公开(公告)号：US20100280078A1

公开(公告)日：2010-11-04

申请号：US12667299

申请日：2008-07-02

申请人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecile Ebuenga

发明人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecile Ebuenga

IPC分类号： A01N43/78 ,  C07D277/18 ,  A61K31/426 ,  C07D417/12 ,  C07D417/14 ,  A61K31/427 ,  C07D263/28 ,  A01N43/76 ,  A61K31/421 ,  A61K31/4439 ,  A61P33/00 ,  A01P7/00 ,  A01P7/02 ,  A01P7/04 ,  A01P5/00

CPC分类号： C07D263/28 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/12 ,  A01N47/16 ,  C07D233/48 ,  C07D277/18 ,  C07D417/06 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

公开(公告)号：US08211924B2

公开(公告)日：2012-07-03

申请号：US12667299

申请日：2008-07-02

申请人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecille Ebuenga

发明人： Markus Kordes ,  Christopher Koradin ,  Ronan Le Vezouet ,  Ernst Baumann ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Cecille Ebuenga

IPC分类号： A01N43/78 ,  A01N43/76 ,  A61K31/425 ,  A61K31/42 ,  C07D277/00 ,  C07D263/00

CPC分类号： C07D263/28 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/12 ,  A01N47/16 ,  C07D233/48 ,  C07D277/18 ,  C07D417/06 ,  C07D417/12

摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, —C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

公开(公告)号：US20110224075A1

公开(公告)日：2011-09-15

申请号：US12934461

申请日：2009-03-24

申请人： Markus Kordes ,  Ronan Le Vezouet ,  Jurgen Langewald ,  Ralph Paulini ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Luiz Antonio Jose ,  Hassan Oloumi-Sadeghi

发明人： Markus Kordes ,  Ronan Le Vezouet ,  Jurgen Langewald ,  Ralph Paulini ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Luiz Antonio Jose ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N25/26 ,  A01N43/78 ,  A61K31/427 ,  A61K31/426 ,  A01N43/42 ,  A61K31/4709 ,  A61K31/4725 ,  A01N43/40 ,  A61K31/4439 ,  A01N43/16 ,  A61K31/7016 ,  A01N43/56 ,  A61K31/415 ,  A01N43/88 ,  A61K31/5395 ,  A61K31/44 ,  A01N37/34 ,  A61K31/277 ,  A01N43/38 ,  A61K31/403 ,  A01N43/58 ,  A61K31/50 ,  A61P33/00 ,  A01P7/02 ,  A01P7/04

CPC分类号： A01N43/78 ,  A01N43/08 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/707 ,  A01N43/88 ,  A01N43/90 ,  A01N47/02 ,  A01N47/06 ,  A01N47/30 ,  A01N47/34 ,  A01N47/40 ,  A01N51/00 ,  A01N53/00 ,  A01N2300/00

摘要： The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one aminothiazoline compound I of formula I: wherein R1 is selected from hydrogen, COCH3, COCH2CH3 or COCH2C(CH3)3; R2 and R3 together with the carbon atoms of the phenyl ring to which they are attached form a ring which, depending on the tautomeric formula I a) or b) is depicted as: a benzene ring, a saturated 5-, 6-, or 7-membered carbocycle, a partially unsaturated 5-, 6-, or 7-membered carbocycle, a 5-, 6-, or 7-membered saturated heterocycle, a partially unsaturated 5-, 6-, or 7-membered heterocycle, which heterocycles contain 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and a 5- or 6-membered heteroaromatic ring which contains 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and wherein the ring is unsubstituted or may carry any combination of 1, 2, 3, or 4 radicals selected from the group consisting of halogen, CH3, CH2CH3, CF3, CH3O, cyano and (═O) (oxo); R4 is selected from hydrogen, fluoro, chloro, bromo, CF3, CH3O or CH3; R5, R6 are selected from hydrogen, chloro, fluoro, bromo, CH3, CH3O or CF3, wherein at least one of R5 or R6 is not hydrogen; with the proviso that R2 and R3 together do not form a —OCH2—O— or a —OCF2O-group; or the tautomers, enantiomers, diastereomers or salts thereof, and 2) at least one active compound II selected from group A as defined in the description, use of these mixtures for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using these mixtures.

摘要翻译： 本发明涉及包含作为活性化合物的杀虫混合物1）至少一种式I的氨基噻唑啉化合物I：其中R 1选自氢，COCH 3，COCH 2 CH 3或COCH 2 C（CH 3）3; R2和R3与它们所连接的苯环的碳原子一起形成环，其取决于互变异构体式a a）或b）被描述为：苯环，饱和的5-，6-或 7元碳环，部分不饱和5-，6-或7-元碳环，5-，6-或7-元饱和杂环，部分不饱和5-，6-或7-元杂环，其中 杂环含有选自O，S和N作为环成员的1,2或3个杂原子，以及含有1,2或3个选自O，S和N作为环成员的杂原子的5或6元杂芳环， 并且其中所述环是未取代的或可以携带选自卤素，CH 3，CH 2 CH 3，CF 3，CH 3 O，氰基和（= O）（氧代）的1,2,3或4个基团的任何组合。 R4选自氢，氟，氯，溴，CF 3，CH 3 O或CH 3; R5，R6选自氢，氯，氟，溴，CH3，CH3O或CF3，其中R5或R6中的至少一个不是氢; 条件是R2和R3一起不形成-OCH2-O-或-OCF2O-基团; 或其互变异构体，对映异构体，非对映异构体或其盐，以及2）选自如说明书中定义的组A的至少一种活性化合物II，这些混合物用于防治昆虫，螨虫或线虫的用途，以及治疗，控制 ，防止或保护动物免受使用这些混合物的寄生虫的感染或感染。

公开(公告)号：US20100167925A1

公开(公告)日：2010-07-01

申请号：US12376455

申请日：2007-08-06

申请人： Christopher Koradin ,  Markus Kordes ,  Ronan Le Vezouet ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

发明人： Christopher Koradin ,  Markus Kordes ,  Ronan Le Vezouet ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

IPC分类号： A01C1/06 ,  A01N43/78 ,  C07D417/02

CPC分类号： C07D417/12 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  C07D277/18

摘要： The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (1.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is —C(R6a)(R6b)—, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, (C1-C6-alkyl)-thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2 are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with Rb may also be ═O, ═NRC or ═CRdRe; or R2a together with R4a may form a bridging bivalent radical.

摘要翻译： 本发明涉及用于对抗动物害虫，特别是节肢动物和线虫的式（Ⅰa）和（Ⅰb）的唑啉-2-基氨基化合物及其盐。 本发明还涉及一种防治这种害虫并防止作物抵抗这种害虫侵染或感染的方法。 此外，本发明涉及用于对抗动物害虫的兽用组合物。 式（Ⅰa），式（Ⅰb）其中n为0-4; X是S，O或NR5; A是-C（R6a）（R6b） - ，O，NR7，S，S（O）或S（O） B是键或CH2; R1是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，C3-C6-环烷基，苯基，苄基等; R2a，R2b是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，（C1-C6-烷基） - 硫代羰基，C（O）NRaRb，C（S）NRaRb，（SO2 ）NRaRb，苯基，苄基，5或6元杂环等; 或R 1与R 2a一起为C 3 -C 5 - 烷二基; 或R 1与R 2一起为C（O）; R3a，R3b，R3c，R3d是H，卤素，CN，C1-C6-烷基，C1-C6-烷基氨基，C3-C6-环烷基，苯基，苄基等; R4a，R4b是H，卤素，C1-C6-烷基，C2-C6-烯基，苯基，苄基，5或6元杂芳基; 或R 4a与R b一起也可以是= O，= NRC或= CRdRe; 或R 2a与R 4a一起形成桥连二价基团。

公开(公告)号：US20100010058A1

公开(公告)日：2010-01-14

申请号：US12305267

申请日：2007-05-25

申请人： Christopher Koradin ,  Markus Kordes ,  Ronan Le Vezouet ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Henry Van Tuyl Cotter

发明人： Christopher Koradin ,  Markus Kordes ,  Ronan Le Vezouet ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Henry Van Tuyl Cotter

IPC分类号： A01N43/78 ,  C07D277/18 ,  A01P5/00 ,  A01P7/00

CPC分类号： C07D277/18

摘要： The present invention relates to azoline compounds and their salts which are useful for combating arthropod pests. The present invention also relates to a method for combating arthropod pests and to agricultural compositions for combating said pests. It has been found that these objectives can be achieved by azoline compounds of the general formulae Ia or Ib, wherein X is S, O or NR4; Ar is phenyl or a 5 or 6 membered heteroaromatic ring; R1 is H, C1-C6-alkyl, C2-C6-alkenyl, phenyl, a heteroaromatic ring etc.; R2a, R2b are H, CN, C1-C6-alkyl etc.; R1 together with R2a may also form a linear C2-C4-alkandiyl; R3a-d are H, halogen, C1-C6-alkyl etc.

摘要翻译： 本发明涉及可用于防治节肢动物害虫的唑啉化合物及其盐。 本发明还涉及一种防治节肢动物害虫的方法和用于对抗所述害虫的农业组合物。 已经发现，这些目的可以通过通式Ia或Ib的唑啉化合物来实现，其中X是S，O或NR 4; Ar是苯基或5或6元杂芳环; R1是H，C1-C6-烷基，C2-C6-烯基，苯基，杂芳环等; R2a，R2b是H，CN，C1-C6-烷基等; R1与R2a一起也可以形成直链C 2 -C 4 - 烷二基; R3a-d为H，卤素，C1-C6烷基等。

公开(公告)号：US20110269770A1

公开(公告)日：2011-11-03

申请号：US13120052

申请日：2009-09-23

申请人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

发明人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

IPC分类号： A01N43/58 ,  A01P7/04 ,  A61P33/00 ,  A01P7/00 ,  C07D403/12 ,  A61K31/501

CPC分类号： A01N43/58 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/82 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

摘要： The present invention relates to pyrazole compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a pyrazole radical of formulae A1, A2 or A3, wherein # denotes the binding site; R41, R42, R43, R51 are H, halogen, CN, NO2, C1-C10-alkyl and the like; R52, R53 are H, halogen, CN, NO2, C1-C10-alkyl, and the like; R61, R62, R63 are H, CN, NO2, C1-C10-alkyl, and the like; T is C(Rt) or N; U is C(Ru) or N; V is C(Rv) or N; W is C(Rw) or N; with the proviso that at least one of the groups T, U, V and W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like.The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

摘要翻译： 本发明涉及式I或II的吡唑化合物及其盐和N-氧化物，其中A是式A1，A2和A3的吡唑基，其中＃表示结合位点; R 41，R 42，R 43，R 51为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R 52，R 53为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R61，R62，R63是H，CN，NO2，C1-C10-烷基等; T为C（Rt）或N; U是C（Ru）或N; V是C（Rv）或N; W是C（Rw）或N; 条件是组T，U，V和W中的至少一个为N; R 1，R u，R v，R w为H，卤素，C 1 -C 4 - 烷基等; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等，或R2b和R2c与它们所结合的氮原子一起形成杂环，R2d是C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基等 ; R1为H，CN，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。

公开(公告)号：US20110173726A1

公开(公告)日：2011-07-14

申请号：US13120208

申请日：2009-09-23

申请人： Steffen Groß ,  Karsten Körber ,  Wolfgang Von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

发明人： Steffen Groß ,  Karsten Körber ,  Wolfgang Von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： A01H5/00 ,  A01N43/40 ,  C07D471/04 ,  A01N43/54 ,  C07D487/04 ,  C07D401/14 ,  A01N43/60 ,  A01N43/58 ,  A01N43/84 ,  C07D498/04 ,  A01N43/42 ,  A01P7/00

CPC分类号： A01N43/90 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04

摘要： The present invention relates to a method for controlling invertebrate pests which method comprises treating the pests, their food supply, their habitat or their breeding ground or a plant, seed, soil, area, material or environment in which the pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from pest attack or infestation with a pesticidally effective amount of a pyrazole compound of formulae I or II or a salt or an N-oxide thereof, wherein A is a pyrazole radical of the formulae A1 or A2, wherein # denotes the binding; D is a 5- or 6-membered heterocyclic radical fused to the pyrazole moiety; Rp1, Rp2 and Rpx are H, halogen, CN, NO2, C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, etc.; n is 0 to 4; or two radicals Rpx bound to the same ring-member may form an oxo substituent, or two radicals Rpx bound to adjacent ring-members may form a 3- to 7-membered fused cyclic radical; B is N or CR4, wherein R4 is H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc.; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl, etc.; X2 is O2a, NR2bR2c or S(O)mR2d, wherein m is 0, 1 or 2; R2a is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R1 is H, CN, C1-C10-alkyl, C1-C10-haloalkyl, C3-C10-cycloalkyl, etc.; R2, R3 and R5 are H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc., to a method for protecting plant propagation material and/or the plants which grow threfrom, to plant propagation material comprising at least one compound of formulae I or II, to a method for treating or protecting and animal from infestation or infection by parasites, to novel pyrazole compounds of formulae I or II and agricultural composition containing those compounds.

公开(公告)号：US20100298138A1

公开(公告)日：2010-11-25

申请号：US12600852

申请日：2008-05-23

申请人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

发明人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

IPC分类号： A01C1/06 ,  A01P7/04 ,  A01P7/02 ,  A01P5/00 ,  A01N43/78 ,  A61K31/426 ,  C07D277/18 ,  A61P33/00 ,  C07C335/12 ,  A61K31/17 ,  A01N47/28 ,  C07C69/347 ,  C07C69/708 ,  C07D261/18 ,  A61K31/42 ,  A01N43/80 ,  C07D213/80 ,  A61K31/44 ,  A01N43/40 ,  C07C69/736 ,  A61K31/216 ,  C07C69/78 ,  C07D307/68 ,  A61K31/341 ,  A01N43/08

CPC分类号： C07D261/18 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N47/32 ,  C07C275/26 ,  C07C279/16 ,  C07C335/14 ,  C07C2602/08 ,  C07C2602/10 ,  C07D213/80 ,  C07D233/50 ,  C07D263/28 ,  C07D277/18 ,  C07D317/60

摘要： The present invention relates to the use of aminoazoline and urea derivatives for com-bating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds and to specific azoline and urea derivatives.

摘要翻译： 本发明涉及氨基唑啉和脲衍生物在动物害虫中的应用。 本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽用组合物以及特定的唑啉和脲衍生物来控制动物害虫的方法。

公开(公告)号：US20100167927A1

公开(公告)日：2010-07-01

申请号：US12601017

申请日：2008-05-13

申请人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

发明人： Christopher Koradin ,  Markus Kordes ,  Ernst Baumann ,  Ronan Le Vezouet ,  Deborah L. Culbertson

IPC分类号： A01N25/26 ,  C07C335/12 ,  A01N47/32 ,  A61K31/17 ,  C07D307/82 ,  A61K31/343 ,  C07D333/66 ,  A61K31/381 ,  A61K31/222 ,  C07D311/68 ,  A61K31/353 ,  C07D335/06 ,  A61K31/382 ,  C07D209/40 ,  A61K31/404 ,  C07D215/46 ,  A61K31/47 ,  A61P33/00 ,  A01P7/02 ,  A01P7/04 ,  A01P5/00

CPC分类号： A01N47/36 ,  A01N47/32 ,  C07C335/14 ,  C07C2602/08 ,  C07C2602/10 ,  C07D307/82 ,  C07D333/66

摘要： The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.

摘要翻译： 本发明涉及式（I）的取代的氨基 - 硫脲化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及取代的氨基 - 硫脲化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。 此外，本发明还涉及应用这些化合物的方法。 取代的氨基 - 硫脲化合物由下式（I）定义：其中A，B，R1，R2，R3，R4，R5.1，R5.2和R6如说明书所定义。

公开(公告)号：US20100041700A1

公开(公告)日：2010-02-18

申请号：US12519985

申请日：2007-12-11

申请人： Markus Kordes ,  Ronan Le Vezouet ,  Christopher Koradin ,  Ernst Baumann ,  Deborah L. Culbertson

发明人： Markus Kordes ,  Ronan Le Vezouet ,  Christopher Koradin ,  Ernst Baumann ,  Deborah L. Culbertson

IPC分类号： A01N43/78 ,  C07D417/14 ,  A01N43/42 ,  A01P7/04 ,  A01P5/00

CPC分类号： C07D409/06 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  C07D401/06 ,  C07D405/06 ,  C07D417/12 ,  C07D417/14

摘要： The present invention relates to 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to methods for combating animal pests and to compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds of the general formula (I): wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur, oxygen or NR7, and HetA, HetB and R1 to R7 are defined as in the description.

摘要翻译： 本发明涉及1-（唑啉-2-基） - 氨基-1,2-杂环基 - 乙烷化合物，其可用于防治昆虫，蜘蛛和线虫。 本发明还涉及用于对抗动物害虫的方法和用于对抗动物害虫的组合物。 已经发现可以通过通式（I）的1-（氮杂-2-基） - 氨基-1,2-杂环基 - 乙烷化合物来对抗动物害虫：其中A是式A1或A2的基团 并且其中X是硫，氧或NR 7，并且HetA，HetB和R 1至R 7如描述中所定义。