摘要:
The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.
摘要:
The present invention relates to the use of aminoazoline and urea derivatives for com-bating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds and to specific azoline and urea derivatives.
摘要:
The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.
摘要:
The present invention relates to 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to methods for combating animal pests and to compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds of the general formula (I): wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur, oxygen or NR7, and HetA, HetB and R1 to R7 are defined as in the description.
摘要:
The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, —C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.
摘要:
The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.
摘要:
The present invention relates to 1-(Azolin-2-yl)-amino-alkane compounds, which are useful for combating insects, arachnids and nematodes.The present invention also relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests.It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-alkane compounds of the general formula I: wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur or oxygen and W, B and R1 to R6 are defined as in the description.
摘要:
The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (1.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is —C(R6a)(R6b)—, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, (C1-C6-alkyl)-thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2 are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with Rb may also be ═O, ═NRC or ═CRdRe; or R2a together with R4a may form a bridging bivalent radical.
摘要:
The present invention relates to azoline compounds and their salts which are useful for combating arthropod pests. The present invention also relates to a method for combating arthropod pests and to agricultural compositions for combating said pests. It has been found that these objectives can be achieved by azoline compounds of the general formulae Ia or Ib, wherein X is S, O or NR4; Ar is phenyl or a 5 or 6 membered heteroaromatic ring; R1 is H, C1-C6-alkyl, C2-C6-alkenyl, phenyl, a heteroaromatic ring etc.; R2a, R2b are H, CN, C1-C6-alkyl etc.; R1 together with R2a may also form a linear C2-C4-alkandiyl; R3a-d are H, halogen, C1-C6-alkyl etc.
摘要:
The present invention relates to 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds (I) and 1-(aminothiocarbonylamino)-2-aryl-1-hetaryl-ethane compounds (II) and their salts which are useful for combating animal pest, in particular insects, arachnids and nematodes. Furthermore, the present invention relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests.