
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