公开(公告)号：US20110195930A1

公开(公告)日：2011-08-11

申请号：US13125582

申请日：2009-11-06

申请人： Takahiro Haga ,  Masayuki Morita ,  Kazuhisa Kiriyama ,  Kumiko Azuma

发明人： Takahiro Haga ,  Masayuki Morita ,  Kazuhisa Kiriyama ,  Kumiko Azuma

IPC分类号： A01N55/10 ,  C07D401/06 ,  A01N43/40 ,  C07F7/18 ,  C07D401/14 ,  A01P7/00

CPC分类号： C07D401/12

摘要： To provide a novel pesticide. The present invention provides a pesticide which contains, as an active ingredient, novel pyridine derivative represented by the formula (I) or its salt: wherein R1 is alkyl, cycloalkyl, alkoxyalkyl or OR3; R2 is 1H-1,2,4-triazol-1-yl which may be substituted, 1H-imidazol-1-yl which may be substituted, 1H-1,2,3-triazol-1-yl which may be substituted, or 4H-1,2,4-triazol-4-yl which may be substituted; X is alkyl which may be substituted, cycloalkyl which may be substituted, halogen, nitro, etc.; R3 is alkyl which may be substituted, cycloalkyl which may be substituted, alkenyl which may be substituted, alkynyl which may be substituted, etc.; m is an integer of from 1 to 4.

摘要翻译： 提供一种新型农药。 本发明提供了含有作为活性成分的由式（I）表示的新型吡啶衍生物或其盐的农药：其中R1是烷基，环烷基，烷氧基烷基或OR3; R2是可以被取代的1H-1,2,4-三唑-1-基，可以被取代的1H-咪唑-1-基，可以被取代的1H-1,2,3-三唑-1-基， 或可被取代的4H-1,2,4-三唑-4-基; X为可被取代的烷基，可被取代的环烷基，卤素，硝基等; R3是可被取代的烷基，可被取代的环烷基，可被取代的链烯基，可被取代的炔基等; m为1〜4的整数。

公开(公告)号：US20100087452A1

公开(公告)日：2010-04-08

申请号：US12526520

申请日：2008-02-07

申请人： Takahiro Haga ,  Hirohiko Kimura ,  Masayuki Morita ,  Tsuyoshi Ueda ,  Toshihiko Ueki ,  Kazuhisa Kiriyama ,  Kotaro Yoshida ,  Taku Hamamoto

发明人： Takahiro Haga ,  Hirohiko Kimura ,  Masayuki Morita ,  Tsuyoshi Ueda ,  Toshihiko Ueki ,  Kazuhisa Kiriyama ,  Kotaro Yoshida ,  Taku Hamamoto

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P7/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： To provide a novel pesticide. The present invention provides a pesticide containing a pyridyl-triazolopyrimidine derivative represented by the formula (I) or its salt as an active ingredient: wherein R1 is substitutable alkyl, substitutable cycloalkyl, substitutable alkenyl, substitutable alkynyl, halogen, cyano, aryl, a heterocyclic group which may be substituted by alkyl, OR2, S(O)n#191R3? or NR4R5; R2 is hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, alkoxyalkyl, acetyl or aryl; R3 is alkyl or acetyl; R4 is hydrogen or alkyl; R5 is hydrogen, alkyl or the like; X is alkyl, alkenyl, alkynyl, halogen, haloalkyl, cyano, nitro or the like; m is an integer of from 1 to 4; and n is an integer of from 0 to 2.

摘要翻译： 提供一种新型农药。 本发明提供含有式（I）表示的吡啶基 - 三唑并嘧啶衍生物或其盐作为活性成分的农药：其中R1是可取代的烷基，可取代的环烷基，可取代的烯基，可取代的炔基，卤素，氰基，芳基，杂环 可以被烷基取代的基团，OR 2，S（O）n＃191R 3 或NR4R5; R2是氢，烷基，烯基，炔基，卤代烷基，烷氧基烷基，乙酰基或芳基; R3是烷基或乙酰基; R4是氢或烷基; R5是氢，烷基等; X为烷基，烯基，炔基，卤素，卤代烷基，氰基，硝基等; m为1〜4的整数， n为0〜2的整数。

公开(公告)号：US06300323B1

公开(公告)日：2001-10-09

申请号：US09634630

申请日：2000-08-08

申请人： Takahiro Haga ,  Kevin E. Crosby ,  Jeffrey R. Schussler

发明人： Takahiro Haga ,  Kevin E. Crosby ,  Jeffrey R. Schussler

IPC分类号： A01N5712

CPC分类号： C07D213/64 ,  A01N25/30 ,  A01N33/08 ,  A01N39/02 ,  A01N39/04 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/84 ,  A01N57/20 ,  C07C215/08 ,  C07C215/14 ,  C07C215/18 ,  C07C217/08 ,  C07C217/16 ,  C07C217/28 ,  C07C217/42 ,  C07C219/04 ,  C07C219/08 ,  C07D213/80 ,  C07D231/20 ,  C07D239/34 ,  C07D295/088 ,  C07F9/3813 ,  C08G65/33306

摘要： A compound Wherein x, y, and z are integers from 0 to 3; and the (poly)ethereal amine is at least one selected from compounds of formula II1 through II5:

摘要翻译： 复合物，其中x，y和z是0至3的整数; 和（多）醚胺是选自式II1至II5的化合物中的至少一种：

公开(公告)号：US6133521A

公开(公告)日：2000-10-17

申请号：US38134

申请日：1998-03-11

申请人： Takahiro Haga ,  Nobuo Hanehira ,  Hiroyuki Mori ,  Masanori Kaji ,  Masayoshi Ono ,  Masato Nishikuni ,  Yoshinobu Takabatake

发明人： Takahiro Haga ,  Nobuo Hanehira ,  Hiroyuki Mori ,  Masanori Kaji ,  Masayoshi Ono ,  Masato Nishikuni ,  Yoshinobu Takabatake

IPC分类号： H01L21/60 ,  H01L27/142 ,  H01L31/02 ,  H01L31/0224 ,  H01L31/04 ,  H01L31/048 ,  H01L31/00

CPC分类号： H01L31/022425 ,  H01L31/02008 ,  H01L31/046 ,  H01L31/0465 ,  H01L2924/0002 ,  Y02E10/50

摘要： The solar battery output section has a hole provided through the substrate and through an output terminal formed on the front-side of that substrate. Metal foil is applied covering the hole on the backside of the substrate. The inside of the hole is filled with conducting material to electrically connect the output terminal and the metal foil. Finally, a protective resin film is applied over the substrate, and a wire lead is solder attached to the metal foil on the backside of the substrate.

摘要翻译： 太阳能电池输出部具有通过基板设置的孔，并且形成在该基板的前侧的输出端子。 应用金属箔覆盖基板背面的孔。 孔的内部填充有导电材料以电连接输出端子和金属箔。 最后，将保护性树脂膜施加在基板上，并且将引线焊接在基板背面的金属箔上。

公开(公告)号：US5102884A

公开(公告)日：1992-04-07

申请号：US554449

申请日：1990-07-19

申请人： Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi ,  Hiroshi Okada

发明人： Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi ,  Hiroshi Okada

IPC分类号： A61K31/505 ,  C07C237/42 ,  C07C275/46 ,  C07C311/31 ,  C07D239/34 ,  C07D401/12 ,  C07D403/12 ,  C07D413/12 ,  C07D417/12

CPC分类号： C07D239/34 ,  C07C237/42 ,  C07C311/31

摘要： A substituted benzoylurea compound of the formula (I): ##STR1## wherein R.sup.1 is a hydrogen atom, a halogen atom or a nitro group, each of R.sup.2 and R.sup.3 is a hydrogen atom, an alkyl group, --COR.sup.6 (wherein R.sup.6 is an alkyl group or an alkoxy group) or --SO.sub.2 R.sup.6 (wherein R.sup.6 is as defined above), or R.sup.2 and R.sup.3 may form together with the adjacent nitrogen atom a heterocyclic ring, R.sup.4 is a halogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkoxy group, a substituted or unsubstituted alkylthio group or a nitro group, and R.sup.5 is a halogen atom, a nitro group or a substituted or unsubstituted alkyl group, or its salt.

公开(公告)号：US4987135A

公开(公告)日：1991-01-22

申请号：US324559

申请日：1989-03-16

申请人： Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi ,  Hiroshi Okada

发明人： Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi ,  Hiroshi Okada

IPC分类号： C07D295/12 ,  A61K31/50 ,  A61K31/505 ,  A61P35/00 ,  C07C257/08 ,  C07C275/54 ,  C07C313/34 ,  C07C323/44 ,  C07C327/58 ,  C07C329/04 ,  C07C381/04 ,  C07C381/08 ,  C07D213/64 ,  C07D213/81 ,  C07D237/14 ,  C07D239/34 ,  C07D295/155 ,  C07D401/12 ,  C07F9/24 ,  C07F9/6512

CPC分类号： C07D213/64 ,  C07C257/08 ,  C07C327/58 ,  C07D237/14 ,  C07D239/34 ,  C07D295/155 ,  C07D401/12 ,  C07F9/65127 ,  C07C2101/08 ,  C07C2101/14

摘要： A substituted benzene derivative represented by a formula: ##STR1## where A represents: ##STR2## wherein X is a hydrogen atom, a halogen atom or a nitro group, R.sup.1 is --X.sup.1 Z.sup.1 (X.sup.1 is an oxygen atom or a sulfur atom and Z.sup.1 is a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkenyl group, a substituted or unsubstituted alkynyl group, a substituted or unsubstituted aryl group or a substituted or unsubstituted heteroaryl group), --COZ.sup.1 group (Z.sup.1 is as defined above), ##STR3## group (Z.sup.1 is as defined above, Z.sup.2 is --CO.sub.2 Z.sup.3 wherein Z.sup.3 is the same as Z.sup.1, or --SO.sub.2 Z.sup.3 wherein Z.sup.3 is as defined above and n is 0 or 1), ##STR4## (Z.sup.1 and Z.sup.3 are as defined above) or ##STR5## (X.sup.2, X.sup.3 and X.sup.4 are, respectively, an oxygen atom or a sulfur atom and Z.sup.4 and Z.sup.5 are the same as Z.sup.1), and R.sup.3 is a nitro group or ##STR6## (R.sup.4 and R.sup.5 are, respectively, an alkyl group, or they may form a heterocyclic group together with the adjacent nitrogen atom), or ##STR7## wherein X and R.sup.3 are as defined above and R.sup.2 is --X.sup.1 Z.sup.1 (X.sup.1 and Z.sup.1 are as defined above); Y is a halogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkoxy group, a substituted or unsubstituted alkylthio group, a nitro group or ##STR8## (R.sup.6 and R.sup.7 are, respectively, a substituted or unsubstituted alkyl group); R is ##STR9## (R.sup.8 is the same as Y and q is an integer of 1 to 4), ##STR10## (R.sup.8 is as defined above, and r is an integer of 1 to 3) or ##STR11## (R.sup.8 and r are defined above); and m is an integer, of 1 to 4, or its salt.

公开(公告)号：US4985449A

公开(公告)日：1991-01-15

申请号：US365607

申请日：1989-06-13

申请人： Takahiro Haga ,  Tadaaki Toki ,  Toru Koyanagi ,  Yasuhiro Fujii ,  Kiyomitsu Yoshida ,  Osamu Imai

发明人： Takahiro Haga ,  Tadaaki Toki ,  Toru Koyanagi ,  Yasuhiro Fujii ,  Kiyomitsu Yoshida ,  Osamu Imai

IPC分类号： A01N43/40 ,  A01N47/34 ,  A01N47/36 ,  A01P7/04 ,  C07C275/54 ,  C07D213/64 ,  C07D213/643 ,  C07D213/70 ,  C07D213/74 ,  C07D213/75 ,  C07D333/38

CPC分类号： C07D213/643 ,  A01N47/34 ,  A01N47/36 ,  C07C275/54 ,  C07D213/70 ,  C07D213/74 ,  C07D213/75 ,  C07D333/38

摘要： A benzoylurea compound having the formula: ##STR1## wherein each of X.sub.1 and X.sub.2 is a hydrogen atom, a halogen atom or a methyl group, provided that X.sub.1 and X.sub.2 are not simultanously hydrogen atoms, Y is independently a hydrogen atom, a halogen atom, an alkyl group which may be substituted by halogen, a --CO.sub.2 R.sub.1 group wherein R.sub.1 is a hydrogen atom, a cation or an alkyl group, or a --OR.sub.1 group wherein R.sub.1 is as defined above, A.sub.1 is .dbd.N-- or ##STR2## wherein Y is as defined above, W is an oxygen atom, a sulfur atom or ##STR3## wherein R.sub.1 is as defined above, k is an integer of from 1 to 3, l is 0 or 1, and Ar is ##STR4## wherein Z is independently a hydrogen atom, a halogen atom, an alkyl group which may be substituted by halogen, an alkoxy group which may be substituted by halogen, a nitro group, a cyano group or a --S(O).sub.n R.sub.2 group wherein R.sub.2 is an alkyl group which may be substituted by halogen and n is 0, 1 or 2, A.sub.2 is --S--, ##STR5## wherein Z is as defined above, or ##STR6## wherein Z is as defined above, and m is an integer of from 1 to 3, or a salt thereof.

公开(公告)号：US4983605A

公开(公告)日：1991-01-08

申请号：US110284

申请日：1987-10-20

申请人： Nobuo Kondo ,  Masahiro Kikuchi ,  Tsunetaka Nakajima ,  Masahiro Watanabe ,  Kazumasa Yokoyama ,  Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi

发明人： Nobuo Kondo ,  Masahiro Kikuchi ,  Tsunetaka Nakajima ,  Masahiro Watanabe ,  Kazumasa Yokoyama ,  Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi

IPC分类号： A61K9/14 ,  A61K9/19 ,  A61K31/44 ,  A61K31/50 ,  A61K31/505 ,  A61K47/14 ,  A61K47/26

CPC分类号： A61K31/505 ,  A61K31/44 ,  A61K31/50 ,  A61K9/145 ,  A61K9/146 ,  A61K9/19 ,  A61K47/14 ,  A61K47/26 ,  Y10S514/961 ,  Y10S514/964

摘要： A pharmaceutical composition comprising a benzoyl urea compound (A) selected from the group consisting of a benzoyl urea compound (I) having the formula: ##STR1## wherein X is a halogen atom, a nitro group or a trifluoromethyl group, provided that when Y is a nitro group, X is a halogen atom or a nitro group, Y is a hydrogen atom, a halogen atom, a nitro group or a trifluoromethyl group, Z.sub.1 is a halogen atom or a trifluoromethyl group, Z.sub.2 is a hydrogen atom or a halogen atom, and A is a .dbd.CH-- group or a nitrogen atom, and a benzoyl urea compound (II) having the formula: ##STR2## wherein each of X.sub.1 and X.sub.2 is a hydrogen atom, a halogen atom or a nitro group, provided that when Y is a nitro group, X.sub.1 is a hydrogen atom, Y is a hydrogen atom, a halogen atom, a nitro group or a trifluoromethyl group, and Z is a hydrogen atom, a halogen atom or a trifluoromethyl group, as an active ingredient; a nonionic surfactant as a dispersant; and at least one member selected from the group consisting of a saccharide, a saccharide alcohol, silicic anhydride and a nonionic surfactant, as a disintegrator.

摘要翻译： 提供一种药物组合物，其包含选自具有下式的苯甲酰脲化合物（I）的苯甲酰脲化合物（A）：其中X为卤素原子，硝基或三氟甲基，其提供 当Y为硝基时，X为卤原子或硝基，Y为氢原子，卤原子，硝基或三氟甲基，Z1为卤原子或三氟甲基，Z2为氢 原子或卤素原子，A为= CH-基或氮原子，和具有下式的苯甲酰脲化合物（II）：其中X1和X2各自为氢原子，卤素 原子或硝基，条件是当Y为硝基时，X 1为氢原子，Y为氢原子，卤素原子，硝基或三氟甲基，Z为氢原子，卤素原子或 三氟甲基作为活性成分; 作为分散剂的非离子表面活性剂; 和选自糖，糖醇，硅酸酐和非离子表面活性剂的至少一种作为崩解剂。

公开(公告)号：US4904668A

公开(公告)日：1990-02-27

申请号：US101005

申请日：1987-09-25

申请人： Nobuo Kondo ,  Masahiro Kikuchi ,  Tsunetaka Nakajima ,  Masahiro Watanabe ,  Kazumasa Yokoyama ,  Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi

发明人： Nobuo Kondo ,  Masahiro Kikuchi ,  Tsunetaka Nakajima ,  Masahiro Watanabe ,  Kazumasa Yokoyama ,  Takahiro Haga ,  Nobutoshi Yamada ,  Hideo Sugi ,  Toru Koyanagi

IPC分类号： A61K9/14 ,  C07D213/64 ,  C07D213/643 ,  C07D237/14 ,  C07D239/34

CPC分类号： C07D213/643 ,  A61K9/14 ,  A61K9/145 ,  A61K9/146 ,  C07D237/14 ,  C07D239/34

摘要： A benzoyl urea compound having the formula: ##STR1## wherein X is a halogen atom, a nitro group or a trifluoromethyl group, provided that when Y is a nitro group, X is a halogen atom or a nitro group, Y is a hydrogen atom, a halogen atom, a nitro group or a trifluoromethyl group, Z.sub.1 is a halogen atom or a trifluoromethyl group, Z.sub.2 is a hydrogen atom or a halogen atom, and A is a .dbd.CH-- group or a nitrogen atom, or the formula: ##STR2## wherein each of X.sub.1 is X.sub.2 is a hydrogen atom, a halogen atom or a nitro group, provided that when Y is a nitro group, X.sub.1 is a hydrogen atom, Y is a hydrogen atom, a halogen atom, a nitro group or a trifluoromethyl group, and Z is a hydrogen atom, a halogen atom or a trifluoromethyl group, characterized in that its average particle size is not larger than 1 .mu.m.

摘要翻译： 具有下式的苯甲酰脲化合物：其中X是卤素原子，硝基或三氟甲基，条件是当Y是硝基时，X是卤原子或硝基，Y是 氢原子，卤素原子，硝基或三氟甲基，Z1为卤素原子或三氟甲基，Z2为氢原子或卤素原子，A为a-CH-基或氮原子，或 其中X 1为X 2的每一个为氢原子，卤原子或硝基的式：其中Y为硝基时，X 1为氢原子，Y为氢原子， 卤原子，硝基或三氟甲基，Z为氢原子，卤素原子或三氟甲基，其特征在于，其平均粒径为1μm以下。

公开(公告)号：US4861886A

公开(公告)日：1989-08-29

申请号：US215532

申请日：1988-07-06

申请人： Takahiro Haga ,  Itaru Shigehara ,  Toru Koyanagi ,  Kazutoshi Hara ,  Masaru Maeda

发明人： Takahiro Haga ,  Itaru Shigehara ,  Toru Koyanagi ,  Kazutoshi Hara ,  Masaru Maeda

IPC分类号： C07D497/20

CPC分类号： C07D497/20

摘要： A method for isomerization of trans-form 2-methylspiro(1,3-oxathiolane-5,3')quinuclidine or acid addition salts thereof, which comprises isomerizing said trans-form quinuclidine or acid addition salts thereof to cis-form 2-methylspiro(1,3-oxathiolane-5,3')quinuclidine or acid addition salts thereof in the presence of at least one acid catalyst selected from the group consisting of an organic sulfuric acid, a halide functioning as a Lewis acid, and sulfuric acid.